Page last updated: 2024-09-03

gyki 53655 and tetrodotoxin

gyki 53655 has been researched along with tetrodotoxin in 11 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(tetrodotoxin)
Trials
(tetrodotoxin)
Recent Studies (post-2010) (tetrodotoxin)
11102212,992111,477

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)tetrodotoxin (IC50)
Sodium channel protein type 9 subunit alphaHomo sapiens (human)0.0186

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (45.45)18.2507
2000's3 (27.27)29.6817
2010's3 (27.27)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kombian, SB; Pittman, QJ; Saleh, TM; Zidichouski, JA1
Freund-Mercier, MJ; Jo, YH; Schlichter, R; Stoeckel, ME1
Bureau, I; Mulle, C1
Ben-Ari, Y; Dzhala, V; Khalilov, I; Khazipov, R; Lamsa, K; Leinekugel, X; Medina, I; Melyan, Z1
Ben-Ari, Y; Chevassus-Au-Louis, N; Diabira, D; Gozlan, H; Hennou, S1
Closier, M; Iop, F; Lestage, P; Lockhart, B1
Hartveit, E; Mørkve, SH; Veruki, ML1
Ibarretxe, G; Jaskolski, F; Mulle, C; Perrais, D; Vimeney, A1
Abrahamsson, T; Cathala, L; Digregorio, DA; Matsui, K; Shigemoto, R1
Jiang, L; Kang, D; Kang, J1
Ballanyi, K; Rancic, V; Rawal, B1

Other Studies

11 other study(ies) available for gyki 53655 and tetrodotoxin

ArticleYear
Cholecystokinin and neurotensin inversely modulate excitatory synaptic transmission in the parabrachial nucleus in vitro.
    Neuroscience, 1997, Volume: 77, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cholecystokinin; Devazepide; Electric Conductivity; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hormone Antagonists; Interneurons; N-Methylaspartate; Neural Inhibition; Neurons, Afferent; Neurotensin; Patch-Clamp Techniques; Phenylurea Compounds; Pons; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin

1997
Oxytocin modulates glutamatergic synaptic transmission between cultured neonatal spinal cord dorsal horn neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Apr-01, Volume: 18, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Electric Stimulation; Enkephalin, Methionine; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamate Decarboxylase; Glutamic Acid; Immunohistochemistry; Neurons; Nociceptors; Oxytocin; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Spinal Cord; Synaptic Transmission; Tetrodotoxin

1998
Potentiation of GABAergic synaptic transmission by AMPA receptors in mouse cerebellar stellate cells: changes during development.
    The Journal of physiology, 1998, Jun-15, Volume: 509 ( Pt 3)

    Topics: Age Factors; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Cadmium; Cerebellum; Dose-Response Relationship, Drug; Evoked Potentials; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Kainic Acid; Mice; Neural Inhibition; Neuromuscular Depolarizing Agents; Neurons; Receptors, AMPA; Receptors, Kainic Acid; Synaptic Transmission; Tetrodotoxin

1998
Maturation of kainate-induced epileptiform activities in interconnected intact neonatal limbic structures in vitro.
    The European journal of neuroscience, 1999, Volume: 11, Issue:10

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Electrophysiology; Entorhinal Cortex; Epilepsy; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Limbic System; Male; Organ Culture Techniques; Potassium; Rats; Rats, Wistar; Septal Nuclei; Synapses; Tetrodotoxin

1999
Late embryonic expression of AMPA receptor function in the CA1 region of the intact hippocampus in vitro.
    The European journal of neuroscience, 1999, Volume: 11, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Afferent Pathways; Aging; Animals; Animals, Newborn; Benzodiazepines; Bicuculline; Cations, Divalent; Electric Stimulation; Embryonic and Fetal Development; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; Hippocampus; Hypoxia; Lysine; Pyramidal Cells; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Synapses; Tetrodotoxin

1999
(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide: (S18986-1) a positive modulator of AMPA receptors enhances (S)-AMPA-mediated [3H]noradrenaline release from rat hippocampal and frontal cortex slices.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Frontal Lobe; Hippocampus; In Vitro Techniques; Male; Norepinephrine; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Stereoisomerism; Tetrodotoxin; Tritium

2000
Functional properties of spontaneous EPSCs and non-NMDA receptors in rod amacrine (AII) cells in the rat retina.
    The Journal of physiology, 2003, Jun-15, Volume: 549, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Algorithms; Amacrine Cells; Animals; Benzodiazepines; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; In Vitro Techniques; Kinetics; Membrane Potentials; Patch-Clamp Techniques; Piperazines; Presynaptic Terminals; Rats; Receptors, AMPA; Receptors, Glutamate; Retinal Rod Photoreceptor Cells; Synapses; Tetrodotoxin

2003
Fast regulation of axonal growth cone motility by electrical activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Jul-18, Volume: 27, Issue:29

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Animals, Newborn; Axons; Benzodiazepines; Calcium; Cell Movement; Cells, Cultured; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Growth Cones; Hippocampus; Kainic Acid; Mice; Mice, Knockout; Neurons; Receptors, Glutamate; Tetrodotoxin

2007
Thin dendrites of cerebellar interneurons confer sublinear synaptic integration and a gradient of short-term plasticity.
    Neuron, 2012, Mar-22, Volume: 73, Issue:6

    Topics: Age Factors; Animals; Animals, Newborn; Benzodiazepines; Biophysics; Cadmium Chloride; Cerebellum; Cesium; Chlorides; Dendrites; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; Imaging, Three-Dimensional; In Vitro Techniques; Indoles; Interneurons; Lasers; Mice; Microscopy, Confocal; Microscopy, Electron, Transmission; Models, Neurological; Neuronal Plasticity; Patch-Clamp Techniques; Potassium Channel Blockers; Receptors, AMPA; Sodium Channel Blockers; Statistics, Nonparametric; Synapses; Tetraethylammonium; Tetrodotoxin; Time Factors

2012
Potentiation of tonic GABAergic inhibition by activation of postsynaptic kainate receptors.
    Neuroscience, 2015, Jul-09, Volume: 298

    Topics: Action Potentials; Animals; Animals, Newborn; Benzodiazepines; Biophysics; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agents; GABAergic Neurons; Hippocampus; Humans; In Vitro Techniques; Kainic Acid; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Tetrodotoxin; Valine

2015
TARP mediation of accelerated and more regular locus coeruleus network bursting in neonatal rat brain slices.
    Neuropharmacology, 2019, Volume: 148

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Kynurenic Acid; Locus Coeruleus; Membrane Potentials; Neurons; Rats; Receptors, AMPA; Tetrodotoxin

2019