gyki 53655 has been researched along with cyclothiazide in 23 studies
Studies (gyki 53655) | Trials (gyki 53655) | Recent Studies (post-2010) (gyki 53655) | Studies (cyclothiazide) | Trials (cyclothiazide) | Recent Studies (post-2010) (cyclothiazide) |
---|---|---|---|---|---|
111 | 0 | 22 | 396 | 4 | 51 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 12 (52.17) | 18.2507 |
2000's | 10 (43.48) | 29.6817 |
2010's | 1 (4.35) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
England, PM; Fleming, JJ | 1 |
Burnett, JP; Desai, MA; Ornstein, PL; Schoepp, DD | 1 |
Lodge, D; Palmer, AJ | 1 |
Huettner, JE; Wilding, TJ | 1 |
Feltz, A; Nooney, JM | 1 |
Mayer, ML; Partin, KM | 1 |
Ballyk, BA; Bath, CP; Bleakman, D; Bufton, HR; Kamboj, RK; Lodge, D; Palmer, AJ; Schoepp, DD; Sharpe, EF; Tarnawa, I; Woolley, ML | 1 |
Allen, TG; Waters, DJ | 1 |
Carvalho, AP; Duarte, CB; Ferreira, IL | 1 |
Geurtz, W; Hatt, H; Okada, T; Schultz, K; Weiler, R | 1 |
Bristow, DR; Lock, EA; Savidge, JR; Sturgess, NC | 1 |
Perkinton, MS; Sihra, TS; Williams, RJ | 1 |
Shen, Y; Yang, XL; Zhou, Y | 1 |
Cotton, JL; Partin, KM | 1 |
Dietrich, D; Dybek, A; Schumacher, TB; Seifert, G; Steinhäuser, C; Weiser, T; Wienrich, M; Wilhelm, D; Zhou, M | 1 |
Cebers, G; Kovács, AD; Liljequist, S | 1 |
Closier, M; Iop, F; Lestage, P; Lockhart, B | 1 |
Brorson, JR; Ihle, EC; Patneau, DK; Robberecht, W; Vandenberghe, W | 1 |
Heggelund, P; Kielland, A | 1 |
Allgaier, C; Fischer, W; Franke, H; Illes, P; Scheibler, P | 1 |
Hartveit, E; Mørkve, SH; Veruki, ML | 1 |
Ali, AB | 1 |
Li, W; Massey, SC; Trexler, EB | 1 |
23 other study(ies) available for gyki 53655 and cyclothiazide
Article | Year |
---|---|
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA | 2010 |
Cyclothiazide acts at a site on the alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor complex that does not recognize competitive or noncompetitive AMPA receptor antagonists.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Hippocampus; In Vitro Techniques; Isoquinolines; Kainic Acid; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetrazoles | 1995 |
Cyclothiazide reverses AMPA receptor antagonism of the 2,3-benzodiazepine, GYKI 53655.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cerebral Cortex; Diuretics; Excitatory Amino Acid Antagonists; Ibotenic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors | 1993 |
Differential antagonism of alpha-amino-3-hydroxy-5-methyl-4- isoxazolepropionic acid-preferring and kainate-preferring receptors by 2,3-benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding, Competitive; Cerebral Cortex; Concanavalin A; Electrophysiology; Ganglia, Spinal; Kainic Acid; Membrane Potentials; Neurons; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Kainic Acid; Substrate Specificity | 1995 |
Inhibition by cyclothiazide of neuronal nicotinic responses in bovine chromaffin cells.
Topics: Acetylcholine; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Bungarotoxins; Cattle; Cells, Cultured; Chromaffin System; Dimethylphenylpiperazinium Iodide; Diuretics; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Neurons; Nicotinic Antagonists; Receptors, AMPA; Receptors, Nicotinic; Sodium Chloride Symporter Inhibitors | 1995 |
Negative allosteric modulation of wild-type and mutant AMPA receptors by GYKI 53655.
Topics: Allosteric Regulation; Amino Acid Sequence; Animals; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Molecular Sequence Data; Prosencephalon; Rats; Receptors, AMPA; Recombinant Proteins; RNA Splicing; RNA, Messenger; Xenopus laevis | 1996 |
Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: stereospecificity and selectivity profiles.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Cerebellum; Cerebral Cortex; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Humans; Kidney; Membrane Potentials; Molecular Structure; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Spinal Cord; Structure-Activity Relationship; Transfection | 1996 |
Ca2+-permeable non-NMDA glutamate receptors in rat magnocellular basal forebrain neurones.
Topics: Animals; Basal Ganglia; Benzodiazepines; Benzothiadiazines; Calcium; Cations, Divalent; Cells, Cultured; Concanavalin A; Diuretics; Electrophysiology; Excitatory Amino Acid Antagonists; Membrane Potentials; Neurons; Patch-Clamp Techniques; Prosencephalon; Rats; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sodium Chloride Symporter Inhibitors | 1998 |
Kainate-induced retina amacrine-like cell damage is mediated by AMPA receptors.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium Radioisotopes; Cells, Cultured; Chickens; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Neuromuscular Depolarizing Agents; Receptors, AMPA; Receptors, Kainic Acid; Retina | 1998 |
AMPA-preferring receptors with high Ca2+ permeability mediate dendritic plasticity of retinal horizontal cells.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carps; Dark Adaptation; Dendrites; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Membrane Potentials; Microscopy, Electron; Neuronal Plasticity; Patch-Clamp Techniques; Receptors, AMPA; Receptors, Kainic Acid; Retina | 1999 |
Characterisation of kainate receptor mediated whole-cell currents in rat cultured cerebellar granule cells.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Concanavalin A; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamates; Hippocampus; Kinetics; Neurons; Neurotoxins; Patch-Clamp Techniques; Rats; Receptors, Kainic Acid; Spider Venoms | 1999 |
Ca(2+)-permeable AMPA receptors induce phosphorylation of cAMP response element-binding protein through a phosphatidylinositol 3-kinase-dependent stimulation of the mitogen-activated protein kinase signaling cascade in neurons.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Androstadienes; Animals; Arachidonic Acid; Benzodiazepines; Benzothiadiazines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Membrane Permeability; Cell Survival; Cells, Cultured; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Flavonoids; Genistein; GTP-Binding Proteins; Kinetics; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neurons; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphorylation; Receptors, AMPA; Signal Transduction; Virulence Factors, Bordetella; Wortmannin | 1999 |
Characterization of AMPA receptors on isolated amacrine-like cells in carp retina.
Topics: Alternative Splicing; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Separation; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Ion Channels; Kainic Acid; Membrane Potentials; N-Methylaspartate; Patch-Clamp Techniques; Phenoxyacetates; Receptors, AMPA; Retina | 1999 |
The contributions of GluR2 to allosteric modulation of AMPA receptors.
Topics: Allosteric Regulation; Amino Acid Substitution; Animals; Benzodiazepines; Benzothiadiazines; Cell Membrane; Excitatory Amino Acid Antagonists; Membrane Potentials; Oocytes; Receptors, AMPA; Recombinant Proteins; Xenopus laevis | 2000 |
Developmental regulation of AMPA-receptor properties in CA1 pyramidal neurons of rat hippocampus.
Topics: Alternative Splicing; Animals; Animals, Newborn; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Female; Hippocampus; In Vitro Techniques; Kinetics; Patch-Clamp Techniques; Pyramidal Cells; Quinoxalines; Rats; Receptors, AMPA; Receptors, Kainic Acid | 2000 |
Kainate receptor-mediated activation of the AP-1 transcription factor complex in cultured rat cerebellar granule cells.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Concanavalin A; Dimerization; Excitatory Amino Acid Antagonists; Isoquinolines; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tetrazoles; Transcription Factor AP-1 | 2000 |
(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide: (S18986-1) a positive modulator of AMPA receptors enhances (S)-AMPA-mediated [3H]noradrenaline release from rat hippocampal and frontal cortex slices.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Frontal Lobe; Hippocampus; In Vitro Techniques; Male; Norepinephrine; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Stereoisomerism; Tetrodotoxin; Tritium | 2000 |
AMPA receptor current density, not desensitization, predicts selective motoneuron vulnerability.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Astrocytes; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Membrane Potentials; Motor Neurons; Patch-Clamp Techniques; Posterior Horn Cells; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord | 2000 |
AMPA receptor properties at the synapse between retinal afferents and thalamocortical cells in the dorsal lateral geniculate nucleus of the rat.
Topics: 2-Amino-5-phosphonovalerate; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Geniculate Bodies; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Retinal Ganglion Cells; Synapses; Visual Cortex; Visual Pathways | 2001 |
AMPA-induced Ca(2+) influx in cultured rat cortical nonpyramidal neurones: pharmacological characterization using fura-2 microfluorimetry.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Cerebral Cortex; Cobalt; Diazoxide; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorescence; Fluorometry; Fura-2; gamma-Aminobutyric Acid; Immunohistochemistry; N-Methylaspartate; Neurons; Piperazines; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate | 2002 |
Functional characteristics of non-NMDA-type ionotropic glutamate receptor channels in AII amacrine cells in rat retina.
Topics: Algorithms; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Concanavalin A; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kainic Acid; Membrane Potentials; Patch-Clamp Techniques; Rats; Receptors, AMPA; Receptors, Glutamate; Retina; Sodium | 2002 |
Involvement of post-synaptic kainate receptors during synaptic transmission between unitary connections in rat neocortex.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Dicarboxylic Acids; Drug Interactions; Electric Conductivity; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Membrane Potentials; Neocortex; Neural Pathways; Neurotransmitter Uptake Inhibitors; Patch-Clamp Techniques; Pyramidal Cells; Pyrrolidines; Rats; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission; Time Factors; Valine | 2003 |
Simultaneous contribution of two rod pathways to AII amacrine and cone bipolar cell light responses.
Topics: Amacrine Cells; Animals; Benzodiazepines; Benzothiadiazines; Diagnostic Imaging; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Fluorescein; GABA Antagonists; Glycine Agents; In Vitro Techniques; Light; Male; Membrane Potentials; Models, Biological; Neurons; Patch-Clamp Techniques; Picrotoxin; Quinoxalines; Rabbits; Retina; Retinal Rod Photoreceptor Cells; Strychnine; Synapses; Synaptic Transmission; Visual Pathways | 2005 |