Page last updated: 2024-08-23

halofantrine and sesquiterpenes

halofantrine has been researched along with sesquiterpenes in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.45)18.7374
1990's19 (65.52)18.2507
2000's9 (31.03)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Trigg, PI1
Bourdeau, EF; Childs, GE; Milhous, WK; Pang, L; Wimonwattratee, T1
Coulaud, JP; Ngo Van, P1
Nosten, F; Price, RN1
Ager, A; Andersen, SL; Berman, J; Ellis, W; Kuschner, R; McGreevy, P; Ohrt, C; Rossan, R; Schuster, BG; Wesche, D1
Baric, RS; Bright, P; Handy, J; Peel, SA; Yount, B1
Basco, LK; Le Bras, J2
Hopperus Buma, AP; Kager, PA; Leentvaar-Kuijpers, A; Tendeloo, CH; van Gool, T; van Thiel, PP1
Angus, B; Bates, I; Krishna, S; Kyle, DE; Pipitaporn, B; Pukrittayakamee, S; Suputtamongkol, Y; Udomsangpetch, R; White, NJ1
Watkins, WM1
Ezedinachi, E1
Falade, CO; Fehintola, FA; Kyle, DE; Makler, MT; Milhous, WK; Oduola, AM; Ogundahunsi, OA; Omitowoju, GO; Piper, RC; Schuster, BG; Sowunmi, A1
Doury, JC; Fusai, T; Pradines, B; Rogier, C; Tall, A; Trape, JF1
Kremsner, PG; Philipps, J; Radloff, PD; Wernsdorfer, W1
Doury, JC; Kombila, M; Lebeau, C; Mabika Mamfoumbi, M; Mourou Mbina, JR; Owono Medang, M; Parzy, D; Pradines, B1
Le Bras, J1
Chongsuphajaisiddhi, T; Luxemburger, C; Nosten, F; Phaipun, L; Price, R; Simpson, JA; ter Kuile, F; van Vugt, M; White, NJ1
Barette, S; Bernard, J; Bouchaud, O; Danis, M; Delmont, J; Gathmann, I; Gras, C; Malvy, D; Mull, R; Touze, JE; van Agtmael, M1
Duraisingh, MT; Jones, P; Pinder, M; Sambou, I; von Seidlein, L; Warhurst, DC1
Caruana, SR; Cowman, AF; Kirk, K; Reed, MB; Saliba, KJ1
Bockarie, MJ; Gbakima, AA; Sahr, F; Willoughby, VR1
Bindschedler, M; Degen, P; Lefèvre, G; Sioufi, A1
Brown, ML; Geyer, JA; Terrell, JC; Trotta, RF1
Beg, MA; Khan, MA; Razi, ST; Smego, RA1
Fidock, DA; Sidhu, AB; Valderramos, SG1
Fidock, DA; Krishna, S; Sidhu, AB; Uhlemann, AC; Valderramos, JC; Valderramos, SG1
Brockman, A; Chotivanich, K; Day, NP; Stepniewska, K; White, NJ1
Abuaku, B; Duah, NO; Koram, KA; Quashie, NB1

Reviews

3 review(s) available for halofantrine and sesquiterpenes

ArticleYear
New antimalarials. A risk-benefit analysis.
    Drug safety, 1995, Volume: 12, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; Dose-Response Relationship, Drug; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Pregnancy; Risk Assessment; Sesquiterpenes

1995
Pharmacology and pharmacokinetics of new antimalarials.
    Medecine tropicale : revue du Corps de sante colonial, 1995, Volume: 55, Issue:4 Suppl

    Topics: Africa; Antimalarials; Artemether; Artemisinins; Drug Costs; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Sesquiterpenes; Trimethoprim, Sulfamethoxazole Drug Combination

1995
Emerging drug--resistance and guidelines for treatment of malaria.
    Journal of the College of Physicians and Surgeons--Pakistan : JCPSP, 2004, Volume: 14, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance, Multiple; Drug Therapy, Combination; Follow-Up Studies; Humans; Malaria, Falciparum; Pakistan; Phenanthrenes; Plasmodium falciparum; Quinidine; Quinine; Sesquiterpenes; Time Factors

2004

Trials

3 trial(s) available for halofantrine and sesquiterpenes

ArticleYear
In vivo efficacy of chloroquine, halofantrine, pyrimethamine-sulfadoxine and qinghaosu (artesunate) in the treatment of malaria in Calabar, Nigeria.
    The Central African journal of medicine, 1996, Volume: 42, Issue:4

    Topics: Adolescent; Antimalarials; Artemisinins; Artesunate; Child; Chloroquine; Drug Combinations; Drug Resistance; Humans; Malaria, Falciparum; Nigeria; Phenanthrenes; Pyrimethamine; Sesquiterpenes; Sulfadoxine; Time Factors; Urban Health

1996
The comparative efficacy and tolerability of CGP 56697 (artemether + lumefantrine) versus halofantrine in the treatment of uncomplicated falciparum malaria in travellers returning from the Tropics to The Netherlands and France.
    International journal of antimicrobial agents, 1999, Volume: 12, Issue:2

    Topics: Adolescent; Adult; Africa; Animals; Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Double-Blind Method; Drug Combinations; Ethanolamines; Female; Fluorenes; France; Humans; Malaria, Falciparum; Male; Middle Aged; Netherlands; Parasite Egg Count; Phenanthrenes; Plasmodium falciparum; Sesquiterpenes; Time Factors; Travel; Tropical Climate

1999
Comparison of the cardiac effects of the antimalarials co-artemether and halofantrine in healthy participants.
    The American journal of tropical medicine and hygiene, 2002, Volume: 66, Issue:3

    Topics: Administration, Oral; Adult; Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Cross-Over Studies; Double-Blind Method; Drug Combinations; Electrocardiography; Ethanolamines; Fluorenes; Heart; Heart Rate; Humans; Long QT Syndrome; Male; Phenanthrenes; Sesquiterpenes

2002

Other Studies

23 other study(ies) available for halofantrine and sesquiterpenes

ArticleYear
Drug use and design in the nineties.
    Acta Leidensia, 1991, Volume: 60, Issue:1

    Topics: Aminoquinolines; Amodiaquine; Antimalarials; Artemisinins; Calcium Channel Blockers; Chloroquine; Humans; Malaria; Mefloquine; Naphthoquinones; Phenanthrenes; Primaquine; Quinine; Sesquiterpenes; Sulfadoxine

1991
In vitro and clinical correlates of mefloquine resistance of Plasmodium falciparum in eastern Thailand.
    The American journal of tropical medicine and hygiene, 1991, Volume: 44, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Butylated Hydroxytoluene; Chloroquine; Drug Resistance; Drugs, Chinese Herbal; Mefloquine; Molecular Structure; Phenanthrenes; Plasmodium falciparum; Pyridines; Pyrimethamine; Quinine; Sesquiterpenes; Thailand

1991
[New antiparasitic drugs].
    Annales de dermatologie et de venereologie, 1988, Volume: 115, Issue:4

    Topics: Amebicides; Anthelmintics; Antifungal Agents; Antimalarials; Artemisinins; Fluconazole; Humans; Itraconazole; Ketoconazole; Mefloquine; Phenanthrenes; Quinolines; Sesquiterpenes; Triazoles

1988
Activity of azithromycin as a blood schizonticide against rodent and human plasmodia in vivo.
    The American journal of tropical medicine and hygiene, 1995, Volume: 52, Issue:2

    Topics: Administration, Oral; Animals; Antimalarials; Aotus trivirgatus; Artemisinins; Azithromycin; Disease Models, Animal; Doxycycline; Drug Therapy, Combination; Humans; Injections, Subcutaneous; Malaria; Malaria, Falciparum; Mice; Parasitemia; Phenanthrenes; Plasmodium berghei; Quinine; Sesquiterpenes

1995
A strong association between mefloquine and halofantrine resistance and amplification, overexpression, and mutation in the P-glycoprotein gene homolog (pfmdr) of Plasmodium falciparum in vitro.
    The American journal of tropical medicine and hygiene, 1994, Volume: 51, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Base Sequence; Blotting, Northern; Blotting, Southern; Chloroquine; DNA Primers; DNA, Protozoan; Drug Resistance; Gene Amplification; Gene Expression; Genes, Protozoan; Mefloquine; Molecular Sequence Data; Phenanthrenes; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Quinine; RNA, Messenger; Selection, Genetic; Sequence Homology, Nucleic Acid; Sesquiterpenes

1994
In vitro susceptibility of Cambodian isolates of Plasmodium falciparum to halofantrine, pyronaridine and artemisinin derivatives.
    Annals of tropical medicine and parasitology, 1994, Volume: 88, Issue:2

    Topics: Adult; Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; In Vitro Techniques; Mefloquine; Naphthyridines; Phenanthrenes; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Sesquiterpenes; Triazines

1994
Artemisinin compounds in treatment of malaria.
    Lancet (London, England), 1993, Apr-17, Volume: 341, Issue:8851

    Topics: Adult; Antimalarials; Artemisinins; Artesunate; Cambodia; Drug Approval; Drug Resistance; Humans; Malaria, Falciparum; Male; Military Personnel; Netherlands; Phenanthrenes; Sesquiterpenes

1993
In vitro activity of artemisinin derivatives against African isolates and clones of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1993, Volume: 49, Issue:3

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Drug Resistance; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes

1993
Antimalarial drugs reduce cytoadherence and rosetting Plasmodium falciparum.
    The Journal of infectious diseases, 1996, Volume: 173, Issue:3

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Cell Adhesion; Erythrocytes; Humans; In Vitro Techniques; Malaria, Falciparum; Middle Aged; Phenanthrenes; Plasmodium falciparum; Quinine; Rosette Formation; Sesquiterpenes

1996
Plasmodium falciparum: evaluation of lactate dehydrogenase in monitoring therapeutic responses to standard antimalarial drugs in Nigeria.
    Experimental parasitology, 1997, Volume: 87, Issue:3

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Female; Humans; Infant; L-Lactate Dehydrogenase; Malaria, Falciparum; Male; Monitoring, Physiologic; Nigeria; Phenanthrenes; Pyrimethamine; Sesquiterpenes; Sulfadoxine; Treatment Outcome

1997
In vitro activity of artemether against African isolates (Senegal) of Plasmodium falciparum in comparison with standard antimalarial drugs.
    The American journal of tropical medicine and hygiene, 1998, Volume: 58, Issue:3

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance; Erythrocytes; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Senegal; Sesquiterpenes

1998
Follow-up of the susceptibility of Plasmodium falciparum to antimalarials in Gabon.
    The American journal of tropical medicine and hygiene, 1998, Volume: 58, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Follow-Up Studies; Gabon; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes; Sulfadoxine

1998
In vitro susceptibility of Gabonese wild isolates of Plasmodium falciparum to artemether, and comparison with chloroquine, quinine, halofantrine and amodiaquine.
    Parasitology, 1998, Volume: 117 ( Pt 6)

    Topics: Adolescent; Amodiaquine; Animals; Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Gabon; Humans; Infant; Malaria, Falciparum; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes

1998
In vitro susceptibility of African Plasmodium falciparum isolates to dihydroartemisinin and the risk factors for resistance to qinghaosu.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chloroquine; Cross Reactions; Drug Evaluation, Preclinical; Drug Resistance; France; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Sesquiterpenes; Travel

1998
Risk factors for gametocyte carriage in uncomplicated falciparum malaria.
    The American journal of tropical medicine and hygiene, 1999, Volume: 60, Issue:6

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemisinins; Carrier State; Child; Child, Preschool; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Multivariate Analysis; Parasitemia; Phenanthrenes; Plasmodium falciparum; Prospective Studies; Quinine; Regression Analysis; Risk Factors; Seroepidemiologic Studies; Sesquiterpenes; Thailand

1999
Inoculum effect leads to overestimation of in vitro resistance for artemisinin derivatives and standard antimalarials: a Gambian field study.
    Parasitology, 1999, Volume: 119 ( Pt 5)

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Gambia; Hematocrit; Humans; Malaria, Falciparum; Mefloquine; Parasitemia; Phenanthrenes; Plasmodium falciparum; Quinine; Scintillation Counting; Sensitivity and Specificity; Sesquiterpenes

1999
Pgh1 modulates sensitivity and resistance to multiple antimalarials in Plasmodium falciparum.
    Nature, 2000, Feb-24, Volume: 403, Issue:6772

    Topics: Amino Acid Substitution; Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Chloroquine; Cloning, Molecular; Drug Resistance; Mefloquine; Mutation; Phenanthrenes; Plasmodium falciparum; Protozoan Proteins; Quinine; Sesquiterpenes; Verapamil

2000
Apparent drug failure following artesunate treatment of Plasmodium falciparum malaria in Freetown, Sierra Leone: four case reports.
    Annals of tropical medicine and parasitology, 2001, Volume: 95, Issue:5

    Topics: Adult; Antimalarials; Artemisinins; Artesunate; Child; Drug Administration Schedule; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Phenanthrenes; Quinine; Sesquiterpenes; Sierra Leone; Treatment Failure

2001
Defective DNA repair as a potential mechanism for the rapid development of drug resistance in Plasmodium falciparum.
    Biochemistry, 2004, May-04, Volume: 43, Issue:17

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; DNA Damage; DNA Repair; Drug Resistance; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Pyrimethamine; Quinine; Sesquiterpenes; Sulfanilamide; Sulfanilamides; Ultraviolet Rays

2004
pfmdr1 mutations contribute to quinine resistance and enhance mefloquine and artemisinin sensitivity in Plasmodium falciparum.
    Molecular microbiology, 2005, Volume: 57, Issue:4

    Topics: Alleles; Animals; Antimalarials; Artemisinins; Asparagine; Aspartic Acid; ATP-Binding Cassette Transporters; Drug Resistance; Mefloquine; Phenanthrenes; Plasmodium falciparum; Point Mutation; Protozoan Proteins; Quinine; Sesquiterpenes

2005
Decreasing pfmdr1 copy number in plasmodium falciparum malaria heightens susceptibility to mefloquine, lumefantrine, halofantrine, quinine, and artemisinin.
    The Journal of infectious diseases, 2006, Aug-15, Volume: 194, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; DNA, Protozoan; Drug Resistance, Multiple; Ethanolamines; Fluorenes; Genes, MDR; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Polymerase Chain Reaction; Protozoan Proteins; Quinine; Sesquiterpenes

2006
Overestimating resistance in field testing of malaria parasites: simple methods for estimating high EC50 values using a Bayesian approach.
    Malaria journal, 2007, Jan-17, Volume: 6

    Topics: Algorithms; Animals; Antimalarials; Artemisinins; Artesunate; Bayes Theorem; Chloroquine; Computer Simulation; Dose-Response Relationship, Drug; Drug Resistance; False Positive Reactions; Inhibitory Concentration 50; Mefloquine; Models, Biological; Phenanthrenes; Plasmodium falciparum; Sesquiterpenes

2007
The in-vitro susceptibilities of Ghanaian Plasmodium falciparum to antimalarial drugs.
    Annals of tropical medicine and parasitology, 2007, Volume: 101, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Artesunate; Child, Preschool; Chloroquine; Drug Resistance; Ghana; Humans; Infant; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes

2007