Page last updated: 2024-09-03

gyki 53655 and cp 465,022

gyki 53655 has been researched along with cp 465,022 in 2 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(cp 465,022)
Trials
(cp 465,022)
Recent Studies (post-2010) (cp 465,022)
1110221105

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)cp 465,022 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.0285
Glutamate receptor 2Rattus norvegicus (Norway rat)0.0285
Glutamate receptor 3Rattus norvegicus (Norway rat)0.0285
Glutamate receptor 4Rattus norvegicus (Norway rat)0.0285

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Balannik, V; Lerma, J; Menniti, FS; Paternain, AV; Stern-Bach, Y1
Kurnikova, M; Narangoda, C; Sampson, JM; Singh, AK; Sobolevsky, AI; Yelshanskaya, MV1

Other Studies

2 other study(ies) available for gyki 53655 and cp 465,022

ArticleYear
Molecular mechanism of AMPA receptor noncompetitive antagonism.
    Neuron, 2005, Oct-20, Volume: 48, Issue:2

    Topics: Animals; Benzodiazepines; Binding Sites; Blotting, Western; Brain; Cell Line; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Humans; Membrane Potentials; Models, Neurological; Mutagenesis; Patch-Clamp Techniques; Peptide Fragments; Protein Conformation; Quinazolines; Rats; Receptors, AMPA; Transfection; Tritium; Xenopus laevis

2005
Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
    Neuron, 2016, Sep-21, Volume: 91, Issue:6

    Topics: Animals; Anticonvulsants; Benzodiazepines; Binding Sites; Crystallization; Molecular Docking Simulation; Nitriles; Pyridones; Quinazolines; Rats; Receptors, AMPA

2016