Page last updated: 2024-08-23

halofantrine and lumefantrine

halofantrine has been researched along with lumefantrine in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (38.46)29.6817
2010's7 (53.85)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Du, LP; Li, MY; Tsai, KC; Xia, L; You, QD1
Masseno, V; Muriithi, S; Nzila, A1
Sen, S; Sinha, N1
Avery, VM; Buchholz, M; Delves, MJ; Duffy, S; Fischli, C; Held, J; Knaab, TC; Kuna, K; Kurz, T; Lehmann, U; Leven, M; Lungerich, B; Meister, S; Meitzner, D; Mordmüller, B; Stahlke, P; Winzeler, EA; Wittlin, S1
Go, ML; Li, QT1
Fidock, DA; Krishna, S; Sidhu, AB; Uhlemann, AC; Valderramos, JC; Valderramos, SG1
Jain, GK; Singh, SP1
Abildrup, U; Alifrangis, LH; Alifrangis, M; Bygbjerg, IC; Hoegberg, L; Khalil, IF; Lemnge, MM; Maiga, D; Nyagonde, N; Persson, OP; Theander, TG; Vestergaard, LS1
Angelino, E; Barnes, KG; Becker, JS; Birren, BW; Cortese, JF; Daniels, RF; Eskin, E; Furlotte, NA; Grossman, SR; Happi, C; Hartl, DL; Johnson, CA; Kang, HM; Karlsson, EK; Lander, ES; Lukens, AK; Mboup, S; Milner, DA; Ndiaye, D; Neafsey, DE; Park, DJ; Rosen, DM; Sabeti, PC; Sarr, O; Schaffner, SF; Shlyakhter, I; Van Tyne, D; Volkman, SK; Wiegand, RC; Wirth, DF; Yamins, D1
Cowman, AF; Healer, J; Uboldi, AD; Van Tyne, D; Wirth, DF1
Gayen, JR; Raju, KS; Siddiqui, HH; Singh, SK; Singh, SP; Taneja, I; Wahajuddin, M1
Raju, KS; Singh, SP; Taneja, I; Wahajuddin, M1
Be Rziņš, KR; Beilles, S; Boyd, BJ; Clulow, AJ; Fraser-Miller, SJ; Gordon, KC; Hawley, A; Ramirez, G; Salim, M; Sutton, JJ1

Other Studies

13 other study(ies) available for halofantrine and lumefantrine

ArticleYear
The pharmacophore hypotheses of I(Kr) potassium channel blockers: novel class III antiarrhythmic agents.
    Bioorganic & medicinal chemistry letters, 2004, Sep-20, Volume: 14, Issue:18

    Topics: Anti-Arrhythmia Agents; Models, Biological; Models, Molecular; Potassium Channel Blockers; Potassium Channels; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2004
In vitro chemosensitization of Plasmodium falciparum to antimalarials by verapamil and probenecid.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:7

    Topics: Adjuvants, Pharmaceutic; Animals; Antimalarials; Parasitic Sensitivity Tests; Plasmodium falciparum; Probenecid; Verapamil

2009
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
3-Hydroxy-N'-arylidenepropanehydrazonamides with Halo-Substituted Phenanthrene Scaffolds Cure P. berghei Infected Mice When Administered Perorally.
    Journal of medicinal chemistry, 2017, 07-27, Volume: 60, Issue:14

    Topics: Amides; Animals; Antimalarials; Hep G2 Cells; Humans; Hydrazones; Malaria; Mice; Phenanthrenes; Plasmodium berghei; Stereoisomerism; Structure-Activity Relationship

2017
Interaction of the antimalarial agents halofantrine and lumefantrine with lipid bilayers.
    Chemical & pharmaceutical bulletin, 2003, Volume: 51, Issue:3

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Animals; Antimalarials; Erythrocyte Membrane; Ethanolamines; Fluorenes; Lipid Bilayers; Lumefantrine; Male; Mice; Phenanthrenes; Phosphatidylcholines

2003
Decreasing pfmdr1 copy number in plasmodium falciparum malaria heightens susceptibility to mefloquine, lumefantrine, halofantrine, quinine, and artemisinin.
    The Journal of infectious diseases, 2006, Aug-15, Volume: 194, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; DNA, Protozoan; Drug Resistance, Multiple; Ethanolamines; Fluorenes; Genes, MDR; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Polymerase Chain Reaction; Protozoan Proteins; Quinine; Sesquiterpenes

2006
Determination of lumefantrine in rat plasma by liquid-liquid extraction using LC-MS/MS with electrospray ionization: assay development, validation and application to a pharmacokinetic study.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2009, Apr-15, Volume: 877, Issue:11-12

    Topics: Animals; Antimalarials; Calibration; Chromatography, High Pressure Liquid; Ethanolamines; Fluorenes; Indicators and Reagents; Lumefantrine; Male; Phenanthrenes; Rats; Rats, Sprague-Dawley; Reference Standards; Reproducibility of Results; Spectrometry, Mass, Electrospray Ionization

2009
Measurement of lumefantrine and its metabolite in plasma by high performance liquid chromatography with ultraviolet detection.
    Journal of pharmaceutical and biomedical analysis, 2011, Jan-05, Volume: 54, Issue:1

    Topics: Acetates; Artemether; Artemisinins; Calibration; Chemistry Techniques, Analytical; Chromatography; Chromatography, High Pressure Liquid; Ethanolamines; Fluorenes; Hexanes; Kinetics; Lumefantrine; Models, Chemical; Phenanthrenes; Regression Analysis; Reproducibility of Results; Spectrophotometry, Ultraviolet; Ultraviolet Rays

2011
Identification and functional validation of the novel antimalarial resistance locus PF10_0355 in Plasmodium falciparum.
    PLoS genetics, 2011, Volume: 7, Issue:4

    Topics: Antimalarials; Drug Resistance; Ethanolamines; Fluorenes; Gene Dosage; Gene Expression; Genetic Association Studies; Genetic Loci; Genetic Variation; Genotype; Haplotypes; Linkage Disequilibrium; Lumefantrine; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Polymorphism, Single Nucleotide; Selection, Genetic

2011
Modulation of PF10_0355 (MSPDBL2) alters Plasmodium falciparum response to antimalarial drugs.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:7

    Topics: Antimalarials; Base Sequence; DNA Copy Number Variations; Drug Resistance; Ethanolamines; Fluorenes; Gene Dosage; Gene Frequency; Genes, Protozoan; Lumefantrine; Malaria, Falciparum; Mefloquine; Mutation; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Sequence Analysis, DNA

2013
Simultaneous quantification of proposed anti-malarial combination comprising of lumefantrine and CDRI 97-78 in rat plasma using the HPLC-ESI-MS/MS method: application to drug interaction study.
    Malaria journal, 2015, Apr-22, Volume: 14

    Topics: Animals; Antimalarials; Blood Chemical Analysis; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Drug Combinations; Ethanolamines; Fluorenes; Lumefantrine; Male; Phenanthrenes; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry

2015
Assessment of pharmacokinetic compatibility of short acting CDRI candidate trioxane derivative, 99-411, with long acting prescription antimalarials, lumefantrine and piperaquine.
    Scientific reports, 2015, Nov-25, Volume: 5

    Topics: Animals; Antimalarials; Chromatography, High Pressure Liquid; Ethanolamines; Fluorenes; Half-Life; Heterocyclic Compounds; Humans; Lumefantrine; Microsomes, Liver; Phenanthrenes; Quinolines; Rats; Spiro Compounds; Tandem Mass Spectrometry

2015
Low-Frequency Raman Scattering Spectroscopy as an Accessible Approach to Understand Drug Solubilization in Milk-Based Formulations during Digestion.
    Molecular pharmaceutics, 2020, 03-02, Volume: 17, Issue:3

    Topics: Administration, Oral; Aminoquinolines; Animals; Biological Availability; Clofazimine; Digestion; Drug Compounding; Drug Delivery Systems; Ferrous Compounds; Infant Formula; Lipolysis; Lumefantrine; Metallocenes; Milk; Phenanthrenes; Scattering, Small Angle; Solubility; Spectrum Analysis, Raman; Suspensions; Water; X-Ray Diffraction

2020