Page last updated: 2024-09-03

gyki 53655 and fg 9041

gyki 53655 has been researched along with fg 9041 in 2 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(fg 9041)
Trials
(fg 9041)
Recent Studies (post-2010) (fg 9041)
1110228120122

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)fg 9041 (IC50)
Chain A, GLUTAMATE RECEPTOR SUBUNIT 2Rattus norvegicus (Norway rat)0.998
Chain A, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.998
Chain B, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.998
fatty acid synthaseHomo sapiens (human)7.755
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)5.1
Glutamate receptor 1Homo sapiens (human)1.51
Glutamate receptor 2Homo sapiens (human)1.51
Glutamate receptor 3Homo sapiens (human)1.51
Glutamate receptor 4Homo sapiens (human)1.51
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)5.1
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)5.1
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)5.1
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)5.1
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)5.1
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)5.1

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bardoul, M; Drian, MJ; König, N1
Hays, FA; Menuz, K; Nicoll, RA; Stroud, RM1

Other Studies

2 other study(ies) available for gyki 53655 and fg 9041

ArticleYear
Blockade of AMPA/kainate receptors can either decrease or increase the survival of cultured neocortical cells depending on the stage of maturation.
    Neurochemistry international, 2001, Volume: 38, Issue:6

    Topics: Animals; Benzodiazepines; Cell Survival; Cells, Cultured; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Female; Kainic Acid; N-Methylaspartate; Neocortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid

2001
TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists.
    Science (New York, N.Y.), 2007, Nov-02, Volume: 318, Issue:5851

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Binding, Competitive; Cell Line; Cerebellum; Crystallography, X-Ray; Drug Partial Agonism; Hippocampus; Humans; In Vitro Techniques; Interneurons; Mice; Models, Molecular; Patch-Clamp Techniques; Protein Conformation; Protein Subunits; Pyramidal Cells; Quinoxalines; Receptors, AMPA; Structure-Activity Relationship; Synaptic Transmission; Trichlormethiazide

2007