Page last updated: 2024-09-03

gyki 53655 and ly 293558

gyki 53655 has been researched along with ly 293558 in 3 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(ly 293558)
Trials
(ly 293558)
Recent Studies (post-2010) (ly 293558)
111022103418

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)ly 293558 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)2.7869
Glutamate receptor 2Rattus norvegicus (Norway rat)2.7869
Glutamate receptor 3Rattus norvegicus (Norway rat)2.7869
Glutamate receptor 4Rattus norvegicus (Norway rat)2.7869
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.23
Glutamate receptor ionotropic, kainate 1Homo sapiens (human)0.5
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.23
Glutamate receptor 1Homo sapiens (human)3.075
Glutamate receptor 2Homo sapiens (human)3.075
Glutamate receptor 3Homo sapiens (human)3.075
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.23
Glutamate receptor 4Homo sapiens (human)3.075
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.23
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.23

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burnett, JP; Desai, MA; Ornstein, PL; Schoepp, DD1
Bleakman, D; Bristow, DR; Savidge, JR1
Cebers, G; Kovács, AD; Liljequist, S1

Other Studies

3 other study(ies) available for gyki 53655 and ly 293558

ArticleYear
Cyclothiazide acts at a site on the alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor complex that does not recognize competitive or noncompetitive AMPA receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Hippocampus; In Vitro Techniques; Isoquinolines; Kainic Acid; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetrazoles

1995
Identification of kainate receptor-mediated intracellular calcium increases in cultured rat cerebellar granule cells.
    Journal of neurochemistry, 1997, Volume: 69, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Calcium; Cells, Cultured; Cerebellum; Concanavalin A; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Intracellular Membranes; Isoquinolines; Kainic Acid; Neurons; Rats; Receptors, Kainic Acid; Tetrazoles

1997
Kainate receptor-mediated activation of the AP-1 transcription factor complex in cultured rat cerebellar granule cells.
    Brain research bulletin, 2000, May-15, Volume: 52, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Concanavalin A; Dimerization; Excitatory Amino Acid Antagonists; Isoquinolines; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tetrazoles; Transcription Factor AP-1

2000