haloperidol and n-n-propylnorapomorphine

haloperidol has been researched along with n-n-propylnorapomorphine in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-199027 (67.50)18.7374
1990's11 (27.50)18.2507
2000's2 (5.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH1
Seeman, P; Titeler, M1
Crumly, HJ; Goldberg, LI; Hinshaw, WB; Pinder, RM1
Baldessarini, RJ; Bissette, G; Campbell, A; Kilts, CD; Levant, B; Nemeroff, CB1
Baldessarini, RJ; Campbell, A; Neumeyer, JL; Yeghiayan, S1
Elazar, Z; Fuchs, S1
Bergmeier, S; Caprathe, BW; Heffner, TG; Humblet, CC; Jaen, JC; Meltzer, LT; Pugsley, TA; Tecle, H; Wise, LD1
Cox, RF; Waszczak, BL1
Heyer, EJ1
Fuchs, S; Kanety, H1
Costall, B; Domeney, AM; Naylor, RJ4
Claustre, Y; Fage, D; Scatton, B; Zivkovic, B1
Agnati, LF; Battistini, N; Benfenati, F; Calza, L; Fuxe, K; Giardino, L; Guidolin, D; Ruggeri, M; Vanderhaeghen, JJ; Zoli, M1
Allikmets, L; Maimets, M; Nurk, A; Soosaar, A; Vasar, E1
Battaglia, G; Creese, I; Norman, AB1
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Schweitzer, JW1
DeWald, HA; Hawkins, ES; Heffner, TG; Meltzer, LT; Pugsley, TA; Reynolds, DM; Wise, LD1
Kohjimoto, Y; Kuwaki, T; Nomura, Y; Ono, T; Satoh, H; Shibayama, F; Shirakawa, K1
Cullen, M; Kazmi, SM; Mishra, RK; Rajakumar, G; Ramwani, J; Ross, GM; Srivastava, LK1
Korf, J; Loopuijt, LD; Sebens, JB1
Fleminger, S; Hall, MD; Jenner, P; Kilpatrick, G; Mann, S; Marsden, CD; Rupniak, NM2
Fleminger, S; Hall, MD; Jenner, P; Kerwin, R; Marsden, CD; Murugaiah, K; Rupniak, NM1
Angeby, K; Florvall, L; Hall, H; Köhler, C; Lindbom, LO; Magnusson, O; Ogren, SO1
MacKenzie, RG; Zigmond, MJ1
Cools, AR; van Rossum, JM1
Hall, MD; Jenner, P; Kilpatrick, G; Marsden, CD; Rupniak, NM1
Fratta, W; Gessa, GL; Napoli-Farris, L1
Baggio, G; Ferrari, F1
Leysen, JE; Van Gompel, P1
Baldessarini, RJ; Ben-Jonathan, N; Campbell, A; Ellingboe, J; Neumeyer, JL; Zong, R1
Evans, DL; Figur, LM; Lahti, RA; Stratman, NC1
He, SF; Xie, Z1
Geurts, M; Hermans, E; Maloteaux, JM1
Hwang, DR; Kegeles, LS; Laruelle, M1
Emms, F; Freedman, SB; Knowles, MR; Marwood, R; McAllister, G; Patel, S; Seabrook, GR1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1

Reviews

1 review(s) available for haloperidol and n-n-propylnorapomorphine

ArticleYear
Multiple receptors for brain dopamine in behavior regulation: concept of dopamine-E and dopamine-I receptors.
    Life sciences, 1980, Oct-06, Volume: 27, Issue:14

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Behavior, Animal; Brain; Cats; Corpus Striatum; Dextroamphetamine; Dopamine; Ergot Alkaloids; Fluorescence; Haloperidol; Histocytochemistry; Humans; Hyperkinesis; Hypothermia; Methyltyrosines; Mice; Motor Activity; Naphthalenes; Neurons; Nucleus Accumbens; Rats; Receptors, Adrenergic, alpha; Receptors, Dopamine; Reserpine; Septal Nuclei; Stereotyped Behavior; Tetrahydronaphthalenes

1980

Other Studies

39 other study(ies) available for haloperidol and n-n-propylnorapomorphine

ArticleYear
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
Antiparkinsonian drug doses and neuroleptic receptors.
    Experientia, 1978, Nov-15, Volume: 34, Issue:11

    Topics: Animals; Antiparkinson Agents; Apomorphine; Bromocriptine; Cattle; Caudate Nucleus; Haloperidol; In Vitro Techniques; Receptors, Dopamine; Spiperone; Tritium

1978
Dopamine-like renal and mesenteric vasodilation caused by apomorphine 6-propylnorapomorphine and 2-amino-6, 7-dihydroxy-1,2,3,4-tetrahydronaphthalene.
    Nature, 1976, Feb-19, Volume: 259, Issue:5544

    Topics: Animals; Apomorphine; Dogs; Dopamine; Femoral Artery; Haloperidol; Kidney; Mesenteric Arteries; Naphthols; Receptors, Drug; Regional Blood Flow; Structure-Activity Relationship; Vasodilator Agents

1976
Effects of the isomers of N-n-propylnorapomorphine and haloperidol on regional concentrations of neurotensin in rat brain.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1991, Volume: 4, Issue:1

    Topics: Animals; Apomorphine; Brain; Dopamine Agents; Haloperidol; Isomerism; Male; Neurotensin; Organ Specificity; Rats; Rats, Inbred Strains; Reference Values

1991
Selective antidopaminergic effects of S(+)N-n-propylnoraporphines in limbic versus extrapyramidal sites in rat brain: comparisons with typical and atypical antipsychotic agents.
    Psychopharmacology, 1991, Volume: 103, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Clozapine; Dibenzothiazepines; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Limbic System; Male; Motor Activity; Pyramidal Tracts; Quetiapine Fumarate; Rats; Rats, Inbred Strains

1991
Vanadate inhibits agonist binding to D2 dopamine receptor.
    Journal of molecular neuroscience : MN, 1991, Volume: 3, Issue:1

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Corpus Striatum; Dopamine Agents; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Kinetics; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Vanadates

1991
4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Apomorphine; Chemical Phenomena; Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Haloperidol; Male; Molecular Conformation; Molecular Structure; Motor Activity; Neurons; Pyridines; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Structure-Activity Relationship; Substantia Nigra; Thermodynamics; Thiazoles

1990
Irreversible receptor inactivation reveals differences in dopamine receptor reserve between A9 and A10 dopamine systems: an electrophysiological analysis.
    Brain research, 1990, Nov-26, Volume: 534, Issue:1-2

    Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Dopamine Antagonists; Electrophysiology; Evoked Potentials; Haloperidol; Kinetics; Male; Neurons; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reference Values; Substantia Nigra; Tegmentum Mesencephali

1990
Dopamine antagonists reduce spontaneous electrical activity in cultured mammalian neurons from ventral mesencephalon.
    Brain research, 1986, Sep-24, Volume: 382, Issue:2

    Topics: Action Potentials; Animals; Apomorphine; Butaclamol; Cells, Cultured; Dibenzocycloheptenes; Dopamine Antagonists; Fetus; Haloperidol; Membrane Potentials; Mesencephalon; Mice; Mice, Inbred ICR; Neurons; Receptors, Dopamine; Spinal Cord; Spiperone

1986
Immuno-photoaffinity labeling of the D2-dopamine receptor.
    Biochemical and biophysical research communications, 1988, Sep-15, Volume: 155, Issue:2

    Topics: Affinity Labels; Animals; Apomorphine; Azides; Butaclamol; Cattle; Corpus Striatum; Haloperidol; Immunologic Techniques; Kinetics; Molecular Weight; Photochemistry; Receptors, Dopamine; Spiperone

1988
Desenkephalin-gamma-endorphin is an antagonist of the hyperactivity response induced by infusion of dopamine into the nucleus accumbens of rat and ventral striatum of marmoset.
    Neuropharmacology, 1989, Volume: 28, Issue:11

    Topics: Animals; Apomorphine; beta-Endorphin; Callitrichinae; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Female; Fluphenazine; Haloperidol; Injections; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei

1989
Relative selectivity of 6,7-dihydroxy-2-dimethylaminotetralin, N-n-propyl-3-(3-hydroxyphenyl)piperidine, N-n-propylnorapomorphine and pergolide as agonists at striatal dopamine autoreceptors and postsynaptic dopamine receptors.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:2

    Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Haloperidol; Homovanillic Acid; Male; Naphthalenes; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sodium Oxybate; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase

1985
Evidence for cholecystokinin-dopamine receptor interactions in the central nervous system of the adult and old rat. Studies on their functional meaning.
    Annals of the New York Academy of Sciences, 1985, Volume: 448

    Topics: Aging; Animals; Apomorphine; Brain; Cholecystokinin; Haloperidol; Male; Neurons; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sincalide; Tyrosine 3-Monooxygenase

1985
Comparison of motor depressant effects of caerulein and N-propylnorapomorphine in mice.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Animals; Apomorphine; Ceruletide; Depression, Chemical; Exploratory Behavior; Fenclonine; Haloperidol; Hydroxydopamines; Male; Mice; Motor Activity; Nerve Endings; Oxidopamine; Receptors, Dopamine; Receptors, Serotonin; Sincalide; Spiperone

1986
Differential recovery rates of rat D2 dopamine receptors as a function of aging and chronic reserpine treatment following irreversible modification: a key to receptor regulatory mechanisms.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:5

    Topics: Aging; Animals; Apomorphine; Corpus Striatum; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Kinetics; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Dopamine; Receptors, Dopamine D2; Reserpine; Spiperone

1987
Chronic haloperidol does not alter agonist affinity for dopamine receptors in vitro.
    European journal of pharmacology, 1985, Mar-12, Volume: 109, Issue:3

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Haloperidol; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
6- and 8-hydroxy-3,4-dihydro-3-(dipropylamino)-2H-1-benzopyrans. Dopamine agonists with autoreceptor selectivity.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: 4-Butyrolactone; Animals; Apomorphine; Benzopyrans; Brain; Chromans; Dopamine; Haloperidol; In Vitro Techniques; Neurons; Rats; Receptors, Dopamine; Reserpine

1988
Effect of long-term dosing with tiapride on brain dopamine receptors and metabolism in rats. Comparative study with sulpiride and haloperidol.
    Japanese journal of pharmacology, 1987, Volume: 44, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Apomorphine; Benzamides; Brain Chemistry; Dopamine; Haloperidol; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Sulpiride; Tiapamil Hydrochloride

1987
Characterization of high-affinity dopamine D2 receptors and modulation of affinity states by guanine nucleotides in cholate-solubilized bovine striatal preparations.
    Journal of neurochemistry, 1986, Volume: 47, Issue:5

    Topics: Animals; Apomorphine; Binding, Competitive; Cattle; Cholic Acid; Cholic Acids; Computers; Corpus Striatum; Domperidone; Guanine Nucleotides; Guanylyl Imidodiphosphate; Haloperidol; Kinetics; Receptors, Dopamine; Solubility; Spiperone

1986
In vivo labeling of dopamine receptors: light microscopic localization at the cellular level by means of dipping autoradiography with the agonist (3H)N-n-propylnorapomorphine.
    Journal of neural transmission, 1987, Volume: 68, Issue:1-2

    Topics: Animals; Apomorphine; Autoradiography; Cerebral Cortex; Corpus Striatum; Dopamine; Haloperidol; Male; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine

1987
Chronic treatment with clozapine, unlike haloperidol, does not induce changes in striatal D-2 receptor function in the rat.
    Biochemical pharmacology, 1985, Aug-01, Volume: 34, Issue:15

    Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Male; Mastication; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Thioxanthenes; Tritium

1985
Long-term adaptive changes in striatal dopamine function in response to chronic neuroleptic intake in rats.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Glutamates; Glutamic Acid; Haloperidol; Rats; Receptors, Dopamine; Spiperone; Sulpiride

1983
Long-term consequences of antagonism by neuroleptics of behavioural events occurring during mesolimbic dopamine infusion.
    Neuropharmacology, 1984, Volume: 23, Issue:3

    Topics: Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Dopamine; Dopamine Antagonists; Female; Haloperidol; Injections; Methysergide; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Sulpiride; Time Factors

1984
Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Benzamides; Binding, Competitive; Brain Chemistry; Catalepsy; Chlorpromazine; Dogs; Female; Haloperidol; Histocytochemistry; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Remoxipride; Spiperone; Sulpiride; Thioridazine; Vomiting

1984
High- and low-affinity states of striatal D2 receptors are not affected by 6-hydroxydopamine or chronic haloperidol treatment.
    Journal of neurochemistry, 1984, Volume: 43, Issue:5

    Topics: Animals; Apomorphine; Butaclamol; Cinanserin; Corpus Striatum; Dopamine; Guanylyl Imidodiphosphate; Haloperidol; Hydroxydopamines; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1984
Differential effects of continuous administration for 1 year of haloperidol or sulpiride on striatal dopamine function in the rat.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Acetylcholine; Animals; Apomorphine; Body Weight; Corpus Striatum; Haloperidol; Humans; Kinetics; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride

1984
Differential alterations in striatal dopamine receptor sensitivity induced by repeated administration of clinically equivalent doses of haloperidol, sulpiride or clozapine in rats.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Haloperidol; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sulpiride

1984
A comparison of the behavioural consequences of chronic stimulation of dopamine receptors in the nucleus accumbens of rat brain effected by a continuous infusion or by single daily injections.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:1

    Topics: Animals; Apomorphine; Dopamine; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei

1983
Stimulation of dopamine autoreceptors elicits "premature ejaculation" in rats.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 20, Issue:1

    Topics: Animals; Apomorphine; Copulation; Domperidone; Dopamine Antagonists; Ejaculation; Female; Haloperidol; Lisuride; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal

1984
Influence of lisuride on morphine withdrawal signs in the rat: a dopamine-mimetic effect.
    Psychopharmacology, 1982, Volume: 78, Issue:4

    Topics: Aggression; Animals; Apomorphine; Dopamine; Ergolines; Haloperidol; Humans; Lisuride; Male; Morphine Dependence; Naloxone; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Sulpiride

1982
Stimulation of rat spontaneous locomotion by low doses of haloperidol and (-)-sulpiride: importance of animal selection and measurement technique.
    European journal of pharmacology, 1983, Jun-17, Volume: 90, Issue:4

    Topics: Animals; Apomorphine; Dextroamphetamine; Female; Haloperidol; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride

1983
Effects of proteolytic enzymes and monovalent ions demonstrate protease-sensitive and protease-insensitive stereospecific binding sites on dopaminergic receptors in rat striatum.
    Biochemical pharmacology, 1982, Apr-01, Volume: 31, Issue:7

    Topics: Animals; Apomorphine; Cations, Monovalent; Corpus Striatum; Female; Haloperidol; In Vitro Techniques; Membranes; Peptide Hydrolases; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1982
Effects of aporphine isomers on rat prolactin.
    Neuroscience letters, 1994, Aug-01, Volume: 176, Issue:2

    Topics: Animals; Apomorphine; Aporphines; Dopamine Agonists; Haloperidol; Male; Prolactin; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Stereoisomerism

1994
Dopamine D4 versus D2 receptor selectivity of dopamine receptor antagonists: possible therapeutic implications.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Animals; Apomorphine; Butyrophenones; Cell Line; Chlorpromazine; Clozapine; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Raclopride; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Trifluoperazine

1993
[Inhibition of voltage-dependent K+ currents in rat C6 glioma cells by haloperidol and R(-)-NPA].
    Sheng li xue bao : [Acta physiologica Sinica], 1997, Volume: 49, Issue:1

    Topics: Animals; Apomorphine; Biological Transport, Active; Brain Neoplasms; Dopamine Agonists; Dopamine Antagonists; Glioma; Haloperidol; Potassium Channels; Rats; Tumor Cells, Cultured

1997
Enhanced striatal dopamine D(2) receptor-induced [35S]GTPgammaS binding after haloperidol treatment.
    European journal of pharmacology, 1999, Oct-08, Volume: 382, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Catalepsy; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Sulfur Radioisotopes; Tritium; Up-Regulation

1999
(-)-N-[(11)C]propyl-norapomorphine: a positron-labeled dopamine agonist for PET imaging of D(2) receptors.
    Nuclear medicine and biology, 2000, Volume: 27, Issue:6

    Topics: Animals; Apomorphine; Binding, Competitive; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Magnetic Resonance Imaging; Male; Organometallic Compounds; Papio; Propionates; Radioactive Tracers; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Sensitivity and Specificity; Tissue Distribution; Tomography, Emission-Computed

2000
Expression and pharmacological characterization of the human D3 dopamine receptor.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:1

    Topics: Animals; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dopamine; Dopamine Antagonists; GTP-Binding Proteins; Guanine Nucleotides; Humans; Potassium Channels; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Second Messenger Systems; Sulpiride

1994
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007