gyki 53655 has been researched along with cp 465,022 in 2 studies
Studies (gyki 53655) | Trials (gyki 53655) | Recent Studies (post-2010) (gyki 53655) | Studies (cp 465,022) | Trials (cp 465,022) | Recent Studies (post-2010) (cp 465,022) |
---|---|---|---|---|---|
111 | 0 | 22 | 11 | 0 | 5 |
Protein | Taxonomy | gyki 53655 (IC50) | cp 465,022 (IC50) |
---|---|---|---|
Glutamate receptor 1 | Rattus norvegicus (Norway rat) | 0.0285 | |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.0285 | |
Glutamate receptor 3 | Rattus norvegicus (Norway rat) | 0.0285 | |
Glutamate receptor 4 | Rattus norvegicus (Norway rat) | 0.0285 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Balannik, V; Lerma, J; Menniti, FS; Paternain, AV; Stern-Bach, Y | 1 |
Kurnikova, M; Narangoda, C; Sampson, JM; Singh, AK; Sobolevsky, AI; Yelshanskaya, MV | 1 |
2 other study(ies) available for gyki 53655 and cp 465,022
Article | Year |
---|---|
Molecular mechanism of AMPA receptor noncompetitive antagonism.
Topics: Animals; Benzodiazepines; Binding Sites; Blotting, Western; Brain; Cell Line; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Humans; Membrane Potentials; Models, Neurological; Mutagenesis; Patch-Clamp Techniques; Peptide Fragments; Protein Conformation; Quinazolines; Rats; Receptors, AMPA; Transfection; Tritium; Xenopus laevis | 2005 |
Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
Topics: Animals; Anticonvulsants; Benzodiazepines; Binding Sites; Crystallization; Molecular Docking Simulation; Nitriles; Pyridones; Quinazolines; Rats; Receptors, AMPA | 2016 |