gyki 53655 has been researched along with ly 293558 in 3 studies
Studies (gyki 53655) | Trials (gyki 53655) | Recent Studies (post-2010) (gyki 53655) | Studies (ly 293558) | Trials (ly 293558) | Recent Studies (post-2010) (ly 293558) |
---|---|---|---|---|---|
111 | 0 | 22 | 103 | 4 | 18 |
Protein | Taxonomy | gyki 53655 (IC50) | ly 293558 (IC50) |
---|---|---|---|
Glutamate receptor 1 | Rattus norvegicus (Norway rat) | 2.7869 | |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | 2.7869 | |
Glutamate receptor 3 | Rattus norvegicus (Norway rat) | 2.7869 | |
Glutamate receptor 4 | Rattus norvegicus (Norway rat) | 2.7869 | |
Glutamate receptor ionotropic, kainate 1 | Rattus norvegicus (Norway rat) | 0.23 | |
Glutamate receptor ionotropic, kainate 1 | Homo sapiens (human) | 0.5 | |
Glutamate receptor ionotropic, kainate 2 | Rattus norvegicus (Norway rat) | 0.23 | |
Glutamate receptor 1 | Homo sapiens (human) | 3.075 | |
Glutamate receptor 2 | Homo sapiens (human) | 3.075 | |
Glutamate receptor 3 | Homo sapiens (human) | 3.075 | |
Glutamate receptor ionotropic, kainate 3 | Rattus norvegicus (Norway rat) | 0.23 | |
Glutamate receptor 4 | Homo sapiens (human) | 3.075 | |
Glutamate receptor ionotropic, kainate 4 | Rattus norvegicus (Norway rat) | 0.23 | |
Glutamate receptor ionotropic, kainate 5 | Rattus norvegicus (Norway rat) | 0.23 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (66.67) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Burnett, JP; Desai, MA; Ornstein, PL; Schoepp, DD | 1 |
Bleakman, D; Bristow, DR; Savidge, JR | 1 |
Cebers, G; Kovács, AD; Liljequist, S | 1 |
3 other study(ies) available for gyki 53655 and ly 293558
Article | Year |
---|---|
Cyclothiazide acts at a site on the alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor complex that does not recognize competitive or noncompetitive AMPA receptor antagonists.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Hippocampus; In Vitro Techniques; Isoquinolines; Kainic Acid; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetrazoles | 1995 |
Identification of kainate receptor-mediated intracellular calcium increases in cultured rat cerebellar granule cells.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Calcium; Cells, Cultured; Cerebellum; Concanavalin A; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Intracellular Membranes; Isoquinolines; Kainic Acid; Neurons; Rats; Receptors, Kainic Acid; Tetrazoles | 1997 |
Kainate receptor-mediated activation of the AP-1 transcription factor complex in cultured rat cerebellar granule cells.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Concanavalin A; Dimerization; Excitatory Amino Acid Antagonists; Isoquinolines; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tetrazoles; Transcription Factor AP-1 | 2000 |