haloperidol and preclamol

haloperidol has been researched along with preclamol in 81 studies

Research

Studies (81)

TimeframeStudies, this research(%)All Research%
pre-199023 (28.40)18.7374
1990's49 (60.49)18.2507
2000's6 (7.41)29.6817
2010's3 (3.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
el-Ashmawy, M; Fischer, JB; Glennon, RA; Herndon, JL; Howie, KJ; Ismaiel, AM; Server, AC; Smith, JD; Yousif, M1
Dannals, RF; Ravert, HT; Sonders, MS; Wagner, HN; Weber, E; Wilson, AA1
Chidester, CG; Haadsma-Svensson, SR; Lahti, RA; Lin, CH; McCall, RB; Piercey, MF; Schreur, PJ; Smith, MW; Von Voigtlander, PF1
Chidester, CG; Haadsma-Svensson, SR; Lahti, RA; Lin, CH; McCall, RB; Phillips, G; Piercey, MF; Schreur, PJ; Smith, MW; Von Voigtlander, PF1
Carlsson, A; Meier, E; Piercey, MF; Smith, MW; Sonesson, C; Svensson, K; Waters, N; Wikström, H1
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X1
Fiechtner, B; Glossmann, H; Hoffmann, RD; Laggner, C; Langer, T; Moebius, FF; Poles, G; Schieferer, C1
Carlsson, A; Hansson, L; Lin, CH; Smith, MW; Sonesson, C; Svensson, K; Waters, N; Wikström, H1
Pettersson, F; Pontén, H; Sonesson, C; Waters, N; Waters, S1
DeHaven-Hudkins, DL; Fleissner, LC1
Hudzik, TJ1
Araki, H; Hasegawa, Y; Kaku, S; Otomo, S1
Ericson, H; Ross, SB1
DeHaven-Hudkins, DL; Fleissner, LC; Ford-Rice, FY1
Chavkin, C; Connor, MA2
Blier, P; de Montigny, C; Debonnel, G; Monnet, FP1
Codd, EE; Shank, RP1
Ross, SB1
Musacchio, JM; Zhou, GZ1
Itzhak, Y; Stein, I1
Karbon, EW; Naper, K; Pontecorvo, MJ1
Cler, JA; Contreras, PC; Dilworth, VM; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL1
Battaglia, G; Glennon, RA; Smith, JD1
Fiorica-Howells, E; Spector, S1
Svensson, L1
Church, J; Lodge, D1
Itzhak, Y; Krähling, H; Ruhland, M1
Klein, M; Musacchio, J; Paturzo, JJ; Zhou, GZ1
Bowen, WD; Moses, EL; Tolentino, PJ; Walker, JM1
Duckles, SP; Massamiri, T1
Culp, SG; De Souza, EB; Wolfe, SA1
Bobker, DH; Shen, KZ; Surprenant, A; Williams, JT1
Claustre, Y; Fage, D; Scatton, B; Zivkovic, B1
Itzhak, Y1
Fowler, CJ; Thorell, G1
Ahlenius, S; Hillegaart, V1
Ahlenius, S; Criborn, CO; Henriksson, C; Hillegaart, V1
Bonsall, RW; Michael, RP; Schaefer, GJ1
Clark, D; Elam, M; Svensson, TH1
Broekkamp, CL; Gower, AJ1
Collu, M; Gessa, GL; Serra, G1
Carlsson, A; Löfberg, L1
Gundlach, AL; Largent, BL; Snyder, SH1
Boissard, CG; Delini-Stula, A; Mogilnicka, E1
Daus, FJ; Hansen, HA; Plantjé, JF; Stoof, JC1
Ahlenius, S; Archer, T; Hillegaart, V; Tandberg, B1
Ahlenius, S; Hillegaart, V; Svensson, L; Thorberg, O1
Berendsen, HG; Broekkamp, CL; Gower, AJ; Princen, MM1
Ahlenius, S; Larsson, K1
Fenton, HM; Gerhardt, S; Hall, NR; Liebman, JM; Neale, R; Noreika, L1
Geyer, MA; Lee, EH1
Carlsson, A; Gunne, LM; Häggström, JE; Wikström, H1
Fratta, W; Gessa, GL; Napoli-Farris, L1
Bowen, WD; Carr, DJ; DeCosta, BR; Garza, HH; Mayo, S1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
Arnold, FJ; Murphy, RB; Schuster, DI1
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC1
Bailey, MA; Karbon, EW1
Davies, JA; Ellis, Y1
Cooper, TB; Klein, M; Musacchio, JM1
Barg, J; Eilam, Y; Ela, C; Hasin, Y; Vogel, Z1
Gerlach, J; Peacock, L1
Enomoto, R; Ogita, K; Yoneda, Y1
Callahan, PM; Cunningham, KA1
Matsuno, K; Mita, S; Senda, T1
Brum, JM; Estafanous, FG; Murray, PA; Schubert, A; Tsuchida, H1
Kobayashi, T; Matsuno, K; Mita, S1
Barrett, TW; Chang, S; Ha, BK; Liu, Y; Saini, P; Whitlock, BB; Wolfe, SA1
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA1
Akiyama, K; Kuroda, S; Okumura, K; Ujike, H1
Earley, B; Faherty, CJ; Leonard, BE1
Fang, H; Helmeste, DM; Li, M; Tang, SW1
Curzon, P; Decker, MW1
Carey, JE; Frey, KA; Kilbourn, MR; Kuhl, DE; Mulholland, GK; Sherman, PS; Wieland, DM1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1
Akaike, A; Hashino, A; Kaneko, S; Katsuki, H; Kume, T; Minami, M; Nishikawa, H; Satoh, M; Taguchi, R1
Baeyens, JM; Cobos, EJ; Del Pozo, E1
Burris, KD; Kikuchi, T; Miwa, T; Mori, T; Stark, A; Tadori, Y; Tottori, K1
Calas, AG; Goursaud, S; Hermans, E; Jeanjean, AP; Koener, B; Maloteaux, JM; Van De Stadt, M1
Carlsson, A; Carlsson, ML; Johansson, AM; Rung, E; Rung, JP; Svensson, K1

Other Studies

81 other study(ies) available for haloperidol and preclamol

ArticleYear
Binding of substituted and conformationally restricted derivatives of N-(3-phenyl-n-propyl)-1-phenyl-2-aminopropane at sigma-receptors.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:6

    Topics: Animals; Brain; Guinea Pigs; Microsomes; Phencyclidine; Propylamines; Radioligand Assay; Receptors, Opioid; Receptors, sigma; Substrate Specificity

1991
Radiosynthesis of sigma receptor ligands for positron emission tomography: 11C- and 18F-labeled guanidines.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:6

    Topics: Animals; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Fluorine Radioisotopes; Guanidines; Guinea Pigs; Magnetic Resonance Spectroscopy; Receptors, Opioid; Receptors, sigma; Tomography, Emission-Computed

1991
Centrally acting serotonergic and dopaminergic agents. 1. Synthesis and structure-activity relationships of 2,3,3a,4,5,9b-hexahydro-1H-benz[e]indole derivatives.
    Journal of medicinal chemistry, 1993, Apr-16, Volume: 36, Issue:8

    Topics: Animals; Brain; Cats; Cattle; Dopamine Agents; Indoles; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Stereoisomerism; Structure-Activity Relationship

1993
Centrally acting serotonergic and dopaminergic agents. 2. Synthesis and structure-activity relationships of 2,3,3a,4,9,9a-hexahydro-1H-benz[f]indole derivatives.
    Journal of medicinal chemistry, 1993, Apr-16, Volume: 36, Issue:8

    Topics: Animals; Binding Sites; Brain; Cats; Cattle; Dopamine Agents; Indoles; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes

1993
Substituted 3-phenylpiperidines: new centrally acting dopamine autoreceptor antagonists.
    Journal of medicinal chemistry, 1993, Oct-15, Volume: 36, Issue:21

    Topics: Animals; Binding Sites; Biological Availability; Brain; Dopamine; Dopamine Antagonists; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship

1993
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.
    Journal of medicinal chemistry, 2003, Oct-09, Volume: 46, Issue:21

    Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water

2003
Discovery of high-affinity ligands of sigma1 receptor, ERG2, and emopamil binding protein by pharmacophore modeling and virtual screening.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Animals; Carrier Proteins; Databases, Factual; Guinea Pigs; Humans; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Isomerism; Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Radioligand Assay; Receptors, sigma; Saccharomyces cerevisiae; Sigma-1 Receptor; Steroid Isomerases

2005
Substituted (S)-phenylpiperidines and rigid congeners as preferential dopamine autoreceptor antagonists: synthesis and structure-activity relationships.
    Journal of medicinal chemistry, 1994, Aug-19, Volume: 37, Issue:17

    Topics: Animals; Benzazepines; Brain; CHO Cells; Cricetinae; Dihydroxyphenylalanine; Dopamine D2 Receptor Antagonists; Habituation, Psychophysiologic; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Motor Activity; Optical Rotation; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Serotonin; Reserpine; Serotonin Antagonists; Spiperone; Structure-Activity Relationship; Transfection

1994
Synthesis and evaluation of a set of 4-phenylpiperidines and 4-phenylpiperazines as D2 receptor ligands and the discovery of the dopaminergic stabilizer 4-[3-(methylsulfonyl)phenyl]-1-propylpiperidine (huntexil, pridopidine, ACR16).
    Journal of medicinal chemistry, 2010, Mar-25, Volume: 53, Issue:6

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Binding, Competitive; Cell Line; Corpus Striatum; Dopamine; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Discovery; Drug Evaluation, Preclinical; Humans; Ligands; Male; Models, Chemical; Molecular Structure; Motor Activity; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

2010
Competitive interactions at [3H]1,3-di(2-tolyl)guanidine (DTG)-defined sigma recognition sites in guinea pig brain.
    Life sciences, 1992, Volume: 50, Issue:9

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Carbazoles; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Male; Pentazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma

1992
Sigma ligand-induced emesis in the pigeon.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1

    Topics: Animals; Apomorphine; Columbidae; Dextromethorphan; Dizocilpine Maleate; Dopamine Agents; Guanidines; Haloperidol; Male; Pentobarbital; Phenazocine; Piperidines; Propranolol; Psychotropic Drugs; Pyrimidines; Receptors, Opioid; Receptors, sigma; Vomiting

1992
Sigma receptor modulation of the muscle relaxant action of eperisone.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1992, Volume: 2, Issue:2

    Topics: Animals; Behavior, Animal; Dopamine Agents; Dose-Response Relationship, Drug; Haloperidol; In Vitro Techniques; Mice; Mice, Inbred ICR; Muscle Relaxants, Central; Piperidines; Propiophenones; Receptors, Opioid; Receptors, sigma

1992
Subchronic treatment of rats with remoxipride fails to modify sigma binding sites in the brain.
    European journal of pharmacology, 1992, Jun-05, Volume: 226, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Corpus Striatum; Dopamine Agents; Dopamine Antagonists; Haloperidol; In Vitro Techniques; Liver; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride; Salicylamides

1992
Characterization of the binding of [3H](+)-pentazocine to sigma recognition sites in guinea pig brain.
    European journal of pharmacology, 1992, Dec-01, Volume: 227, Issue:4

    Topics: Animals; Antipsychotic Agents; Binding Sites; Binding, Competitive; Brain; Carbazoles; Dopamine Agents; Guinea Pigs; Haloperidol; Kinetics; Male; Pentazocine; Piperidines; Receptors, sigma

1992
Ionic zinc may function as an endogenous ligand for the haloperidol-sensitive sigma 2 receptor in rat brain.
    Molecular pharmacology, 1992, Volume: 42, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Cations, Divalent; Copper; Electric Stimulation; Guanidines; Haloperidol; Hippocampus; Hydrogen-Ion Concentration; Kinetics; Male; Membranes; Pentazocine; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sensitivity and Specificity; Tritium; Zinc

1992
Modulation by sigma ligands of N-methyl-D-aspartate-induced [3H]noradrenaline release in the rat hippocampus: G-protein dependency.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:1

    Topics: Animals; Calcium; Cinnamates; Cyclopropanes; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanidines; Haloperidol; Hippocampus; In Vitro Techniques; Magnesium; Male; N-Methylaspartate; Norepinephrine; Pertussis Toxin; Piperidines; Rats; Rats, Inbred Strains; Spiperone; Tritium; Virulence Factors, Bordetella

1992
1,3-Di(2-[5-3H]tolyl)guanidine labels more than one site in rat forebrain.
    European journal of pharmacology, 1992, Jul-07, Volume: 217, Issue:2-3

    Topics: Animals; Binding Sites; Binding, Competitive; Carbamazepine; Guanidines; Haloperidol; Male; Pentazocine; Phenytoin; Piperidines; Prosencephalon; Rats; Rats, Wistar; Receptors, sigma; Stereoisomerism

1992
Heterogeneous binding of sigma radioligands in the rat brain and liver: possible relationship to subforms of cytochrome P-450.
    Pharmacology & toxicology, 1991, Volume: 68, Issue:4

    Topics: Animals; Brain; Cytochrome P-450 Enzyme System; Guanidines; Haloperidol; Kinetics; Ligands; Liver; Male; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Subcellular Fractions

1991
Computer-assisted modeling of multiple dextromethorphan and sigma binding sites in guinea pig brain.
    European journal of pharmacology, 1991, Apr-25, Volume: 206, Issue:4

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Computer Simulation; Dextromethorphan; Guanidines; Guinea Pigs; Haloperidol; Kinetics; Male; Models, Biological; Piperidines; Receptors, Opioid; Receptors, sigma; Tritium

1991
Regulation of sigma receptors and responsiveness to guanine nucleotides following repeated exposure of rats to haloperidol: further evidence for multiple sigma binding sites.
    Brain research, 1991, Dec-06, Volume: 566, Issue:1-2

    Topics: Adenosine Triphosphate; Animals; Brain; Cell Membrane; Down-Regulation; Guanidines; Guanine Nucleotides; Guanylyl Imidodiphosphate; Haloperidol; Kinetics; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Reference Values

1991
[3H]DTG and [3H](+)-3-PPP label pharmacologically distinct sigma binding sites in guinea pig brain membranes.
    European journal of pharmacology, 1991, Jan-25, Volume: 193, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Membranes; Phenazocine; Phenytoin; Piperidines; Receptors, Opioid; Receptors, sigma

1991
Focal stimulation of specific pathways in the rat hippocampus causes a reduction in radioligand binding to the haloperidol-sensitive sigma receptor.
    Experimental brain research, 1991, Volume: 85, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Electric Stimulation; Guanidines; Haloperidol; Hippocampus; Male; Piperidines; Quinoxalines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1991
Neurochemical characterization of dopaminergic effects of opipramol, a potent sigma receptor ligand, in vivo.
    Neuropharmacology, 1990, Volume: 29, Issue:12

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Ligands; Male; Mice; Opipramol; Organ Specificity; Phencyclidine; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
(-)PPAP: a new and selective ligand for sigma binding sites.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Animals; Catalysis; Dextroamphetamine; Discrimination, Psychological; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Piperidines; Propylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
Selectivity of some "specific" opioid ligands?
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Benzomorphans; Binding, Competitive; Brain; Dynorphins; Female; Haloperidol; In Vitro Techniques; Mice; Morphinans; Peptide Fragments; Phencyclidine; Piperidines; Receptors, Opioid

1990
The role of the dopaminergic system in the modulation of the acoustic startle response in the rat.
    European journal of pharmacology, 1990, Jan-03, Volume: 175, Issue:1

    Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Reflex, Startle; Stereoisomerism

1990
Failure of sigma-receptor ligands to reduce the excitatory actions of N-methyl-DL-aspartate on rat spinal neurons in-vivo.
    The Journal of pharmacy and pharmacology, 1990, Volume: 42, Issue:1

    Topics: Animals; Aspartic Acid; Haloperidol; In Vitro Techniques; Kainic Acid; Ligands; N-Methylaspartate; Neurons; Oxadiazoles; Piperidines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Spinal Cord; Stereoisomerism

1990
Binding of umespirone to the sigma receptor: evidence for multiple affinity states.
    Neuropharmacology, 1990, Volume: 29, Issue:2

    Topics: Animals; Antipsychotic Agents; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorpromazine; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine

1990
The effect of sigma ligands on dextromethorphan binding sites in the guinea pig.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Binding Sites; Dextromethorphan; Guinea Pigs; Hallucinogens; Haloperidol; In Vitro Techniques; Kinetics; Levorphanol; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
Metabolites of haloperidol display preferential activity at sigma receptors compared to dopamine D-2 receptors.
    European journal of pharmacology, 1990, Feb-27, Volume: 177, Issue:3

    Topics: Animals; Brain; Haloperidol; In Vitro Techniques; Male; Motor Activity; Parasympathetic Nervous System; Pentazocine; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Receptors, sigma

1990
Multiple vascular effects of sigma and PCP ligands: inhibition of amine uptake and contractile responses.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:1

    Topics: Animals; Cocaine; Desoxycorticosterone; Haloperidol; Male; Norepinephrine; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Serotonin; Vasoconstriction

1990
Sigma-receptors in endocrine organs: identification, characterization, and autoradiographic localization in rat pituitary, adrenal, testis, and ovary.
    Endocrinology, 1989, Volume: 124, Issue:3

    Topics: Adrenal Glands; Animals; Autoradiography; Brain Chemistry; Cell Membrane; Dibenzocycloheptenes; Dizocilpine Maleate; Female; Haloperidol; Hypophysectomy; Male; Ovary; Phencyclidine; Piperidines; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Testis; Tissue Distribution

1989
DTG and (+)-3-PPP inhibit a ligand-activated hyperpolarization in mammalian neurons.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:3

    Topics: Animals; Brimonidine Tartrate; Dopamine Agents; Enkephalin, Methionine; Guanidines; Haloperidol; Male; Membrane Potentials; Neurons; Norepinephrine; Piperidines; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Serotonin

1989
Relative selectivity of 6,7-dihydroxy-2-dimethylaminotetralin, N-n-propyl-3-(3-hydroxyphenyl)piperidine, N-n-propylnorapomorphine and pergolide as agonists at striatal dopamine autoreceptors and postsynaptic dopamine receptors.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:2

    Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Haloperidol; Homovanillic Acid; Male; Naphthalenes; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sodium Oxybate; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase

1985
Pharmacological specificity of some psychotomimetic and antipsychotic agents for the sigma and PCP binding sites.
    Life sciences, 1988, Volume: 42, Issue:7

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Haloperidol; In Vitro Techniques; Male; Phenazocine; Phencyclidine; Piperidines; Psychotropic Drugs; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1988
Antagonist effects of the enantiomers of 3-PPP towards alpha 1-adrenoceptors coupled to inositol phospholipid breakdown in the rat cerebral cortex.
    Pharmacology & toxicology, 1987, Volume: 60, Issue:5

    Topics: Animals; Antiparkinson Agents; Atropine; Carbachol; Cerebral Cortex; Haloperidol; In Vitro Techniques; Inositol Phosphates; Male; Norepinephrine; Phenoxybenzamine; Piperidines; Prazosin; Raclopride; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Salicylamides; Stereoisomerism; Sugar Phosphates

1987
Effects of raclopride on exploratory locomotor activity, treadmill locomotion, conditioned avoidance behaviour and catalepsy in rats: behavioural profile comparisons between raclopride, haloperidol and preclamol.
    Pharmacology & toxicology, 1987, Volume: 60, Issue:5

    Topics: Animals; Avoidance Learning; Behavior, Animal; Catalepsy; Exploratory Behavior; Haloperidol; Male; Motor Activity; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Salicylamides; Scopolamine

1987
Partial protection against hyperbaric oxygen induced convulsions by dopaminergic agents in mice: possible involvement of autoreceptors?
    Journal of neural transmission, 1987, Volume: 69, Issue:3-4

    Topics: Animals; Antiparkinson Agents; Apomorphine; Body Temperature; Dose-Response Relationship, Drug; Haloperidol; Hyperbaric Oxygenation; Levodopa; Male; Mice; Mice, Inbred CBA; Piperidines; Reaction Time; Receptors, Dopamine; Respiration; Seizures

1987
An automatic device for measuring speed of movement and time spent at rest: its application to testing dopaminergic drugs.
    Physiology & behavior, 1986, Volume: 37, Issue:1

    Topics: Animals; Dextroamphetamine; Dose-Response Relationship, Drug; Female; Haloperidol; Motor Activity; Neurophysiology; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1986
Electrophysiological effects of the enantiomers of 3-PPP on neurons in the locus coeruleus of the rat.
    Neuropharmacology, 1986, Volume: 25, Issue:9

    Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Haloperidol; Injections, Intravenous; Iontophoresis; Locus Coeruleus; Male; Neurons; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Stereoisomerism; Yohimbine

1986
Dopaminergic agents including 3-PPP and its enantiomers on medial septal self-stimulation.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Appetite Depressants; Benzazepines; Dextroamphetamine; Drug Interactions; Haloperidol; Male; Nomifensine; Piperidines; Rats; Receptors, Dopamine; Self Stimulation; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes

1985
Dopamine receptors mediating yawning: are they autoreceptors?
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: Animals; Domperidone; Drug Synergism; Haloperidol; Male; Methyltyrosines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reflex; Reserpine; Stereoisomerism; Sulpiride

1986
In vivo displacement by 3-PPP enantiomers of N,N-dipropyl-5,6-ADTN from dopamine receptor-binding sites in rat striatum.
    Journal of neural transmission, 1985, Volume: 64, Issue:3-4

    Topics: Animals; Binding, Competitive; Brain; Cerebellum; Corpus Striatum; Haloperidol; Isomerism; Male; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tetrahydronaphthalenes

1985
Psychotomimetic opiate receptors labeled and visualized with (+)-[3H]3-(3-hydroxyphenyl)-N-(1-propyl)piperidine.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:15

    Topics: Animals; Brain Mapping; Brain Stem; Cerebellum; Guinea Pigs; Haloperidol; Hypothalamus; Limbic System; Mesencephalon; Piperidines; Rats; Receptors, Dopamine; Receptors, Opioid; Stereoisomerism

1984
Effects of apomorphine, TL-99 and 3-PPP on yawning in rats.
    Neuropharmacology, 1984, Volume: 23, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apomorphine; Behavior, Animal; Haloperidol; Male; Naphthalenes; Piperidines; Rats; Tetrahydronaphthalenes

1984
The effects of SCH 23390, YM 09151-2, (+)- and (-)-3-PPP and some classical neuroleptics on D-1 and D-2 receptors in rat neostriatum in vitro.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Antipsychotic Agents; Aporphines; Benzamides; Benzazepines; Caudate Nucleus; Chlorpromazine; Clozapine; Flupenthixol; Haloperidol; In Vitro Techniques; Male; Piperidines; Potassium; Putamen; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1984
Effects of (-)3-PPP on acquisition and retention of a conditioned avoidance response in the rat.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Discrimination Learning; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains

1984
Antagonism by haloperidol of the suppression of exploratory locomotor activity induced by the local application of (-)3-(3-hydroxyphenyl)-N-n-propylpiperidine into the nucleus accumbens of the rat.
    Experientia, 1984, Aug-15, Volume: 40, Issue:8

    Topics: Animals; Exploratory Behavior; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Septal Nuclei

1984
The yawning-penile erection syndrome as a model for putative dopamine autoreceptor activity.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Apomorphine; Drug Interactions; Haloperidol; Inhalation; Isomerism; Male; Models, Psychological; Penis; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Respiration; Sexual Behavior, Animal; Syndrome

1984
Apomorphine and haloperidol-induced effects on male rat sexual behavior: no evidence for actions due to stimulation of central dopamine autoreceptors.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:3

    Topics: Animals; Apomorphine; Brain; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal

1984
Avoidance and ICSS behavioral models dissociate TL-99 and 3-PPP from dopamine receptor antagonists.
    European journal of pharmacology, 1983, Aug-05, Volume: 91, Issue:4

    Topics: Animals; Avoidance Learning; Haloperidol; Male; Models, Psychological; Naphthalenes; Piperidines; Rats; Rats, Inbred F344; Receptors, Dopamine; Saimiri; Self Stimulation; Tetrahydronaphthalenes

1983
Similarities of the effects of apomorphine and 3-PPP on serotonin neurons.
    European journal of pharmacology, 1983, Oct-28, Volume: 94, Issue:3-4

    Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Corpus Striatum; Haloperidol; Hippocampus; Male; Neurons; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spectrometry, Fluorescence

1983
Antidyskinetic action of 3-PPP, a selective dopaminergic autoreceptor agonist, in Cebus monkeys with persistent neuroleptic-induced dyskinesias.
    Journal of neural transmission, 1983, Volume: 58, Issue:3-4

    Topics: Animals; Cebus; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Female; Fluphenazine; Haloperidol; Male; Piperidines; Stereoisomerism

1983
Stimulation of dopamine autoreceptors elicits "premature ejaculation" in rats.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 20, Issue:1

    Topics: Animals; Apomorphine; Copulation; Domperidone; Dopamine Antagonists; Ejaculation; Female; Haloperidol; Lisuride; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal

1984
Characterization of a (+)-azidophenazocine-sensitive sigma receptor on splenic lymphocytes.
    Journal of immunology (Baltimore, Md. : 1950), 1993, Nov-01, Volume: 151, Issue:9

    Topics: Affinity Labels; Animals; Binding Sites; Binding, Competitive; Female; Haloperidol; Interferons; Lymphocytes; Mice; Mice, Inbred C57BL; Phenazocine; Piperidines; Receptors, sigma; Spleen

1993
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
Purification, pharmacological characterization and photoaffinity labeling of sigma receptors from rat and bovine brain.
    Brain research, 1995, Jan-23, Volume: 670, Issue:1

    Topics: Animals; Binding Sites; Cattle; Cerebellum; Dopamine Agonists; Haloperidol; Male; Phenazocine; Piperidines; Rats; Receptors, sigma

1995
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
    Brain research, 1995, Feb-06, Volume: 671, Issue:1

    Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma

1995
Haloperidol treatment differentially regulates [3H]DTG and [3H](+)-3-PPP labeled sigma binding sites.
    European journal of pharmacology, 1993, Aug-24, Volume: 240, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Binding Sites; Brain; Dopamine Agents; Drug Administration Schedule; Guanidines; Guinea Pigs; Haloperidol; Male; Phenytoin; Piperidines; Receptors, sigma

1993
The effects of sigma ligands on the release of glutamate from rat striatal slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 350, Issue:2

    Topics: Animals; Corpus Striatum; Female; Glutamic Acid; Haloperidol; In Vitro Techniques; Ligands; Neuropeptide Y; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, sigma

1994
Effects of haloperidol and reduced haloperidol on binding to sigma sites.
    European journal of pharmacology, 1994, Mar-21, Volume: 254, Issue:3

    Topics: Animals; Binding Sites; Brain; Dextromethorphan; Guinea Pigs; Haloperidol; Male; Oxidation-Reduction; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma

1994
Sigma receptor ligands modulate contractility, Ca++ influx and beating rate in cultured cardiac myocytes.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:3

    Topics: Animals; Calcium; Cells, Cultured; GTP-Binding Proteins; Guanidines; Haloperidol; Heart Rate; Myocardial Contraction; Pentazocine; Piperidines; Rats; Receptors, sigma; Sarcoplasmic Reticulum

1994
Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: Administration, Oral; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Benzothiazoles; Cebus; Disease Models, Animal; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dyskinesia, Drug-Induced; Dystonia; Ergolines; Female; Haloperidol; Lisuride; Male; Piperidines; Pramipexole; Quinpirole; Raclopride; Salicylamides; Thiazoles

1993
Multiplicity of [3H]1,3-di-o-tolylguanidine binding sites with low affinity for haloperidol in rat brain.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:10

    Topics: Animals; Binding Sites; Brain; Guanidines; Haloperidol; Male; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma

1993
Discriminative stimulus properties of cocaine in relation to dopamine D2 receptor function in rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Animals; Bromocriptine; Cocaine; Discrimination Learning; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

1993
Correlation between potentiation of neurogenic twitch contraction and benzomorphan sigma receptor binding potency in the mouse vas deferens.
    European journal of pharmacology, 1993, Feb-16, Volume: 231, Issue:3

    Topics: Animals; Antiparkinson Agents; Brain; Drug Synergism; Guinea Pigs; Haloperidol; Ligands; Male; Mice; Phenazocine; Piperidines; Receptors, sigma; Spasm; Vas Deferens

1993
Sigma receptor activation does not mediate fentanyl-induced attenuation of muscarinic coronary contraction.
    Anesthesia and analgesia, 1996, Volume: 82, Issue:5

    Topics: Acetylcholine; Anesthetics, Intravenous; Animals; Coronary Vessels; Cyclazocine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fentanyl; Guanidines; Haloperidol; Muscarine; Muscarinic Agonists; Narcotic Antagonists; Narcotics; Pentazocine; Phencyclidine; Piperidines; Potassium Channel Blockers; Receptors, Dopamine; Receptors, sigma; Signal Transduction; Swine; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

1996
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:1

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens

1996
Initial characterization and autoradiographic localization of a novel sigma/opioid binding site in immune tissues.
    Journal of neuroimmunology, 1996, Volume: 67, Issue:2

    Topics: Animals; Anticonvulsants; Autoradiography; Binding Sites; Binding, Competitive; Brain Chemistry; Cytochrome P-450 Enzyme System; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Hydrogen-Ion Concentration; Kinetics; Leukocytes; Monoamine Oxidase; Naltrexone; Narcotic Antagonists; Narcotics; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Spleen; Tritium

1996
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
    Journal of neuroimmunology, 1997, Volume: 72, Issue:1

    Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium

1997
BMY-14802 reversed the sigma receptor agonist-induced neck dystonia in rats.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:10

    Topics: Animals; Antipsychotic Agents; Dibenzothiepins; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dystonia; Guanidines; Haloperidol; Male; Microinjections; Nerve Tissue Proteins; Perphenazine; Piperidines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Red Nucleus; Sulpiride; Torticollis

1996
Behavioural effects of selective serotonin reuptake inhibitors following direct micro injection into the left red nucleus of the rat.
    Journal of psychopharmacology (Oxford, England), 1997, Volume: 11, Issue:1

    Topics: 1-Naphthylamine; Animals; Behavior, Animal; Chlorpromazine; Citalopram; Fluoxetine; Fluvoxamine; Guanidines; Haloperidol; Male; Microinjections; Motor Activity; Paroxetine; Piperidines; Posture; Rats; Rats, Sprague-Dawley; Receptors, sigma; Red Nucleus; Selective Serotonin Reuptake Inhibitors; Sertraline

1997
Multiple [3H]-nemonapride binding sites in calf brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Benzamides; Binding, Competitive; Brain; Cattle; Cerebellum; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine Agonists; Dopamine Antagonists; Guanidines; Haloperidol; In Vitro Techniques; Isotope Labeling; Narcotic Antagonists; Pentazocine; Piperidines; Propylamines; Pyrrolidines; Receptors, Dopamine D2; Receptors, sigma; Sulpiride; Tritium

1997
Effects of phencyclidine (PCP) and (+)MK-801 on sensorimotor gating in CD-1 mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 1998, Volume: 22, Issue:1

    Topics: Acoustic Stimulation; Animals; Apomorphine; Clozapine; Dextroamphetamine; Dizocilpine Maleate; Dopamine Agonists; Dose-Response Relationship, Drug; Haloperidol; Male; Mice; Mice, Inbred Strains; Phencyclidine; Piperidines; Rats; Receptors, sigma; Reflex, Startle; Species Specificity

1998
[18F]fluoroethoxy-benzovesamicol, a PET radiotracer for the vesicular acetylcholine transporter and cholinergic synapses.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:3

    Topics: Acetylcholine; Animals; Autoradiography; Brain; Calibration; Carrier Proteins; Cholinesterase Inhibitors; Donepezil; Dopamine Agonists; Female; Fluorine Radioisotopes; Haloperidol; Humans; Indans; Kinetics; Male; Membrane Transport Proteins; Mice; Organ Specificity; Piperidines; Rats; Rats, Sprague-Dawley; Stereoisomerism; Synapses; Tissue Distribution; Tomography, Emission-Computed; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

1998
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001
Antagonism of NMDA receptors by sigma receptor ligands attenuates chemical ischemia-induced neuronal death in vitro.
    European journal of pharmacology, 2002, Nov-29, Volume: 455, Issue:2-3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Calcium; Cell Hypoxia; Cell Survival; Cells, Cultured; Cerebral Cortex; Cyclopentanes; Deoxyglucose; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fetus; Glucose; Glutamates; Haloperidol; Neurons; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sodium Azide

2002
Phenytoin differentially modulates the affinity of agonist and antagonist ligands for sigma 1 receptors of guinea pig brain.
    Synapse (New York, N.Y.), 2005, Mar-01, Volume: 55, Issue:3

    Topics: Allosteric Regulation; Animals; Anisoles; Anticonvulsants; Binding, Competitive; Brain; Dextromethorphan; Drug Interactions; Ethylenediamines; Guinea Pigs; Haloperidol; Ligands; Male; Morpholines; Neurons; Phenazocine; Phenytoin; Piperazines; Piperidines; Progesterone; Propylamines; Receptors, sigma; Synaptic Transmission

2005
Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.
    European journal of pharmacology, 2005, May-16, Volume: 515, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Humans; Lisuride; Piperazines; Piperidines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Risperidone; Transfection; Tritium

2005
Pharmacological blockade of dopamine D2 receptors by aripiprazole is not associated with striatal sensitization.
    Naunyn-Schmiedeberg's archives of pharmacology, 2011, Volume: 383, Issue:1

    Topics: Animals; Apomorphine; Aripiprazole; Buffers; Catalepsy; Cell Membrane; Cerebral Cortex; Corpus Striatum; Domperidone; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Antagonism; Drug Partial Agonism; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Hippocampus; Male; Piperazines; Piperidines; Pyridines; Quinolones; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Stereotyped Behavior; Up-Regulation

2011
Effects of the dopamine stabilizers (S)-(-)-OSU6162 and ACR16 on prolactin secretion in drug-naive and monoamine-depleted rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2011, Volume: 384, Issue:1

    Topics: Animals; Aripiprazole; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Hyperprolactinemia; Lactotrophs; Male; Methyltyrosines; Piperazines; Piperidines; Prolactin; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reserpine

2011