haloperidol has been researched along with e-52862 in 10 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 5 (50.00) | 24.3611 |
| 2020's | 5 (50.00) | 2.80 |
| Authors | Studies |
|---|---|
| Almansa, C; Berrocal, J; Burgueño, J; Buschmann, H; Christmann, U; Contijoch, M; Cuberes, R; Díaz, JL; Fernández, A; Holenz, J; Laggner, C; Merlos, M; Port, A; Serafini, MT; Vela, JM; Zamanillo, D | 1 |
| Almansa, C; Benet-Buchholz, J; Bordas, M; Burgueño, J; Carro, M; Cerón-Bertran, J; Christmann, U; Díaz, JL; Enrech, R; Fernández de Henestrosa, AR; Fernández, A; Luengo, M; Merlos, M; Pascual, R; Ramírez, J; Reinoso, RF; Vela, JM | 1 |
| Chen, Y; Lan, Y; Liu, BF; Liu, S; Liu, X; Qiu, Y; Xu, X; Zhang, G | 1 |
| Cao, X; Chen, Y; Lan, Y; Liu, BF; Liu, X; Qiu, Y; Xu, X; Zhang, G; Zhang, J; Zhang, Y; Zhao, S | 1 |
| Iyamu, ID; Lv, W; Malik, N; Mishra, RK; Schiltz, GE | 1 |
| Alegret, C; Almansa, C; Alonso, M; Fernández, B; García, M; Monroy, X; Pascual, R; Port, A; Serafini, MT; Vela, JM; Vidal-Torres, A; Virgili, M | 1 |
| Agard, DA; Ashworth, A; Barrio-Hernandez, I; Batra, J; Beltrao, P; Bennett, MJ; Bohn, M; Bouhaddou, M; Braberg, H; Broadhurst, DJ; Cai, Y; Cakir, M; Calviello, L; Cavero, DA; Chang, JCJ; Chorba, JS; Craik, CS; d'Enfert, C; Dai, SA; Eckhardt, M; Emerman, M; Fabius, JM; Fletcher, SJ; Floor, SN; Foussard, H; Frankel, AD; Fraser, JS; Fujimori, DG; Ganesan, SJ; García-Sastre, A; Gordon, DE; Gross, JD; Guo, JZ; Haas, K; Haas, P; Hernandez-Armenta, C; Hiatt, J; Huang, XP; Hubert, M; Hüttenhain, R; Ideker, T; Jacobson, M; Jang, GM; Jura, N; Kaake, RM; Kim, M; Kirby, IT; Klippsten, S; Koh, C; Kortemme, T; Krogan, NJ; Kuzuoglu-Ozturk, D; Li, Q; Liboy-Lugo, J; Lin, Y; Liu, X; Liu, Y; Lou, K; Lyu, J; Mac Kain, A; Malik, HS; Mathy, CJP; McGregor, MJ; Melnyk, JE; Memon, D; Meyer, B; Miorin, L; Modak, M; Moreno, E; Mukherjee, S; Naing, ZZC; Noack, J; O'Meara, MJ; O'Neal, MC; Obernier, K; Ott, M; Peng, S; Perica, T; Pilla, KB; Polacco, BJ; Rakesh, R; Rathore, U; Rezelj, VV; Richards, AL; Roesch, F; Rosenberg, OS; Rosenthal, SB; Roth, BL; Roth, TL; Ruggero, D; Safari, M; Sali, A; Saltzberg, DJ; Savar, NS; Schwartz, O; Sharp, PP; Shen, W; Shengjuler, D; Shi, Y; Shoichet, BK; Shokat, KM; Soucheray, M; Stroud, RM; Subramanian, A; Swaney, DL; Taunton, J; Tran, QD; Trenker, R; Tummino, TA; Tutuncuoglu, B; Ugur, FS; Vallet, T; Venkataramanan, S; Verba, KA; Verdin, E; Vignuzzi, M; von Zastrow, M; Wang, HY; Wankowicz, SA; Wenzell, NA; White, KM; Xu, J; Young, JM; Zhang, Z; Zhou, Y | 1 |
| Almansa, C; Álvarez, I; Caamaño, AM; Cendán, CM; de la Puente, B; Díaz, JL; Enjo, J; García, M; Lorente, A; Maldonado, R; Martín, M; Montero, A; Port, A; Sicre, C; Torrens, A; Vela, JM; Vidal-Torres, A; Yeste, S | 1 |
| Peng, Y; Welsh, WJ; Zhang, Q | 1 |
| Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M | 1 |
10 other study(ies) available for haloperidol and e-52862
| Article | Year |
|---|---|
Synthesis and biological evaluation of the 1-arylpyrazole class of σ(1) receptor antagonists: identification of 4-{2-[5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862).
Topics: Animals; Brain; Female; Guinea Pigs; HEK293 Cells; Humans; Hyperalgesia; In Vitro Techniques; Male; Mice; Microsomes, Liver; Morpholines; Motor Activity; Neuralgia; Patch-Clamp Techniques; Pyrazoles; Radioligand Assay; Receptors, sigma; Sciatic Neuropathy; Sigma-1 Receptor; Structure-Activity Relationship | 2012 |
Synthesis and biological evaluation of a new series of hexahydro-2H-pyrano[3,2-c]quinolines as novel selective σ1 receptor ligands.
Topics: Analgesics; Animals; Chemical Phenomena; Chemistry Techniques, Synthetic; Drug Evaluation, Preclinical; Female; Guinea Pigs; High-Throughput Screening Assays; Humans; Ligands; Male; Mice; Models, Molecular; Protein Conformation; Quinolines; Receptors, sigma; Structure-Activity Relationship | 2013 |
Synthesis and biological evaluation of a novel sigma-1 receptor antagonist based on 3,4-dihydro-2(1H)-quinolinone scaffold as a potential analgesic.
Topics: Analgesics; Animals; Brain; Dose-Response Relationship, Drug; Formaldehyde; Guinea Pigs; Hydroquinones; Mice; Mice, Inbred Strains; Molecular Structure; Nociceptive Pain; Pain Measurement; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship | 2014 |
Synthesis and Biological Evaluation of Novel σ1 Receptor Ligands for Treating Neuropathic Pain: 6-Hydroxypyridazinones.
Topics: Analgesics, Non-Narcotic; Animals; Chemistry Techniques, Synthetic; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Formaldehyde; Guinea Pigs; Ligands; Mice; Neuralgia; Pain Measurement; Pyridazines; Rats, Sprague-Dawley; Receptors, Opioid, delta; Rotarod Performance Test; Structure-Activity Relationship | 2016 |
Discovery of a novel class of potent and selective tetrahydroindazole-based sigma-1 receptor ligands.
Topics: Animals; Binding Sites; Indazoles; Ligands; Mice; Microsomes, Liver; Molecular Docking Simulation; Protein Structure, Tertiary; Receptors, sigma; Sigma-1 Receptor; Solubility; Structure-Activity Relationship | 2019 |
4-Aryl-1-oxa-4,9-diazaspiro[5.5]undecane Derivatives as Dual μ-Opioid Receptor Agonists and σ
Topics: Alkanes; Analgesics; Analgesics, Opioid; Animals; Humans; Male; Mice; Models, Molecular; Pain; Pain Management; Receptors, Opioid, mu; Receptors, sigma; Sigma-1 Receptor; Spiro Compounds | 2020 |
A SARS-CoV-2 protein interaction map reveals targets for drug repurposing.
Topics: Animals; Antiviral Agents; Betacoronavirus; Chlorocebus aethiops; Cloning, Molecular; Coronavirus Infections; COVID-19; COVID-19 Drug Treatment; Drug Evaluation, Preclinical; Drug Repositioning; HEK293 Cells; Host-Pathogen Interactions; Humans; Immunity, Innate; Mass Spectrometry; Molecular Targeted Therapy; Pandemics; Pneumonia, Viral; Protein Binding; Protein Biosynthesis; Protein Domains; Protein Interaction Mapping; Protein Interaction Maps; Receptors, sigma; SARS-CoV-2; SKP Cullin F-Box Protein Ligases; Vero Cells; Viral Proteins | 2020 |
EST64454: a Highly Soluble σ
Topics: Analgesics; Animals; Caco-2 Cells; Humans; Mice; Molecular Structure; Pain; Piperazines; Pyrazoles; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship | 2020 |
Novel Sigma 1 Receptor Antagonists as Potential Therapeutics for Pain Management.
Topics: Animals; Binding Sites; Blood-Brain Barrier; Drug Design; Guinea Pigs; Half-Life; Humans; Microsomes, Liver; Molecular Dynamics Simulation; Neuralgia; Pain Management; Protein Structure, Tertiary; Quantitative Structure-Activity Relationship; Rats; Receptors, sigma; Sigma-1 Receptor; Triazoles | 2021 |
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries | 2023 |