Compounds > haloperidol

haloperidol and eliprodil

haloperidol has been researched along with eliprodil in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (15.38)18.2507
2000's2 (15.38)29.6817
2010's7 (53.85)24.3611
2020's2 (15.38)2.80

Authors

AuthorsStudies
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Frehland, B; Schepmann, D; Schmidtke, KU; Tewes, B; Winckler, T; Wünsch, B1
Bonifazi, A; Gawaskar, S; Schepmann, D; Wünsch, B1
Bonifazi, A; Gawaskar, S; Robaa, D; Schepmann, D; Sippl, W; Wünsch, B1
Lütnant, I; Schepmann, D; Wünsch, B1
Dey, S; Frehland, B; Lehmkuhl, K; Schepmann, D; Schreiber, JA; Seebohm, G; Strutz-Seebohm, N; Temme, L; Wünsch, B1
Kitamura, M; Schepmann, D; Shuto, Y; Temme, L; Thum, S; Wünsch, B1
Ametamey, SM; Schepmann, D; Wagner, M; Wünsch, B1
Baumeister, S; Schepmann, D; Wünsch, B1
Bechthold, E; Daniliuc, C; Ritter, N; Schepmann, D; Schreiber, JA; Seebohm, G; Wünsch, B1
Cordon, JJ; Coughenour, LL1
Pahk, AJ; Williams, K1
Lanis, A; Schmidt, WJ1

Other Studies

13 other study(ies) available for haloperidol and eliprodil

ArticleYear
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Conformationally constrained NR2B selective NMDA receptor antagonists derived from ifenprodil: Synthesis and biological evaluation of tetrahydro-3-benzazepine-1,7-diols.
    Bioorganic & medicinal chemistry, 2010, Nov-15, Volume: 18, Issue:22

    Topics: Analgesics; Animals; Benzazepines; Humans; Mice; Microsomes, Liver; Neuralgia; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2010
Synthesis, GluN2B affinity and selectivity of benzo[7]annulen-7-amines.
    Bioorganic & medicinal chemistry, 2014, Dec-01, Volume: 22, Issue:23

    Topics: Benzocycloheptenes; Dose-Response Relationship, Drug; Humans; Molecular Structure; Piperazines; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2014
Benzo[7]annulene-based GluN2B selective NMDA receptor antagonists: Surprising effect of a nitro group in 2-position.
    Bioorganic & medicinal chemistry letters, 2015, Dec-15, Volume: 25, Issue:24

    Topics: Amines; Binding Sites; Molecular Docking Simulation; Phenols; Piperidines; Protein Binding; Protein Structure, Tertiary; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2015
Benzimidazolone bioisosteres of potent GluN2B selective NMDA receptor antagonists.
    European journal of medicinal chemistry, 2016, Jun-30, Volume: 116

    Topics: Benzimidazoles; Drug Design; Humans; Receptors, N-Methyl-D-Aspartate

2016
Deconstruction - reconstruction approach to analyze the essential structural elements of tetrahydro-3-benzazepine-based antagonists of GluN2B subunit containing NMDA receptors.
    European journal of medicinal chemistry, 2017, Sep-29, Volume: 138

    Topics: Benzazepines; Dose-Response Relationship, Drug; Humans; Models, Molecular; Molecular Structure; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2017
Do GluN2B subunit containing NMDA receptors tolerate a fluorine atom in the phenylalkyl side chain?
    MedChemComm, 2017, May-01, Volume: 8, Issue:5

    Topics:

2017
Modification of the 4-phenylbutyl side chain of potent 3-benzazepine-based GluN2B receptor antagonists.
    Bioorganic & medicinal chemistry, 2019, 08-15, Volume: 27, Issue:16

    Topics: Benzazepines; Binding Sites; Models, Molecular; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

2019
Thiophene bioisosteres of GluN2B selective NMDA receptor antagonists: Synthesis and pharmacological evaluation of [7]annuleno[b]thiophen-6-amines.
    Bioorganic & medicinal chemistry, 2020, 01-15, Volume: 28, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Molecular Structure; Rats; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Thiophenes

2020
Synthesis and biological evaluation of conformationally restricted GluN2B ligands derived from eliprodil.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Ligands; Piperidines; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Tropanes

2022
Characterization of haloperidol and trifluperidol as subtype-selective N-methyl-D-aspartate (NMDA) receptor antagonists using [3H]TCP and [3H]ifenprodil binding in rat brain membranes.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Female; Haloperidol; Illicit Drugs; Kinetics; Oocytes; Phencyclidine; Piperidines; Radioligand Assay; Rats; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Trifluperidol; Xenopus

1997
Influence of extracellular pH on inhibition by ifenprodil at N-methyl-D-aspartate receptors in Xenopus oocytes.
    Neuroscience letters, 1997, Mar-28, Volume: 225, Issue:1

    Topics: Animals; Excitatory Amino Acid Antagonists; Haloperidol; Hydrogen-Ion Concentration; Neuroprotective Agents; Nylidrin; Oocytes; Patch-Clamp Techniques; Piperidines; Receptors, N-Methyl-D-Aspartate; Xenopus laevis

1997
NMDA receptor antagonists do not block the development of sensitization of catalepsy, but make its expression state-dependent.
    Behavioural pharmacology, 2001, Volume: 12, Issue:2

    Topics: Animals; Conditioning, Classical; Drug Interactions; Excitatory Amino Acid Antagonists; Haloperidol; Male; Phenols; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate

2001