haloperidol has been researched along with quinpirole in 193 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 36 (18.65) | 18.7374 |
1990's | 92 (47.67) | 18.2507 |
2000's | 34 (17.62) | 29.6817 |
2010's | 28 (14.51) | 24.3611 |
2020's | 3 (1.55) | 2.80 |
Authors | Studies |
---|---|
Andrieux, M; Besançon, R; Giros, B; Martres, MP; Pilon, C; Schwartz, JC; Sokoloff, P | 1 |
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P | 1 |
Chio, CL; Ensinger, HA; Huff, RM; Lajiness, ME; Mierau, J; Schneider, FJ | 1 |
Foulon, C; Kung, HF; Kung, MP | 1 |
Berardi, F; Colabufo, NA; Contino, M; Lacivita, E; Leopoldo, M; Perrone, R | 1 |
Allouchi, H; Argiolas, A; El Hakmaoui, A; Enguehard-Gueiffier, C; Gmeiner, P; Gueiffier, A; Hübner, H; Melis, MR | 1 |
Berardi, F; Contino, M; De Giorgio, P; Lacivita, E; Leopoldo, M; Perrone, R | 1 |
Babic, S; Calvin, W; Cui, J; Luedtke, RR; Mach, RH; Taylor, M; Vangveravong, S; Xu, J | 1 |
Cui, J; Ho, D; Li, S; Luedtke, RR; Mach, RH; Taylor, M; Tu, Z; Xu, J | 1 |
Gmeiner, P; Götz, A; Hübner, H; Kühhorn, J; Thompson, D; Whistler, J | 1 |
Gmeiner, P; Hübner, H; Kling, RC; Leuner, K; Möller, D; Skultety, M | 1 |
Guo, L; Huang, J; Li, Z; Liu, H; Sun, H; Zhen, X; Zhou, S; Zhou, Y | 1 |
Bernhardt, G; Biselli, S; Bresinsky, M; Buschauer, A; Forster, L; Honisch, C; Pockes, S; Tropmann, K | 1 |
Cheng, J; Fan, L; Liu, R; Tan, L; Wang, H; Wang, S; Yan, W; Yu, J | 1 |
Destrade, C; Messier, C; Mrabet, O | 1 |
Damsma, G; De Boer, P; Schram, Q; Stoof, JC; Westerink, BH; Zaagsma, J | 1 |
Bernardi, G; Calabresi, P; De Murtas, M; Mercuri, NB | 1 |
LaHoste, GJ; Marshall, JF | 1 |
Akaoka, H; Buda, M; Charléty, P; Chouvet, G; Saunier, CF | 1 |
Gerlach, J; Lublin, H; Peacock, L | 1 |
Levin, ED; Rose, JE | 1 |
Artz, MT; Cools, AR; Ellenbroek, BA | 1 |
Edinger, H; Siegel, A; Sweidan, S | 1 |
Berry, SA; Gudelsky, GA | 1 |
Cory-Slechta, DA; Widzowski, DV | 1 |
Guenaneche, F; Lefebvre, RA; Schuurkes, JA | 1 |
Eichelman, B; Pucilowski, O | 1 |
Geyer, MA; Paulus, MP | 1 |
Abraini, JH; Rostain, JC; Tomei, C | 1 |
Schaus, JM; Seeman, P | 1 |
Brent, PJ | 1 |
Miller, JC | 1 |
Gonon, F; Ponec, J; Suaud-Chagny, MF | 1 |
Courtney, ND; Howlett, AC; Westfall, TC | 1 |
Goldberg, SR; Schindler, CW; Tella, SR; Witkin, JM | 1 |
Axelrod, J; Briley, EM; Felder, CC; Kanterman, RY; Mahan, LC; Monsma, FJ; Sibley, DR | 1 |
Glowinski, J; Godbout, R; Mantz, J; Pirot, S; Thierry, AM | 1 |
Linseman, MA | 1 |
Altar, CA; Jiang, LH; Kasser, RJ; Wang, RY | 1 |
Bruno, JP; Hadjiconstantinou, M; Weihmuller, FB | 1 |
Altar, CA; Boyar, WC; Kim, HS | 1 |
Bunney, BS; Shi, WS | 1 |
Appel, JB; Callahan, PM; Cunningham, KA | 2 |
Bull, DR; Humphrey, PP; Kruk, ZL; Millar, J; Palij, P; Sheehan, MJ; Stamford, J | 1 |
Dowling, JE; Rodrigues, Pdos S | 1 |
Barnes, DE; Bellows, EP; Csernansky, JG; Lombrozo, L | 1 |
Freedman, JE; Weight, FF | 1 |
de Chaffoy de Courcelles, D; Eens, A; Gommeren, W; Janssen, PA; Leysen, JE; Stoof, JC | 1 |
Adamovage, LA; Kreamer, LD; Salama, AI; Saller, CF | 1 |
Bijak, M; Smiałowski, A | 2 |
McKenzie, GM; Warenycia, MW | 1 |
Farah, JM; Mueller, GP | 1 |
Ashby, CR; Hitzemann, R; Rubinstein, JE; Wang, RY | 1 |
Asin, KE; Montana, WE | 1 |
Chiodo, LA; Freeman, AS; Kelland, MD | 1 |
Hu, XT; Wang, RY | 1 |
Dimpfel, W; Koch, R; Schatton, W; Spüler, M | 1 |
Gerlach, J; Kistrup, K | 1 |
Fitten, J; Gordon, LI; Kodama, CK; Menon, MK | 1 |
Ahlenius, S; Criborn, CO; Hillegaart, V; Muren, A | 1 |
Di Chiara, G; Imperato, A | 1 |
Ellison, G; Gunne, L; Johansson, P; Levin, E; See, R | 1 |
Bradshaw, CM; Sheridan, RD; Szabadi, E | 1 |
Bergstrom, DA; Carlson, JH; Walters, JR | 1 |
Cubeddu, LX; Hoffmann, IS; Talmaciu, RK | 2 |
Altar, CA; Boyar, WC | 1 |
Appel, JB; Weathersby, RT | 1 |
Caporali, MG; Ongini, E | 1 |
Ahlenius, S; Fernández-Guasti, A; Hjorth, S; Larsson, K | 1 |
Millington, WR; Mueller, GP; O'Donohue, TL | 1 |
Heikkila, RE; Manzino, L; Sonsalla, PK | 1 |
Cameron, DL; Crocker, AD | 1 |
Burchill, SA; Thody, AJ | 1 |
Gerlach, J; Lublin, H | 1 |
Anderson, D; Gordon, J; Herbster, G; Koller, W; Wack, R | 1 |
Jenks, BG; Tonon, MC; Vaudry, H; Verburg-Van Kemenade, BM | 1 |
Breese, GR; Mueller, RA; Napier, TC | 1 |
Baumeister, A; Breese, GR; Frye, GD; Mueller, RA; Napier, TC | 1 |
Ahlenius, S; Larsson, K | 1 |
Chio, CL; Drong, RF; Gill, GS; Huff, RM; Riley, DT; Slightom, JL | 1 |
Middlemiss, DN; Reavill, C; Storey, VJ | 1 |
Diaz, J; Dimitriadou, V; Griffon, N; Lammers, CH; Levesque, D; Martres, MP; Pilon, C; Schwartz, JC; Sokoloff, P | 1 |
Artigas, F; Ferré, S | 1 |
Barrett, RJ; Caul, WF; Huffman, EM; Jones, JR; Strand, EJ | 1 |
Castellano, C; Cestari, V; Mele, A; Oliverio, A | 1 |
Barrett, JE; Rosenzweig-Lipson, S | 1 |
Bodnar, RJ; Hobbs, DJ; Koch, JE | 1 |
Bodnar, RJ; Koch, JE; Schaefer, LA | 1 |
Swerdlow, NR; Wan, FJ | 1 |
Katz, JL; Witkin, JM | 1 |
Goldstein, M; Ogren, SO | 1 |
Hashimoto, T; Obata, K; Stork, O | 2 |
Schmidt, WJ; Zadow, B | 1 |
Bernard, A; Cavegn, C; Chabert, C; Mills, A | 1 |
Bennett, JP; Richard, MG | 1 |
Mittleman, G; Rosner, AL; Schaub, CL | 1 |
Hasegawa, T; Kameyama, T; Kinoshita, H; Nabeshima, T; Yamamoto, I | 1 |
Burnham, P; Louis, JC; Magal, E; Varon, S | 1 |
Chase, TN; Marin, C | 1 |
Dietze, S; Kleim, J; Kuschinsky, K; Welsch-Kunze, S | 1 |
Kameyama, T; Mori, E; Ukai, M | 1 |
Dorsa, DM; Merchant, KM | 1 |
Landwehrmeyer, B; Mengod, G; Palacios, JM | 1 |
Lamm, MC; Russell, VA; Taljaard, JJ | 1 |
Ichihara, K; Kameyama, T; Nabeshima, T | 1 |
Gerlach, J; Peacock, L | 1 |
Lundström, J; Nilsson, LB; Ogren, SO; Widman, M | 1 |
Abercrombie, ED; DeBoer, P | 1 |
Ellerbrock, BR; Sethy, VH; Wu, H | 1 |
Cabib, S; Caccia, S; Castellano, C; Felici, A; Mele, A; Oliverio, A | 1 |
Bargas, J; Galarraga, E; Hernández-López, S; Pacheco-Cano, MT; Tapia, D | 1 |
Alzheimer, C; Chesi, AJ; Feasey-Truger, KJ; ten Bruggencate, G | 1 |
Desiraju, T; Raju, TR; Singh, J | 1 |
Ellerbrock, BR; Fici, GJ; Sethy, VH; Wu, H | 1 |
Obuchowicz, E | 2 |
Ishibashi, T; Ishida, K; Nakamura, M; Ohno, Y | 1 |
Griffon, N; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P | 1 |
Inoue, A; Kikuchi, T; Miki, S; Misu, Y; Morita, S; Nakata, Y; Seto, M; Ueda, H | 1 |
Cho, S; Hadjiconstantinou, M; Neff, NH | 1 |
Hoffmann, WE; Hyslop, DK; Piercey, MF | 1 |
Marin, C; Tolosa, E | 1 |
Abercrombie, ED; DeBoer, P; Heeringa, MJ | 1 |
Mohell, N | 1 |
Dalia, A; Uretsky, NJ; Wallace, LJ | 1 |
Davidkova, G; Morabito, M; Weiss, B; Zhang, SP; Zhou, LW | 1 |
Barrientos, A; Cardellach, F; Casademont, J; Gómez, M; Marín, C; Miró, O; Nunes, V; Tolosa, E; Urbano-Márquez, A | 1 |
Goeders, NE; Ikemoto, S | 1 |
Grace, AA; Lavin, A | 1 |
Pehek, EA | 1 |
Fass, DM; Levitan, ES; Mains, RE; Takimoto, K | 1 |
Annoh, N; Harano, M; Tanaka, M; Yamada, S | 1 |
Maj, J; Rogóz, Z; Skuza, G | 1 |
Adachi, K; Cools, AR; Hasegawa, M; Hirose, N; Ikeda, H; Koshikawa, N; Sato, M | 1 |
Alper, RH; Gilliland, SL; Levant, B | 1 |
Armogida, M; Chiacchio, S; Colzi, A; Corsini, GU; DeMontis, MG; Maggio, R; Scarselli, M | 1 |
Bonci, A; Malenka, RC; Thomas, MJ | 1 |
Hillefors, M; von Euler, G | 1 |
Moore, CC; Smith, B; Thompson, TL | 1 |
Kung, MP; Sankoorikal, EB; Sasaoka, T; Tonegawa, S; Wang, Y; Xu, R | 1 |
Baik, JH; Borrelli, E; Dierich, A; LeMeur, M; Piazza, PV; Picetti, R; Rougé-Pont, F; Usiello, A | 1 |
Badia, A; Clos, MV; García-Sanz, A | 1 |
Corsini, G; Fumagalli, F; Gennarelli, M; Maggio, R; Molteni, R; Racagni, G; Riva, M; Roceri, M | 1 |
Cools, AR; de Bruin, NM; Ellenbroek, BA; Stevens, KE; van Luijtelaar, EL | 1 |
Schlicker, E; Sokoloff, P; Stark, H; Weber, B | 1 |
Devoto, P; Flore, G; Gessa, GL; Pani, L | 1 |
Fraeyman, NH; Vermis, K | 1 |
Lau, YS; Meredith, GE; Petroske, E; Wang, JQ | 1 |
Meredith, GE; Napier, TC; Switzer, RC | 1 |
Al'perina, EL; Cheĭdo, MA; Devoĭno, LV; Gevorgian, MM | 1 |
Axelrod, JD; Barghshoon, S; Chen, CK; Cheyette, BN; Ebert, J; Kovoor, A; Lester, HA; Schwarz, J; Schwarz, S; Seyffarth, P; Simon, MI | 1 |
Copeland, BJ; Hadjiconstantinou, M; Neff, NH | 1 |
Alimohamad, H; Mouyal, J; Rajakumar, N; Rushlow, WJ; Sutton, L | 1 |
Herman, ZS; Krysiak, R; Obuchowicz, E; Smialowska, M; Wieronska, JM | 1 |
Kuhn, CM; Ray, R; Walker, QD | 1 |
Fisone, G; Galdi, S; Greengard, P; Håkansson, K; Hendrick, J; Snyder, G | 1 |
Baella, SA; Crawford, CA; McDougall, SA; Stuebner, NM; Yoshida, ST | 1 |
Claytor, R; Martelle, JL; Nader, MA; Newman, AH; Reboussin, BA; Ross, JT | 1 |
Bezzina, G; Body, S; Bradshaw, CM; Cheung, TH; Fone, KC; Hampson, CL; Szabadi, E | 1 |
Gabriele, J; Mishra, R; N-Marandi, S; Thomas, N | 1 |
Cheido, MA; Idova, GV; Zhukova, EN | 1 |
Amato, D; Borsini, F; Nencini, P; Stasi, MA | 1 |
Benaliouad, F; Kapur, S; Natesan, S; Rompré, PP | 1 |
Li, M; Zhao, C | 2 |
Dunham, JH; Garcia, EL; Hall, RA; Meyer, RC | 1 |
Charntikov, S; Crawford, CA; Der-Ghazarian, T; McDougall, SA; Varela, FA | 1 |
Dubrovina, NI; Kostyunina, NV; Loskutova, LV | 1 |
De Carolis, L; Milella, MS; Nativio, P; Nencini, P; Passarelli, F; Scaccianoce, S; Schepisi, C | 1 |
Akagawa, K; Fujiwara, T; Kofuji, T; Snada, M; Yoshikawa, T | 1 |
Borsini, F; De Carolis, L; Nencini, P; Serlupi-Crescenzi, O; Stasi, MA | 1 |
De Carolis, L; Milella, MS; Nencini, P; Schepisi, C | 1 |
Bini, V; Bortolato, M; Devoto, P; Frau, R; Pillolla, G; Tambaro, S | 1 |
Panagis, G; Rea, E; Schmidt, TT; Shababi-Klein, J; Winter, C | 1 |
Brodnik, Z; Double, M; Jaskiw, GE | 1 |
Abdulla, ZI; Crawford, CA; Kaplan, GJ; Lee, RJ; McDougall, SA; Mohd-Yusof, A | 1 |
Brandao, ML; Muthuraju, S; Nobre, MJ; Saito, VM | 1 |
Creighton, AE; Wilczynski, W | 1 |
Gao, J; Li, M | 1 |
Artigas, F; Bortolozzi, A; Gomez-Sintes, R; Lucas, JJ | 1 |
Amato, D; Carey, RJ; de Souza Silva, MA; Groos, D; Huston, JP; Lauber, AC; Müller, CP; Pum, ME | 1 |
Caraci, F; Cathala, A; Devroye, C; Di Marco, B; Drago, F; Piazza, PV; Spampinato, U | 1 |
Akimoto, N; Furue, H; Ikeda, A; Naitou, K; Nakamori, H; Nozue, Y; Sano, Y; Shiina, T; Shimizu, Y; Yamada, A; Yamamoto, Y; Yokoyama, T | 1 |
Engmann, O; Giralt, A; Girault, JA | 1 |
Cavalli, J; Corvino, ME; Izídio, GS; Marchette, RCN; Pavesi, E; Pértile, RAN; Ramos, A | 1 |
Boeckers, T; Hengerer, B; Nespoli, E; Rizzo, F; Schulze, U | 1 |
Cao, T; Chen, J; Jiang, Y; Waddington, JL; Wang, C; Wang, P; Zhen, X | 1 |
Alemany-González, M; Chanovas, J; Delgado-Sallent, C; Gener, T; Nebot, P; Puig, MV; Tauste Campo, A | 1 |
Kumar Yadav, R; Mallick, BN | 1 |
1 review(s) available for haloperidol and quinpirole
Article | Year |
---|---|
Neurophysiological evidence that D-1 dopamine receptor blockade attenuates postsynaptic but not autoreceptor-mediated effects of dopamine agonists.
Topics: Animals; Apomorphine; Basal Ganglia; Benzazepines; Dextroamphetamine; Dopamine Antagonists; Electrophysiology; Ergolines; Globus Pallidus; Haloperidol; Ketanserin; Neurons; Pergolide; Piperidines; Quinpirole; Rats; Receptors, Dopamine; Substantia Nigra | 1986 |
192 other study(ies) available for haloperidol and quinpirole
Article | Year |
---|---|
Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor.
Topics: Animals; Chlorides; CHO Cells; Cricetinae; Dopamine; Dopamine Agents; Dopamine Antagonists; Guanylyl Imidodiphosphate; Humans; Lithium; Lithium Chloride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sodium Chloride; Sulpiride; Transfection | 1992 |
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.
Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution | 1990 |
Pramipexole binding and activation of cloned and expressed dopamine D2, D3 and D4 receptors.
Topics: Animals; Benzothiazoles; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dopamine Agonists; Humans; Pramipexole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Spiperone; Thiazoles | 1995 |
Synthesis of (R,S)-2'-trans-7-hydroxy-2-[N-n-propyl-N-(3'-iodo-2'- propenyl)-amino]tetralin (trans-7-OH-PIPAT): a new D3 dopamine receptor ligand.
Topics: Binding Sites; Dopamine Agents; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Stereoisomerism; Tetrahydronaphthalenes | 1993 |
First structure-activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure.
Topics: Amides; Animals; CHO Cells; Cricetinae; Cricetulus; Humans; Piperazines; Radioligand Assay; Receptors, Dopamine D3; Stereoisomerism; Structure-Activity Relationship | 2005 |
2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist.
Topics: Animals; Cattle; CHO Cells; Cricetinae; Cricetulus; Erectile Dysfunction; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Imidazoles; Ligands; Male; Mitosis; Penile Erection; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Rats; Receptors, Dopamine D4; Structure-Activity Relationship | 2006 |
Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands with optimal lipophilicity for brain imaging of the dopamine D3 receptor. Part II.
Topics: Amides; Drug Design; Humans; Ligands; Piperazines; Positron-Emission Tomography; Protein Binding; Radiopharmaceuticals; Receptors, Dopamine D3 | 2009 |
Synthesis and characterization of selective dopamine D2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626.
Topics: Adenylyl Cyclases; Benzofurans; Cell Line; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Indoles; Protein Binding; Receptors, Dopamine D2; Thiophenes | 2010 |
Synthesis and pharmacological evaluation of fluorine-containing D₃ dopamine receptor ligands.
Topics: Benzamides; Cyclic AMP; Fluorine; HEK293 Cells; Humans; Ligands; Molecular Conformation; Piperazines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Receptors, sigma; Structure-Activity Relationship | 2011 |
Development of a bivalent dopamine D₂ receptor agonist.
Topics: Animals; Benzamides; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Partial Agonism; HEK293 Cells; Humans; Ligands; Models, Molecular; Piperazines; Protein Multimerization; Radioligand Assay; Receptors, Dopamine D2; Signal Transduction; Structure-Activity Relationship; Swine; Triazoles | 2011 |
Functionally selective dopamine D₂, D₃ receptor partial agonists.
Topics: Animals; Antipsychotic Agents; Arrestins; beta-Arrestin 2; beta-Arrestins; CHO Cells; Cricetulus; Drug Partial Agonism; GTP-Binding Protein alpha Subunits, Gi-Go; HEK293 Cells; Heterocyclic Compounds, 2-Ring; Humans; Mice; Molecular Docking Simulation; Oximes; Piperazines; Pyrazoles; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereoisomerism; Structure-Activity Relationship; Swine | 2014 |
Design, synthesis and evaluation of benzo[a]thieno[3,2-g]quinolizines as novel l-SPD derivatives possessing dopamine D1, D2 and serotonin 5-HT1A multiple action profiles.
Topics: Antipsychotic Agents; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Drug Design; Humans; Molecular Docking Simulation; Protein Binding; Protein Structure, Tertiary; Quinolizines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2014 |
Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H
Topics: Animals; Cells, Cultured; Dopamine Agonists; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; HEK293 Cells; Humans; Ligands; Molecular Structure; Receptors, Dopamine D3; Receptors, Histamine H2; Structure-Activity Relationship | 2021 |
2-Phenylcyclopropylmethylamine Derivatives as Dopamine D
Topics: Animals; Cell Line, Tumor; Disease Models, Animal; Dopamine Agonists; Drug Design; Drug Evaluation, Preclinical; Half-Life; Humans; Mice; Mice, Inbred ICR; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 2021 |
Locomotor bias produced by intra-accumbens injection of dopamine agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dextroamphetamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Injections; Male; Metoclopramide; Mice; Mice, Inbred BALB C; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior | 1992 |
The effect of intrastriatal application of directly and indirectly acting dopamine agonists and antagonists on the in vivo release of acetylcholine measured by brain microdialysis. The importance of the post-surgery interval.
Topics: Acetylcholine; Amphetamine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Indoles; Male; Oxidopamine; Phenanthridines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1992 |
Chronic neuroleptic treatment: D2 dopamine receptor supersensitivity and striatal glutamatergic transmission.
Topics: Aging; Animals; Antipsychotic Agents; Corpus Striatum; Ergolines; Glutamine; Haloperidol; Parasympathomimetics; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, GABA-A; Receptors, Muscarinic; Synaptic Transmission; Time Factors | 1992 |
Dopamine supersensitivity and D1/D2 synergism are unrelated to changes in striatal receptor density.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Oxidopamine; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone; Stereotyped Behavior; Time Factors; Tritium | 1992 |
Inhibition of nigral dopamine neurons by systemic and local apomorphine: possible contribution of dendritic autoreceptors.
Topics: Animals; Apomorphine; Benzazepines; Bicuculline; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Evoked Potentials; gamma-Aminobutyric Acid; Haloperidol; Injections, Intravenous; Lidocaine; Male; Microinjections; Neurons; Phenethylamines; Quinpirole; Rats; Rats, Wistar; Substantia Nigra | 1992 |
Effect of D1 and D2 agonists in primates withdrawn from long-term treatment with haloperidol: the potential role of dopamine D1 receptors in dyskinesia.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Cebus; Dopamine Agents; Dyskinesia, Drug-Induced; Ergolines; Female; Grooming; Haloperidol; Hypnotics and Sedatives; Male; Motor Activity; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Substance Withdrawal Syndrome | 1992 |
Interactive effects of D1 and D2 agonists with scopolamine on radial-arm maze performance.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cognition; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Exploratory Behavior; Female; Haloperidol; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Scopolamine | 1991 |
The involvement of dopamine D1 and D2 receptors in the effects of the classical neuroleptic haloperidol and the atypical neuroleptic clozapine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Clozapine; Dopamine Agents; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1991 |
D2 dopamine receptor-mediated mechanisms in the medial preoptic-anterior hypothalamus regulate effective defense behavior in the cat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Affect; Aggression; Analysis of Variance; Animals; Apomorphine; Benzazepines; Cats; Dopamine Agents; Dose-Response Relationship, Drug; Electric Stimulation; Ergolines; Female; Haloperidol; Hypothalamus, Anterior; Male; Organ Specificity; Preoptic Area; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1991 |
Effect of D2 dopamine agonists on tuberoinfundibular dopamine neurons.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Arcuate Nucleus of Hypothalamus; Benzazepines; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Neurons; Quinolines; Quinpirole; Rats; Rats, Inbred Strains | 1991 |
Low level lead exposure increases sensitivity to the stimulus properties of dopamine D1 and D2 agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Cocaine; Dextroamphetamine; Discrimination Learning; Dizocilpine Maleate; Dopamine Agents; Drug Synergism; Ergolines; Generalization, Psychological; Haloperidol; Lead; Male; Morphine; N-Methylaspartate; Pentobarbital; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid; Receptors, Opioid, mu | 1991 |
Influence of fenoldopam and quinpirole in the guinea-pig stomach.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Clonidine; Dopamine; Dopamine Agents; Electric Stimulation; Ergolines; Female; Fenoldopam; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Methysergide; Muscle Contraction; Muscle Relaxation; Prazosin; Quinpirole; Stomach; Yohimbine | 1991 |
Diltiazem suppresses quinpirole-induced oral stereotypies in haloperidol withdrawn rats.
Topics: Analysis of Variance; Animals; Diltiazem; Dopamine Agents; Dyskinesia, Drug-Induced; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substance Withdrawal Syndrome | 1991 |
A scaling approach to find order parameters quantifying the effects of dopaminergic agents on unconditioned motor activity in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Cocaine; Dextroamphetamine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Haloperidol; Motor Activity; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Yawning | 1991 |
Role of dopamine receptors in the occurrence of the behavioral motor disturbances in rats exposed to high pressure.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Atmospheric Pressure; Behavior, Animal; Dopamine Agents; Epilepsies, Myoclonic; Ergolines; Haloperidol; High Pressure Neurological Syndrome; Injections, Intraventricular; Male; Motor Activity; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Tremor | 1991 |
Dopamine receptors labelled by [3H]quinpirole.
Topics: Animals; Corpus Striatum; Dogs; Dopamine Agents; Dopamine Antagonists; Ergolines; Guanine Nucleotides; Haloperidol; In Vitro Techniques; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1991 |
Similar behavioural effects of sigma agonists and PCP-like non-competitive NMDA antagonists in guinea-pigs.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Dizocilpine Maleate; Dopamine Agents; Dopamine Antagonists; Ergolines; Female; Guanidines; Guinea Pigs; Haloperidol; Ketamine; Male; Motor Activity; N-Methylaspartate; Pentazocine; Phenazocine; Phencyclidine; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride | 1991 |
Induction of c-fos mRNA expression in rat striatum by neuroleptic drugs.
Topics: Animals; Antipsychotic Agents; Butaclamol; Corpus Striatum; DNA-Binding Proteins; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Quinpirole; Rats; Rats, Inbred Strains; RNA, Messenger; Stereoisomerism | 1990 |
Presynaptic autoinhibition of the electrically evoked dopamine release studied in the rat olfactory tubercle by in vivo electrochemistry.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dopamine; Electric Stimulation; Ergolines; Evoked Potentials; Haloperidol; Male; Microelectrodes; Olfactory Bulb; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Secretory Rate; Sulpiride | 1991 |
Dopaminergic regulation of dopamine release from PC12 cells via a pertussis toxin-sensitive G protein.
Topics: Adrenal Gland Neoplasms; Animals; Apomorphine; Cell Line; Dopamine; Dopamine Antagonists; Ergolines; GTP-Binding Proteins; Haloperidol; Nicotine; Pertussis Toxin; Pheochromocytoma; Potassium; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Virulence Factors, Bordetella | 1991 |
Interaction of haloperidol and SCH 23390 with cocaine and dopamine receptor subtype-selective agonists on schedule-controlled behavior of squirrel monkeys.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Cocaine; Conditioning, Operant; Ergolines; Female; Haloperidol; Male; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Saimiri | 1991 |
Transfected D2 dopamine receptors mediate the potentiation of arachidonic acid release in Chinese hamster ovary cells.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Apomorphine; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine; Drug Synergism; Ergolines; Haloperidol; In Vitro Techniques; Melitten; Pertussis Toxin; Protein Kinase C; Quinpirole; Receptors, Dopamine; Sulpiride; Tetradecanoylphorbol Acetate; Transfection; Virulence Factors, Bordetella | 1991 |
Inhibitory influence of the mesocortical dopaminergic neurons on their target cells: electrophysiological and pharmacological characterization.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine; Electric Stimulation; Ergolines; Frontal Lobe; Haloperidol; Iontophoresis; Isoproterenol; Male; Norepinephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Sulpiride | 1991 |
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone | 1990 |
One year of continuous treatment with haloperidol or clozapine fails to induce a hypersensitive response of caudate putamen neurons to dopamine D1 and D2 receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Oral; Animals; Clozapine; Dibenzazepines; Dopamine Agents; Drug Interactions; Ergolines; Haloperidol; Male; Neurons; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1990 |
Dopamine receptors and sensorimotor behavior in MPTP-treated mice.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arousal; Benzazepines; Discrimination Learning; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Mice; Mice, Inbred Strains; Motor Activity; Orientation; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1990 |
Discriminatory roles for D1 and D2 dopamine receptor subtypes in the in vivo control of neostriatal cyclic GMP.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Cyclic GMP; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Haloperidol; Male; Mice; Quinpirole; Receptors, Dopamine; Sulpiride | 1990 |
Neurotensin attenuates dopamine D2 agonist quinpirole-induced inhibition of midbrain dopamine neurons.
Topics: Animals; Cerebral Ventricles; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Injections, Intraventricular; Male; Mesencephalon; Neurons; Neurotensin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Substantia Nigra; Tegmentum Mesencephali | 1990 |
Dopamine D1 and D2 mediation of the discriminative stimulus properties of d-amphetamine and cocaine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Dextroamphetamine; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Ergolines; Generalization, Psychological; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1991 |
Presynaptic regulation of dopamine release in corpus striatum monitored in vitro in real time by fast cyclic voltammetry.
Topics: Animals; Corpus Striatum; Dopamine; Electric Stimulation; Electrochemistry; Ergolines; Haloperidol; In Vitro Techniques; Nerve Endings; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2 | 1990 |
Dopamine induces neurite retraction in retinal horizontal cells via diacylglycerol and protein kinase C.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alkaloids; Animals; Axons; Benzazepines; Catfishes; Cells, Cultured; Diglycerides; Dopamine; Ergolines; Haloperidol; Kainic Acid; Kinetics; Protein Kinase C; Quinpirole; Receptors, Dopamine; Retina; Staurosporine; Tetradecanoylphorbol Acetate | 1990 |
Sensitization versus tolerance to the dopamine turnover-elevating effects of haloperidol: the effect of regular/intermittent dosing.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Brain Chemistry; Corpus Striatum; Dopamine; Drug Tolerance; Ergolines; Haloperidol; Homovanillic Acid; Male; Motor Activity; Nucleus Accumbens; Olfactory Bulb; Quinpirole; Rats; Rats, Inbred Strains | 1990 |
Single K+ channels activated by D2 dopamine receptors in acutely dissociated neurons from rat corpus striatum.
Topics: Action Potentials; Animals; Corpus Striatum; Electric Conductivity; Ergolines; Haloperidol; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Neurons; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2 | 1988 |
Biochemical profile of risperidone, a new antipsychotic.
Topics: Animals; Antipsychotic Agents; Blood Platelets; Cerebral Cortex; Dopamine; Ergolines; Female; Haloperidol; Isoxazoles; Models, Molecular; Norepinephrine; Oxazoles; Phosphatidic Acids; Piperidines; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Serotonin; Risperidone; Ritanserin; X-Ray Diffraction | 1988 |
Dopamine receptor occupancy in vivo: measurement using N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Clozapine; Corpus Striatum; Ergolines; Haloperidol; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1989 |
Functional supersensitivity of the hippocampal dopaminergic system after prolonged treatment with haloperidol.
Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Hippocampus; In Vitro Techniques; Male; Neurons; Quinpirole; Rats; Rats, Inbred Strains; Sulpiride; Time Factors | 1989 |
Pharmacological activity profiles of dopamine D-1 and D-2 reception agonists and antagonists on striatal neuronal activity and the response to dexamphetamine in freely moving rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Corpus Striatum; Dextroamphetamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Male; Neurons; Quinpirole; Rats; Sulpiride | 1989 |
A D-2 dopaminergic agonist stimulates secretion of anterior pituitary immunoreactive beta-endorphin in rats.
Topics: Animals; beta-Endorphin; Chromatography, Gel; Culture Techniques; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Pituitary Gland, Anterior; Prolactin; Quinpirole; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors | 1989 |
One year treatment with haloperidol or clozapine fails to alter neostriatal D1- and D2-dopamine receptor sensitivity in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Colforsin; Corpus Striatum; Cyclic AMP; Dibenzazepines; Drug Synergism; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1989 |
Studies on D1 and D2 dopamine receptor involvement in conditioned taste aversions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cerebral Ventricles; Conditioning, Classical; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Taste | 1989 |
(+/-)-3,4-Methylenedioxymethamphetamine-induced changes in the basal activity and pharmacological responsiveness of nigrostriatal dopamine neurons.
Topics: 3,4-Methylenedioxyamphetamine; Amphetamines; Animals; Apomorphine; Biogenic Amines; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; N-Methyl-3,4-methylenedioxyamphetamine; Neurons; Quinpirole; Rats; Rats, Inbred Strains; Serotonin; Substantia Nigra | 1989 |
Haloperidol and clozapine: differential effects on the sensitivity of caudate-putamen neurons to dopamine agonists and cholecystokinin following one month continuous treatment.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Benzazepines; Cholecystokinin; Clozapine; Corpus Striatum; Dibenzazepines; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sincalide | 1989 |
Radioelectroencephalographic comparison of memantine with receptor-specific drugs acting on dopaminergic transmission in freely moving rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amantadine; Animals; Benzazepines; Brain; Corpus Striatum; Electroencephalography; Ergolines; Evoked Potentials; Frontal Lobe; Haloperidol; Hippocampus; Male; Memantine; Quinpirole; Rats; Rats, Inbred F344; Receptors, Dopamine; Reticular Formation; Synaptic Transmission; Telemetry | 1987 |
Selective D1 and D2 receptor manipulation in Cebus monkeys: relevance for dystonia and dyskinesia in humans.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biperiden; Cebus; Dystonia; Ergolines; Haloperidol; Male; Movement Disorders; Quinpirole; Raclopride; Receptors, Dopamine; Salicylamides; Stereotyped Behavior | 1987 |
Influence of D-1 receptor system on the D-2 receptor-mediated hypothermic response in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1988 |
Effects of lisuride and quinpirole on convulsions induced by hyperbaric oxygen in the mouse.
Topics: Animals; Body Temperature; Diazepam; Dopamine Agents; Drug Interactions; Ergolines; Haloperidol; Hyperbaric Oxygenation; Lisuride; Lung Volume Measurements; Male; Mice; Mice, Inbred CBA; Quinpirole; Seizures | 1988 |
Effects of locally applied D-1 and D-2 receptor agonists and antagonists studied with brain dialysis.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Azepines; Benzazepines; Brain; Dialysis; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1988 |
Chronic neuroleptics alter the effects of the D1 agonist SK&F 38393 and the D2 agonist LY171555 on oral movements in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Behavior, Animal; Benzazepines; Dopamine Agents; Ergolines; Female; Fluphenazine; Haloperidol; Mouth; Quinpirole; Rats; Rats, Inbred Strains | 1988 |
Excitatory neuronal responses to dopamine in the cerebral cortex: involvement of D2 but not D1 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetite Depressants; Benzazepines; Cerebral Cortex; Dopamine; Ergolines; Haloperidol; In Vitro Techniques; Male; Neurons; Phenylephrine; Prazosin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1985 |
Dopamine D1 receptor mediation of the discriminative stimulus properties of SKF 38393.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Discrimination Learning; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1 | 1985 |
Interactions between endogenous dopamine and dopamine agonists at release modulatory receptors: multiple effects of neuronal uptake inhibitors on transmitter release.
Topics: Acetylcholine; alpha-Methyltyrosine; Animals; Apomorphine; Bromocriptine; Cocaine; Corpus Striatum; Dopamine; Electric Stimulation; Ergolines; Haloperidol; In Vitro Techniques; Methyltyrosines; Neurotransmitter Uptake Inhibitors; Nomifensine; Quinpirole; Rabbits; Receptors, Dopamine; Reserpine | 1986 |
Modulation of in vivo dopamine release by D2 but not D1 receptor agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Benzopyrans; Brain; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Homovanillic Acid; Kinetics; Male; Metoclopramide; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1987 |
Dopamine D2 receptor mediation of the discriminative stimulus properties of LY 171555 (quinpirole).
Topics: Animals; Apomorphine; Benzazepines; Discrimination Learning; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2 | 1986 |
Differential effects of dopamine D-1 and D-2 receptor agonists on EEG activity and behaviour in the rabbit.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Electroencephalography; Ergolines; Haloperidol; Male; Quinpirole; Rabbits; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Sulpiride | 1987 |
Separation of dopaminergic and serotonergic inhibitory mechanisms in the mediation of estrogen-induced lordosis behaviour in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Dopamine; Ergolines; Estradiol; Female; Haloperidol; Lisuride; Male; Ovariectomy; Posture; Quinpirole; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Sexual Behavior, Animal; Tetrahydronaphthalenes | 1987 |
Dopaminergic agents selectively alter the post-translational processing of beta-endorphin in the intermediate pituitary of the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; beta-Endorphin; Bromocriptine; Domperidone; Dopamine Antagonists; Ergolines; Haloperidol; Male; Pituitary Gland; Protein Processing, Post-Translational; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1987 |
Interactions of D1 and D2 dopamine receptors on the ipsilateral vs. contralateral side in rats with unilateral lesions of the dopaminergic nigrostriatal pathway.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Basal Ganglia; Benzazepines; Corpus Striatum; Denervation; Dextroamphetamine; Ergolines; Female; Flunarizine; Functional Laterality; Haloperidol; Levodopa; Neural Pathways; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Rotation; Substantia Nigra | 1988 |
Evidence for post-synaptic changes mediating increased behavioural sensitivity to dopamine receptor agonists in hypothyroid rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Brain; Dopamine Antagonists; Ergolines; Haloperidol; Hypothyroidism; Male; Motor Activity; Propylthiouracil; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reference Values; Stereotyped Behavior; Synapses | 1988 |
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride | 1986 |
The effect of acute and prolonged treatment with citalopram on the action of dopamine and SKF 38393 in rat hippocampal slices.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Appetite Depressants; Benzazepines; Citalopram; Dopamine; Ergolines; Haloperidol; Hippocampus; In Vitro Techniques; Male; Motor Activity; Neurons; Propylamines; Quinpirole; Rats; Rats, Inbred Strains; Sulpiride | 1988 |
Behavioural effects of dopamine D-1 and D-2 receptor agonists in monkeys previously treated with haloperidol.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Cebus; Dyskinesia, Drug-Induced; Ergolines; Female; Haloperidol; Quinpirole; Receptors, Dopamine | 1988 |
Quinpirole hydrochloride, a potential anti-parkinsonism drug.
Topics: Animals; Benzazepines; Corpus Striatum; Dogs; Dose-Response Relationship, Drug; Ergolines; Grooming; Haloperidol; Male; Motor Activity; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Sulpiride | 1987 |
Dopamine autoreceptors modulate dopamine release from the prefrontal cortex.
Topics: Animals; Apomorphine; Calcium; Desipramine; Dopamine; Electric Stimulation; Ergolines; Female; Frontal Lobe; Haloperidol; Male; Nomifensine; Quinpirole; Rabbits; Receptors, Dopamine | 1986 |
Characteristics of receptors for dopamine in the pars intermedia of the amphibian Xenopus laevis.
Topics: Animals; Apomorphine; Benzamides; Domperidone; Dopamine; Drug Interactions; Ergolines; Haloperidol; Melanocyte-Stimulating Hormones; Pituitary Gland, Anterior; Quinpirole; Receptors, Dopamine; Sulpiride; Xenopus laevis | 1986 |
Dopamine agonist-induced locomotor activity in rats treated with 6-hydroxydopamine at differing ages: functional supersensitivity of D-1 dopamine receptors in neonatally lesioned rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Age Factors; Animals; Animals, Newborn; Apomorphine; Benzazepines; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Flupenthixol; Haloperidol; Hydroxydopamines; Male; Motor Activity; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1985 |
Evidence that D-1 dopamine receptors contribute to the supersensitive behavioral responses induced by L-dihydroxyphenylalanine in rats treated neonatally with 6-hydroxydopamine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Dihydroxyphenylalanine; Drug Interactions; Ergolines; Female; Flupenthixol; Haloperidol; Hydroxydopamines; Levodopa; Male; Motor Activity; Oxidopamine; Pregnancy; Quinpirole; Rats; Receptors, Dopamine; Self Mutilation; Stereotyped Behavior | 1985 |
Lisuride, LY-141865, and 8-OH-DPAT facilitate male rat sexual behavior via a non-dopaminergic mechanism.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Haloperidol; Lisuride; Male; Naphthalenes; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal; Tetrahydronaphthalenes | 1984 |
D4 dopamine receptor-mediated signaling events determined in transfected Chinese hamster ovary cells.
Topics: Amiloride; Animals; Arachidonic Acid; Base Sequence; Butaclamol; CHO Cells; Cloning, Molecular; Clozapine; Cricetinae; Cyclic AMP; DNA; Dopamine; Dopamine Antagonists; Ergolines; Genes, Synthetic; Haloperidol; Humans; Kinetics; Molecular Sequence Data; Pertussis Toxin; Protein Kinase C; Quinpirole; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Signal Transduction; Sodium-Hydrogen Exchangers; Transfection; Virulence Factors, Bordetella | 1994 |
Effect of haloperidol and (-)-sulpiride on dopamine agonist-induced hypoactivity.
Topics: Animals; Apomorphine; Benzopyrans; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Motor Activity; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Tetrahydronaphthalenes | 1995 |
Novel dopamine receptor subtypes as targets for antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; Bradykinin; Brain; Carbachol; Cell Division; Cyclic AMP; Dopamine; Dopamine Agonists; Ergolines; Gene Expression; Genes, fos; Haloperidol; Humans; Inositol Phosphates; Neurotensin; Oxidopamine; Quinpirole; Receptors, Dopamine; Second Messenger Systems; Signal Transduction; Virulence Factors, Bordetella | 1995 |
Clozapine decreases serotonin extracellular levels in the nucleus accumbens by a dopamine receptor-independent mechanism.
Topics: Animals; Clozapine; Dopamine; Dopamine Agonists; Ergolines; Haloperidol; Microdialysis; Nucleus Accumbens; Quinpirole; Raclopride; Rats; Receptors, Dopamine; Salicylamides; Serotonin; Time Factors | 1995 |
D2-specific discriminative stimuli: parameters, blocking, and rebound.
Topics: Animals; Cues; Discrimination, Psychological; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Food Deprivation; Haloperidol; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Spiperone | 1995 |
Interaction between the NMDA competitive antagonist CPP and the dopaminergic system in one-trial inhibitory avoidance in C57BL/6 mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Avoidance Learning; Brain; Dopamine Agonists; Dose-Response Relationship, Drug; Electroshock; Ergolines; Haloperidol; Male; Mice; Mice, Inbred C57BL; Neural Inhibition; Piperazines; Quinpirole; Reaction Time; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Retention, Psychology | 1995 |
K-channel blockers attenuate the presynaptic effects of the D2/D3 agonist quinpirole in monkeys.
Topics: 4-Aminopyridine; Amodiaquine; Animals; Apamin; Behavior, Animal; Catalepsy; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Potassium Channels; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Presynaptic; Saimiri | 1995 |
Naltrexone, dopamine receptor agonists and antagonists, and food intake in rats: 1. Food deprivation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Eating; Ergolines; Food Deprivation; Haloperidol; Male; Naltrexone; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1994 |
Naltrexone, dopamine receptor agonists and antagonists, and food intake in rats: 2. 2-deoxy-D-glucose.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Deoxyglucose; Dopamine Agonists; Dopamine Antagonists; Eating; Ergolines; Haloperidol; Male; Naltrexone; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1994 |
Intra-accumbens infusion of quinpirole impairs sensorimotor gating of acoustic startle in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acoustic Stimulation; Animals; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Injections; Male; Nucleus Accumbens; Quinpirole; Rats; Rats, Sprague-Dawley; Reflex, Startle | 1993 |
Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Reinforcement Schedule; Saimiri; Spiperone | 1993 |
Phencyclidine- and dizocilpine-induced hyperlocomotion are differentially mediated.
Topics: Analysis of Variance; Animals; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Ergolines; Haloperidol; Male; Motor Activity; Phencyclidine; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Remoxipride; Salicylamides | 1994 |
Haloperidol activates tyrosine hydroxylase gene-expression in the rat substantia nigra, pars reticulata.
Topics: Animals; Benzoxazines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Enzyme Activation; Ergolines; Gene Expression; Haloperidol; Immunohistochemistry; In Situ Hybridization; Male; Oxazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Substantia Nigra; Tyrosine 3-Monooxygenase | 1994 |
The AMPA antagonists NBQX and GYKI 52466 do not counteract neuroleptic-induced catalepsy.
Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Benzodiazepines; Catalepsy; Dizocilpine Maleate; Drug Interactions; Ergolines; Haloperidol; Levodopa; Male; Pilot Projects; Quinoxalines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, AMPA | 1994 |
Characterization of the functional activity of dopamine ligands at human recombinant dopamine D4 receptors.
Topics: Animals; Cell Line; Clozapine; DNA; Dopamine; Dopamine Agents; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Ligands; Moths; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Sulfur Radioisotopes; Tritium | 1994 |
Increase of tyrosine hydroxylase and its mRNA in the rat substantia nigra pars reticulata by diazepam and picrotoxin.
Topics: Animals; Diazepam; Dopamine Agents; Ergolines; Haloperidol; Male; Picrotoxin; Quinpirole; Rats; Rats, Wistar; RNA, Messenger; Substantia Nigra; Tyrosine 3-Monooxygenase | 1994 |
Regulation by D2 dopamine receptors of in vivo dopamine synthesis in striata of rats and mice with experimental parkinsonism.
Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Ergolines; Haloperidol; Hydrazines; Kinetics; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Oxidopamine; Parkinson Disease, Secondary; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reference Values | 1994 |
Polydipsia and dopamine: behavioral effects of dopamine D1 and D2 receptor agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Diazepam; Dopamine Agonists; Dopamine Antagonists; Drinking; Eating; Ergolines; Haloperidol; Male; Motor Activity; Quinpirole; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Thirst | 1994 |
Competitive NMDA antagonists enhance the catalepsy induced by delta 9-tetrahydrocannabinol in mice.
Topics: 2-Amino-5-phosphonovalerate; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amantadine; Amino Acids; Animals; Anticonvulsants; Catalepsy; Dizocilpine Maleate; Dopamine Agonists; Dose-Response Relationship, Drug; Dronabinol; Drug Synergism; Ergolines; Haloperidol; Male; Mice; Mice, Inbred Strains; Motor Activity; Piperazines; Quinpirole; Receptors, N-Methyl-D-Aspartate; Scopolamine | 1994 |
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase | 1993 |
Dopamine D1 receptor stimulation but not dopamine D2 receptor stimulation attenuates haloperidol-induced behavioral supersensitivity and receptor up-regulation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Dopamine Agents; Ergolines; Grooming; Haloperidol; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Up-Regulation | 1993 |
Recordings of extracellular glutamate and gamma-aminobutyric acid in the striatum of non-anesthetized rats. K(+)-stimulation, its Ca(2+)-dependence and lack of effects of drugs acting on dopamine receptors.
Topics: Animals; Apomorphine; Calcium; Corpus Striatum; Dialysis; Ergolines; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Haloperidol; Male; Potassium; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Stimulation, Chemical | 1993 |
Discriminative stimulus properties of cocaine in the rat using a two-choice discrete-trial avoidance paradigm.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Avoidance Learning; Benzazepines; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine Agents; Dose-Response Relationship, Drug; Electroshock; Ergolines; Haloperidol; Male; Methamphetamine; Neurotransmitter Uptake Inhibitors; Piperazines; Quinpirole; Rats; Sulpiride | 1993 |
Differential induction of neurotensin and c-fos gene expression by typical versus atypical antipsychotics.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Atropine; Benzazepines; Corpus Striatum; Ergolines; Gene Expression; Genes; Genes, fos; Haloperidol; In Situ Hybridization; Male; Neurons; Neurotensin; Nucleus Accumbens; Peptide Fragments; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; RNA, Messenger | 1993 |
Dopamine D3 receptor mRNA and binding sites in human brain.
Topics: Aminoquinolines; Binding Sites; Binding, Competitive; Brain Chemistry; Corpus Striatum; DNA; Domperidone; Dopamine; Dopamine Agents; Ergolines; Gene Expression Regulation; Haloperidol; Humans; Nerve Tissue Proteins; Organ Specificity; Protein Binding; Quinpirole; Receptors, Dopamine; RNA, Messenger; Sulpiride | 1993 |
Lack of interaction between alpha 2-adrenoceptors and dopamine D2-receptors in mediating their inhibitory effects on [3H]dopamine release from rat nucleus accumbens slices.
Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Binding, Competitive; Brimonidine Tartrate; Dopamine; Electric Stimulation; Ergolines; GTP-Binding Proteins; Haloperidol; In Vitro Techniques; Male; Nucleus Accumbens; Pergolide; Quinoxalines; Quinpirole; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Dopamine D2; Signal Transduction; Sulpiride | 1993 |
Mediation of dopamine D1 and D2 receptors in the effects of GBR 12909 on latent learning and locomotor activity in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Drinking Behavior; Ergolines; Exploratory Behavior; Haloperidol; Learning; Male; Mice; Mice, Inbred Strains; Motor Activity; Neurotransmitter Uptake Inhibitors; Piperazines; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1993 |
Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.
Topics: Administration, Oral; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Benzothiazoles; Cebus; Disease Models, Animal; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dyskinesia, Drug-Induced; Dystonia; Ergolines; Female; Haloperidol; Lisuride; Male; Piperidines; Pramipexole; Quinpirole; Raclopride; Salicylamides; Thiazoles | 1993 |
Dopamine D2 blocking activity and plasma concentrations of remoxipride and its main metabolites in the rat.
Topics: Animals; Body Temperature; Chromatography, High Pressure Liquid; Dopamine D2 Receptor Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Pergolide; Quinpirole; Rats; Rats, Sprague-Dawley; Remoxipride; Salicylamides | 1993 |
Physiological release of striatal acetylcholine in vivo: modulation by D1 and D2 dopamine receptor subtypes.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Corpus Striatum; Ergolines; Haloperidol; Male; Neostigmine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1996 |
Comparative dopaminergic and muscarinic antagonist activity of clozapine and haloperidol.
Topics: Acetylcholine; Animals; Cerebellum; Clozapine; Corpus Striatum; Cyclic GMP; Dopamine Antagonists; Ergolines; Haloperidol; Male; Mice; Muscarinic Antagonists; Oxotremorine; Quinpirole; Rats; Rats, Sprague-Dawley | 1996 |
Dopamine-N-methyl-D-aspartate interactions in the modulation of locomotor activity and memory consolidation in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Avoidance Learning; Benzazepines; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Haloperidol; Male; Memory; Mice; Mice, Inbred Strains; Motor Activity; Piperazines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Sulpiride | 1996 |
Inhibitory action of dopamine involves a subthreshold Cs(+)-sensitive conductance in neostriatal neurons.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Benzazepines; Cesium; Cyclic AMP; Dopamine; Dopamine Agonists; Electric Stimulation; Electrophysiology; Evoked Potentials; Haloperidol; In Vitro Techniques; Ion Channels; Membrane Potentials; Neostriatum; Neurons; Patch-Clamp Techniques; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride; Tetrodotoxin | 1996 |
Dopamine autoreceptor sensitivity is unchanged in rat nucleus accumbens after chronic haloperidol treatment: an in vivo and in vitro voltammetric study.
Topics: Animals; Autoreceptors; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Nucleus Accumbens; Quinpirole; Rats; Sulpiride; Time Factors | 1995 |
Dose-response functions of apomorphine, SKF 38393, LY 171555, haloperidol and clonidine on the self-stimulation evoked from lateral hypothalamus and ventral tegmentum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apomorphine; Clonidine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electrodes, Implanted; Haloperidol; Hypothalamic Area, Lateral; Male; Medial Forebrain Bundle; Quinpirole; Rats; Rats, Wistar; Self Stimulation; Tegmentum Mesencephali | 1996 |
D2 and D1 dopaminergic activity of 7-OH-DPAT.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Cells, Cultured; Cerebellum; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Indans; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes | 1996 |
Long-term treatment with chlorpromazine and haloperidol but not with sulpiride and clozapine markedly elevates neuropeptide Y-like immunoreactivity in the rat hypothalamus.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Benzazepines; Chlorpromazine; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gene Expression Regulation; Haloperidol; Hypothalamus; Male; Neuropeptide Y; Prazosin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Sulpiride | 1996 |
Effects of SM-9018, a novel 5-HT2 and D2 receptor antagonist, on electrically-evoked [3H]acetylcholine release from rat striatal slices.
Topics: Acetylcholine; Animals; Antipsychotic Agents; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electric Stimulation; Haloperidol; In Vitro Techniques; Indoles; Isoindoles; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Serotonin Antagonists; Thiazoles | 1996 |
Antipsychotics with inverse agonist activity at the dopamine D3 receptor.
Topics: Animals; Antipsychotic Agents; Calcium; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; DNA Replication; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Glioma; Haloperidol; Humans; Hybrid Cells; Naphthalenes; Neuroblastoma; Pertussis Toxin; Phenothiazines; Pimozide; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Risperidone; Salicylamides; Second Messenger Systems; Sulpiride; Tetrahydronaphthalenes; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1996 |
Aripiprazole, a novel antipsychotic drug, inhibits quinpirole-evoked GTPase activity but does not up-regulate dopamine D2 receptor following repeated treatment in the rat striatum.
Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Dopamine Agonists; GTP Phosphohydrolases; Haloperidol; Male; Membranes; Neostriatum; Oligonucleotides, Antisense; Piperazines; Quinolones; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Up-Regulation | 1997 |
Regulation of tyrosine hydroxylase and aromatic L-amino acid decarboxylase by dopaminergic drugs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aromatic-L-Amino-Acid Decarboxylases; Benzazepines; Brain; Bromocriptine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Mesencephalon; Mice; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase | 1997 |
Excitation of type II anterior caudate neurons by stimulation of dopamine D3 receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminoquinolines; Animals; Benzothiazoles; Caudate Nucleus; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Haloperidol; Imidazoles; Neurons; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Tetrahydronaphthalenes; Thiazoles | 1997 |
Striatal synaptophysin levels are not indicative of dopaminergic supersensitivity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Blotting, Western; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Haloperidol; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Synaptophysin | 1997 |
Biochemistry of somatodendritic dopamine release in substantia nigra: an in vivo comparison with striatal dopamine release.
Topics: Amphetamine; Animals; Corpus Striatum; Dendrites; Dopamine; Haloperidol; Nerve Endings; Quinpirole; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Substantia Nigra; Tetrodotoxin | 1998 |
Agonist and inverse agonist activity at the dopamine D3 receptor measured by guanosine 5'--gamma-thio-triphosphate--35S- binding.
Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Mice; Pertussis Toxin; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Tetrahydronaphthalenes; Virulence Factors, Bordetella | 1998 |
Dopaminergic agonists administered into the nucleus accumbens: effects on extracellular glutamate and on locomotor activity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Caffeine; Central Nervous System Stimulants; Dopamine Agonists; Dopamine Antagonists; Glutamic Acid; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Quinpirole; Rats; Rats, Sprague-Dawley; Salicylamides | 1998 |
D2 dopamine antisense RNA expression vector, unlike haloperidol, produces long-term inhibition of D2 dopamine-mediated behaviors without causing Up-regulation of D2 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Catalepsy; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Tolerance; Fluphenazine; Genetic Vectors; Grooming; Haloperidol; Male; Mice; Quinpirole; Receptors, Dopamine D2; RNA, Antisense; Stereotyped Behavior; Up-Regulation | 1998 |
Biochemical and molecular effects of chronic haloperidol administration on brain and muscle mitochondria of rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Brain; DNA, Mitochondrial; Drug Administration Schedule; Haloperidol; Male; Mitochondria; Mitochondria, Muscle; Mutagenesis; Oxygen Consumption; Point Mutation; Protein Biosynthesis; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Sequence Deletion; Time Factors | 1998 |
Microinjections of dopamine agonists and cocaine elevate plasma corticosterone: dissociation effects among the ventral and dorsal striatum and medial prefrontal cortex.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Corpus Striatum; Corticosterone; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Microinjections; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley | 1998 |
Dopamine modulates the responsivity of mediodorsal thalamic cells recorded in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Antipsychotic Agents; Cell Size; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; In Vitro Techniques; Membrane Potentials; Patch-Clamp Techniques; Quinpirole; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Thalamus | 1998 |
Comparison of effects of haloperidol administration on amphetamine-stimulated dopamine release in the rat medial prefrontal cortex and dorsal striatum.
Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Dextroamphetamine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Haloperidol; Male; Microdialysis; Neostriatum; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2 | 1999 |
Tonic dopamine inhibition of L-type Ca2+ channel activity reduces alpha1D Ca2+ channel gene expression.
Topics: Animals; Bromocriptine; Calcium Channels; Calcium Channels, L-Type; Cells, Cultured; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Gene Expression Regulation; Haloperidol; Patch-Clamp Techniques; Pituitary Gland, Posterior; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA, Messenger; Transcription, Genetic | 1999 |
Dopamine D(3) receptors modulate evoked dopamine release from slices of rat nucleus accumbens via muscarinic receptors, but not from the striatum.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; Haloperidol; In Vitro Techniques; Indans; Male; Muscarinic Antagonists; Neostriatum; Nucleus Accumbens; Pirenzepine; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Muscarinic | 1999 |
Differential behavioural effect of quinpirole in neuroleptic-pretreated rats - role of alpha(1)-adrenoceptor.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Behavior, Animal; Chlorpromazine; Dopamine Agonists; Drug Synergism; Haloperidol; Injections, Intraperitoneal; Male; Motor Activity; Prazosin; Quinpirole; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sodium Chloride; Sulpiride | 1999 |
The anticataleptic effect of 7-OH-DPAT: are dopamine D3 receptors involved?
Topics: Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dextroamphetamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Fluphenazine; Haloperidol; Hyperkinesis; Levodopa; Locomotion; Male; Naphthalenes; Pyrrolidines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reserpine; Tetrahydronaphthalenes | 1999 |
Effects of chronic haloperidol and clozapine on vacuous chewing and dopamine-mediated jaw movements in rats: evaluation of a revised animal model of tardive dyskinesia.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Clozapine; Disease Models, Animal; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dyskinesia, Drug-Induced; Haloperidol; Jaw; Male; Mastication; Quinpirole; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Serotonin Antagonists | 1999 |
Pharmacology of quinpirole-stimulated [35S]GTPgammaS binding: discrepancy with receptor binding profile.
Topics: Animals; Benzazepines; Binding, Competitive; Clorgyline; Clozapine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Membranes; Monoamine Oxidase Inhibitors; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Selegiline; Spiperone; Sulfur Radioisotopes; Thiazoles | 2000 |
Reconstitution of functional dopamine D(2s) receptor by co-expression of amino- and carboxyl-terminal receptor fragments.
Topics: Animals; Apomorphine; Binding, Competitive; Clozapine; Colforsin; COS Cells; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gene Expression; Haloperidol; Membranes; Peptide Fragments; Pergolide; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Transfection; Tritium | 2000 |
Modulation of long-term depression by dopamine in the mesolimbic system.
Topics: Animals; Benzazepines; Conditioning, Psychological; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Limbic System; Long-Term Potentiation; Mesencephalon; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Neural Inhibition; Neuronal Plasticity; Neurons; Nucleus Accumbens; Patch-Clamp Techniques; Quinpirole; Salicylamides; Substance-Related Disorders; Sulpiride; Ventral Tegmental Area | 2000 |
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes | 2001 |
Estrogen priming modulates autoreceptor-mediated potentiation of dopamine uptake.
Topics: Animals; Antifungal Agents; Autoreceptors; Benzazepines; Biological Transport; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrogens; Female; Haloperidol; Kinetics; Ovariectomy; Phosphoprotein Phosphatases; Protein Phosphatase 1; Pyrans; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiro Compounds; Synaptosomes; Time Factors | 2000 |
Dopamine D2 long receptor-deficient mice display alterations in striatum-dependent functions.
Topics: Animals; Anxiety; Behavior, Animal; Catalepsy; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gait Disorders, Neurologic; Gene Targeting; Haloperidol; Homozygote; In Vitro Techniques; Male; Maze Learning; Mice; Mice, Knockout; Motor Activity; Mutagenesis, Site-Directed; Protein Isoforms; Psychomotor Performance; Quinpirole; Radioligand Assay; Receptors, Dopamine D2 | 2000 |
Distinct functions of the two isoforms of dopamine D2 receptors.
Topics: Animals; Apomorphine; Benzazepines; Catalepsy; Chimera; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Mice; Mice, Inbred C57BL; Mice, Knockout; Mutagenesis; Protein Isoforms; Quinpirole; Receptors, Dopamine D2; Signal Transduction; Spiperone; Synapses | 2000 |
Differential effect of quinpirole and 7-OH-DPAT on the spontaneous [(3)H]-dopamine efflux from rat striatal synaptosomes.
Topics: Animals; Benzopyrans; Calcium; Calcium Channels; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Neostriatum; Oxazines; Presynaptic Terminals; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Synaptosomes; Tetrahydronaphthalenes; Tetrodotoxin; Tritium | 2001 |
Stimulatory role of dopamine on fibroblast growth factor-2 expression in rat striatum.
Topics: Animals; Apomorphine; Benzazepines; Corpus Striatum; Dizocilpine Maleate; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fibroblast Growth Factor 2; Haloperidol; Male; Nicotine; Nicotinic Agonists; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Stereoisomerism | 2001 |
Hippocampal and cortical sensory gating in rats: effects of quinpirole microinjections in nucleus accumbens core and shell.
Topics: Acoustic Stimulation; Animals; Auditory Perception; Cerebral Cortex; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electroencephalography; Evoked Potentials, Auditory; Haloperidol; Hippocampus; Male; Neural Inhibition; Neural Pathways; Neurons; Nucleus Accumbens; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Schizophrenia | 2001 |
Identification of the dopamine autoreceptor in the guinea-pig retina as D(2) receptor using novel subtype-selective antagonists.
Topics: Animals; Azepines; Binding Sites; CHO Cells; Cricetinae; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guinea Pigs; Haloperidol; Male; Naphthalenes; Norepinephrine; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Retina; Substrate Specificity | 2001 |
Evidence for co-release of noradrenaline and dopamine from noradrenergic neurons in the cerebral cortex.
Topics: 4-Butyrolactone; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cerebellum; Clonidine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Extracellular Space; Haloperidol; Idazoxan; Male; Microdialysis; Motor Cortex; Neurons; Norepinephrine; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Solvents | 2001 |
Cellular activity of dopamine DA2 receptor splice variants and mutants.
Topics: Animals; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Extracellular Space; Genetic Variation; Haloperidol; Humans; Hydrogen-Ion Concentration; Mutation; Protein Kinase C; Quinpirole; Receptors, Dopamine D2 | 2003 |
Elevated neuronal nitric oxide synthase expression in chronic haloperidol-treated rats.
Topics: Animals; Basal Ganglia; Behavior, Animal; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Immunohistochemistry; In Situ Hybridization; Male; Neostriatum; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA, Messenger; Spiperone | 2003 |
Short-term, D2 receptor blockade induces synaptic degeneration, reduces levels of tyrosine hydroxylase and brain-derived neurotrophic factor, and enhances D2-mediated firing in the ventral pallidum.
Topics: Animals; Antipsychotic Agents; Brain-Derived Neurotrophic Factor; Cell Survival; Disease Models, Animal; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Administration Schedule; Dyskinesia, Drug-Induced; Haloperidol; Immunohistochemistry; Male; Microscopy, Electron; Nerve Degeneration; Presynaptic Terminals; Prosencephalon; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Salicylamides; Synaptic Transmission; Tyrosine 3-Monooxygenase | 2004 |
[Contribution of D2 dopamine receptors of the rat dorsolateral caudate nucleus to immunomodulation].
Topics: Adjuvants, Immunologic; Animals; Antibody-Producing Cells; Caudate Nucleus; Dopamine D2 Receptor Antagonists; Erythrocytes; Haloperidol; Immunization; Male; Neuroimmunomodulation; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Sheep | 2004 |
D2 dopamine receptors colocalize regulator of G-protein signaling 9-2 (RGS9-2) via the RGS9 DEP domain, and RGS9 knock-out mice develop dyskinesias associated with dopamine pathways.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Mice; Mice, Knockout; Movement Disorders; Parkinson Disease; Patch-Clamp Techniques; Protein Interaction Mapping; Protein Structure, Tertiary; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, G-Protein-Coupled; Recombinant Fusion Proteins; Reserpine; RGS Proteins; Subcellular Fractions; Sulpiride; Transfection | 2005 |
Enhanced dopamine uptake in the striatum following repeated restraint stress.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenalectomy; Animals; Behavior, Animal; Biogenic Amines; Chromatography, High Pressure Liquid; Corpus Striatum; Corticosterone; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Electrochemistry; Haloperidol; Hormone Antagonists; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mifepristone; Nerve Tissue Proteins; Protein Binding; Quinpirole; Restraint, Physical; RNA, Messenger; Stress, Physiological; Time Factors; Tritium; Tyrosine | 2005 |
The effects of antipsychotics on beta-catenin, glycogen synthase kinase-3 and dishevelled in the ventral midbrain of rats.
Topics: Adaptor Proteins, Signal Transducing; Amphetamine; Animals; Antipsychotic Agents; Benzazepines; beta Catenin; Blotting, Western; Central Nervous System Stimulants; Clozapine; Cytoskeletal Proteins; Dishevelled Proteins; Dopamine Agonists; Female; Glycogen Synthase Kinase 3; Haloperidol; Immunohistochemistry; Intercellular Signaling Peptides and Proteins; Male; Mesencephalon; Phosphoproteins; Quinpirole; Rats; Rats, Sprague-Dawley; Risperidone; Signal Transduction; Trans-Activators; Wnt Proteins; Wnt1 Protein | 2005 |
Alterations in striatal neuropeptide Y system activity of rats with haloperidol-induced behavioral supersensitivity.
Topics: Animals; Behavior, Animal; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Haloperidol; In Situ Hybridization; Male; Motor Activity; Neuropeptide Y; Quinpirole; Rats; Rats, Wistar; RNA, Messenger | 2005 |
Sex differences in neurochemical effects of dopaminergic drugs in rat striatum.
Topics: Analysis of Variance; Animals; Brain Chemistry; Cocaine; Corpus Striatum; Dopamine; Dopamine Agents; Dose-Response Relationship, Radiation; Electric Stimulation; Electrochemistry; Female; Haloperidol; Male; Quinpirole; Rats; Sex Characteristics; Synaptosomes; Time Factors | 2006 |
Regulation of phosphorylation of the GluR1 AMPA receptor by dopamine D2 receptors.
Topics: Adenosine A2 Receptor Antagonists; Amino Acid Sequence; Animals; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Haloperidol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Phosphorylation; Purines; Quinpirole; Receptors, AMPA; Receptors, Dopamine D2; Serine; Threonine | 2006 |
Effects of a partial D2-like receptor agonist on striatal dopamine autoreceptor functioning in preweanling rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Animals, Newborn; Autoreceptors; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Enzyme Inhibitors; Haloperidol; Hydrazines; Lisuride; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reserpine | 2006 |
Effects of two novel D3-selective compounds, NGB 2904 [N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-9H-fluorene-2-carboxamide] and CJB 090 [N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(pyridin-2-yl)benzamide], on the reinforcing and discrimin
Topics: Animals; Cocaine; Conditioning, Psychological; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Fluorenes; Haloperidol; Macaca mulatta; Male; Piperazines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology | 2007 |
Effect of quinpirole on timing behaviour in the free-operant psychophysical procedure: evidence for the involvement of D2 dopamine receptors.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Female; Haloperidol; Quinpirole; Rats; Rats, Wistar; Reaction Time; Salicylamides; Sulpiride | 2007 |
Differential modulation of a 40 kDa catecholamine regulated protein in the core and shell subcompartments of the nucleus accumbens following chronic quinpirole and haloperidol administration in the rat.
Topics: Analysis of Variance; Animals; Dopamine Agonists; Dopamine Antagonists; Drug Administration Schedule; Gene Expression Regulation; Haloperidol; HSP70 Heat-Shock Proteins; Male; Nerve Tissue Proteins; Nucleus Accumbens; Quinpirole; Rats; Rats, Long-Evans | 2007 |
Effects of activation and blockade of dopamine D(2) receptors on the immune response in mice with different types of behavior.
Topics: Animals; Antibody Formation; Behavior, Animal; Dominance-Subordination; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Erythrocytes; Haloperidol; Immunization; Male; Mice; Mice, Inbred C57BL; Neuroimmunomodulation; Quinpirole; Receptors, Dopamine D2 | 2007 |
Haloperidol both prevents and reverses quinpirole-induced nonregulatory water intake, a putative animal model of psychogenic polydipsia.
Topics: Administration, Oral; Animals; Antipsychotic Agents; Benzodiazepines; Clomipramine; Clozapine; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking; Haloperidol; Male; Olanzapine; Piperazines; Pyrroles; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Thiazepines | 2008 |
Effects of the dopamine stabilizer, OSU-6162, on brain stimulation reward and on quinpirole-induced changes in reward and locomotion.
Topics: Analysis of Variance; Animals; Behavior, Animal; Brain; Conditioning, Operant; Deep Brain Stimulation; Dopamine Agents; Haloperidol; Locomotion; Male; Piperidines; Quinpirole; Rats; Rats, Sprague-Dawley; Reward; Self Administration; Time Factors | 2009 |
The receptor mechanisms underlying the disruptive effects of haloperidol and clozapine on rat maternal behavior: a double dissociation between dopamine D(2) and 5-HT(2A/2C) receptors.
Topics: Amphetamines; Animals; Antipsychotic Agents; Clozapine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Female; Haloperidol; Maternal Behavior; Nesting Behavior; Postpartum Period; Pregnancy; Quinpirole; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine D2; Serotonin Receptor Agonists | 2009 |
GPR37 surface expression enhancement via N-terminal truncation or protein-protein interactions.
Topics: Blotting, Western; Cell Line; Cell Membrane; Dopamine; Dopamine D2 Receptor Antagonists; Flow Cytometry; Haloperidol; Humans; Immunoprecipitation; Microscopy, Confocal; Protein Binding; Quinpirole; Receptors, Dopamine D2; Receptors, G-Protein-Coupled; Syntenins | 2009 |
c-Fos identification of neuroanatomical sites associated with haloperidol and clozapine disruption of maternal behavior in the rat.
Topics: Amphetamines; Animals; Animals, Newborn; Antipsychotic Agents; Biomarkers; Brain; Clozapine; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Immunohistochemistry; Male; Maternal Behavior; Neostriatum; Nucleus Accumbens; Proto-Oncogene Proteins c-fos; Quinpirole; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Septum of Brain; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists | 2010 |
Effects of repeated and acute aripiprazole or haloperidol treatment on dopamine synthesis in the dorsal striatum of young rats: comparison to adult rats.
Topics: Aging; Animals; Animals, Newborn; Antipsychotic Agents; Aripiprazole; Autoreceptors; Brain Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Drug Administration Schedule; Drug Interactions; Female; Haloperidol; Male; Piperazines; Quinolones; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2 | 2010 |
Involvement of different types of dopamine receptors in the formation of latent inhibition of a conditioned passive avoidance reaction in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Avoidance Learning; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Haloperidol; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2010 |
Opposite roles of dopamine and orexin in quinpirole-induced excessive drinking: a rat model of psychotic polydipsia.
Topics: Animals; Benzoxazoles; Cerebral Cortex; Conditioning, Operant; Corticosterone; Disease Models, Animal; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Drinking; Drug Synergism; Haloperidol; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexins; Psychotic Disorders; Quinpirole; Rats; Rats, Sprague-Dawley; Urea | 2010 |
HPC-1/syntaxin 1A gene knockout mice show abnormal behavior possibly related to a disruption in 5-HTergic systems.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Amphetamines; Animals; Behavior, Animal; Desipramine; Dopamine Agonists; Dopamine Antagonists; Fluoxetine; Haloperidol; Hippocampus; Humans; Hypothalamus; Inhibition, Psychological; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Phenotype; Piperazines; Quinpirole; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Social Behavior; Syntaxin 1 | 2010 |
The effects of clozapine on quinpirole-induced non-regulatory drinking and prepulse inhibition disruption in rats.
Topics: Animals; Antipsychotic Agents; Brain; Brain-Derived Neurotrophic Factor; Clozapine; Disease Models, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Drinking; Gene Expression Regulation; Haloperidol; Male; Proto-Oncogene Proteins c-fos; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Schizophrenia | 2010 |
Clomipramine, but not haloperidol or aripiprazole, inhibits quinpirole-induced water contrafreeloading, a putative animal model of compulsive behavior.
Topics: Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Aripiprazole; Clomipramine; Compulsive Behavior; Conditioning, Operant; Disease Models, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Drinking Behavior; Haloperidol; Male; Piperazines; Quinolones; Quinpirole; Rats; Rats, Sprague-Dawley | 2011 |
Inhibition of 5α-reductase attenuates behavioral effects of D1-, but not D2-like receptor agonists in C57BL/6 mice.
Topics: 5-alpha Reductase Inhibitors; Animals; Apomorphine; Benzazepines; Catalepsy; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Finasteride; Haloperidol; Male; Mice; Mice, Inbred C57BL; Motor Activity; Quinpirole; Sensory Gating; Stereotyped Behavior | 2013 |
Enhanced reward-facilitating effects of d-amphetamine in rats in the quinpirole model of obsessive-compulsive disorder.
Topics: Analysis of Variance; Animals; Central Nervous System Stimulants; Conditioning, Operant; Dextroamphetamine; Disease Models, Animal; Dopamine Antagonists; Electric Stimulation; Haloperidol; Male; Obsessive-Compulsive Disorder; Quinpirole; Rats; Rats, Wistar; Reward; Self Administration | 2013 |
Presynaptic regulation of extracellular dopamine levels in the medial prefrontal cortex and striatum during tyrosine depletion.
Topics: Amino Acids; Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Microdialysis; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Tyrosine | 2013 |
Postnatal manganese exposure does not alter dopamine autoreceptor sensitivity in adult and adolescent male rats.
Topics: Aging; Animals; Animals, Newborn; Apomorphine; Autoreceptors; Behavior, Animal; Corpus Striatum; Dopamine; Haloperidol; Male; Manganese; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine | 2013 |
Distinct effects of haloperidol in the mediation of conditioned fear in the mesolimbic system and processing of unconditioned aversive information in the inferior colliculus.
Topics: Animals; Catalepsy; Conditioning, Classical; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Evoked Potentials, Auditory; Fear; Haloperidol; Inferior Colliculi; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Reflex, Startle; Stress, Physiological | 2014 |
Influence of dopamine D2-type receptors on motor behaviors in the green tree frog, Hyla cinerea.
Topics: Animals; Anura; Dopamine Agonists; Dopamine Antagonists; Female; Haloperidol; Learning; Male; Motor Activity; Quinpirole; Receptors, Dopamine D2; Swimming; Task Performance and Analysis; Time Factors; Water | 2014 |
Differential effects of intermittent versus continuous haloperidol treatment throughout adolescence on haloperidol sensitization and social behavior in adulthood.
Topics: Aging; Animals; Antipsychotic Agents; Avoidance Learning; Drug Delivery Systems; Haloperidol; Male; Memory; Neuropsychological Tests; Psychomotor Agitation; Quinpirole; Random Allocation; Rats, Sprague-Dawley; Social Behavior | 2014 |
Reduced striatal dopamine DA D2 receptor function in dominant-negative GSK-3 transgenic mice.
Topics: Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Gene Expression Regulation; Glycogen Synthase Kinase 3; Haloperidol; Mice; Mice, Inbred C57BL; Mice, Transgenic; Microdialysis; Motor Activity; Neurons; Quinpirole; Receptors, Dopamine D2; Time Factors; Tyrosine 3-Monooxygenase | 2014 |
Neuropharmacology of light-induced locomotor activation.
Topics: Animals; Dopamine Agents; Dose-Response Relationship, Drug; Excitatory Amino Acid Agents; Haloperidol; Indoles; Ketamine; Light; Male; Motor Activity; Naphthyridines; Phencyclidine; Photic Stimulation; Piperazines; Piperidines; Pyridines; Quinpirole; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Ritanserin; Serotonin Antagonists | 2015 |
Central serotonin(2B) receptor blockade inhibits cocaine-induced hyperlocomotion independently of changes of subcortical dopamine outflow.
Topics: Animals; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Haloperidol; Male; Motor Activity; Pyrimidines; Quinpirole; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Serotonin 5-HT2 Receptor Antagonists | 2015 |
Stimulation of dopamine D2-like receptors in the lumbosacral defaecation centre causes propulsive colorectal contractions in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Anesthetics, Local; Animals; Benzazepines; Colon; Defecation; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dopaminergic Neurons; Gastrointestinal Motility; Haloperidol; Injections, Spinal; Lumbosacral Region; Male; Muscle Contraction; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2; Rectum; Spinal Cord; Tetrodotoxin | 2016 |
Acute drug-induced spine changes in the nucleus accumbens are dependent on β-adducin.
Topics: Animals; Caffeine; Cytoskeletal Proteins; Dendritic Spines; Dopamine and cAMP-Regulated Phosphoprotein 32; Female; Haloperidol; Male; Mice, Inbred C57BL; Mice, Transgenic; Microfilament Proteins; Nucleus Accumbens; Phosphorylation; Psychotropic Drugs; Quinpirole | 2016 |
The Quinpirole Hypolocomotive Effects are Strain and Route of Administration Dependent in SHR and SLA16 Isogenic Rats.
Topics: Animals; Anxiety; Behavior, Animal; Dopamine; Dopamine D2 Receptor Antagonists; Drug Administration Routes; Haloperidol; Hippocampus; Locomotion; Male; Motor Activity; Quinpirole; Rats; Rats, Inbred SHR; Rats, Mutant Strains; Receptors, Dopamine D2 | 2017 |
Altered dopaminergic regulation of the dorsal striatum is able to induce tic-like movements in juvenile rats.
Topics: Animals; Corpus Striatum; Disease Models, Animal; Dopamine Agonists; Down-Regulation; Haloperidol; Male; Motor Activity; Oxidopamine; Phenotype; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Tourette Syndrome | 2018 |
D2 receptor-mediated miRNA-143 expression is associated with the effects of antipsychotic drugs on phencyclidine-induced schizophrenia-related locomotor hyperactivity and with Neuregulin-1 expression in mice.
Topics: Animals; Benzazepines; Clozapine; Dopamine D2 Receptor Antagonists; Haloperidol; Hippocampus; Male; Mice; Mice, Transgenic; MicroRNAs; Motor Activity; Neuregulin-1; Phencyclidine; Prefrontal Cortex; Primary Cell Culture; Quinpirole; Receptors, Dopamine D2; Salicylamides | 2019 |
Serotonin 5-HT
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Antipsychotic Agents; Brain Waves; Cortical Synchronization; Dopamine Agonists; Dopamine Antagonists; Electroencephalography; Fluorobenzenes; Gamma Rhythm; Haloperidol; Hippocampus; Locomotion; Mice; Neural Pathways; Piperazines; Piperidines; Prefrontal Cortex; Pyridines; Quinpirole; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Risperidone; Serotonin Antagonists; Serotonin Receptor Agonists | 2019 |
Dopaminergic- and cholinergic-inputs from substantia nigra and pedunculo-pontine tegmentum, respectively, converge in amygdala to modulate rapid eye movement sleep in rats.
Topics: Amygdala; Animals; Carbachol; Cholinergic Neurons; Dopaminergic Neurons; Electric Stimulation; Haloperidol; Male; Pontine Tegmentum; Quinpirole; Rats; Rats, Wistar; Scopolamine; Sleep, REM; Substantia Nigra; Wakefulness | 2021 |