haloperidol and rimcazole

haloperidol has been researched along with rimcazole in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-19907 (25.00)18.7374
1990's15 (53.57)18.2507
2000's4 (14.29)29.6817
2010's1 (3.57)24.3611
2020's1 (3.57)2.80

Authors

AuthorsStudies
Campbell, BG; Kimes, AS; London, ED; Scheffel, U; Wilson, AA1
Abou-Gharbia, M; Moyer, JA; Muth, EA; Patel, UR1
Abou-Gharbia, M; Andree, TH; Moyer, JA; Muth, EA; Patel, UR; Webb, MB1
Meier, E; Moltzen, EK; Perregaard, J; Sánchez, C1
Meier, E; Moltzen, EK; Perregaard, J1
Baldessarini, RJ; Booth, RG; Charifson, PS; Kula, NS; McPhail, AT; Myers, AM; Owens, CE; Wyrick, SD1
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD1
Lever, JR; Lever, SZ; Nahas, RI1
Agard, DA; Ashworth, A; Barrio-Hernandez, I; Batra, J; Beltrao, P; Bennett, MJ; Bohn, M; Bouhaddou, M; Braberg, H; Broadhurst, DJ; Cai, Y; Cakir, M; Calviello, L; Cavero, DA; Chang, JCJ; Chorba, JS; Craik, CS; d'Enfert, C; Dai, SA; Eckhardt, M; Emerman, M; Fabius, JM; Fletcher, SJ; Floor, SN; Foussard, H; Frankel, AD; Fraser, JS; Fujimori, DG; Ganesan, SJ; García-Sastre, A; Gordon, DE; Gross, JD; Guo, JZ; Haas, K; Haas, P; Hernandez-Armenta, C; Hiatt, J; Huang, XP; Hubert, M; Hüttenhain, R; Ideker, T; Jacobson, M; Jang, GM; Jura, N; Kaake, RM; Kim, M; Kirby, IT; Klippsten, S; Koh, C; Kortemme, T; Krogan, NJ; Kuzuoglu-Ozturk, D; Li, Q; Liboy-Lugo, J; Lin, Y; Liu, X; Liu, Y; Lou, K; Lyu, J; Mac Kain, A; Malik, HS; Mathy, CJP; McGregor, MJ; Melnyk, JE; Memon, D; Meyer, B; Miorin, L; Modak, M; Moreno, E; Mukherjee, S; Naing, ZZC; Noack, J; O'Meara, MJ; O'Neal, MC; Obernier, K; Ott, M; Peng, S; Perica, T; Pilla, KB; Polacco, BJ; Rakesh, R; Rathore, U; Rezelj, VV; Richards, AL; Roesch, F; Rosenberg, OS; Rosenthal, SB; Roth, BL; Roth, TL; Ruggero, D; Safari, M; Sali, A; Saltzberg, DJ; Savar, NS; Schwartz, O; Sharp, PP; Shen, W; Shengjuler, D; Shi, Y; Shoichet, BK; Shokat, KM; Soucheray, M; Stroud, RM; Subramanian, A; Swaney, DL; Taunton, J; Tran, QD; Trenker, R; Tummino, TA; Tutuncuoglu, B; Ugur, FS; Vallet, T; Venkataramanan, S; Verba, KA; Verdin, E; Vignuzzi, M; von Zastrow, M; Wang, HY; Wankowicz, SA; Wenzell, NA; White, KM; Xu, J; Young, JM; Zhang, Z; Zhou, Y1
DeHaven-Hudkins, DL; Fleissner, LC1
DeHaven-Hudkins, DL; Fleissner, LC; Ford-Rice, FY1
Berger, P; Butman, M; Graham, SH; Koistinaho, J; Longo, FM; Noble, L; Sagar, SM; Sharp, FR; Wang, S1
Bissette, G; Levant, B; Nemeroff, CB; Widerlöv, E1
Balestra, B; Candura, SM; Coccini, T; Costa, LG; Iapadre, N; Manzo, L; Tonini, M1
Iwamoto, ET1
Brunn, RD; Mann, JJ; Shaw, ED; Sinsheimer, LM; Weiden, PJ1
Salama, AI; Saller, CF1
Su, TP; Vaupel, DB1
Ford-Rice, FY; London, ED; Schell, SE; Su, TP1
Bastianetto, S; Perrault, G; Sanger, DJ1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
Hara, H; Harada, Y; Sukamoto, T; Tanaka, K1
Kobayashi, T; Matsuno, K; Mita, S1
Kamei, J1
Bridges, S; Miller, C; Thompson, TL1
Kambara, T; Masuzawa, M; Miyamoto, E; Nakao, S; Shingu, K1
Appleyard, MV; Box, G; Campbell, LA; Cooper, MA; Downes, CP; Eccles, S; Ferguson, MJ; Hayes, A; Howie, J; Lambert, JJ; Leslie, NR; McLean, D; McTavish, N; Murray, K; Nutley, B; O'Neill, M; Peters, JA; Prescott, AR; Raynaud, F; Safrany, ST; Samson, J; Spruce, BA; Thompson, AM; Watt, S1
Chen, D; Ding, W; Li, N; Qiao, L; Shi, Y; Sun, Y; Zhang, H; Zhang, Y1

Reviews

1 review(s) available for haloperidol and rimcazole

ArticleYear
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases

1999

Trials

1 trial(s) available for haloperidol and rimcazole

ArticleYear
A case of suicidal and homicidal ideation and akathisia in a double-blind neuroleptic crossover study.
    Journal of clinical psychopharmacology, 1986, Volume: 6, Issue:3

    Topics: Adult; Akathisia, Drug-Induced; Antipsychotic Agents; Carbazoles; Clinical Trials as Topic; Double-Blind Method; Haloperidol; Homicide; Humans; Male; Suicide

1986

Other Studies

26 other study(ies) available for haloperidol and rimcazole

ArticleYear
Radiosynthesis, cerebral distribution, and binding of [125I]-1-(p-iodophenyl)-3-(1-adamantyl)guanidine, a ligand for sigma binding sites.
    Journal of medicinal chemistry, 1992, Dec-11, Volume: 35, Issue:25

    Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Guanidines; Guinea Pigs; Iodobenzenes; Male; Mice; Receptors, sigma; Tissue Distribution

1992
Psychotropic agents: synthesis and antipsychotic activity of substituted beta-carbolines.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:6

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Carbolines; Male; Mice; Rats; Stereotyped Behavior; Structure-Activity Relationship

1987
Antipsychotic activity of substituted gamma-carbolines.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:10

    Topics: Animals; Antipsychotic Agents; Apomorphine; Avoidance Learning; Carbolines; Male; Mice; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Structure-Activity Relationship

1987
Sigma ligands with subnanomolar affinity and preference for the sigma 2 binding site. 1. 3-(omega-aminoalkyl)-1H-indoles.
    Journal of medicinal chemistry, 1995, May-26, Volume: 38, Issue:11

    Topics: Animals; Binding Sites; Indoles; Ligands; Male; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Sensitivity and Specificity; Structure-Activity Relationship

1995
Sigma ligands with subnanomolar affinity and preference for the sigma 2 binding site. 2. Spiro-joined benzofuran, isobenzofuran, and benzopyran piperidines.
    Journal of medicinal chemistry, 1995, May-26, Volume: 38, Issue:11

    Topics: Animals; Benzofurans; Benzopyrans; Binding Sites; Binding, Competitive; Brain; Male; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Sensitivity and Specificity; Structure-Activity Relationship

1995
Conformational analysis, pharmacophore identification, and comparative molecular field analysis of ligands for the neuromodulatory sigma 3 receptor.
    Journal of medicinal chemistry, 1994, Nov-25, Volume: 37, Issue:24

    Topics: Animals; Ligands; Models, Molecular; Molecular Conformation; Receptors, sigma; Rodentia; Structure-Activity Relationship; Tetrahydronaphthalenes

1994
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
    Journal of medicinal chemistry, 1999, Aug-12, Volume: 42, Issue:16

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes

1999
Synthesis and structure-activity relationships of N-(3-phenylpropyl)-N'-benzylpiperazines: Potent ligands for sigma1 and sigma2 receptors.
    Bioorganic & medicinal chemistry, 2008, Jan-15, Volume: 16, Issue:2

    Topics: Combinatorial Chemistry Techniques; Ligands; Molecular Structure; Piperazines; Quantitative Structure-Activity Relationship; Receptors, sigma

2008
A SARS-CoV-2 protein interaction map reveals targets for drug repurposing.
    Nature, 2020, Volume: 583, Issue:7816

    Topics: Animals; Antiviral Agents; Betacoronavirus; Chlorocebus aethiops; Cloning, Molecular; Coronavirus Infections; COVID-19; COVID-19 Drug Treatment; Drug Evaluation, Preclinical; Drug Repositioning; HEK293 Cells; Host-Pathogen Interactions; Humans; Immunity, Innate; Mass Spectrometry; Molecular Targeted Therapy; Pandemics; Pneumonia, Viral; Protein Binding; Protein Biosynthesis; Protein Domains; Protein Interaction Mapping; Protein Interaction Maps; Receptors, sigma; SARS-CoV-2; SKP Cullin F-Box Protein Ligases; Vero Cells; Viral Proteins

2020
Competitive interactions at [3H]1,3-di(2-tolyl)guanidine (DTG)-defined sigma recognition sites in guinea pig brain.
    Life sciences, 1992, Volume: 50, Issue:9

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Carbazoles; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Male; Pentazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma

1992
Characterization of the binding of [3H](+)-pentazocine to sigma recognition sites in guinea pig brain.
    European journal of pharmacology, 1992, Dec-01, Volume: 227, Issue:4

    Topics: Animals; Antipsychotic Agents; Binding Sites; Binding, Competitive; Brain; Carbazoles; Dopamine Agents; Guinea Pigs; Haloperidol; Kinetics; Male; Pentazocine; Piperidines; Receptors, sigma

1992
Haloperidol prevents induction of the hsp70 heat shock gene in neurons injured by phencyclidine (PCP), MK801, and ketamine.
    Journal of neuroscience research, 1992, Volume: 33, Issue:4

    Topics: Amygdala; Animals; Base Sequence; Carbazoles; Cerebral Cortex; Dizocilpine Maleate; Dose-Response Relationship, Drug; Female; Gene Expression; Haloperidol; Heat-Shock Proteins; Humans; Immunohistochemistry; Ketamine; Kinetics; Microscopy, Electron; Molecular Sequence Data; Neurons; Oligodeoxyribonucleotides; Oligonucleotides, Antisense; Phencyclidine; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Reference Values; Restriction Mapping; RNA, Messenger

1992
Alterations in regional brain neurotensin concentrations produced by atypical antipsychotic drugs.
    Regulatory peptides, 1991, Feb-01, Volume: 32, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Carbazoles; Caudate Nucleus; Haloperidol; Male; Neurotensin; Nucleus Accumbens; Radioimmunoassay; Rats; Rats, Inbred Strains; Remoxipride; Sulpiride

1991
Two subtypes of enteric non-opioid sigma receptors in guinea-pig cholinergic motor neurons.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Carbazoles; Dextromethorphan; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Motor Neurons; Myenteric Plexus; Parasympathetic Nervous System; Phenazocine; Pyrimidines; Receptors, Opioid; Receptors, sigma

1991
Evidence for a model of activation of central sigma systems.
    Life sciences, 1989, Volume: 44, Issue:21

    Topics: Animals; Benzazepines; Benzomorphans; Butaclamol; Carbazoles; Dopamine Antagonists; Haloperidol; Kinetics; Male; Models, Biological; Motor Activity; Naltrexone; Narcotic Antagonists; Phenazocine; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Sulpiride

1989
3-Methoxytyramine accumulation: effects of typical neuroleptics and various atypical compounds.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 334, Issue:2

    Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Buspirone; Carbazoles; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Fluphenazine; Haloperidol; Male; Molindone; Pargyline; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Regression Analysis

1986
Guinea-pig vas deferens preparation may contain both receptors and phencyclidine receptors.
    European journal of pharmacology, 1987, Jul-02, Volume: 139, Issue:1

    Topics: Animals; Antipsychotic Agents; Carbazoles; Electric Stimulation; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pentazocine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Vas Deferens

1987
Correlation of inhibitory potencies of putative antagonists for sigma receptors in brain and spleen.
    European journal of pharmacology, 1988, Apr-13, Volume: 148, Issue:3

    Topics: Animals; Antipsychotic Agents; Brain Chemistry; Carbazoles; Guinea Pigs; Haloperidol; In Vitro Techniques; Isoquinolines; Male; Phenazocine; Piperazines; Pyrimidines; Receptors, Opioid; Receptors, sigma; Spleen; Tritium

1988
Pharmacological evidence for the involvement of sigma sites in DTG-induced contralateral circling in rats.
    Neuropharmacology, 1995, Volume: 34, Issue:1

    Topics: Animals; Anticonvulsants; Behavior, Animal; Carbazoles; Dose-Response Relationship, Drug; Guanidines; Haloperidol; Injections, Spinal; Male; Motor Activity; Phenazocine; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, sigma; Salicylamides

1995
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
Sigma receptor-mediated effects of a new antiulcer agent, KB-5492, on experimental gastric mucosal lesions and gastric alkaline secretion in rats.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:2

    Topics: Animals; Anti-Ulcer Agents; Autoradiography; Carbazoles; Ethanol; Gastric Mucosa; Guanidines; Haloperidol; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stomach Ulcer; Stress, Physiological

1994
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:1

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens

1996
Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands.
    Neuroscience letters, 2001, Oct-26, Volume: 312, Issue:3

    Topics: Animals; Antipsychotic Agents; Carbazoles; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Haloperidol; Ligands; Neurons; Nomifensine; Nucleus Accumbens; Phenazocine; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, sigma; Spiperone; Sulpiride; Synaptosomes; Tritium

2001
Ketamine-induced c-Fos expression in the mouse posterior cingulate and retrosplenial cortices is mediated not only via NMDA receptors but also via sigma receptors.
    Brain research, 2002, Feb-01, Volume: 926, Issue:1-2

    Topics: Animals; Anticonvulsants; Carbazoles; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Gyrus Cinguli; Haloperidol; Ketamine; Male; Mice; Mice, Inbred Strains; Mice, Knockout; Presynaptic Terminals; Proto-Oncogene Proteins c-fos; Receptors, N-Methyl-D-Aspartate; Receptors, sigma

2002
Small molecule antagonists of the sigma-1 receptor cause selective release of the death program in tumor and self-reliant cells and inhibit tumor growth in vitro and in vivo.
    Cancer research, 2004, Jul-15, Volume: 64, Issue:14

    Topics: Animals; Antineoplastic Agents; Apoptosis; Breast Neoplasms; Calcium Signaling; Carbazoles; Caspases; Cattle; Cell Division; Cell Line, Tumor; Enzyme Activation; Ethylenediamines; Haloperidol; Humans; Isoenzymes; Lung Neoplasms; Male; Mice; Mice, Nude; Phospholipase C delta; Piperazines; Prostatic Neoplasms; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Receptors, sigma; Sigma-1 Receptor; Type C Phospholipases; Xenograft Model Antitumor Assays

2004
Sigma-1 receptor agonists provide neuroprotection against gp120 via a change in bcl-2 expression in mouse neuronal cultures.
    Brain research, 2012, Jan-11, Volume: 1431

    Topics: Animals; Apoptosis; bcl-2-Associated X Protein; Brain; Carbazoles; Cell Survival; Cells, Cultured; DNA Fragmentation; Dose-Response Relationship, Drug; Embryo, Mammalian; Gene Expression Regulation; Haloperidol; HIV Envelope Protein gp120; Mice; Mice, Inbred BALB C; Microtubule-Associated Proteins; Neurites; Neurons; Neuroprotective Agents; Proto-Oncogene Proteins c-bcl-2; Receptors, sigma; RNA, Messenger; Sigma-1 Receptor; Statistics, Nonparametric

2012