haloperidol has been researched along with metoclopramide in 142 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 79 (55.63) | 18.7374 |
1990's | 25 (17.61) | 18.2507 |
2000's | 20 (14.08) | 29.6817 |
2010's | 17 (11.97) | 24.3611 |
2020's | 1 (0.70) | 2.80 |
Authors | Studies |
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Hasegawa, O; Hirata, Y; Iwanami, S; Takashima, M; Usuda, S | 1 |
Calderó, JM; del Río, J; García, E; Lasheras, B; Monge, A; Palop, JA; Peña, MC; Roca, J; Romero, G | 1 |
Topliss, JG; Yoshida, F | 1 |
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA | 1 |
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY | 2 |
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X | 1 |
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL | 1 |
Bergström, F; Giordanetto, F; Rehngren, M; Tunek, A; Wan, H | 1 |
Andricopulo, AD; Moda, TL; Montanari, CA | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Ahman, M; Holmén, AG; Wan, H | 1 |
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Boriss, H; Braggio, S; Corbioli, S; Fontana, S; Helmdach, L; Longhi, R; Schiller, J; Vinco, F | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Bellman, K; Knegtel, RM; Settimo, L | 1 |
Artursson, P; Mateus, A; Matsson, P | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Bateman, DN; Dutta, DK; McClelland, HA; Rawlins, MD | 2 |
Beckett, PR; Nahorski, SR; Roberts, DJ; Salazar, W | 1 |
Hope, W; Majewski, H; McCulloch, MW; Rand, MJ; Story, DF | 2 |
Fozard, JR; Palfreyman, MG | 1 |
Buyniski, JP; Doran, KM; Gylys, JA | 1 |
Besser, GM; Delitala, G; Jones, A; Stubbs, WA; Thorner, MO; Yeo, T | 1 |
Ba, A; Diop Mar, I; Sow, A | 1 |
Berry, MS; MacDonald, JF | 1 |
Costall, B; Naylor, RJ | 3 |
Roufogalis, BD; Thornton, M; Wade, DN | 1 |
Baxter, MG; Miller, AA; Wheatley, PL | 1 |
Miller, R | 1 |
Cassimos, C; Danielides, B; Malaka-Zafiriu, K; Tsiuris, J | 1 |
Lincoln, DW; Mason, CA | 1 |
Marsden, CD; Pycock, C; Tarsy, D | 1 |
Cianchetti, C; Corsini, GU; Mangoni, A; Zompo, MD | 1 |
Gu, SF | 1 |
Destrade, C; Messier, C; Mrabet, O | 2 |
Joshi, RS; Marco, LA | 1 |
Monrad, L; Ottesen, S | 1 |
Lauterbach, EC | 1 |
Borzecki, Z; Kaliszuk, S; Swies, Z | 1 |
Iakimovskiĭ, AF | 2 |
Gupta, PP; Srivastava, AK; Srivastava, YP; Verma, RB | 1 |
Décio, RC; Francischetti, I; Frussa-Filho, R; Haber, VA; Onimaru, AT; Soares, CG | 1 |
Cabib, S; Castellano, C; Cestari, V; Filibeck, U; Puglisi-Allegra, S | 1 |
Francom, M | 1 |
Evans, AM; Green, KL | 2 |
O'Neill, WM | 1 |
Cohen, PR; Cowen, PJ; McCance, SL | 1 |
Ljungberg, T | 2 |
Pfaus, JG; Phillips, AG | 1 |
Davis, KL; Guerin, JJ; Halperin, R | 1 |
Blackburn, JR; Phillips, AG | 1 |
Copeland, PA; Thomas, P | 1 |
Berényi, E; Kiss, E | 1 |
Ståhle, L; Ungerstedt, U | 1 |
Blaha, CD; Lane, RF | 1 |
Cools, AR; Ellenbroek, BA; Honig, WM; Peeters, BW | 1 |
Altar, CA; Boyar, WC | 1 |
Barrett, RJ; Proakis, AG; Taylor, DR; Wright, KF | 1 |
Starr, BS; Starr, MS | 1 |
Costall, B; Gunning, SJ; Naylor, RJ; Tyers, MB | 1 |
Murakami, M; Ota, K | 1 |
Fujiwara, M; Nishikawa, H; Yokotani, K | 1 |
Cui, XW; Li, BH; Shen, DL; Yang, XY | 1 |
Bhalla, S; Mehta, VL; Wafai, ZA | 1 |
Rogers, J; Venning, M | 1 |
Aziz, L; Forsling, ML; Matziari, C | 1 |
Henke, PG; Ray, A; Sullivan, RM | 1 |
Calvo Fernández, J; Castro-Gago, M; Couce Pico, M; López Rois, F; Novo, I | 1 |
Clopton, JK; Curtin, JC; Gordon, JH; Koller, WC | 1 |
Cvitanović, B; Geber, J; Gjuris, V; Ivanović, D; Mise, S; Rotkvić, I; Sikirić, P; Suchanek, E; Tućan-Foretić, M | 1 |
Fahn, S; Hassan, MN; Higgins, D; Kuhn, C; Reches, A | 1 |
Gerber, R; Gerhardt, S; Liebman, JM | 1 |
Hellenbrecht, D; Saller, R | 1 |
Crammer, JL; Crane, G; Rosser, RM | 1 |
Boublik, JH; Funder, JW | 1 |
Besser, GM; Delitala, G; Grossman, A; Stubbs, WA; Yeo, T | 1 |
Hall, N; Liebman, JM; Prowse, J | 1 |
Bracha, HS; Davis, KL; Kendler, KS | 1 |
Anderson, RJ; Carp, JS | 1 |
Azuma, H; Iwai, K; Kikuta, M; Liu, HJ; Oshino, N; Sato, K | 1 |
Pi, EH; Simpson, GM | 1 |
Borsini, F; Nowakowska, E; Samanin, R | 1 |
Davis, KL; Kendler, KS | 1 |
Jungmann, E; Schöffling, K; Schwedes, U; Usadel, KH; Wächtler, M | 1 |
Fang, VS; Shian, LR | 1 |
Costall, B; Naylor, RJ; Tan, CC | 1 |
Bernardi, MM; Palermo-Neto, J | 1 |
Daw, NW; Jensen, RJ | 1 |
Bernardi, MM; Palermo-Neto, J; Saban, R | 1 |
Cariffe, P; Gala, KV; Grunberg, SM; Jamin, D; Johnson, K; Krailo, M; Lampenfeld, M; Strych, D | 1 |
Bendesky, RJ; Hichens, M; King, SW; Mangel, AW; Martin, GE; Remy, DC; Robinson, JL; Taylor, DA; Williams, M; Yarbrough, GG | 1 |
Idoipe, A; Idoipe, C; Sanz, F | 1 |
Bruera, ED; Chacón, RD; Roca, E | 1 |
Benson, DI; Kuhn, CM; Meyerson, LR; Stanley, M; Virgilio, J; Wazer, D | 1 |
Angrist, BM | 1 |
Fenton, HM; Liebman, JM | 1 |
Arushanian, EB; Smirnova, LE; Tolpyshev, BA | 1 |
Kim, HS; Liebman, J; Welch, JJ | 1 |
Besser, GM; Delitala, G; Grossman, A; Hathway, NR; Yeo, T | 1 |
Barbieri, C; Caldara, R; Ferrari, C; Romussi, M | 1 |
Golub, M; Sowers, DK; Sowers, JR; Tuck, M | 1 |
Asin, KE; Wirtshafter, D | 1 |
Archer, T | 1 |
Demenge, P; Duarte, GP; Lahlou, S | 1 |
Lynch, AM; See, RE; Sorg, BA | 1 |
Barbosa-Coutinho, LM; Barros, HM; Moraes, JT; Oliveira, MC | 1 |
Deutch, AY; Elsworth, JD; Iadarola, MJ; Lewis, DA; Redmond, DE; Roth, RH; Whitehead, RE | 1 |
Graybiel, AM; Hiroi, N | 1 |
Frussa-Filho, R; Palermo-Neto, J; Vital, MB | 1 |
Chinen, CC; Frussa-Filho, R | 1 |
Li, Y; Matsuda, H; Yoshikawa, M | 1 |
Azuara, ML; Barcia, E; Negro, S; Reyes, R; Sánchez, Y | 1 |
Arnold, RM; Buss, MK | 1 |
Weschules, DJ | 1 |
Andersen, D; Gottrup, F; Hovendal, CP | 1 |
Davidson, A; Hunter, C; Jankovic, J; Kenney, C | 1 |
Agovic, MS; Banerjee, SP; Lidsky, TI; Yablonsky-Alter, E | 1 |
Apfel, CC; Kolodzie, K | 1 |
Feng, YB; McAlonan, GM; Sze, SC; Wang, D; Wang, XM; Wong, HK; Zhang, L; Zhang, ZJ | 1 |
Brunetti, AE; Nardulli, P; Russano, M; Silvestris, N | 1 |
Agar, M; Currow, DC; To, TH; Yates, P | 1 |
Brosnan, EA; Landman, WJ; Mittal, A; Mittal, DL | 1 |
Baker, TW; Beninger, RJ; Florczynski, MM | 1 |
Kaminska, E; Leppert, W; Mikolajczak, P; Okulicz-Kozaryn, I; Szulc, M | 1 |
Bruner, DI; Frumkin, K; Gaffigan, ME; Pritchard, A; Wason, C | 1 |
Fisher, H | 1 |
Grześkowiak, T; Jeszka-Skowron, M; Rusińska-Roszak, D; Zaporowska-Stachowiak, I; Zgoła-Grześkowiak, A | 1 |
Hirai, T; Kose, E; Seki, T; Yasuno, N | 1 |
4 review(s) available for haloperidol and metoclopramide
Article | Year |
---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
[Recent advances in the management of chemotherapy-induced emesis].
Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Domperidone; Dronabinol; Drug Therapy, Combination; Haloperidol; Humans; Metoclopramide; Nausea; Neoplasms; Prochlorperazine; Vomiting | 1986 |
Atypical neuroleptics: clozapine and the benzamides in the prevention and treatment of tardive dyskinesia.
Topics: Antipsychotic Agents; Benzamides; Clinical Trials as Topic; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Prospective Studies; Schizophrenia; Sulpiride; Tiapamil Hydrochloride | 1983 |
Nausea and vomiting after office-based anesthesia.
Topics: Anesthesia; Antiemetics; Droperidol; Haloperidol; Humans; Incidence; Metoclopramide; Neurokinin-1 Receptor Antagonists; Postoperative Nausea and Vomiting; Risk Factors; Scopolamine; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists | 2009 |
7 trial(s) available for haloperidol and metoclopramide
Article | Year |
---|---|
Metoclopramide and haloperidol in tardive dyskinesia.
Topics: Aged; Antipsychotic Agents; Dose-Response Relationship, Drug; Double-Blind Method; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Male; Metoclopramide; Middle Aged; Receptors, Dopamine | 1979 |
[A double-blind study of metoclopramide in the treatment of schizophrenia and determination of prolactin].
Topics: Adolescent; Adult; Basal Ganglia Diseases; Double-Blind Method; Female; Haloperidol; Humans; Male; Metoclopramide; Middle Aged; Prolactin; Schizophrenia | 1992 |
[Benefit and risk of high-dose metoclopramide in comparison to high-dose haloperidol or triflupromazine in cisplatin-induced vomiting].
Topics: Cisplatin; Dose-Response Relationship, Drug; Haloperidol; Humans; Metoclopramide; Neoplasms; Risk; Triflupromazine; Vomiting | 1985 |
Atypical neuroleptics: clozapine and the benzamides in the prevention and treatment of tardive dyskinesia.
Topics: Antipsychotic Agents; Benzamides; Clinical Trials as Topic; Clozapine; Dibenzazepines; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Prospective Studies; Schizophrenia; Sulpiride; Tiapamil Hydrochloride | 1983 |
Comparison of the antiemetic effect of high-dose intravenous metoclopramide and high-dose intravenous haloperidol in a randomized double-blind crossover study.
Topics: Adult; Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Double-Blind Method; Drug Evaluation; Female; Haloperidol; Humans; Injections, Intravenous; Male; Metoclopramide; Neoplasms; Random Allocation; Vomiting | 1984 |
Optimal control of nausea and vomiting with a three-drug antiemetic regimen with aprepitant in metastatic pancreatic cancer patients treated with first-line modified FOLFIRINOX.
Topics: Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Aprepitant; Benztropine; Camptothecin; Dexamethasone; Drug Combinations; Female; Fluorouracil; Haloperidol; Humans; Leucovorin; Male; Metoclopramide; Morpholines; Nausea; Organoplatinum Compounds; Pancreatic Neoplasms; Vomiting | 2013 |
A Randomized Controlled Trial of Intravenous Haloperidol vs. Intravenous Metoclopramide for Acute Migraine Therapy in the Emergency Department.
Topics: Acute Disease; Adolescent; Adult; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Double-Blind Method; Emergency Service, Hospital; Female; Haloperidol; Humans; Injections, Intravenous; Male; Metoclopramide; Middle Aged; Migraine Disorders; Pain Measurement; Prospective Studies; Severity of Illness Index; Treatment Outcome | 2015 |
132 other study(ies) available for haloperidol and metoclopramide
Article | Year |
---|---|
Synthesis and neuroleptic activity of benzamides. Cis-N-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-(methylamino)benzamide and related compounds.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Benzamides; Catalepsy; Humans; Rats; Stereotyped Behavior; Structure-Activity Relationship | 1981 |
Synthesis of 2-piperazinylbenzothiazole and 2-piperazinylbenzoxazole derivatives with 5-HT3 antagonist and 5-HT4 agonist properties.
Topics: Animals; Benzothiazoles; Binding, Competitive; Cerebral Cortex; Female; Gastric Emptying; Granisetron; Guinea Pigs; Ileum; Male; Molecular Structure; Mucous Membrane; Ondansetron; Piperazines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles | 1994 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water | 2001 |
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding | 2002 |
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.
Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water | 2003 |
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution | 2004 |
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration | 2004 |
High-throughput screening of drug-brain tissue binding and in silico prediction for assessment of central nervous system drug delivery.
Topics: Animals; Brain; Central Nervous System Agents; Dialysis; Hydrophobic and Hydrophilic Interactions; In Vitro Techniques; Mice; Models, Statistical; Protein Binding; Quantitative Structure-Activity Relationship; Rats | 2007 |
Hologram QSAR model for the prediction of human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2007 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship | 2008 |
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry | 2009 |
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
Brain tissue binding of drugs: evaluation and validation of solid supported porcine brain membrane vesicles (TRANSIL) as a novel high-throughput method.
Topics: Absorption; Albumins; Animals; Brain; Brain Chemistry; Cell Membrane; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; In Vitro Techniques; Lipids; Male; Microdialysis; Pharmaceutical Preparations; Protein Binding; Rats; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Swine; Tissue Distribution | 2011 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation | 2014 |
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization | 2014 |
[Clebopride, a new orthopramide with potent and selective central antidopaminergic properties].
Topics: Alprenolol; Animals; Benzamides; Dihydroergotoxine; Haloperidol; Metoclopramide; Piperidines; Rats; Receptors, Dopamine; Sulpiride | 1978 |
Modulation of sympathetic transmission by neuronally-released dopamine.
Topics: Animals; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Dopamine; Ergonovine; Haloperidol; In Vitro Techniques; Metoclopramide; Neurons; Norepinephrine; Phentolamine; Rabbits; Stimulation, Chemical; Sympathetic Nervous System; Synaptic Transmission | 1979 |
Metoclopramide antagonism of 5-hydroxytryptophan-induced "wet-dog" shake behaviour in the rat.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Brain Chemistry; Carbidopa; Haloperidol; Male; Methysergide; Metoclopramide; Quipazine; Rats; Serotonin; Time Factors | 1979 |
Antagonism of cisplatin induced emesis in the dog.
Topics: Animals; Antiemetics; Chlorpromazine; Cisplatin; Dogs; Dronabinol; Female; Haloperidol; Indoles; Male; Metoclopramide; Piperidines; Vomiting | 1979 |
Action of dopamine receptor agonists and antagonists, and a serotonin antagonist on prolactin release from isolated rat pituitary cell columns [proceedings].
Topics: Animals; Chlorpromazine; Dopamine; Ergot Alkaloids; Haloperidol; In Vitro Techniques; Metoclopramide; Pituitary Gland; Prolactin; Rats; Receptors, Dopamine | 1979 |
The effect of metoclopramide and haloperidol on tardive dyskinesia [proceedings].
Topics: Aged; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Male; Metoclopramide; Middle Aged | 1979 |
[Rare and unusual drug intolerances, apropos of 6 cases].
Topics: Adolescent; Adult; Basal Ganglia Diseases; Chemical and Drug Induced Liver Injury; Child; Drug Hypersensitivity; Erythromycin; Female; Haloperidol; Humans; Liver; Male; Metoclopramide; Trismus | 1977 |
Further identification of multiple responses mediated by dopamine in the CNS of Planorbis corneus.
Topics: Animals; Apomorphine; Central Nervous System; Dopamine; Evoked Potentials; Fluphenazine; Ganglia; Haloperidol; In Vitro Techniques; Lysergic Acid Diethylamide; Metoclopramide; Mollusca; Tubocurarine | 1978 |
A comparison of the abilities of typical neuroleptic agents and of thioridazine, clozapine, sulpiride and metoclopramide to antagonise the hyperactivity induced by dopamine applied intracerebrally to areas of the extrapyramidal and mesolimbic systems.
Topics: Animals; Brain; Clozapine; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Fluphenazine; Haloperidol; Limbic System; Male; Metoclopramide; Pimozide; Rats; Stereotaxic Techniques; Sulpiride; Thioridazine; Tranquilizing Agents | 1976 |
Specificity of the dopamine sensitive adenylate cyclase for antipsychotic antagonists.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Haloperidol; Male; Metoclopramide; Rats; Sulpiride | 1976 |
Comparative studies on the effects of metoclopramide and some known neuroleptics on the EEG of the conscious rat [proceedings].
Topics: Animals; Chlorpromazine; Dextroamphetamine; Electroencephalography; Haloperidol; Male; Metoclopramide; Pimozide; Rats; Tranquilizing Agents | 1976 |
Metoclopramide and dopamine receptor blockade.
Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Dopamine; Haloperidol; Injections; Male; Metoclopramide; Mice; Procaine; Receptors, Drug; Stimulation, Chemical | 1976 |
Urinary D-glucaric acid excretion in children with dystonic reactions caused by antiemetic drugs.
Topics: Adolescent; Antiemetics; Child; Chlorpromazine; Dimenhydrinate; Glucaric Acid; Haloperidol; Humans; Metoclopramide; Muscle Tonus; Sugar Acids; Thiethylperazine | 1975 |
Proceedings: Visualization of retino-hypothalamic projections in the rat.
Topics: Animals; Dopamine; Female; Haloperidol; Lactation; Metoclopramide; Milk Ejection; Pregnancy; Rats | 1975 |
Inhibition of circling behavior by neuroleptic drugs in mice with unilateral 6-hydroxydopamine lesions of the striatum.
Topics: Animals; Apomorphine; Basal Ganglia Diseases; Behavior; Biogenic Amines; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Chlorpromazine; Clozapine; Corpus Striatum; Dextroamphetamine; Diazepam; Dopamine; Haloperidol; Humans; Hydroxydopamines; Levodopa; Male; Metoclopramide; Mice; Motor Activity; Pentobarbital; Phenoxybenzamine; Pimozide; Promethazine; Stereotyped Behavior; Tranquilizing Agents | 1975 |
Therapeutical efficacy of a combination of apomorphine with sulpiride or metoclopramide in Parkinsonism.
Topics: Adult; Apomorphine; Drug Therapy, Combination; Haloperidol; Humans; Male; Metoclopramide; Parkinson Disease; Sleep; Sulpiride; Vomiting | 1976 |
Locomotor bias produced by intra-accumbens injection of dopamine agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dextroamphetamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Injections; Male; Metoclopramide; Mice; Mice, Inbred BALB C; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior | 1992 |
A ketamine-induced rat model of tardive dyskinesia.
Topics: Animals; Antipsychotic Agents; Clozapine; Dizocilpine Maleate; Dyskinesia, Drug-Induced; Haloperidol; Ketamine; Metoclopramide; Pharynx; Rats; Rats, Inbred Strains; Stereotyped Behavior; Tongue | 1992 |
[Morphine-antiemetics mixtures for continuous subcutaneous infusion in terminal cancer].
Topics: Antiemetics; Drug Combinations; Drug Stability; Haloperidol; Humans; Infusion Pumps, Implantable; Metoclopramide; Morphine; Neoplasms; Pain, Intractable; Palliative Care; Terminal Care | 1992 |
Haloperidol-induced dystonia and parkinsonism on discontinuing metoclopramide: implications for differential thalamocortical activity.
Topics: Adult; Brain; Drug Therapy, Combination; Dystonia; Female; Haloperidol; Humans; Metoclopramide; Parkinson Disease, Secondary; Substance Withdrawal Syndrome | 1992 |
The influence of agonists and antagonists of dopaminergic system on the formation of audiogenic seizures in rats during the ethanol abstinence period.
Topics: Amantadine; Animals; Bromocriptine; Dopamine Agents; Dopamine Antagonists; Ethanol; Haloperidol; Male; Metoclopramide; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Sulpiride | 1990 |
[Neuropharmacological activity of cerucal and haloperidol by intraperitoneal and intrastriatal administration in rats].
Topics: Animals; Avoidance Learning; Catalepsy; Corpus Striatum; Haloperidol; Injections; Injections, Intraperitoneal; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains | 1991 |
Characterization of dopamine receptors involved in central thermoregulation in rabbits.
Topics: Animals; Body Temperature Regulation; Female; Haloperidol; Male; Metoclopramide; Rabbits; Receptors, Dopamine | 1991 |
Antitumor effects of dopaminergic blockers in mice bearing Ehrlich tumors.
Topics: Analysis of Variance; Animals; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Ehrlich Tumor; Domperidone; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Haloperidol; Metoclopramide; Mice | 1991 |
D1 and D2 receptor antagonists differently affect cocaine-induced locomotor hyperactivity in the mouse.
Topics: Animals; Benzazepines; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Metoclopramide; Mice; Mice, Inbred C57BL; Motor Activity; Receptors, Dopamine D1; Receptors, Dopamine D2; Stimulation, Chemical; Sulpiride | 1991 |
Compounding nausea aid.
Topics: Benztropine; Chemistry, Pharmaceutical; Dexamethasone; Diphenhydramine; Drug Combinations; Drug Compounding; Haloperidol; Humans; Lorazepam; Metoclopramide; Nausea; Suppositories; Vomiting | 1991 |
The action of dopamine receptor antagonists on the secretory response of the cockroach salivary gland in vitro.
Topics: Animals; Benzazepines; Binding, Competitive; Chlorpromazine; Cockroaches; Domperidone; Dopamine; Dopamine Antagonists; Haloperidol; Metoclopramide; Salivary Glands; Sulpiride | 1990 |
The neuroleptic malignant syndrome.
Topics: Adult; Female; Haloperidol; Humans; Metoclopramide; Neuroleptic Malignant Syndrome; Postoperative Complications; Uterine Cervical Neoplasms; Vomiting | 1990 |
Characterization of the dopamine receptor mediating the hyperpolarization of cockroach salivary gland acinar cells in vitro.
Topics: Animals; Benzazepines; Chlorpromazine; Cockroaches; Domperidone; Electric Stimulation; Haloperidol; In Vitro Techniques; Kinetics; Metoclopramide; Receptors, Dopamine; Salivary Glands; Sulpiride | 1990 |
[Circling behavior produced by the unilateral intra-accumbens injection of dopaminergic agonist and two dopaminergic antagonists in mice].
Topics: Animals; Apomorphine; Behavior, Animal; Haloperidol; Male; Metoclopramide; Mice; Mice, Inbred BALB C; Motor Activity; Nucleus Accumbens; Septal Nuclei | 1989 |
Lithium increases 5-HT-mediated prolactin release.
Topics: Clomipramine; Haloperidol; Humans; Hydrocortisone; Infusions, Intravenous; Lithium; Male; Metoclopramide; Prolactin; Serotonin; Time Factors | 1989 |
Dopamine D-2 antagonists reverse apomorphine-induced decreased water intake in the rat: prediction of antipsychotic drugs with few extrapyramidal side-effects?
Topics: Animals; Antipsychotic Agents; Apomorphine; Domperidone; Dose-Response Relationship, Drug; Drinking Behavior; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1989 |
Differential effects of dopamine receptor antagonists on the sexual behavior of male rats.
Topics: Animals; Antipsychotic Agents; Clozapine; Ejaculation; Female; Haloperidol; Male; Metoclopramide; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal; Sulpiride | 1989 |
Regional differences in the induction of behavioral supersensitivity by prolonged treatment with atypical neuroleptics.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Body Weight; Clozapine; Corpus Striatum; Dopamine; Haloperidol; Humans; Injections; Metoclopramide; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride | 1989 |
Blockade of acquisition of one-way conditioned avoidance responding by haloperidol and metoclopramide but not by thioridazine or clozapine: implications for screening new antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; Avoidance Learning; Clozapine; Dibenzazepines; Drug Evaluation, Preclinical; Haloperidol; Male; Metoclopramide; Rats; Thioridazine | 1989 |
Control of gonadotropin release in the Atlantic croaker (Micropogonias undulatus): evidence for lack of dopaminergic inhibition.
Topics: Animals; Bromocriptine; Domperidone; Dopamine; Female; Fishes; Gonadotropin-Releasing Hormone; Gonadotropins; Haloperidol; Male; Metoclopramide; Pimozide; Sex Factors | 1989 |
[Management of vomiting induced by polychemotherapy in Hodgkin's disease].
Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Dose-Response Relationship, Drug; Haloperidol; Hodgkin Disease; Humans; Methylprednisolone; Metoclopramide; Vomiting | 1989 |
Effects of neuroleptic drugs on the inhibition of exploratory behaviour induced by a low dose of apomorphine: implications for the identity of dopamine receptors.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Drug Interactions; Exploratory Behavior; Flupenthixol; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1986 |
Chronic treatment with classical and atypical antipsychotic drugs differentially decreases dopamine release in striatum and nucleus accumbens in vivo.
Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Haloperidol; Male; Metoclopramide; Nucleus Accumbens; Promethazine; Rats; Rats, Inbred Strains; Septal Nuclei; Thioridazine | 1987 |
Blockade by neuroleptics of water intake and operant responding for water in the rat: anhedonia, motor deficit, or both?
Topics: Animals; Antipsychotic Agents; Conditioning, Operant; Consummatory Behavior; Drinking; Haloperidol; Male; Metoclopramide; Motivation; Motor Activity; Rats; Rats, Inbred Strains; Sulpiride | 1987 |
The paw test: a behavioural paradigm for differentiating between classical and atypical neuroleptic drugs.
Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Desipramine; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Forelimb; Haloperidol; Hindlimb; Male; Metoclopramide; Morphine; Motor Activity; Rats; Rats, Inbred Strains; Thioridazine | 1987 |
Modulation of in vivo dopamine release by D2 but not D1 receptor agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Benzopyrans; Brain; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Homovanillic Acid; Kinetics; Male; Metoclopramide; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1987 |
Involvement of dopamine receptor subtypes in dopaminergic modulation of aldosterone secretion in rats.
Topics: Aldosterone; Animals; Blood; Domperidone; Dopamine; Haloperidol; Male; Metoclopramide; Osmolar Concentration; Potassium; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sodium; Sulpiride | 1987 |
Behavioural interactions involving D1 and D2 dopamine receptors in non-habituated mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Drug Interactions; Haloperidol; Male; Metoclopramide; Mice; Motor Activity; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1987 |
The effect of GR38032F, novel 5-HT3-receptor antagonist on gastric emptying in the guinea-pig.
Topics: Animals; Gastric Emptying; Guinea Pigs; Haloperidol; Imidazoles; Metoclopramide; Ondansetron; Serotonin Antagonists | 1987 |
Catecholamine receptors involved in the inhibitory effects of dopamine on vagally stimulated gastric acid secretion and mucosal blood flow in rats.
Topics: Animals; Domperidone; Dopamine; Gastric Acid; Gastric Mucosa; Haloperidol; Male; Metoclopramide; Phentolamine; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Catecholamine; Regional Blood Flow; Sulpiride; Vagus Nerve | 1987 |
[Effects of haloperidol, chlorpromazine, metoclopramide and ascorbic acid on adrenergic salivation and lacrimation in mice at an ambient temperature of 30 degrees C].
Topics: Animals; Ascorbic Acid; Chlorpromazine; Epinephrine; Female; Haloperidol; Male; Metoclopramide; Mice; Norepinephrine; Salivation; Tears; Temperature | 1985 |
Attenuation of pentylenetetrazol kindling of epileptogenesis in rats by dopaminergic agents.
Topics: Amantadine; Amphetamine; Animals; Epilepsy; Haloperidol; Kindling, Neurologic; Levodopa; Male; Metoclopramide; Pentylenetetrazole; Rats | 1988 |
Continuous subcutaneous infusion: flexible option in symptom control.
Topics: Anxiety; Female; Haloperidol; Humans; Infusion Pumps; Infusions, Parenteral; Metoclopramide; Middle Aged; Morphine; Nausea; Pain; Rectal Neoplasms; Spinal Neoplasms | 1988 |
A comparison of the vasopressin response of rats to intraperitoneal and intravenous administration of hypertonic saline, and the effect of opioid and aminergic antagonists.
Topics: Animals; Haloperidol; Infusions, Intravenous; Injections, Intraperitoneal; Male; Metoclopramide; Narcotic Antagonists; Osmolar Concentration; Rats; Rats, Inbred Strains; Saline Solution, Hypertonic; Sodium Chloride; Sympatholytics; Vasopressins | 1988 |
Effects of intra-amygdalar dopamine agonists and antagonists on gastric stress lesions in rats.
Topics: Amygdala; Animals; Apomorphine; Cold Temperature; Dopamine; Dopamine Antagonists; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Restraint, Physical; Stomach Ulcer; Stress, Psychological | 1988 |
[Drug-induced extrapyramidal syndrome. Apropos of 22 cases].
Topics: Adolescent; Antiemetics; Basal Ganglia Diseases; Benzamides; Child; Child, Preschool; Female; Haloperidol; Humans; Infant; Male; Metoclopramide; Syndrome | 1987 |
Chronic autoreceptor blockade and neuroleptic-induced dopamine receptor hypersensitivity.
Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; Haloperidol; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Synapses | 1987 |
Dopamine antagonists induce gastric lesions in rats.
Topics: Animals; Bromocriptine; Domperidone; Dopamine Antagonists; Female; Haloperidol; Levodopa; Male; Metoclopramide; Rats; Rats, Inbred Strains; Stomach Ulcer | 1986 |
Pharmacologic evaluation of dopaminergic receptor blockade by metoclopramide.
Topics: Animals; Behavior, Animal; Catalepsy; Dopamine; Haloperidol; Male; Metoclopramide; Motor Activity; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior | 1986 |
SCH 23390 dissociated from conventional neuroleptics in apomorphine climbing and primate acute dyskinesia models.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Benzimidazoles; Chlorpromazine; Chlorprothixene; Drug Synergism; Dyskinesia, Drug-Induced; Haloperidol; Male; Metoclopramide; Mice; Motor Activity; Saimiri; Stereotyped Behavior | 1985 |
The nucleus amygdaloideus centralis and neuroleptic activity in the rat.
Topics: Amygdala; Animals; Behavior; Benzoates; Butyrophenones; Catalepsy; Dextroamphetamine; Dibenzazepines; Dibenzothiazepines; Dose-Response Relationship, Drug; Fluphenazine; Haloperidol; Humans; Male; Metoclopramide; Piperidines; Rats; Stereotyped Behavior; Time Factors; Tranquilizing Agents | 1974 |
Blood levels and management of lithium treatment.
Topics: Administration, Oral; Adult; Aged; Carbimazole; Delayed-Action Preparations; Dementia; Depression; Diabetes Insipidus; Female; Gastrointestinal Motility; Haloperidol; Humans; Hypothyroidism; Lithium; Male; Metoclopramide; Middle Aged; Obesity; Polyuria; Propantheline; Tablets; Thirst; Thyroxine; Time Factors | 1974 |
Mesolimbic involvement with behavioural effects indicating antipsychotic activity.
Topics: Animals; Behavior, Animal; Catalepsy; Dextroamphetamine; Dibenzothiazepines; Dose-Response Relationship, Drug; Electrodes, Implanted; Fluphenazine; Haloperidol; Humans; Limbic System; Male; Metoclopramide; Morphine; Piperidines; Rats; Spiro Compounds; Stereotaxic Techniques; Stereotyped Behavior; Tranquilizing Agents | 1974 |
Interaction of dopamine receptor ligands with subtypes of the opiate receptor.
Topics: Animals; Binding, Competitive; Brain; Bromocriptine; Dopamine Antagonists; Drug Interactions; Haloperidol; In Vitro Techniques; Ligands; Male; Membranes; Metoclopramide; Naloxone; Pimozide; Prochlorperazine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Tritium | 1984 |
Chlorpromazine, haloperidol, metoclopramide and domperidone release prolactin through dopamine antagonism at low concentrations but paradoxically inhibit prolactin release at high concentrations.
Topics: Animals; Antipsychotic Agents; Benzimidazoles; Cells, Cultured; Chlorpromazine; Domperidone; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Metoclopramide; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats | 1980 |
Effects of various catecholamine receptor antagonists, muscle relaxation and physical hindrance on shuttlebox self-stimulation.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Clozapine; Haloperidol; Male; Methocarbamol; Metoclopramide; Muscle Relaxants, Central; Prazosin; Rats; Rats, Inbred F344; Reaction Time; Receptors, Dopamine; Self Stimulation | 1982 |
Dopamine autoreceptor and postsynaptic receptor blocking potency of neuroleptics.
Topics: Animals; Antipsychotic Agents; Apomorphine; Fluphenazine; Haloperidol; Male; Metoclopramide; Mice; Molindone; Motor Activity; Receptors, Dopamine; Sulpiride; Synapses | 1982 |
Dopamine receptor-mediated depression of spinal monosynaptic transmission.
Topics: Action Potentials; Animals; Apomorphine; Cats; Ergolines; Female; Haloperidol; Lisuride; Male; Metoclopramide; Phentolamine; Receptors, Dopamine; Spinal Cord; Synapses; Synaptic Transmission | 1982 |
[Suppressive effects of lisuride on the synthesis, release and metabolism of dopamine in rat brain].
Topics: Animals; Apomorphine; Brain; Depression, Chemical; Dihydroergotoxine; Dopamine; Ergolines; Female; Haloperidol; Histocytochemistry; Homovanillic Acid; Lisuride; Metoclopramide; Nucleus Accumbens; Olfactory Bulb; Rats; Sulpiride; Tyrosine 3-Monooxygenase | 1982 |
Effect of repeated treatment with desipramine in the behavioral "despair" test in rats: antagonism by "atypical" but not "classical" neuroleptics or antiadrenergic drugs.
Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Butyrophenones; Chlorpromazine; Clonidine; Clozapine; Depressive Disorder; Desipramine; Dibenzazepines; Haloperidol; Humans; Male; Metoclopramide; Phentolamine; Prazosin; Propranolol; Rats; Sulpiride | 1984 |
Acute and chronic effects of neuroleptic drugs on plasma and brain homovanillic acid in the rat.
Topics: Animals; Antipsychotic Agents; Brain Chemistry; Chlorpromazine; Fluphenazine; Haloperidol; Homovanillic Acid; Loxapine; Male; Metoclopramide; Molindone; Phenylacetates; Rats; Rats, Inbred Strains; Sulpiride | 1984 |
Evidence for a modulatory role of dopamine in sympathetic transmission.
Topics: Animals; Arteries; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Dopamine; Ear; Ergonovine; Haloperidol; Metoclopramide; Norepinephrine; Phentolamine; Rabbits; Receptors, Dopamine; Sympathetic Nervous System; Synaptic Transmission; Time Factors; Tritium | 1980 |
The effect of metoclopramide and haloperidol on plasma renin activity and aldosterone levels in rats.
Topics: Aldosterone; Animals; Diet, Sodium-Restricted; Drug Administration Schedule; Furosemide; Haloperidol; Kinetics; Male; Metoclopramide; Rats; Rats, Inbred Strains; Renin | 1983 |
A serotonergic mechanism of the prolactin-stimulating action of metoclopramide.
Topics: Adrenalectomy; Animals; Blood Proteins; Dopamine; Dose-Response Relationship, Drug; Fenclonine; Haloperidol; Hypothalamus; Male; Metoclopramide; Prolactin; Rats; Serotonin | 1981 |
Neuronally mediated contraction responses of guinea-pig stomach smooth muscle preparations: modification by benzamide derivatives does not reflect a dopamine antagonist action.
Topics: Animals; Benzamides; Domperidone; Electric Stimulation; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Receptors, Dopamine; Stomach | 1984 |
Kinetic analysis of central nervous system supersensitivity induced in rats by long-term haloperidol administration. Part II: KB determination.
Topics: Animals; Central Nervous System; Haloperidol; Kinetics; Metoclopramide; Rats | 1984 |
Effects of dopamine antagonists on receptive fields of brisk cells and directionally selective cells in the rabbit retina.
Topics: Animals; Dopamine Antagonists; Flupenthixol; Fluphenazine; Haloperidol; Metoclopramide; Rabbits; Receptors, Dopamine; Retina; Retinal Ganglion Cells; Sulpiride | 1984 |
Kinetic analysis of central nervous system supersensitivity induced in rats by long-term haloperidol administration. I. pA2 determination.
Topics: Animals; Apomorphine; Brain; Dose-Response Relationship, Drug; Haloperidol; Humans; Kinetics; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior | 1984 |
L-646,462, a cyproheptadine-related antagonist of dopamine and serotonin with selectivity for peripheral systems.
Topics: Animals; Apomorphine; Cyproheptadine; Domperidone; Dopamine Antagonists; Gastrointestinal Motility; Haloperidol; Homovanillic Acid; Male; Metoclopramide; Prolactin; Receptors, Serotonin; Serotonin Antagonists | 1984 |
Dopaminergic receptors in guinea-pig bladder.
Topics: Animals; Domperidone; Dopamine; Guinea Pigs; Haloperidol; In Vitro Techniques; Metoclopramide; Radioligand Assay; Receptors, Dopamine; Spiperone; Urinary Bladder | 1983 |
[Emesis due to cytostatic drugs. Update and review of our experiences].
Topics: Antineoplastic Agents; Dexamethasone; Haloperidol; Humans; Metoclopramide; Prochlorperazine; Vomiting | 1983 |
Lack of potency of metoclopramide's metabolites in various dopaminergic models.
Topics: Animals; Apomorphine; Dopamine; Fluphenazine; Haloperidol; Homovanillic Acid; Humans; Male; Metoclopramide; Prolactin; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes | 1983 |
The neurobiologically active benzamides and related compounds: some historical aspects.
Topics: Benzamides; Chlorpromazine; Haloperidol; History, 20th Century; Humans; Metoclopramide; Nervous System; Procainamide; Sulpiride | 1982 |
Self-stimulation response decrement patterns differentiate clonidine, baclofen and dopamine antagonists from drugs causing performance deficit.
Topics: Animals; Baclofen; Clonidine; Conditioning, Operant; Dopamine Antagonists; Extinction, Psychological; Haloperidol; Male; Methocarbamol; Metoclopramide; Prazosin; Rats; Rats, Inbred F344; Receptors, Dopamine; Self Stimulation | 1982 |
[Possible discrepancy between behavioral adequacy and motor automatisms in cats with phenamine-induced stereotypy].
Topics: Amphetamine; Animals; Cats; Clozapine; Dibenzazepines; Female; Haloperidol; Humans; Male; Metoclopramide; Stereotyped Behavior | 1981 |
Amphetamine-induced increases in dopaminergic single cell firing rate after haloperidol pretreatment. Correlation with extrapyramidal side effects.
Topics: Animals; Apomorphine; Brain; Clozapine; Dextroamphetamine; Dopamine; Drug Interactions; Extrapyramidal Tracts; Haloperidol; Male; Metoclopramide; Neurons; Rats; Substantia Nigra; Thioridazine | 1980 |
A comparison of the effects of four ergot derivatives on prolactin secretion by dispersed rat pituitary cells.
Topics: Animals; Dopamine; Dose-Response Relationship, Drug; Ergot Alkaloids; Female; Haloperidol; In Vitro Techniques; Metoclopramide; Perfusion; Pituitary Gland, Anterior; Prolactin; Rats | 1980 |
Effect of four dopamine receptor antagonists on gastrin secretion in healthy subjects.
Topics: Adult; Female; Gastrins; Haloperidol; Humans; Male; Metoclopramide; Middle Aged; Pimozide; Receptors, Dopamine; Secretory Rate; Sulpiride; Time Factors | 1980 |
Role of prolactin and the renin-angiotensin system in mediating dopaminergic control of aldosterone secretion in the rat.
Topics: Aldosterone; Angiotensin II; Animals; Dopamine; Dopamine Antagonists; Haloperidol; Hypophysectomy; Levodopa; Male; Metoclopramide; Prolactin; Rats; Saralasin | 1981 |
Dopamine antagonists induce fos-like-immunoreactivity in the substantia nigra and entopeduncular nucleus of the rat.
Topics: Animals; Benzazepines; Globus Pallidus; Haloperidol; Immunohistochemistry; Male; Metoclopramide; Nerve Tissue Proteins; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Substantia Nigra | 1995 |
Behavioural retardation in the neuropathology of mental retardation.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Dihydroxyphenylalanine; Dopamine Agents; Female; Haloperidol; Intellectual Disability; Learning; Male; Mercury Poisoning; Methylazoxymethanol Acetate; Metoclopramide; Mice; Motor Activity; Organotin Compounds; Pregnancy; Rats; Rats, Sprague-Dawley | 1993 |
Central dopaminergic origin of bromocriptine induced tachycardia in normotensive rats.
Topics: Adrenalectomy; Animals; Blood Pressure; Bromocriptine; Domperidone; Dopamine D2 Receptor Antagonists; Haloperidol; Heart Rate; Male; Metoclopramide; Rats; Rats, Wistar; Sulpiride; Tachycardia | 1993 |
[The effect of the activation and blockade of the neostriatal dopaminergic system on the hyperkinesis evoked in rats by the intrastriatal administration of picrotoxin].
Topics: Amphetamine; Animals; Chorea; Haloperidol; Hyperkinesis; Male; Metoclopramide; Microinjections; Myoclonus; Neostriatum; Picrotoxin; Rats; Rats, Wistar; Receptors, Dopamine; Time Factors | 1993 |
Subchronic administration of clozapine, but not haloperidol or metoclopramide, decreases dopamine D2 receptor messenger RNA levels in the nucleus accumbens and caudate-putamen in rats.
Topics: Actins; Animals; Antipsychotic Agents; Blotting, Northern; Brain Chemistry; Caudate Nucleus; Clozapine; Dopamine Antagonists; Haloperidol; Male; Metoclopramide; Nucleus Accumbens; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA, Messenger; Spiperone | 1996 |
Effect of estrogen and neuroleptics on prolactin secretion and immunoreactive prolactin cells.
Topics: Animals; Antipsychotic Agents; Estrogens; Fluphenazine; Haloperidol; Male; Metoclopramide; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Sulpiride | 1996 |
Effects of D2 dopamine receptor antagonists on Fos protein expression in the striatal complex and entorhinal cortex of the nonhuman primate.
Topics: Animals; Basal Ganglia Diseases; Caudate Nucleus; Chlorocebus aethiops; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Entorhinal Cortex; Haloperidol; Homovanillic Acid; Immunohistochemistry; Metoclopramide; Neostriatum; Proto-Oncogene Proteins c-fos; Putamen | 1996 |
Atypical and typical neuroleptic treatments induce distinct programs of transcription factor expression in the striatum.
Topics: Analysis of Variance; Animals; Antipsychotic Agents; Clozapine; Corpus Striatum; Haloperidol; Immunoblotting; Immunohistochemistry; Male; Metoclopramide; Neurons; Phenotype; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Transcription Factors | 1996 |
Monosialoganglioside increased the in vivo affinity of D2 receptors for apomorphine in supersensitive rats.
Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; G(M1) Ganglioside; Haloperidol; Kinetics; Metoclopramide; Rats; Receptors, Dopamine D2; Stereotyped Behavior; Substance Withdrawal Syndrome | 1998 |
Conditioning to injection procedures and repeated testing increase SCH 23390-induced catalepsy in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Catalepsy; Conditioning, Psychological; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Locomotion; Male; Metoclopramide; Mice; Mice, Inbred Strains; Time Factors | 1999 |
Possible involvement of dopamine and dopamine2 receptors in the inhibitions of gastric emptying by escin Ib in mice.
Topics: alpha-Methyltyrosine; Animals; Benzazepines; Domperidone; Dopamine; Dose-Response Relationship, Drug; Escin; Gastric Emptying; Haloperidol; Male; Metoclopramide; Mice; Oxidopamine; Receptors, Dopamine; Reserpine; Spiperone | 2000 |
Physical compatibility and in vivo evaluation of drug mixtures for subcutaneous infusion to cancer patients in palliative care.
Topics: Adult; Aged; Aged, 80 and over; Analgesics; Butylscopolammonium Bromide; Dexamethasone; Drug Evaluation; Drug Therapy, Combination; Female; Follow-Up Studies; Haloperidol; Humans; Infusion Pumps; Male; Metoclopramide; Midazolam; Middle Aged; Morphine; Neoplasms; Palliative Care; Spain; Tramadol; Treatment Outcome | 2002 |
Challenges in palliative care research: one experience.
Topics: Antiemetics; Attitude of Health Personnel; Diphenhydramine; Drug Combinations; Ethics Committees, Research; Haloperidol; Hospice Care; Humans; Lorazepam; Metoclopramide; Nausea; Palliative Care; Patient Selection; Randomized Controlled Trials as Topic | 2004 |
Tolerability of the compound ABHR in hospice patients.
Topics: Aged; Antiemetics; Cohort Studies; Diphenhydramine; Drug Combinations; Female; Haloperidol; Hospice Care; Humans; Lorazepam; Male; Metoclopramide; Nausea; Retrospective Studies; United States; Vomiting | 2005 |
Dopamine receptors do not influence beta2-sympathomimetic-mediated inhibition of gastric acid secretion in the dog.
Topics: Adrenergic beta-2 Receptor Agonists; Animals; Dogs; Dopamine Antagonists; Ethanolamines; Female; Gastric Acid; Gastric Mucosa; Haloperidol; Male; Metoclopramide; Pentagastrin; Stomach; Sympathomimetics | 1981 |
Metoclopramide, an increasingly recognized cause of tardive dyskinesia.
Topics: Adverse Drug Reaction Reporting Systems; Aged; Amitriptyline; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Middle Aged; Perphenazine; Retrospective Studies; Texas; Thioridazine; Time Factors | 2008 |
Mechanisms for metoclopramide-mediated sensitization and haloperidol-induced catalepsy in rats.
Topics: Animals; Behavior, Animal; Binding, Competitive; Catalepsy; Cerebral Cortex; Dizocilpine Maleate; Dopamine Antagonists; Haloperidol; Male; Metoclopramide; Neostriatum; Rats; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Spiperone | 2008 |
Not only dopamine D2 receptors involved in Peony-Glycyrrhiza Decoction, an herbal preparation against antipsychotic-associated hyperprolactinemia.
Topics: Animals; Bromocriptine; Cell Line; Disease Models, Animal; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Estradiol; Female; Glycyrrhiza; Haloperidol; Herb-Drug Interactions; Hyperprolactinemia; Metoclopramide; Paeonia; PC12 Cells; Phytotherapy; Plant Extracts; Progesterone; Prolactin; Rabbits; Rats, Sprague-Dawley; Receptors, Dopamine D2 | 2012 |
Prescribing for nausea in palliative care: a cross-sectional national survey of Australian palliative medicine doctors.
Topics: Adult; Antiemetics; Australia; Cross-Sectional Studies; Female; Haloperidol; Humans; Male; Metoclopramide; Middle Aged; Nausea; Palliative Care; Practice Patterns, Physicians'; Quality of Health Care; Surveys and Questionnaires | 2014 |
Nonopioid pharmacological management of malignant bowel obstruction: a New Zealand-wide survey.
Topics: Aged; Aged, 80 and over; Antiemetics; Cholinergic Antagonists; Dexamethasone; Enema; Female; Gastrointestinal Neoplasms; Guideline Adherence; Haloperidol; Humans; Intestinal Obstruction; Laxatives; Male; Metoclopramide; Middle Aged; New Zealand; Palliative Care; Practice Patterns, Physicians'; Scopolamine; Surveys and Questionnaires | 2014 |
Differential effects of clozapine, metoclopramide, haloperidol and risperidone on acquisition and performance of operant responding in rats.
Topics: Animals; Antipsychotic Agents; Clozapine; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Haloperidol; Male; Metoclopramide; Prefrontal Cortex; Rats; Rats, Wistar; Risperidone | 2015 |
Analgesic effects of morphine in combination with adjuvant drugs in rats.
Topics: Adjuvants, Pharmaceutic; Analgesics, Opioid; Animals; Butylscopolammonium Bromide; Drug Interactions; Drug Therapy, Combination; Haloperidol; Male; Methotrimeprazine; Metoclopramide; Midazolam; Morphine; Pain; Rats, Wistar | 2014 |
Comment on a Randomized Controlled Trial of Intravenous Haloperidol versus Intravenous Metoclopramide for Acute Migraine Therapy in the Emergency Department.
Topics: Emergency Service, Hospital; Haloperidol; Humans; Metoclopramide; Migraine Disorders | 2017 |
Fragmentation studies of selected drugs utilized in palliative care.
Topics: Adjuvants, Anesthesia; Analgesics, Opioid; Anticonvulsants; Antiemetics; Antipsychotic Agents; Clonazepam; Fentanyl; Haloperidol; Humans; Methotrimeprazine; Metoclopramide; Midazolam; Palliative Care; Pharmaceutical Preparations; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Tramadol | 2018 |
Anticholinergic Load and Nutritional Status in Older Individuals.
Topics: Aged; Aged, 80 and over; Chlorpromazine; Cholinergic Antagonists; Female; Geriatric Assessment; Haloperidol; Hospitalization; Humans; Hydroxyzine; Japan; Linear Models; Longitudinal Studies; Male; Malnutrition; Metoclopramide; Multivariate Analysis; Nutrition Assessment; Nutritional Status; Patient Discharge; Regression Analysis; Retrospective Studies; Risperidone | 2020 |