Page last updated: 2024-09-03

gyki 53655 and cyclothiazide

gyki 53655 has been researched along with cyclothiazide in 23 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(cyclothiazide)
Trials
(cyclothiazide)
Recent Studies (post-2010) (cyclothiazide)
111022396451

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (52.17)18.2507
2000's10 (43.48)29.6817
2010's1 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
England, PM; Fleming, JJ1
Burnett, JP; Desai, MA; Ornstein, PL; Schoepp, DD1
Lodge, D; Palmer, AJ1
Huettner, JE; Wilding, TJ1
Feltz, A; Nooney, JM1
Mayer, ML; Partin, KM1
Ballyk, BA; Bath, CP; Bleakman, D; Bufton, HR; Kamboj, RK; Lodge, D; Palmer, AJ; Schoepp, DD; Sharpe, EF; Tarnawa, I; Woolley, ML1
Allen, TG; Waters, DJ1
Carvalho, AP; Duarte, CB; Ferreira, IL1
Geurtz, W; Hatt, H; Okada, T; Schultz, K; Weiler, R1
Bristow, DR; Lock, EA; Savidge, JR; Sturgess, NC1
Perkinton, MS; Sihra, TS; Williams, RJ1
Shen, Y; Yang, XL; Zhou, Y1
Cotton, JL; Partin, KM1
Dietrich, D; Dybek, A; Schumacher, TB; Seifert, G; Steinhäuser, C; Weiser, T; Wienrich, M; Wilhelm, D; Zhou, M1
Cebers, G; Kovács, AD; Liljequist, S1
Closier, M; Iop, F; Lestage, P; Lockhart, B1
Brorson, JR; Ihle, EC; Patneau, DK; Robberecht, W; Vandenberghe, W1
Heggelund, P; Kielland, A1
Allgaier, C; Fischer, W; Franke, H; Illes, P; Scheibler, P1
Hartveit, E; Mørkve, SH; Veruki, ML1
Ali, AB1
Li, W; Massey, SC; Trexler, EB1

Other Studies

23 other study(ies) available for gyki 53655 and cyclothiazide

ArticleYear
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
Cyclothiazide acts at a site on the alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor complex that does not recognize competitive or noncompetitive AMPA receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Hippocampus; In Vitro Techniques; Isoquinolines; Kainic Acid; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetrazoles

1995
Cyclothiazide reverses AMPA receptor antagonism of the 2,3-benzodiazepine, GYKI 53655.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cerebral Cortex; Diuretics; Excitatory Amino Acid Antagonists; Ibotenic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1993
Differential antagonism of alpha-amino-3-hydroxy-5-methyl-4- isoxazolepropionic acid-preferring and kainate-preferring receptors by 2,3-benzodiazepines.
    Molecular pharmacology, 1995, Volume: 47, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding, Competitive; Cerebral Cortex; Concanavalin A; Electrophysiology; Ganglia, Spinal; Kainic Acid; Membrane Potentials; Neurons; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Kainic Acid; Substrate Specificity

1995
Inhibition by cyclothiazide of neuronal nicotinic responses in bovine chromaffin cells.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Acetylcholine; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Bungarotoxins; Cattle; Cells, Cultured; Chromaffin System; Dimethylphenylpiperazinium Iodide; Diuretics; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Neurons; Nicotinic Antagonists; Receptors, AMPA; Receptors, Nicotinic; Sodium Chloride Symporter Inhibitors

1995
Negative allosteric modulation of wild-type and mutant AMPA receptors by GYKI 53655.
    Molecular pharmacology, 1996, Volume: 49, Issue:1

    Topics: Allosteric Regulation; Amino Acid Sequence; Animals; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Molecular Sequence Data; Prosencephalon; Rats; Receptors, AMPA; Recombinant Proteins; RNA Splicing; RNA, Messenger; Xenopus laevis

1996
Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: stereospecificity and selectivity profiles.
    Neuropharmacology, 1996, Volume: 35, Issue:12

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Cerebellum; Cerebral Cortex; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Humans; Kidney; Membrane Potentials; Molecular Structure; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Spinal Cord; Structure-Activity Relationship; Transfection

1996
Ca2+-permeable non-NMDA glutamate receptors in rat magnocellular basal forebrain neurones.
    The Journal of physiology, 1998, Apr-15, Volume: 508 ( Pt 2)

    Topics: Animals; Basal Ganglia; Benzodiazepines; Benzothiadiazines; Calcium; Cations, Divalent; Cells, Cultured; Concanavalin A; Diuretics; Electrophysiology; Excitatory Amino Acid Antagonists; Membrane Potentials; Neurons; Patch-Clamp Techniques; Prosencephalon; Rats; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sodium Chloride Symporter Inhibitors

1998
Kainate-induced retina amacrine-like cell damage is mediated by AMPA receptors.
    Neuroreport, 1998, Oct-26, Volume: 9, Issue:15

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium Radioisotopes; Cells, Cultured; Chickens; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Neuromuscular Depolarizing Agents; Receptors, AMPA; Receptors, Kainic Acid; Retina

1998
AMPA-preferring receptors with high Ca2+ permeability mediate dendritic plasticity of retinal horizontal cells.
    The European journal of neuroscience, 1999, Volume: 11, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carps; Dark Adaptation; Dendrites; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Membrane Potentials; Microscopy, Electron; Neuronal Plasticity; Patch-Clamp Techniques; Receptors, AMPA; Receptors, Kainic Acid; Retina

1999
Characterisation of kainate receptor mediated whole-cell currents in rat cultured cerebellar granule cells.
    Neuropharmacology, 1999, Volume: 38, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Concanavalin A; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamates; Hippocampus; Kinetics; Neurons; Neurotoxins; Patch-Clamp Techniques; Rats; Receptors, Kainic Acid; Spider Venoms

1999
Ca(2+)-permeable AMPA receptors induce phosphorylation of cAMP response element-binding protein through a phosphatidylinositol 3-kinase-dependent stimulation of the mitogen-activated protein kinase signaling cascade in neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-15, Volume: 19, Issue:14

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Androstadienes; Animals; Arachidonic Acid; Benzodiazepines; Benzothiadiazines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Membrane Permeability; Cell Survival; Cells, Cultured; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Flavonoids; Genistein; GTP-Binding Proteins; Kinetics; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neurons; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphorylation; Receptors, AMPA; Signal Transduction; Virulence Factors, Bordetella; Wortmannin

1999
Characterization of AMPA receptors on isolated amacrine-like cells in carp retina.
    The European journal of neuroscience, 1999, Volume: 11, Issue:12

    Topics: Alternative Splicing; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Separation; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Ion Channels; Kainic Acid; Membrane Potentials; N-Methylaspartate; Patch-Clamp Techniques; Phenoxyacetates; Receptors, AMPA; Retina

1999
The contributions of GluR2 to allosteric modulation of AMPA receptors.
    Neuropharmacology, 2000, Volume: 39, Issue:1

    Topics: Allosteric Regulation; Amino Acid Substitution; Animals; Benzodiazepines; Benzothiadiazines; Cell Membrane; Excitatory Amino Acid Antagonists; Membrane Potentials; Oocytes; Receptors, AMPA; Recombinant Proteins; Xenopus laevis

2000
Developmental regulation of AMPA-receptor properties in CA1 pyramidal neurons of rat hippocampus.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: Alternative Splicing; Animals; Animals, Newborn; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Female; Hippocampus; In Vitro Techniques; Kinetics; Patch-Clamp Techniques; Pyramidal Cells; Quinoxalines; Rats; Receptors, AMPA; Receptors, Kainic Acid

2000
Kainate receptor-mediated activation of the AP-1 transcription factor complex in cultured rat cerebellar granule cells.
    Brain research bulletin, 2000, May-15, Volume: 52, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Concanavalin A; Dimerization; Excitatory Amino Acid Antagonists; Isoquinolines; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tetrazoles; Transcription Factor AP-1

2000
(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide: (S18986-1) a positive modulator of AMPA receptors enhances (S)-AMPA-mediated [3H]noradrenaline release from rat hippocampal and frontal cortex slices.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Frontal Lobe; Hippocampus; In Vitro Techniques; Male; Norepinephrine; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Stereoisomerism; Tetrodotoxin; Tritium

2000
AMPA receptor current density, not desensitization, predicts selective motoneuron vulnerability.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Oct-01, Volume: 20, Issue:19

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Astrocytes; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Membrane Potentials; Motor Neurons; Patch-Clamp Techniques; Posterior Horn Cells; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord

2000
AMPA receptor properties at the synapse between retinal afferents and thalamocortical cells in the dorsal lateral geniculate nucleus of the rat.
    Neuroscience letters, 2001, Volume: 316, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Geniculate Bodies; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Retinal Ganglion Cells; Synapses; Visual Cortex; Visual Pathways

2001
AMPA-induced Ca(2+) influx in cultured rat cortical nonpyramidal neurones: pharmacological characterization using fura-2 microfluorimetry.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Cerebral Cortex; Cobalt; Diazoxide; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorescence; Fluorometry; Fura-2; gamma-Aminobutyric Acid; Immunohistochemistry; N-Methylaspartate; Neurons; Piperazines; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2002
Functional characteristics of non-NMDA-type ionotropic glutamate receptor channels in AII amacrine cells in rat retina.
    The Journal of physiology, 2002, Jul-01, Volume: 542, Issue:Pt 1

    Topics: Algorithms; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Concanavalin A; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kainic Acid; Membrane Potentials; Patch-Clamp Techniques; Rats; Receptors, AMPA; Receptors, Glutamate; Retina; Sodium

2002
Involvement of post-synaptic kainate receptors during synaptic transmission between unitary connections in rat neocortex.
    The European journal of neuroscience, 2003, Volume: 17, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Dicarboxylic Acids; Drug Interactions; Electric Conductivity; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Membrane Potentials; Neocortex; Neural Pathways; Neurotransmitter Uptake Inhibitors; Patch-Clamp Techniques; Pyramidal Cells; Pyrrolidines; Rats; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission; Time Factors; Valine

2003
Simultaneous contribution of two rod pathways to AII amacrine and cone bipolar cell light responses.
    Journal of neurophysiology, 2005, Volume: 93, Issue:3

    Topics: Amacrine Cells; Animals; Benzodiazepines; Benzothiadiazines; Diagnostic Imaging; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Fluorescein; GABA Antagonists; Glycine Agents; In Vitro Techniques; Light; Male; Membrane Potentials; Models, Biological; Neurons; Patch-Clamp Techniques; Picrotoxin; Quinoxalines; Rabbits; Retina; Retinal Rod Photoreceptor Cells; Strychnine; Synapses; Synaptic Transmission; Visual Pathways

2005