haloperidol and l 745870

haloperidol has been researched along with l 745870 in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (33.33)18.2507
2000's4 (44.44)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, R; Broughton, HB; Curtis, NR; Emms, F; Freedman, SB; Kulagowski, JJ; Leeson, PD; Marwood, R; Mawer, IM; Patel, S; Ragan, CI; Ridgill, MP1
Berardi, F; Colabufo, NA; Leopoldo, M; Perrone, R; Tortorella, V1
Akunne, HC; Belliotti, TR; Brink, WA; Corbin, AE; Georgic, LM; Heffner, TG; Pugsley, TA; Shih, YH; Whetzel, SZ; Wise, LD; Wustrow, DJ; Zoski, KT1
Allouchi, H; Argiolas, A; El Hakmaoui, A; Enguehard-Gueiffier, C; Gmeiner, P; Gueiffier, A; Hübner, H; Melis, MR1
Boeckler, F; Gmeiner, P; Hocke, C; Hübner, H; Kuwert, T; Prante, O; Salama, I; Utz, W1
Ablordeppey, SY; Altundas, R; Nkansah, NT; Roth, BL; Setola, V; Sikazwe, DM; Zhu, XY1
Hopkins, CR; Lindsley, CW1
Nadelhaft, I; Vera, PL1
Arai, Y; Kikuchi, T; Mitazaki, S; Nakagawasai, O; Nakaya, K; Niijima, F; Onogi, H; Sato, A; Tadano, T; Tan-No, K1

Reviews

1 review(s) available for haloperidol and l 745870

ArticleYear
Return of D
    Journal of medicinal chemistry, 2017, 09-14, Volume: 60, Issue:17

    Topics: Animals; Drug Discovery; Humans; Ligands; Molecular Targeted Therapy; Neoplasms; Parkinson Disease; Receptors, Dopamine D4; Small Molecule Libraries; Substance-Related Disorders

2017

Other Studies

8 other study(ies) available for haloperidol and l 745870

ArticleYear
3-((4-(4-Chlorophenyl)piperazin-1-yl)-methyl)-1H-pyrrolo-2,3-b-pyridine: an antagonist with high affinity and selectivity for the human dopamine D4 receptor.
    Journal of medicinal chemistry, 1996, May-10, Volume: 39, Issue:10

    Topics: Animals; Cell Line; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Pyridines; Pyrroles; Receptors, Dopamine D4

1996
N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: a potent and selective dopamine D4 ligand.
    Journal of medicinal chemistry, 1998, Nov-19, Volume: 41, Issue:24

    Topics: Animals; Benzamides; Cell Line; Cerebral Cortex; Humans; Insecta; Ligands; Piperazines; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4; Structure-Activity Relationship

1998
A series of 6- and 7-piperazinyl- and -piperidinylmethylbenzoxazinones with dopamine D4 antagonist activity: discovery of a potential atypical antipsychotic agent.
    Journal of medicinal chemistry, 1999, Dec-16, Volume: 42, Issue:25

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; CHO Cells; Corpus Striatum; Cricetinae; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Hippocampus; Magnetic Resonance Spectroscopy; Oxazines; Rats; Receptors, Dopamine D4

1999
2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist.
    Journal of medicinal chemistry, 2006, Jun-29, Volume: 49, Issue:13

    Topics: Animals; Cattle; CHO Cells; Cricetinae; Cricetulus; Erectile Dysfunction; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Imidazoles; Ligands; Male; Mitosis; Penile Erection; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Rats; Receptors, Dopamine D4; Structure-Activity Relationship

2006
Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands.
    Journal of medicinal chemistry, 2007, Feb-08, Volume: 50, Issue:3

    Topics: Animals; Benzamides; Fluorine Radioisotopes; In Vitro Techniques; Ligands; Models, Molecular; Molecular Conformation; Piperazines; Positron-Emission Tomography; Quantitative Structure-Activity Relationship; Radioligand Assay; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Swine

2007
Synthesis and evaluation of ligands for D2-like receptors: the role of common pharmacophoric groups.
    Bioorganic & medicinal chemistry, 2009, Feb-15, Volume: 17, Issue:4

    Topics: Antipsychotic Agents; Binding Sites; Butyrophenones; Haloperidol; Humans; Indoles; Kinetics; Ligands; Receptors, Dopamine D2; Structure-Activity Relationship

2009
Effects of the atypical neuroleptic clozapine on micturition parameters in anesthetized rats.
    Neurourology and urodynamics, 2001, Volume: 20, Issue:5

    Topics: Anesthesia; Animals; Antipsychotic Agents; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electric Stimulation; Female; Haloperidol; Hypogastric Plexus; Pyridines; Pyrroles; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D4; Urinary Bladder; Urination; Urination Disorders

2001
p-Hydroxyamphetamine causes prepulse inhibition disruptions in mice: contribution of dopamine neurotransmission.
    Behavioural brain research, 2010, Dec-25, Volume: 214, Issue:2

    Topics: Animals; Benzazepines; Clozapine; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Indoles; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Oxidopamine; p-Hydroxyamphetamine; Piperazines; Piperidines; Pyridines; Pyrroles; Reflex, Startle; Salicylamides; Sensory Gating; Sympathomimetics; Synaptic Transmission

2010