haloperidol and flunarizine

haloperidol has been researched along with flunarizine in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19905 (23.81)18.7374
1990's5 (23.81)18.2507
2000's6 (28.57)29.6817
2010's5 (23.81)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ1
Brouillette, WJ; Brown, GB; Zha, C1
Bennis, K; Ducki, S; Lesage, F; Vivier, D1
Bertolucci, PH; De Andrade, LA; Ferraz, HB; Pereira, JS1
Ahlemeyer, B; Krieglstein, J1
Fadda, F; Gessa, GL; Mosca, E; Stefanini, E1
Heikkila, RE; Manzino, L; Sonsalla, PK1
Heikkila, RE; Manzino, L1
Calder, L; Clikeman, J; Finnegan, KT; Karler, R; Wei, S1
Camargos, ST; Cardoso, F; Silva Júnior, GA1
Petkov, VD; Petkova, B1
Amorim, SC; Costa, PG; Futuro-Neto, HA; Pires, JG; Ribeiro, CA; Saraiva, FP1
Matsuo, H; Nasu, R; Ohtani, H; Sawada, Y1
Armando, I; Belforte, JE; Buño, W; Magariños-Azcone, C; Pazo, JH1
Cayabyab, FS; Hamming, KS; McRory, JE; Mezeyova, J; Parker, D; Santi, CM; Snutch, TP; Stea, A; Sutton, KG1
Dall'Igna, OP; de Oliveira, RV; Fett, P; Gomes, MW; Lara, DR; Mantese, CE; Schuh, J; Souza, DO; Tort, AB1
Bisol, LW; Borba, DL; Bressan, RA; Brunstein, MG; Daltio, CS; de Oliveira, RV; de Souza, SE; Lara, DR; Ottoni, GL; Paz, GE; Ramos, FL1
Munhoz, RP; Teive, HA; Werneck, LC1

Reviews

1 review(s) available for haloperidol and flunarizine

ArticleYear
Perspectives on the Two-Pore Domain Potassium Channel TREK-1 (TWIK-Related K(+) Channel 1). A Novel Therapeutic Target?
    Journal of medicinal chemistry, 2016, 06-09, Volume: 59, Issue:11

    Topics: Arrhythmias, Cardiac; Depression; Epilepsy; Humans; Inflammation; Models, Molecular; Molecular Structure; Neuroprotective Agents; Pain; Potassium Channels, Tandem Pore Domain; Structure-Activity Relationship

2016

Trials

1 trial(s) available for haloperidol and flunarizine

ArticleYear
Is flunarizine a long-acting oral atypical antipsychotic? A randomized clinical trial versus haloperidol for the treatment of schizophrenia.
    The Journal of clinical psychiatry, 2008, Volume: 69, Issue:10

    Topics: Administration, Oral; Adult; Analysis of Variance; Antipsychotic Agents; Dopamine Antagonists; Double-Blind Method; Drug Administration Schedule; Drug-Related Side Effects and Adverse Reactions; Female; Flunarizine; Haloperidol; Humans; Male; Metabolic Clearance Rate; Schizophrenia

2008

Other Studies

19 other study(ies) available for haloperidol and flunarizine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:1

    Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity

2013
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
A study on the action of two calcium channel blockers (verapamil and flunarizine) upon an experimental model of tardive dyskinesia in rats.
    Arquivos de neuro-psiquiatria, 1992, Volume: 50, Issue:3

    Topics: Animals; Apomorphine; Drug Evaluation, Preclinical; Dyskinesia, Drug-Induced; Flunarizine; Haloperidol; Male; Rats; Rats, Wistar; Stereotyped Behavior; Verapamil

1992
Testing drug effects against hypoxic damage of cultured neurons during long-term recovery.
    Life sciences, 1989, Volume: 45, Issue:9

    Topics: Adenosine Triphosphate; Animals; Anticonvulsants; Brain Ischemia; Cell Count; Cell Survival; Cells, Cultured; Chick Embryo; Clonazepam; Diazepam; Dibenzocycloheptenes; Dizocilpine Maleate; Flunarizine; Haloperidol; Imipramine; Ketamine; Lidocaine; Nafronyl; Neurons; Pyrithioxin; Telencephalon

1989
Different effects of the calcium antagonists nimodipine and flunarizine on dopamine metabolism in the rat brain.
    Journal of neural transmission, 1989, Volume: 75, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Calcium Channel Blockers; Caudate Nucleus; Dopamine; Dose-Response Relationship, Drug; Flunarizine; Haloperidol; Male; Nimodipine; Rats; Rats, Inbred Strains

1989
Interactions of D1 and D2 dopamine receptors on the ipsilateral vs. contralateral side in rats with unilateral lesions of the dopaminergic nigrostriatal pathway.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Basal Ganglia; Benzazepines; Corpus Striatum; Denervation; Dextroamphetamine; Ergolines; Female; Flunarizine; Functional Laterality; Haloperidol; Levodopa; Neural Pathways; Parkinson Disease; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Rotation; Substantia Nigra

1988
Behavioral properties of GBR 12909, GBR 13069 and GBR 13098: specific inhibitors of dopamine uptake.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Behavior, Animal; Biogenic Amines; Cerebral Cortex; Corpus Striatum; Dopamine; Female; Flunarizine; Haloperidol; Humans; Hydroxydopamines; In Vitro Techniques; Male; Mice; Motor Activity; Neurotransmitter Uptake Inhibitors; Oxidopamine; Piperazines; Rats; Rats, Inbred Strains; Stereotyped Behavior

1984
Effects of L-type calcium channel antagonists on the serotonin-depleting actions of MDMA in rats.
    Brain research, 1993, Feb-12, Volume: 603, Issue:1

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Flunarizine; Haloperidol; Hippocampus; Male; Methamphetamine; N-Methyl-3,4-methylenedioxyamphetamine; Nifedipine; Rats; Rats, Sprague-Dawley; Seizures; Serotonin; Stereotyped Behavior; Verapamil

1993
Etiology of parkinsonism in a Brazilian movement disorders clinic.
    Arquivos de neuro-psiquiatria, 1998, Volume: 56, Issue:2

    Topics: Aged; Anti-Dyskinesia Agents; Brazil; Calcium Channel Blockers; Cinnarizine; Female; Flunarizine; Haloperidol; Histamine H1 Antagonists; Humans; Male; Middle Aged; Parkinson Disease; Parkinson Disease, Secondary

1998
Behavioral changes as a result of dotarizine or flunarizine influence on dopaminergic neurotransmission in the striatum.
    Acta physiologica et pharmacologica Bulgarica, 1998, Volume: 23, Issue:1

    Topics: Administration, Oral; Animals; Area Under Curve; Benzhydryl Compounds; Calcium Channel Blockers; Catalepsy; Corpus Striatum; Dopamine Antagonists; Flunarizine; Haloperidol; Injections, Intraperitoneal; Male; Piperazines; Rats; Rats, Wistar; Stereotypic Movement Disorder; Synaptic Transmission

1998
Evidence of sex related differences in the effects of calcium channel blockers on neuroleptic-induced catalepsy in mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 1999, Volume: 23, Issue:2

    Topics: Animals; Antipsychotic Agents; Basal Ganglia Diseases; Calcium Channel Blockers; Catalepsy; Dose-Response Relationship, Drug; Female; Flunarizine; Haloperidol; Male; Mice; Nimodipine; Sex Factors; Verapamil

1999
Relationship between structure and drug-induced parkinsonism.
    The Annals of pharmacotherapy, 2000, Volume: 34, Issue:5

    Topics: Antipsychotic Agents; Catalepsy; Cinnarizine; Drug Design; Flunarizine; Haloperidol; Humans; Parkinson Disease, Secondary; Structure-Activity Relationship; Vasodilator Agents

2000
Pharmacological involvement of the calcium channel blocker flunarizine in dopamine transmission at the striatum.
    Parkinsonism & related disorders, 2001, Volume: 8, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Calcium Channel Blockers; Calcium Channels, L-Type; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Flunarizine; Haloperidol; Male; Microinjections; Neostriatum; Nifedipine; Parkinson Disease, Secondary; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Synapses; Synaptic Transmission

2001
Differential inhibition of T-type calcium channels by neuroleptics.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Jan-15, Volume: 22, Issue:2

    Topics: Antipsychotic Agents; Calcium Channel Blockers; Calcium Channels, T-Type; Cell Line; Dose-Response Relationship, Drug; Flunarizine; Haloperidol; Humans; Ion Channel Gating; Kidney; Patch-Clamp Techniques; Penfluridol; Pimozide; Piperidines; Transfection

2002
Atypical antipsychotic profile of flunarizine in animal models.
    Psychopharmacology, 2005, Volume: 177, Issue:3

    Topics: Administration, Oral; Animals; Catalepsy; Dextroamphetamine; Disease Models, Animal; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Flunarizine; Haloperidol; Mice; Motor Activity; Receptors, N-Methyl-D-Aspartate; Time Factors

2005
The differential diagnoses of parkinsonism: findings from a cohort of 1528 patients and a 10 years comparison in tertiary movement disorders clinics.
    Clinical neurology and neurosurgery, 2010, Volume: 112, Issue:5

    Topics: Aged; Antipsychotic Agents; Cinnarizine; Cohort Studies; Diagnosis, Differential; Female; Flunarizine; Haloperidol; Humans; Male; Methotrimeprazine; Movement Disorders; Outpatient Clinics, Hospital; Parkinsonian Disorders; Psychotic Disorders; Risperidone; Severity of Illness Index; Time Factors; Valproic Acid

2010