Page last updated: 2024-09-03

gyki 53655 and quinazolines

gyki 53655 has been researched along with quinazolines in 2 studies

Compound Research Comparison

Studies (gyki 53655)	Trials (gyki 53655)	Recent Studies (post-2010) (gyki 53655)	Studies (quinazolines)	Trials (quinazolines)	Recent Studies (post-2010) (quinazolines)
111	0	22	19,235	2,417	8,835

Protein Interaction Comparison

Protein	Taxonomy	gyki 53655 (IC50)	quinazolines (IC50)
Epidermal growth factor receptor	Homo sapiens (human)		0.027

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	1 (50.00)	29.6817
2010's	1 (50.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Balannik, V; Lerma, J; Menniti, FS; Paternain, AV; Stern-Bach, Y	1
Kurnikova, M; Narangoda, C; Sampson, JM; Singh, AK; Sobolevsky, AI; Yelshanskaya, MV	1

Other Studies

2 other study(ies) available for gyki 53655 and quinazolines

Article	Year
Molecular mechanism of AMPA receptor noncompetitive antagonism. Neuron, 2005, Oct-20, Volume: 48, Issue:2 Topics: Animals; Benzodiazepines; Binding Sites; Blotting, Western; Brain; Cell Line; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Humans; Membrane Potentials; Models, Neurological; Mutagenesis; Patch-Clamp Techniques; Peptide Fragments; Protein Conformation; Quinazolines; Rats; Receptors, AMPA; Transfection; Tritium; Xenopus laevis	2005
Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs. Neuron, 2016, Sep-21, Volume: 91, Issue:6 Topics: Animals; Anticonvulsants; Benzodiazepines; Binding Sites; Crystallization; Molecular Docking Simulation; Nitriles; Pyridones; Quinazolines; Rats; Receptors, AMPA	2016

Article

Year

Molecular mechanism of AMPA receptor noncompetitive antagonism.

Neuron, 2005, Oct-20, Volume: 48, Issue:2

Topics: Animals; Benzodiazepines; Binding Sites; Blotting, Western; Brain; Cell Line; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Humans; Membrane Potentials; Models, Neurological; Mutagenesis; Patch-Clamp Techniques; Peptide Fragments; Protein Conformation; Quinazolines; Rats; Receptors, AMPA; Transfection; Tritium; Xenopus laevis

2005

Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.

Neuron, 2016, Sep-21, Volume: 91, Issue:6

Topics: Animals; Anticonvulsants; Benzodiazepines; Binding Sites; Crystallization; Molecular Docking Simulation; Nitriles; Pyridones; Quinazolines; Rats; Receptors, AMPA

2016