haloperidol has been researched along with phenazocine in 72 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 23 (31.94) | 18.7374 |
1990's | 41 (56.94) | 18.2507 |
2000's | 7 (9.72) | 29.6817 |
2010's | 1 (1.39) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Clarke, IM; Tempest, SM | 1 |
Hudzik, TJ | 1 |
McCann, DJ; Su, TP | 4 |
Hitosugi, H; Iwamoto, Y; Kamei, J; Kasuya, Y; Kawashima, N; Misawa, M | 1 |
Borsini, F; Ceci, A; Volonté, M | 1 |
Ross, SB | 1 |
deCosta, BR; Hardwick, WC; McMillan, DE; Rice, KC | 1 |
Karbon, EW; Naper, K; Pontecorvo, MJ | 1 |
Balestra, B; Candura, SM; Coccini, T; Costa, LG; Iapadre, N; Manzo, L; Tonini, M | 1 |
Pèzzola, A; Popoli, P; Sagratella, S; Scotti de Carolis, A | 1 |
Brent, PJ | 1 |
Connick, JH; Fox, PK; France, L; Hanlon, GM; Nicholson, CD | 1 |
Duckles, SP; Massamiri, T | 1 |
Kesingland, AC; Singh, L; Tricklebank, MD; Wong, EH | 1 |
Defaux, JP; Junien, JL; Pascaud, X; Rozé, C | 1 |
Katki, AG; Rodbard, D; Schwarz, S; Zhou, GZ | 1 |
Balster, RL | 1 |
Iwamoto, ET | 1 |
Alerhand, S; Itzhak, Y | 1 |
Allikmets, LKh; Kharro, IaE; Lang, AE; Vasar, EE | 1 |
Duffy, O; Junien, JL; Martin, B; Pascaud, X; Roman, FJ; Vauche, D | 1 |
Cook, L; Steinfels, GF; Tam, SW | 1 |
Iversen, SD; Oles, RJ; Singh, L; Tricklebank, MD; Wong, EH | 1 |
Jaffe, JH; London, ED; Su, TP | 1 |
Junien, JL; Pascaud, X; Roman, F; Vauché, D | 1 |
Downes, CP; Lewis, PE; Stone, MA | 1 |
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K | 1 |
Itzhak, Y | 2 |
Ford-Rice, FY; London, ED; Schell, SE; Su, TP | 1 |
Lahti, RA; Mickelson, MM | 1 |
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR | 1 |
Clark, RD; Katz, JL; Spealman, RD | 1 |
Bunney, BS; Freeman, AS | 1 |
Cook, L; Tam, SW | 1 |
Billington, CJ; Gerritsen, GC; Levine, AS; Morley, JE | 1 |
Holtzman, SG; Teal, JJ | 1 |
Johnson, KM; Leventer, SM | 1 |
Bastianetto, S; Perrault, G; Sanger, DJ | 1 |
Brent, PJ; Dunkley, PR; Haynes, H; Jarvie, PE; Mudge, L; Sim, AT | 1 |
Bowen, WD; Carr, DJ; DeCosta, BR; Garza, HH; Mayo, S | 1 |
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA | 1 |
Arnold, FJ; Murphy, RB; Schuster, DI | 1 |
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC | 1 |
Hara, H; Harada, Y; Sukamoto, T | 1 |
Chaki, S; Imagawa, Y; Muramatsu, M; Okuyama, S; Otomo, S; Tanaka, M | 1 |
London, ED | 1 |
Shi, GG; Xu, SF | 1 |
Bouchard, P; Dumont, Y; Fournier, A; Quirion, R; St-Pierre, S | 1 |
Matsuno, K; Mita, S; Senda, T | 1 |
Bergeron, R; Bouchard, P; de Montigny, C; Debonnel, G; Junien, JL; Monnet, F; Quirion, R; Roman, F | 1 |
Kobayashi, T; Matsuno, K; Mita, S; Senda, T | 1 |
Kobayashi, T; Matsuno, K; Mita, S | 1 |
Bowen, WD; Torrence-Campbell, C | 1 |
Kobayashi, T; Matsuno, K; Mita, S; Nakata, K | 1 |
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA | 1 |
Su, TP; Tsao, LI | 1 |
Ahmed, MS; Enna, SJ; Mather, A | 1 |
Baulieu, EE; Collin, T; Denavit-Saubié, M; Monnet, FP; Morin-Surun, MP | 1 |
Horikomi, K; Iizuka, K; Mita, N; Miwa, T; Nagase, H; Sakai, K; Sonehara, K; Takagi, K; Takahashi, S | 1 |
Kamei, J | 1 |
Akaike, A; Hashino, A; Kaneko, S; Katsuki, H; Kume, T; Nishikawa, H | 1 |
Bridges, S; Miller, C; Thompson, TL | 1 |
Horikomi, K; Karasawa, J; Takagi, K; Takahashi, S | 1 |
Akaike, A; Hashino, A; Kaneko, S; Katsuki, H; Kume, T; Minami, M; Nishikawa, H; Satoh, M; Taguchi, R | 1 |
Chen, CF; Chou, YC; Liao, JF; Wang, HH | 1 |
Baeyens, JM; Cobos, EJ; Del Pozo, E | 1 |
Jackson, MB; Johannessen, M; Ramachandran, S; Ramos-Serrano, A; Riemer, L; Ruoho, AE | 1 |
Kim, FJ; Marino, JC; Pasternak, GW; Schrock, JM; Spino, CM | 1 |
2 review(s) available for haloperidol and phenazocine
Article | Year |
---|---|
Studies of sigma receptors and metabolic responses to sigma ligands in the brain.
Topics: Animals; Brain; Glucose; Haloperidol; Humans; Ligands; Phenazocine; Receptors, Phencyclidine; Receptors, sigma | 1993 |
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases | 1999 |
70 other study(ies) available for haloperidol and phenazocine
Article | Year |
---|---|
Analgesia in terminal malignant disease.
Topics: Administration, Oral; Haloperidol; Humans; Palliative Care; Phenazocine; Terminal Care | 1979 |
Sigma ligand-induced emesis in the pigeon.
Topics: Animals; Apomorphine; Columbidae; Dextromethorphan; Dizocilpine Maleate; Dopamine Agents; Guanidines; Haloperidol; Male; Pentobarbital; Phenazocine; Piperidines; Propranolol; Psychotropic Drugs; Pyrimidines; Receptors, Opioid; Receptors, sigma; Vomiting | 1992 |
Tris inhibits (+)-[3H]SKF-10,047 binding to sigma receptors.
Topics: Animals; Dizocilpine Maleate; Haloperidol; Liver; Male; Phenazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stereoisomerism; Tritium; Tromethamine | 1992 |
Involvement of haloperidol-sensitive sigma-sites in antitussive effects.
Topics: Animals; Antitussive Agents; Capsaicin; Cough; Dose-Response Relationship, Drug; Drug Interactions; Guanidines; Haloperidol; Injections, Intraperitoneal; Male; Phenazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stereoisomerism | 1992 |
Effect of haloperidol and clozapine on (+)SKF 10,047-induced dopamine release: role of 5-HT3 receptors.
Topics: Animals; Brain; Clozapine; Corpus Striatum; Dopamine; Haloperidol; Male; Nucleus Accumbens; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1992 |
Heterogeneous binding of sigma radioligands in the rat brain and liver: possible relationship to subforms of cytochrome P-450.
Topics: Animals; Brain; Cytochrome P-450 Enzyme System; Guanidines; Haloperidol; Kinetics; Ligands; Liver; Male; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Subcellular Fractions | 1991 |
Effects of drugs that bind to PCP and sigma receptors on punished responding.
Topics: Animals; Buspirone; Dizocilpine Maleate; Haloperidol; Learning; Male; Pentobarbital; Phenazocine; Phencyclidine; Punishment; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1991 |
[3H]DTG and [3H](+)-3-PPP label pharmacologically distinct sigma binding sites in guinea pig brain membranes.
Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Membranes; Phenazocine; Phenytoin; Piperidines; Receptors, Opioid; Receptors, sigma | 1991 |
Two subtypes of enteric non-opioid sigma receptors in guinea-pig cholinergic motor neurons.
Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Carbazoles; Dextromethorphan; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Motor Neurons; Myenteric Plexus; Parasympathetic Nervous System; Phenazocine; Pyrimidines; Receptors, Opioid; Receptors, sigma | 1991 |
Behavioural and electoencephalographic interactions between haloperidol and PCP/sigma ligands in the rat.
Topics: 2-Amino-5-phosphonovalerate; Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Catalepsy; Electroencephalography; Haloperidol; Isoquinolines; Kinetics; Male; Phenazocine; Phencyclidine; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Spiperone | 1991 |
Similar behavioural effects of sigma agonists and PCP-like non-competitive NMDA antagonists in guinea-pigs.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Dizocilpine Maleate; Dopamine Agents; Dopamine Antagonists; Ergolines; Female; Guanidines; Guinea Pigs; Haloperidol; Ketamine; Male; Motor Activity; N-Methylaspartate; Pentazocine; Phenazocine; Phencyclidine; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride | 1991 |
Solubilization and characterization of haloperidol-sensitive (+)-[3H]SKF-10,047 binding sites (sigma sites) from rat liver membranes.
Topics: Animals; Binding Sites; Cell Membrane; Cholic Acids; Culture Techniques; Haloperidol; Liver; Male; Phenazocine; Rats; Rats, Inbred F344; Receptors, Opioid; Receptors, sigma; Tritium | 1991 |
The lack of utility of the rat vas deferens as a functional bioassay for sigma ligands.
Topics: Animals; Binding Sites; Biological Assay; Electric Stimulation; Guanidines; Guinea Pigs; Haloperidol; Male; Muscle Contraction; Pentazocine; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Vas Deferens | 1991 |
Multiple vascular effects of sigma and PCP ligands: inhibition of amine uptake and contractile responses.
Topics: Animals; Cocaine; Desoxycorticosterone; Haloperidol; Male; Norepinephrine; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Serotonin; Vasoconstriction | 1990 |
Evidence against an involvement of the haloperidol-sensitive sigma recognition site in the discriminative stimulus properties of (+)-N-allylnormetazocine ((+)-SKF 10,047).
Topics: Animals; Aspartic Acid; Binding, Competitive; Dibenzocycloheptenes; Discrimination, Psychological; Dizocilpine Maleate; Guanidines; Haloperidol; Male; Mice; N-Methylaspartate; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Seizures | 1990 |
Haloperidol competitively inhibits the binding of (+)-[3H]SKF-10,047 to sigma sites.
Topics: Animals; Binding, Competitive; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Male; Phenazocine; Rats; Receptors, Opioid; Receptors, sigma | 1990 |
Haloperidol-sensitive (+)[3H]SKF-10,047 binding sites (sigma sites) exhibit a unique distribution in rat brain subcellular fractions.
Topics: 5'-Nucleotidase; Animals; Brain; Choline O-Acetyltransferase; Haloperidol; In Vitro Techniques; Male; Ouabain; Phenazocine; Rats; Rats, Inbred F344; Receptors, Opioid; Receptors, sigma; Subcellular Fractions; Synaptosomes | 1990 |
Effect of selective sigma ligands on duodenal alkaline secretion in the rat.
Topics: Animals; Atropine; Bicarbonates; Dose-Response Relationship, Drug; Duodenum; Guanidines; Haloperidol; Injections, Intravenous; Intestinal Mucosa; Intestinal Secretions; Male; Naloxone; Phenazocine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Yohimbine | 1990 |
Differential modulation by cations of sigma and phencyclidine binding sites in rat brain.
Topics: Animals; Binding Sites; Brain; Cations; Dose-Response Relationship, Drug; Haloperidol; Ligands; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Sigma Factor; Tritium | 1990 |
Substitution and antagonism in rats trained to discriminate (+)-N-allylnormetazocine from saline.
Topics: Animals; Binding Sites; Butaclamol; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Haloperidol; Male; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1989 |
Evidence for a model of activation of central sigma systems.
Topics: Animals; Benzazepines; Benzomorphans; Butaclamol; Carbazoles; Dopamine Antagonists; Haloperidol; Kinetics; Male; Models, Biological; Motor Activity; Naltrexone; Narcotic Antagonists; Phenazocine; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Sulpiride | 1989 |
Differential regulation of sigma and PCP receptors after chronic administration of haloperidol and phencyclidine in mice.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Hallucinogens; Haloperidol; Male; Mice; Mice, Inbred Strains; Phenazocine; Phencyclidine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Time Factors | 1989 |
[Adaptive changes in sigma and phencyclidine receptors during the long-term use of haloperidol and raclopride in rats].
Topics: Adaptation, Physiological; Animals; Apomorphine; Behavior, Animal; Drug Interactions; Haloperidol; Ketamine; Phenazocine; Phencyclidine; Raclopride; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Salicylamides; Time Factors; Tritium | 1989 |
Neuropeptide Y and peptide YY interact with rat brain sigma and PCP binding sites.
Topics: Animals; Brain Chemistry; Haloperidol; In Vitro Techniques; Male; Neuropeptide Y; Pentazocine; Peptide YY; Peptides; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1989 |
Discriminative stimulus properties of a sigma receptor agonist in the rat: role of monoamine systems.
Topics: Animals; Apomorphine; Biogenic Amines; Brain Chemistry; Discrimination, Psychological; Haloperidol; Male; Methysergide; Phenazocine; Rats; Rats, Inbred F344; Receptors, Opioid; Receptors, Opioid, delta; Yohimbine | 1987 |
A role for receptors of N-methyl-D-aspartic acid in the discriminative stimulus properties of phencyclidine.
Topics: Animals; Discrimination, Psychological; Generalization, Stimulus; Haloperidol; Male; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter | 1987 |
Steroid binding at sigma receptors suggests a link between endocrine, nervous, and immune systems.
Topics: Animals; Brain; Endocrine Glands; Guinea Pigs; Haloperidol; Immunity; Male; Nervous System Physiological Phenomena; Phenazocine; Receptors, Opioid; Receptors, sigma; Spleen; Steroids | 1988 |
Evidence for a non-opioid sigma binding site in the guinea-pig myenteric plexus.
Topics: Animals; Binding, Competitive; Cell Membrane; Chlorpromazine; Cyclazocine; Ethylketocyclazocine; Guinea Pigs; Haloperidol; Imipramine; Male; Myenteric Plexus; Phenazocine; Propranolol; Receptors, Opioid; Receptors, sigma | 1988 |
A comparison of the binding of sigma opioids and phencyclidine, and the interaction with antipsychotic drugs in rat brain membranes.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Brain; Corpus Striatum; Endorphins; Haloperidol; In Vitro Techniques; Male; Membranes; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, delta | 1986 |
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice.
Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid | 1987 |
Pharmacological specificity of some psychotomimetic and antipsychotic agents for the sigma and PCP binding sites.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Haloperidol; In Vitro Techniques; Male; Phenazocine; Phencyclidine; Piperidines; Psychotropic Drugs; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma | 1988 |
Correlation of inhibitory potencies of putative antagonists for sigma receptors in brain and spleen.
Topics: Animals; Antipsychotic Agents; Brain Chemistry; Carbazoles; Guinea Pigs; Haloperidol; In Vitro Techniques; Isoquinolines; Male; Phenazocine; Piperazines; Pyrimidines; Receptors, Opioid; Receptors, sigma; Spleen; Tritium | 1988 |
Demonstration of non-opioid sigma binding with (d)3H-SKF 10047 in guinea pig brain.
Topics: Animals; Binding Sites; Brain; Brain Chemistry; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Phenazocine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism; Tritium | 1985 |
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism | 1987 |
[3H]PCP-3-OH and (+)[3H]SKF 10047 binding sites in rat brain membranes: evidence of multiplicity.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Haloperidol; In Vitro Techniques; Phenazocine; Phencyclidine; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine | 1987 |
Stereoselective behavioral effects of N-allylnormetazocine in pigeons and squirrel monkeys.
Topics: Animals; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Morphine; Naloxone; Phenazocine; Phencyclidine; Reinforcement Schedule; Saimiri; Stereoisomerism | 1985 |
The effects of phencyclidine and N-allylnormetazocine on midbrain dopamine neuronal activity.
Topics: Animals; Haloperidol; Iontophoresis; Male; Mesencephalon; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Stereoisomerism | 1984 |
Sigma opiates and certain antipsychotic drugs mutually inhibit (+)-[3H] SKF 10,047 and [3H]haloperidol binding in guinea pig brain membranes.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Brain; Cell Membrane; Corpus Striatum; Guinea Pigs; Haloperidol; Kinetics; Male; Narcotics; Phenazocine; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Spiperone | 1984 |
Feeding systems in Chinese hamsters.
Topics: Animals; Brain; Calcitonin; Circadian Rhythm; Cricetinae; Cyclazocine; Diabetes Mellitus; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Feeding Behavior; Haloperidol; Mesocricetus; Naloxone; Peptide Fragments; Phenazocine; Sincalide; Starvation | 1984 |
Discriminative stimulus effects of prototype opiate receptor agonists in monkeys.
Topics: Animals; Apomorphine; Cyclazocine; Ethylketocyclazocine; Female; Generalization, Stimulus; Haloperidol; Male; Models, Biological; Morphine; Naltrexone; Phenazocine; Prejudice; Receptors, Opioid; Saimiri | 1980 |
Phencyclidine-induced inhibition of striatal acetylcholine release: comparisons with mu, kappa, and sigma opiate agonists.
Topics: Acetylcholine; Animals; Corpus Striatum; Cyclazocine; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains | 1984 |
Pharmacological evidence for the involvement of sigma sites in DTG-induced contralateral circling in rats.
Topics: Animals; Anticonvulsants; Behavior, Animal; Carbazoles; Dose-Response Relationship, Drug; Guanidines; Haloperidol; Injections, Spinal; Male; Motor Activity; Phenazocine; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, sigma; Salicylamides | 1995 |
Phosphorylation of synapsin I and dynamin in rat forebrain synaptosomes: modulation by sigma (sigma) ligands.
Topics: Animals; Anticonvulsants; Dynamins; GTP Phosphohydrolases; Guanidines; Haloperidol; In Vitro Techniques; Microtubules; Pentazocine; Phenazocine; Phosphorylation; Prosencephalon; Rats; Receptors, sigma; Synapsins; Synaptosomes | 1995 |
Characterization of a (+)-azidophenazocine-sensitive sigma receptor on splenic lymphocytes.
Topics: Affinity Labels; Animals; Binding Sites; Binding, Competitive; Female; Haloperidol; Interferons; Lymphocytes; Mice; Mice, Inbred C57BL; Phenazocine; Piperidines; Receptors, sigma; Spleen | 1993 |
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc | 1994 |
Purification, pharmacological characterization and photoaffinity labeling of sigma receptors from rat and bovine brain.
Topics: Animals; Binding Sites; Cattle; Cerebellum; Dopamine Agonists; Haloperidol; Male; Phenazocine; Piperidines; Rats; Receptors, sigma | 1995 |
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma | 1995 |
Characterization of specific (+)-[3H]N-allylnormetazocine and [3H]1,3-di(2-tolyl)guanidine binding sites in porcine gastric fundic mucosa.
Topics: Animals; Binding Sites; Gastric Fundus; Gastric Mucosa; Guanidines; Haloperidol; Phenazocine; Receptors, sigma; Swine | 1994 |
FH-510, a potent and selective ligand for rat brain sigma recognition sites.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain; Carbazoles; Dopamine; Haloperidol; Male; Mice; Phenazocine; Phencyclidine; Propylamines; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma; Stereotyped Behavior | 1993 |
Effect of phencyclidine on contraction of porcine coronary vessel strips.
Topics: Animals; Biological Assay; Coronary Vessels; Dextromethorphan; Dizocilpine Maleate; Haloperidol; In Vitro Techniques; Muscle, Smooth, Vascular; Myocardial Contraction; Phenazocine; Phencyclidine; Receptors, Phencyclidine; Receptors, sigma; Swine | 1993 |
Evidence for in vivo interactions between neuropeptide Y-related peptides and sigma receptors in the mouse hippocampal formation.
Topics: Animals; Binding, Competitive; Epinephrine; Gastrointestinal Hormones; Haloperidol; Hippocampus; Kinetics; Male; Mice; Mice, Inbred Strains; Neuropeptide Y; Neurotensin; Peptide YY; Peptides; Phenazocine; Receptors, sigma; Vasoactive Intestinal Peptide | 1993 |
Correlation between potentiation of neurogenic twitch contraction and benzomorphan sigma receptor binding potency in the mouse vas deferens.
Topics: Animals; Antiparkinson Agents; Brain; Drug Synergism; Guinea Pigs; Haloperidol; Ligands; Male; Mice; Phenazocine; Piperidines; Receptors, sigma; Spasm; Vas Deferens | 1993 |
In vivo modulation of sigma receptor sites by calcitonin gene-related peptide in the mouse and rat hippocampal formation: radioligand binding and electrophysiological studies.
Topics: Animals; Antipsychotic Agents; Calcitonin Gene-Related Peptide; Dopamine Antagonists; Electrophysiology; Haloperidol; Hippocampus; In Vitro Techniques; Iontophoresis; Male; Membranes; Mice; Narcotics; Neuropeptide Y; Pentazocine; Phenazocine; Pyramidal Cells; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma | 1995 |
Involvement of sigma 1 receptor in (+)-N-allylnormetazocine-stimulated hippocampal cholinergic functions in rats.
Topics: Acetylcholine; Amnesia; Analysis of Variance; Animals; Haloperidol; Hippocampus; Male; Muscarinic Antagonists; Phenazocine; Rats; Rats, Wistar; Receptors, sigma; Scopolamine; Stereoisomerism; Stimulation, Chemical; Synaptic Transmission | 1995 |
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens | 1996 |
Differential solubilization of rat liver sigma 1 and sigma 2 receptors: retention of sigma 2 sites in particulate fractions.
Topics: Animals; Binding, Competitive; Cell Fractionation; Cell Membrane; Cholic Acids; Detergents; Guanidines; Haloperidol; In Vitro Techniques; Liver; Male; Pentazocine; Phenazocine; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Solubility; Subcellular Fractions | 1996 |
Enhancement of acetylcholine release by SA4503, a novel sigma 1 receptor agonist, in the rat brain.
Topics: Acetylcholine; Animals; Brain; Haloperidol; Male; Phenazocine; Piperazines; Rats; Rats, Wistar; Receptors, sigma; Tacrine; Tetrodotoxin | 1996 |
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium | 1997 |
Naloxone-sensitive, haloperidol-sensitive, [3H](+)SKF-10047-binding protein partially purified from rat liver and rat brain membranes: an opioid/sigma receptor?
Topics: Animals; Antipsychotic Agents; Brain; Haloperidol; Liver; Naloxone; Phenazocine; Radioligand Assay; Rats; Receptors, Opioid | 1997 |
Binding of [3H]desglycinyl remacemide to rat brain membranes: association with the benzomorphan attachment site of the N-methyl-D-aspartic acid receptor channel.
Topics: Animals; Antipsychotic Agents; Benzomorphans; Binding Sites; Brain Chemistry; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Haloperidol; Male; Membrane Proteins; Neurons; Phenazocine; Phencyclidine; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Subcellular Fractions; Tritium | 1999 |
Intracellular sigma1 receptor modulates phospholipase C and protein kinase C activities in the brainstem.
Topics: Action Potentials; Animals; Antipsychotic Agents; Brain Stem; Cell Membrane; Cytoplasm; GTP-Binding Proteins; Guinea Pigs; Haloperidol; In Vitro Techniques; Isoenzymes; Ligands; Male; Pentazocine; Pertussis Toxin; Phenazocine; Protein Kinase C; Protein Kinase C beta; Receptors, sigma; Respiratory Mechanics; Reverse Transcriptase Polymerase Chain Reaction; Type C Phospholipases; Virulence Factors, Bordetella | 1999 |
Pharmacological profile of MS-377, a novel antipsychotic agent with selective affinity for sigma receptors.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Dopamine Agonists; Free Radical Scavengers; Guinea Pigs; Haloperidol; Head Movements; Male; Mice; Phenazocine; Phencyclidine; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, sigma; Risperidone; Serotonin; Serotonin Antagonists; Stereotyped Behavior; Sulpiride; Tartrates | 1999 |
Involvement of direct inhibition of NMDA receptors in the effects of sigma-receptor ligands on glutamate neurotoxicity in vitro.
Topics: Animals; Cells, Cultured; Cerebral Cortex; Glutamic Acid; Haloperidol; Ligands; Neurons; Neuroprotective Agents; Phenazocine; Propylamines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, delta; RNA, Messenger | 2000 |
Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands.
Topics: Animals; Antipsychotic Agents; Carbazoles; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Haloperidol; Ligands; Neurons; Nomifensine; Nucleus Accumbens; Phenazocine; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, sigma; Spiperone; Sulpiride; Synaptosomes; Tritium | 2001 |
Effects of sigma(1) receptor ligand MS-377 on D(2) antagonists-induced behaviors.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Catalepsy; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Female; Haloperidol; Male; Mice; Nootropic Agents; Phenazocine; Piperazines; Pyridines; Pyrrolidines; Rats; Receptors, sigma; Serotonin Antagonists; Sigma-1 Receptor; Sulpiride; Tartrates | 2002 |
Antagonism of NMDA receptors by sigma receptor ligands attenuates chemical ischemia-induced neuronal death in vitro.
Topics: 2-Amino-5-phosphonovalerate; Animals; Calcium; Cell Hypoxia; Cell Survival; Cells, Cultured; Cerebral Cortex; Cyclopentanes; Deoxyglucose; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fetus; Glucose; Glutamates; Haloperidol; Neurons; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sodium Azide | 2002 |
Dimemorfan enhances acetylcholine release from rat hippocampal slices.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Antipsychotic Agents; Atropine; Carbachol; Cholinergic Agonists; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Hippocampus; In Vitro Techniques; Male; Morphinans; Muscarinic Antagonists; Phenazocine; Potassium Chloride; Rats; Tritium | 2004 |
Phenytoin differentially modulates the affinity of agonist and antagonist ligands for sigma 1 receptors of guinea pig brain.
Topics: Allosteric Regulation; Animals; Anisoles; Anticonvulsants; Binding, Competitive; Brain; Dextromethorphan; Drug Interactions; Ethylenediamines; Guinea Pigs; Haloperidol; Ligands; Male; Morpholines; Neurons; Phenazocine; Phenytoin; Piperazines; Piperidines; Progesterone; Propylamines; Receptors, sigma; Synaptic Transmission | 2005 |
Voltage-gated sodium channel modulation by sigma-receptors in cardiac myocytes and heterologous systems.
Topics: Adenosine Triphosphate; Animals; Antipsychotic Agents; Cell Line; Chlorocebus aethiops; COS Cells; Guanosine Triphosphate; Haloperidol; Humans; Kidney; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Proteins; Myocytes, Cardiac; Narcotics; NAV1.5 Voltage-Gated Sodium Channel; Patch-Clamp Techniques; Pentazocine; Phenazocine; Receptors, sigma; RNA, Small Interfering; Sodium; Sodium Channels | 2009 |
Inhibition of tumor cell growth by Sigma1 ligand mediated translational repression.
Topics: Cell Line, Tumor; Cell Proliferation; Cell Size; Haloperidol; Humans; Ligands; Morpholines; Neoplasms; Phenazocine; Protein Biosynthesis; Receptors, sigma; RNA Cap-Binding Proteins; Sigma-1 Receptor | 2012 |