gyki 53655 has been researched along with glutamic acid in 17 studies
Studies (gyki 53655) | Trials (gyki 53655) | Recent Studies (post-2010) (gyki 53655) | Studies (glutamic acid) | Trials (glutamic acid) | Recent Studies (post-2010) (glutamic acid) |
---|---|---|---|---|---|
111 | 0 | 22 | 41,757 | 452 | 12,876 |
Protein | Taxonomy | gyki 53655 (IC50) | glutamic acid (IC50) |
---|---|---|---|
Chain A, GLUTAMATE RECEPTOR SUBUNIT 2 | Rattus norvegicus (Norway rat) | 0.821 | |
Chain A, Glutamate Receptor Subunit 2 | Rattus norvegicus (Norway rat) | 0.821 | |
Chain B, Glutamate Receptor Subunit 2 | Rattus norvegicus (Norway rat) | 0.821 | |
Metabotropic glutamate receptor 8 | Homo sapiens (human) | 0.0057 | |
Glutamate receptor ionotropic, NMDA 2D | Homo sapiens (human) | 0.07 | |
Glutamate receptor ionotropic, NMDA 3B | Homo sapiens (human) | 0.07 | |
Glutamate receptor 1 | Rattus norvegicus (Norway rat) | 0.5885 | |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.5885 | |
Glutamate receptor 3 | Rattus norvegicus (Norway rat) | 0.5885 | |
Glutamate receptor 4 | Rattus norvegicus (Norway rat) | 0.5885 | |
Glutamate receptor ionotropic, kainate 1 | Rattus norvegicus (Norway rat) | 0.38 | |
Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | 0.1533 | |
Glutamate receptor ionotropic, kainate 2 | Rattus norvegicus (Norway rat) | 0.38 | |
Glutamate receptor 1 | Homo sapiens (human) | 0.613 | |
Glutamate receptor 2 | Homo sapiens (human) | 0.613 | |
Glutamate receptor 3 | Homo sapiens (human) | 0.613 | |
Glutamate receptor ionotropic, kainate 3 | Rattus norvegicus (Norway rat) | 0.38 | |
Excitatory amino acid transporter 1 | Homo sapiens (human) | 207 | |
Glutamate receptor 4 | Homo sapiens (human) | 0.613 | |
Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | 0.1533 | |
Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | 0.1533 | |
Glutamate receptor ionotropic, NMDA 2C | Rattus norvegicus (Norway rat) | 0.1533 | |
Glutamate receptor ionotropic, kainate 4 | Rattus norvegicus (Norway rat) | 0.38 | |
Glutamate receptor ionotropic, NMDA 1 | Homo sapiens (human) | 0.07 | |
Glutamate receptor ionotropic, NMDA 2A | Homo sapiens (human) | 0.07 | |
Glutamate receptor ionotropic, NMDA 2B | Homo sapiens (human) | 0.07 | |
Glutamate receptor ionotropic, NMDA 2C | Homo sapiens (human) | 0.07 | |
Glutamate receptor ionotropic, NMDA 2D | Rattus norvegicus (Norway rat) | 0.1533 | |
Glutamate receptor ionotropic, kainate 5 | Rattus norvegicus (Norway rat) | 0.38 | |
Glutamate receptor ionotropic, NMDA 3A | Homo sapiens (human) | 0.07 | |
Glutamate receptor ionotropic, NMDA 3B | Rattus norvegicus (Norway rat) | 0.1533 | |
Glutamate receptor ionotropic, NMDA 3A | Rattus norvegicus (Norway rat) | 0.1533 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (35.29) | 18.2507 |
2000's | 8 (47.06) | 29.6817 |
2010's | 3 (17.65) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
England, PM; Fleming, JJ | 1 |
Huettner, JE; Wilding, TJ | 1 |
Castillo, PE; Malenka, RC; Nicoll, RA | 1 |
Freund-Mercier, MJ; Jo, YH; Schlichter, R; Stoeckel, ME | 1 |
Lu, T; Shen, Y; Yang, XL | 1 |
Baranyi, M; Milusheva, E; Nakai, T; Satoh, T; Uchihashi, Y; Vizi, ES | 1 |
Shen, Y; Yang, XL; Zhou, Y | 1 |
Lerma, J; López-García, JC; Rodríguez-Moreno, A | 1 |
Cull-Candy, SG; Liu, SQ | 1 |
Brorson, JR; Ihle, EC; Patneau, DK; Robberecht, W; Vandenberghe, W | 1 |
Akiba, I; Barsoumian, E; Brenner, M; Iizuka, M; Nishimura, S; Palluk, R; Steinhäuser, C; Weiser, T; Wienrich, M; Zhou, M | 1 |
Baumbarger, PJ; Muhlhauser, M; Nisenbaum, ES; Yang, CR; Zhai, J | 1 |
Alberdi, E; Marino, A; Matute, C; Sánchez-Gómez, MV | 1 |
Clarke, VR; Collingridge, GL | 1 |
Cathala, L; Cull-Candy, SG; DiGregorio, DA; Holderith, NB; Nusser, Z | 1 |
Rodríguez-Moreno, A; Sihra, TS | 1 |
Babai, N; Feigenspan, A | 1 |
17 other study(ies) available for gyki 53655 and glutamic acid
Article | Year |
---|---|
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA | 2010 |
Activation and desensitization of hippocampal kainate receptors.
Topics: Animals; Animals, Newborn; Benzodiazepines; Cells, Cultured; Dizocilpine Maleate; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamates; Glutamic Acid; Hippocampus; Kainic Acid; Lanthanum; Membrane Potentials; Neurons; Rats; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate | 1997 |
Kainate receptors mediate a slow postsynaptic current in hippocampal CA3 neurons.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamic Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Kainic Acid; Nerve Fibers; Neurons; Receptors, AMPA; Receptors, Kainic Acid; Synapses | 1997 |
Oxytocin modulates glutamatergic synaptic transmission between cultured neonatal spinal cord dorsal horn neurons.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Electric Stimulation; Enkephalin, Methionine; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamate Decarboxylase; Glutamic Acid; Immunohistochemistry; Neurons; Nociceptors; Oxytocin; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Spinal Cord; Synaptic Transmission; Tetrodotoxin | 1998 |
Desensitization of AMPA receptors on horizontal cells isolated from crucian carp retina.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Cells, Cultured; Drug Tolerance; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Kainic Acid; Patch-Clamp Techniques; Receptors, AMPA; Retina | 1998 |
Excessive release of [3H]noradrenaline and glutamate in response to simulation of ischemic conditions in rat spinal cord slice preparation: effect of NMDA and AMPA receptor antagonists.
Topics: Animals; Benzodiazepines; Dizocilpine Maleate; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Glucose; Glutamic Acid; Hypoxia; In Vitro Techniques; Ischemia; Male; Norepinephrine; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Stereoisomerism; Tritium | 1999 |
Characterization of AMPA receptors on isolated amacrine-like cells in carp retina.
Topics: Alternative Splicing; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Separation; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Ion Channels; Kainic Acid; Membrane Potentials; N-Methylaspartate; Patch-Clamp Techniques; Phenoxyacetates; Receptors, AMPA; Retina | 1999 |
Two populations of kainate receptors with separate signaling mechanisms in hippocampal interneurons.
Topics: 2-Amino-5-phosphonovalerate; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Bicuculline; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Indoles; Interneurons; Isoxazoles; Kainic Acid; Lidocaine; Maleimides; Naphthalenes; Nerve Tissue Proteins; Patch-Clamp Techniques; Propionates; Protein Kinase C; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Kainic Acid; Receptors, Presynaptic; Signal Transduction; Staurosporine; Virulence Factors, Bordetella | 2000 |
Synaptic activity at calcium-permeable AMPA receptors induces a switch in receptor subtype.
Topics: Animals; Benzodiazepines; Calcium; Cell Membrane Permeability; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Ion Channel Gating; Neuronal Plasticity; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Synapses; Synaptic Membranes | 2000 |
AMPA receptor current density, not desensitization, predicts selective motoneuron vulnerability.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Astrocytes; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Membrane Potentials; Motor Neurons; Patch-Clamp Techniques; Posterior Horn Cells; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord | 2000 |
Characterization of the anticonvulsant and neuroprotectant BIIR 561 CL in vitro: effects on native and recombinant alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptors.
Topics: Animals; Anticonvulsants; Benzodiazepines; Cells, Cultured; Dose-Response Relationship, Drug; Female; Glutamic Acid; Humans; Hydrogen-Ion Concentration; Neuroprotective Agents; Oxadiazoles; Rats; Receptors, AMPA; Recombinant Proteins | 2000 |
Positive modulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid (AMPA) receptors in prefrontal cortical pyramidal neurons by a novel allosteric potentiator.
Topics: Allosteric Regulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Dioxoles; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Sulfonamides | 2001 |
Ca(2+) influx through AMPA or kainate receptors alone is sufficient to initiate excitotoxicity in cultured oligodendrocytes.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Calcium; Calcium Channel Blockers; Cell Death; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Lanthanum; Neurotoxins; Nifedipine; Oligodendroglia; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid | 2002 |
Characterisation of the effects of ATPA, a GLU(K5) kainate receptor agonist, on GABAergic synaptic transmission in the CA1 region of rat hippocampal slices.
Topics: Animals; Benzodiazepines; Dose-Response Relationship, Drug; Drug Interactions; Electric Impedance; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agents; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Kainic Acid; Membrane Potentials; Neural Inhibition; Propionates; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission; Valine | 2004 |
Changes in synaptic structure underlie the developmental speeding of AMPA receptor-mediated EPSCs.
Topics: Age Factors; Animals; Animals, Newborn; Benzodiazepines; Cerebellum; Dose-Response Relationship, Radiation; Electric Conductivity; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Imaging, Three-Dimensional; Immunohistochemistry; In Vitro Techniques; Kynurenic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Microscopy, Electron, Transmission; Models, Neurological; Nerve Fibers; Neurons; Patch-Clamp Techniques; Receptors, AMPA; Synapses; Synaptic Transmission; Temperature; Ultrasonography | 2005 |
Presynaptic kainate receptor-mediated facilitation of glutamate release involves Ca2+-calmodulin and PKA in cerebrocortical synaptosomes.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzodiazepines; Calcium; Calmodulin; Cerebral Cortex; Cyclic AMP-Dependent Protein Kinases; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Isoquinolines; Kainic Acid; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Receptors, Presynaptic; Sulfonamides; Synaptic Transmission; Synaptosomes; Thionucleotides | 2013 |
Functional properties of spontaneous excitatory currents and encoding of light/dark transitions in horizontal cells of the mouse retina.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Dendrites; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; Glutamic Acid; Mice; Mice, Transgenic; Neural Pathways; Photic Stimulation; Receptors, AMPA; Receptors, Kainic Acid; Retinal Cone Photoreceptor Cells; Retinal Horizontal Cells | 2015 |