haloperidol has been researched along with enkephalin, ala(2)-mephe(4)-gly(5)- in 24 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 11 (45.83) | 18.2507 |
2000's | 6 (25.00) | 29.6817 |
2010's | 5 (20.83) | 24.3611 |
2020's | 2 (8.33) | 2.80 |
Authors | Studies |
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Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG | 1 |
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L | 1 |
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S | 1 |
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L | 1 |
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E | 1 |
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E | 1 |
Amata, E; Artacho-Cordón, A; Barbaraci, C; Cobos, EJ; Dichiara, M; Gómez-Guzmán, M; González-Cano, R; Marrazzo, A; Pasquinucci, L; Rodríguez-Gómez, I; Santos-Caballero, M; Turnaturi, R | 1 |
Amata, E; Dichiara, M; Fortuna, S; Mamolo, MG; Marrazzo, A; Pasquinucci, L; Romano, M; Turnaturi, R; Zampieri, D | 1 |
Austin, MC; Churchill, L; Kalivas, PW | 1 |
Napier, TC | 1 |
Austin, MC; Kalivas, PW | 1 |
De Vries, TJ; Jonker, AJ; Mulder, AH; Schoffelmeer, AN; Voorn, P | 1 |
Kalivas, PW; Klitenick, MA | 1 |
Chiou, GC; Li, BH; Rohde, BH | 1 |
Cheĭdo, MA; Idova, GV | 4 |
Kennedy, JL; Nobrega, JN; Sasaki, T | 1 |
Capasso, A; Sorrentino, L | 1 |
Dun, NJ; Hwang, BH; Mizoguchi, H; Nagase, H; Narita, M; Oji, DE; Tseng, LF | 1 |
Baca, SM; Bower, CM; Egan, MF; Hamid, EH; Hyde, TM; Zaka, M | 1 |
Alperina, E; Cheido, M; Devoino, L; Idova, G | 1 |
Cadet, P | 1 |
24 other study(ies) available for haloperidol and enkephalin, ala(2)-mephe(4)-gly(5)-
Article | Year |
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cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship | 2008 |
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship | 2013 |
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2013 |
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship | 2013 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine | 2016 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship | 2017 |
Dual Sigma-1 receptor antagonists and hydrogen sulfide-releasing compounds for pain treatment: Design, synthesis, and pharmacological evaluation.
Topics: Animals; Guinea Pigs; Hydrogen; Hydrogen Sulfide; Ligands; Male; Morpholines; Pain; Piperazines; Rats, Sprague-Dawley; Receptors, sigma; Sigma-1 Receptor | 2022 |
Design, synthesis and biological evaluation of novel aminopropylcarboxamide derivatives as sigma ligands.
Topics: Haloperidol; Ligands; Piperidines; Quinolines; Receptors, sigma; Structure-Activity Relationship | 2022 |
Dopamine and endogenous opioid regulation of picrotoxin-induced locomotion in the ventral pallidum after dopamine depletion in the nucleus accumbens.
Topics: Animals; Dopamine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Globus Pallidus; Haloperidol; Male; Microinjections; Motor Activity; Naloxone; Nucleus Accumbens; Picrotoxin; Rats; Rats, Sprague-Dawley; Sympathectomy, Chemical | 1992 |
Dopamine receptors in the ventral pallidum regulate circling induced by opioids injected into the ventral pallidum.
Topics: Amphetamine; Animals; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Globus Pallidus; Haloperidol; Injections; Male; Parasympatholytics; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Stereotyped Behavior | 1992 |
Dopaminergic involvement in locomotion elicited from the ventral pallidum/substantia innominata.
Topics: Animals; Biogenic Amines; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fluphenazine; Globus Pallidus; Haloperidol; Male; Motor Activity; Osmolar Concentration; Picrotoxin; Rats; Rats, Inbred Strains; Substantia Innominata | 1991 |
Adaptive changes in rat striatal preproenkephalin expression and dopamine-opioid interactions upon chronic haloperidol treatment during different developmental stages.
Topics: Aging; Animals; Corpus Striatum; Dopamine; Embryonic and Fetal Development; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Fetus; Gene Expression; Guanylate Cyclase; Haloperidol; In Situ Hybridization; Maternal-Fetal Exchange; Pregnancy; Protein Precursors; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger | 1994 |
Behavioral and neurochemical studies of opioid effects in the pedunculopontine nucleus and mediodorsal thalamus.
Topics: Amino Acid Sequence; Animals; Baclofen; Behavior, Animal; Dopamine; Dorsomedial Hypothalamic Nucleus; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Extracellular Space; Haloperidol; Male; Microinjections; Molecular Sequence Data; Motor Activity; Nucleus Accumbens; Pons; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Synaptic Transmission; Ventral Tegmental Area | 1994 |
Effects of melatonin and haloperidol given via vortex vein on the intraocular pressure.
Topics: Analgesics; Animals; Ciliary Body; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Haloperidol; Injections, Intravenous; Intraocular Pressure; Iris; Ketamine; Melatonin; Rabbits; Retina; Sclera; Veins; Xylazine | 1993 |
[Dopaminergic mechanisms in the immunostimulating effect of mu-opioid receptors].
Topics: Animals; Dopamine Antagonists; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Haloperidol; Immunoglobulin M; Male; Mice; Mice, Inbred CBA; Pituitary Gland; Receptors, Dopamine; Receptors, Opioid, mu; Rosette Formation | 1996 |
Autoradiographic mapping of mu opioid receptor changes in rat brain after long-term haloperidol treatment: relationship to the development of vacuous chewing movements.
Topics: Animals; Antipsychotic Agents; Autoradiography; Brain; Dopamine Antagonists; Dyskinesia, Drug-Induced; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Haloperidol; Male; Mastication; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Opioid, mu; Salicylamides | 1996 |
Differential influence of D1 and D2 dopamine receptors on acute opiate withdrawal in guinea-pig isolated ileum.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Apomorphine; Dopamine Agents; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Guinea Pigs; Haloperidol; Ileum; In Vitro Techniques; Male; Morphine; Muscle, Smooth; Pyrrolidines; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substance Withdrawal Syndrome | 1997 |
[Effect of opioid peptides on immunomodulation].
Topics: Animals; Cyproheptadine; Dopamine D2 Receptor Antagonists; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Haloperidol; Male; Mice; Mice, Inbred CBA; Neuroimmunomodulation; Pituitary Gland; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Serotonin; Spleen | 1998 |
Identification of the G-protein-coupled ORL1 receptor in the mouse spinal cord by [35S]-GTPgammaS binding and immunohistochemistry.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Autoradiography; Baclofen; Binding, Competitive; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Haloperidol; Immunohistochemistry; In Vitro Techniques; Male; Membranes; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Propranolol; Receptors, Opioid; Somatostatin; Spinal Cord; Sulfur Radioisotopes; Yohimbine | 1999 |
Decreased mu-opioid receptor binding in the globus pallidus of rats treated with chronic haloperidol.
Topics: Animals; Antipsychotic Agents; Autoradiography; Behavior, Animal; Dyskinesia, Drug-Induced; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Globus Pallidus; Haloperidol; Male; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Time Factors | 2000 |
Evidence for a role of dopaminergic mechanisms in the immunostimulating effect of mu-opioid receptor agonist DAGO.
Topics: Analgesics, Opioid; Animals; Cerebellar Nuclei; Dopamine; Dopamine Antagonists; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Erythrocytes; Haloperidol; Hemolytic Plaque Technique; Hypothalamus; Immunization; Immunoglobulin M; Male; Mice; Mice, Inbred CBA; Neuroimmunomodulation; Nucleus Accumbens; Pituitary Gland; Rats; Rats, Wistar; Receptors, Opioid, mu; Rosette Formation; Sheep; Species Specificity; Spleen | 2003 |
Nitric oxide modulates the physiological control of ciliary activity in the marine mussel Mytilus edulis via morphine: novel mu opiate receptor splice variants.
Topics: Alternative Splicing; Animals; Base Sequence; Bivalvia; Cilia; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ganglia, Invertebrate; Genetic Variation; Haloperidol; Molecular Sequence Data; Morphine; NG-Nitroarginine Methyl Ester; Nitric Oxide; Receptors, Opioid, mu; Reverse Transcriptase Polymerase Chain Reaction; S-Nitroso-N-Acetylpenicillamine | 2004 |
[Differential contribution of dopamine D1 and D2 receptors in the mu-opioidergic immunomodulation].
Topics: Analgesics, Opioid; Animals; Antibody Formation; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Haloperidol; Male; Mice; Mice, Inbred CBA; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, mu | 2006 |
The differential contribution of dopamine D(1) and D (2) receptors to mu-opioidergic immunomodulation.
Topics: Analgesics, Opioid; Animals; Antibody Formation; Benzazepines; Dopamine Antagonists; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Haloperidol; Male; Mice; Mice, Inbred CBA; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, mu | 2007 |