Page last updated: 2024-09-03

gyki 53655 and alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid

gyki 53655 has been researched along with alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid in 32 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid)
Trials
(alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid)
Recent Studies (post-2010) (alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid)
1110222,89911609

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.157
Glutamate receptor 2Rattus norvegicus (Norway rat)0.1765
Glutamate receptor 3Rattus norvegicus (Norway rat)0.1765
Glutamate receptor 4Rattus norvegicus (Norway rat)0.1765
Glutamate receptor 1Mus musculus (house mouse)0.04
Glutamate receptor 2Mus musculus (house mouse)0.04
Glutamate receptor 1Homo sapiens (human)0.1353
Glutamate receptor 2Homo sapiens (human)0.1353
Glutamate receptor 3Homo sapiens (human)0.1353
Glutamate receptor 4Homo sapiens (human)0.1353
Glutamate receptor 4Mus musculus (house mouse)0.04
Glutamate receptor 3Mus musculus (house mouse)0.04

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's18 (56.25)18.2507
2000's12 (37.50)29.6817
2010's2 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
England, PM; Fleming, JJ1
Chizh, BA; Cumberbatch, MJ; Headley, PM2
Burnett, JP; Desai, MA; Ornstein, PL; Schoepp, DD1
Lodge, D; Palmer, AJ1
Parks, TN; Taylor, DA; Zhou, N1
Borsini, F; Brambilla, A; Grippa, N; Prudentino, A1
Kombian, SB; Pittman, QJ; Saleh, TM; Zidichouski, JA1
Ballyk, BA; Bath, CP; Bleakman, D; Bufton, HR; Kamboj, RK; Lodge, D; Palmer, AJ; Schoepp, DD; Sharpe, EF; Tarnawa, I; Woolley, ML1
Kovács, AD; Szabó, G1
Bleakman, D; Bristow, DR; Savidge, JR1
Barks, JD; Liu, XH; Wang, P1
Bureau, I; Mulle, C1
Lu, T; Shen, Y; Yang, XL1
Carvalho, AP; Duarte, CB; Ferreira, IL1
Dai, WM; Ebert, B; Lambert, JD; Madsen, U1
Geurtz, W; Hatt, H; Okada, T; Schultz, K; Weiler, R1
Bristow, DR; Lock, EA; Savidge, JR; Sturgess, NC1
Perkinton, MS; Sihra, TS; Williams, RJ1
Lerma, J; López-García, JC; Rodríguez-Moreno, A1
Durand, J; Ruiz, A1
Cebers, G; Kovács, AD; Liljequist, S1
Closier, M; Iop, F; Lestage, P; Lockhart, B1
Brorson, JR; Ihle, EC; Patneau, DK; Robberecht, W; Vandenberghe, W1
Baumbarger, PJ; Muhlhauser, M; Nisenbaum, ES; Yang, CR; Zhai, J1
Christensen, KV; Dai, WM; Ebert, B; Egebjerg, J; Lambert, JD1
Alberdi, E; Marino, A; Matute, C; Sánchez-Gómez, MV1
Allgaier, C; Fischer, W; Franke, H; Illes, P; Scheibler, P1
Hartveit, E; Mørkve, SH; Veruki, ML1
Arai, AC; Kessler, M1
Anderson, RL; Daniele, C; Engelman, HS; Macdermott, AB1
Kimura, H; Kunugi, A; Suzuki, A; Tajima, Y1

Other Studies

32 other study(ies) available for gyki 53655 and alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid

ArticleYear
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
AMPA receptors have an equal role in spinal nociceptive and non-nociceptive transmission.
    Neuroreport, 1994, Apr-14, Volume: 5, Issue:8

    Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Dose-Response Relationship, Drug; Iontophoresis; Male; N-Methylaspartate; Nociceptors; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Spinal Cord; Synapses; Synaptic Transmission

1994
A comparison of intravenous NBQX and GYKI 53655 as AMPA antagonists in the rat spinal cord.
    British journal of pharmacology, 1994, Volume: 112, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Hot Temperature; Injections, Intravenous; Iontophoresis; Male; N-Methylaspartate; Neurons; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Spinal Cord

1994
Cyclothiazide acts at a site on the alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid receptor complex that does not recognize competitive or noncompetitive AMPA receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Hippocampus; In Vitro Techniques; Isoquinolines; Kainic Acid; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetrazoles

1995
Cyclothiazide reverses AMPA receptor antagonism of the 2,3-benzodiazepine, GYKI 53655.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cerebral Cortex; Diuretics; Excitatory Amino Acid Antagonists; Ibotenic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1993
Cobalt-permeable non-NMDA receptors in developing chick brainstem auditory nuclei.
    Neuroreport, 1995, Nov-27, Volume: 6, Issue:17

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Auditory Pathways; Benzodiazepines; Brain Stem; Cell Membrane Permeability; Chick Embryo; Cobalt; Evoked Potentials, Auditory, Brain Stem; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Neurons; Receptors, N-Methyl-D-Aspartate

1995
Pharmacological characterization of AMPA-induced biting behaviour in mice.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Behavior, Animal; Benzodiazepines; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Hyperalgesia; Injections, Spinal; Male; Mice; Mice, Inbred Strains; Nociceptors; Quinoxalines; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

1996
Cholecystokinin and neurotensin inversely modulate excitatory synaptic transmission in the parabrachial nucleus in vitro.
    Neuroscience, 1997, Volume: 77, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cholecystokinin; Devazepide; Electric Conductivity; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hormone Antagonists; Interneurons; N-Methylaspartate; Neural Inhibition; Neurons, Afferent; Neurotensin; Patch-Clamp Techniques; Phenylurea Compounds; Pons; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin

1997
Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: stereospecificity and selectivity profiles.
    Neuropharmacology, 1996, Volume: 35, Issue:12

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Cerebellum; Cerebral Cortex; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Humans; Kidney; Membrane Potentials; Molecular Structure; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Spinal Cord; Structure-Activity Relationship; Transfection

1996
GYKI 53665, a 2,3-benzodiazepine, non-competitively protects cultured neurones against AMPA toxicity.
    European journal of pharmacology, 1997, Jul-16, Volume: 331, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Brain; Cells, Cultured; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Neuroprotective Agents; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA

1997
Identification of kainate receptor-mediated intracellular calcium increases in cultured rat cerebellar granule cells.
    Journal of neurochemistry, 1997, Volume: 69, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Calcium; Cells, Cultured; Cerebellum; Concanavalin A; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Intracellular Membranes; Isoquinolines; Kainic Acid; Neurons; Rats; Receptors, Kainic Acid; Tetrazoles

1997
The non-competitive AMPA antagonist LY 300168 (GYKI 53655) attenuates AMPA-induced hippocampal injury in neonatal rodents.
    Neuroscience letters, 1997, Oct-10, Volume: 235, Issue:1-2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analysis of Variance; Animals; Animals, Newborn; Atrophy; Benzodiazepines; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Hippocampus; Injections, Intraperitoneal; N-Methylaspartate; Pyramidal Cells; Rats; Rats, Sprague-Dawley

1997
Potentiation of GABAergic synaptic transmission by AMPA receptors in mouse cerebellar stellate cells: changes during development.
    The Journal of physiology, 1998, Jun-15, Volume: 509 ( Pt 3)

    Topics: Age Factors; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Cadmium; Cerebellum; Dose-Response Relationship, Drug; Evoked Potentials; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Kainic Acid; Mice; Neural Inhibition; Neuromuscular Depolarizing Agents; Neurons; Receptors, AMPA; Receptors, Kainic Acid; Synaptic Transmission; Tetrodotoxin

1998
Desensitization of AMPA receptors on horizontal cells isolated from crucian carp retina.
    Neuroscience research, 1998, Volume: 31, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Cells, Cultured; Drug Tolerance; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Kainic Acid; Patch-Clamp Techniques; Receptors, AMPA; Retina

1998
Kainate-induced retina amacrine-like cell damage is mediated by AMPA receptors.
    Neuroreport, 1998, Oct-26, Volume: 9, Issue:15

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium Radioisotopes; Cells, Cultured; Chickens; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Neuromuscular Depolarizing Agents; Receptors, AMPA; Receptors, Kainic Acid; Retina

1998
Studies of the antagonist actions of (RS)-2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl] propionic acid (ATPO) on non-NMDA receptors in cultured rat neurones.
    British journal of pharmacology, 1998, Volume: 125, Issue:7

    Topics: Adrenal Cortex Hormones; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Cells, Cultured; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamates; Isoxazoles; Kainic Acid; Neurons; Organophosphonates; Rats; Rats, Sprague-Dawley; Receptors, AMPA

1998
AMPA-preferring receptors with high Ca2+ permeability mediate dendritic plasticity of retinal horizontal cells.
    The European journal of neuroscience, 1999, Volume: 11, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carps; Dark Adaptation; Dendrites; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Membrane Potentials; Microscopy, Electron; Neuronal Plasticity; Patch-Clamp Techniques; Receptors, AMPA; Receptors, Kainic Acid; Retina

1999
Characterisation of kainate receptor mediated whole-cell currents in rat cultured cerebellar granule cells.
    Neuropharmacology, 1999, Volume: 38, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Concanavalin A; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamates; Hippocampus; Kinetics; Neurons; Neurotoxins; Patch-Clamp Techniques; Rats; Receptors, Kainic Acid; Spider Venoms

1999
Ca(2+)-permeable AMPA receptors induce phosphorylation of cAMP response element-binding protein through a phosphatidylinositol 3-kinase-dependent stimulation of the mitogen-activated protein kinase signaling cascade in neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-15, Volume: 19, Issue:14

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Androstadienes; Animals; Arachidonic Acid; Benzodiazepines; Benzothiadiazines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Membrane Permeability; Cell Survival; Cells, Cultured; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Flavonoids; Genistein; GTP-Binding Proteins; Kinetics; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neurons; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphorylation; Receptors, AMPA; Signal Transduction; Virulence Factors, Bordetella; Wortmannin

1999
Two populations of kainate receptors with separate signaling mechanisms in hippocampal interneurons.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Feb-01, Volume: 97, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Bicuculline; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Indoles; Interneurons; Isoxazoles; Kainic Acid; Lidocaine; Maleimides; Naphthalenes; Nerve Tissue Proteins; Patch-Clamp Techniques; Propionates; Protein Kinase C; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Kainic Acid; Receptors, Presynaptic; Signal Transduction; Staurosporine; Virulence Factors, Bordetella

2000
Blocking the trigeminal EPSP in rat abducens motoneurons in vivo with the AMPA antagonists NBQX and GYKI 53655.
    Brain research bulletin, 2000, May-15, Volume: 52, Issue:2

    Topics: Abducens Nerve; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Male; Motor Neurons; N-Methylaspartate; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Trigeminal Nerve

2000
Kainate receptor-mediated activation of the AP-1 transcription factor complex in cultured rat cerebellar granule cells.
    Brain research bulletin, 2000, May-15, Volume: 52, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Cerebellum; Concanavalin A; Dimerization; Excitatory Amino Acid Antagonists; Isoquinolines; Kainic Acid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Tetrazoles; Transcription Factor AP-1

2000
(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide: (S18986-1) a positive modulator of AMPA receptors enhances (S)-AMPA-mediated [3H]noradrenaline release from rat hippocampal and frontal cortex slices.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Frontal Lobe; Hippocampus; In Vitro Techniques; Male; Norepinephrine; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Stereoisomerism; Tetrodotoxin; Tritium

2000
AMPA receptor current density, not desensitization, predicts selective motoneuron vulnerability.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Oct-01, Volume: 20, Issue:19

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Astrocytes; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Membrane Potentials; Motor Neurons; Patch-Clamp Techniques; Posterior Horn Cells; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord

2000
Positive modulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid (AMPA) receptors in prefrontal cortical pyramidal neurons by a novel allosteric potentiator.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:1

    Topics: Allosteric Regulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Dioxoles; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Sulfonamides

2001
Correlation of the expression of kainate receptor subtypes to responses evoked in cultured cortical and spinal cord neurones.
    Brain research, 2002, Feb-01, Volume: 926, Issue:1-2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Concanavalin A; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression; Kainic Acid; Membrane Potentials; Neurons; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord

2002
Ca(2+) influx through AMPA or kainate receptors alone is sufficient to initiate excitotoxicity in cultured oligodendrocytes.
    Neurobiology of disease, 2002, Volume: 9, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Calcium; Calcium Channel Blockers; Cell Death; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Lanthanum; Neurotoxins; Nifedipine; Oligodendroglia; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid

2002
AMPA-induced Ca(2+) influx in cultured rat cortical nonpyramidal neurones: pharmacological characterization using fura-2 microfluorimetry.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Cerebral Cortex; Cobalt; Diazoxide; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorescence; Fluorometry; Fura-2; gamma-Aminobutyric Acid; Immunohistochemistry; N-Methylaspartate; Neurons; Piperazines; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2002
Functional characteristics of non-NMDA-type ionotropic glutamate receptor channels in AII amacrine cells in rat retina.
    The Journal of physiology, 2002, Jul-01, Volume: 542, Issue:Pt 1

    Topics: Algorithms; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Concanavalin A; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kainic Acid; Membrane Potentials; Patch-Clamp Techniques; Rats; Receptors, AMPA; Receptors, Glutamate; Retina; Sodium

2002
Use of [3H]fluorowillardiine to study properties of AMPA receptor allosteric modulators.
    Brain research, 2006, Mar-03, Volume: 1076, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alanine; Allosteric Site; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Membranes; Peptides, Cyclic; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tritium

2006
Presynaptic alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptors modulate release of inhibitory amino acids in rat spinal cord dorsal horn.
    Neuroscience, 2006, May-12, Volume: 139, Issue:2

    Topics: Age Factors; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Newborn; Benzodiazepines; Cadmium Chloride; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Kainic Acid; Neural Inhibition; Patch-Clamp Techniques; Posterior Horn Cells; Rats; Receptors, AMPA; Receptors, Presynaptic; Spinal Cord

2006
Electrophysiological characterization of a novel AMPA receptor potentiator, TAK-137, in rat hippocampal neurons.
    Neuroscience letters, 2019, 11-01, Volume: 712

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Evoked Potentials; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Male; Neurons; Patch-Clamp Techniques; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Thiadiazines

2019