Page last updated: 2024-09-03

gyki 53655 and 6-cyano-7-nitroquinoxaline-2,3-dione

gyki 53655 has been researched along with 6-cyano-7-nitroquinoxaline-2,3-dione in 18 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(6-cyano-7-nitroquinoxaline-2,3-dione)
Trials
(6-cyano-7-nitroquinoxaline-2,3-dione)
Recent Studies (post-2010) (6-cyano-7-nitroquinoxaline-2,3-dione)
1110222,6981353

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)6-cyano-7-nitroquinoxaline-2,3-dione (IC50)
Glutamate receptor 1Homo sapiens (human)1.02
Glutamate receptor 2Homo sapiens (human)1.02
Glutamate receptor 3Homo sapiens (human)1.02
Glutamate receptor 4Homo sapiens (human)1.02

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (33.33)18.2507
2000's9 (50.00)29.6817
2010's3 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Parks, TN; Taylor, DA; Zhou, N1
Kombian, SB; Pittman, QJ; Saleh, TM; Zidichouski, JA1
Castillo, PE; Malenka, RC; Nicoll, RA1
Freund-Mercier, MJ; Jo, YH; Schlichter, R; Stoeckel, ME1
Ben-Ari, Y; Dzhala, V; Khalilov, I; Khazipov, R; Lamsa, K; Leinekugel, X; Medina, I; Melyan, Z1
Ben-Ari, Y; Chevassus-Au-Louis, N; Diabira, D; Gozlan, H; Hennou, S1
Alberdi, E; Marino, A; Matute, C; Sánchez-Gómez, MV1
Allgaier, C; Fischer, W; Franke, H; Illes, P; Scheibler, P1
Hartveit, E; Mørkve, SH; Veruki, ML1
Ali, AB1
Breustedt, J; Schmitz, D1
Ko, SW; Toyoda, H; Wu, LJ; Zhao, MG; Zhuo, M1
Arai, AC; Kessler, M1
Ibarretxe, G; Jaskolski, F; Mulle, C; Perrais, D; Vimeney, A1
Hays, FA; Menuz, K; Nicoll, RA; Stroud, RM1
Eggers, ED; Lukasiewicz, PD; Purgert, R; Sagdullaev, BT1
Babai, N; Feigenspan, A1
Ballanyi, K; Rancic, V; Rawal, B1

Other Studies

18 other study(ies) available for gyki 53655 and 6-cyano-7-nitroquinoxaline-2,3-dione

ArticleYear
Cobalt-permeable non-NMDA receptors in developing chick brainstem auditory nuclei.
    Neuroreport, 1995, Nov-27, Volume: 6, Issue:17

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Auditory Pathways; Benzodiazepines; Brain Stem; Cell Membrane Permeability; Chick Embryo; Cobalt; Evoked Potentials, Auditory, Brain Stem; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Neurons; Receptors, N-Methyl-D-Aspartate

1995
Cholecystokinin and neurotensin inversely modulate excitatory synaptic transmission in the parabrachial nucleus in vitro.
    Neuroscience, 1997, Volume: 77, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cholecystokinin; Devazepide; Electric Conductivity; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hormone Antagonists; Interneurons; N-Methylaspartate; Neural Inhibition; Neurons, Afferent; Neurotensin; Patch-Clamp Techniques; Phenylurea Compounds; Pons; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin

1997
Kainate receptors mediate a slow postsynaptic current in hippocampal CA3 neurons.
    Nature, 1997, Jul-10, Volume: 388, Issue:6638

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamic Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Kainic Acid; Nerve Fibers; Neurons; Receptors, AMPA; Receptors, Kainic Acid; Synapses

1997
Oxytocin modulates glutamatergic synaptic transmission between cultured neonatal spinal cord dorsal horn neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Apr-01, Volume: 18, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Electric Stimulation; Enkephalin, Methionine; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamate Decarboxylase; Glutamic Acid; Immunohistochemistry; Neurons; Nociceptors; Oxytocin; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Spinal Cord; Synaptic Transmission; Tetrodotoxin

1998
Maturation of kainate-induced epileptiform activities in interconnected intact neonatal limbic structures in vitro.
    The European journal of neuroscience, 1999, Volume: 11, Issue:10

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Electrophysiology; Entorhinal Cortex; Epilepsy; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Limbic System; Male; Organ Culture Techniques; Potassium; Rats; Rats, Wistar; Septal Nuclei; Synapses; Tetrodotoxin

1999
Late embryonic expression of AMPA receptor function in the CA1 region of the intact hippocampus in vitro.
    The European journal of neuroscience, 1999, Volume: 11, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Afferent Pathways; Aging; Animals; Animals, Newborn; Benzodiazepines; Bicuculline; Cations, Divalent; Electric Stimulation; Embryonic and Fetal Development; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; Hippocampus; Hypoxia; Lysine; Pyramidal Cells; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Synapses; Tetrodotoxin

1999
Ca(2+) influx through AMPA or kainate receptors alone is sufficient to initiate excitotoxicity in cultured oligodendrocytes.
    Neurobiology of disease, 2002, Volume: 9, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Calcium; Calcium Channel Blockers; Cell Death; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Kainic Acid; Lanthanum; Neurotoxins; Nifedipine; Oligodendroglia; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid

2002
AMPA-induced Ca(2+) influx in cultured rat cortical nonpyramidal neurones: pharmacological characterization using fura-2 microfluorimetry.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Cerebral Cortex; Cobalt; Diazoxide; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorescence; Fluorometry; Fura-2; gamma-Aminobutyric Acid; Immunohistochemistry; N-Methylaspartate; Neurons; Piperazines; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2002
Functional properties of spontaneous EPSCs and non-NMDA receptors in rod amacrine (AII) cells in the rat retina.
    The Journal of physiology, 2003, Jun-15, Volume: 549, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Algorithms; Amacrine Cells; Animals; Benzodiazepines; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; In Vitro Techniques; Kinetics; Membrane Potentials; Patch-Clamp Techniques; Piperazines; Presynaptic Terminals; Rats; Receptors, AMPA; Receptors, Glutamate; Retinal Rod Photoreceptor Cells; Synapses; Tetrodotoxin

2003
Involvement of post-synaptic kainate receptors during synaptic transmission between unitary connections in rat neocortex.
    The European journal of neuroscience, 2003, Volume: 17, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Dicarboxylic Acids; Drug Interactions; Electric Conductivity; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Membrane Potentials; Neocortex; Neural Pathways; Neurotransmitter Uptake Inhibitors; Patch-Clamp Techniques; Pyramidal Cells; Pyrrolidines; Rats; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission; Time Factors; Valine

2003
Assessing the role of GLUK5 and GLUK6 at hippocampal mossy fiber synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Nov-10, Volume: 24, Issue:45

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids, Dicarboxylic; Animals; Benzodiazepines; Cyclopropanes; Excitatory Postsynaptic Potentials; Gene Deletion; GluK2 Kainate Receptor; Glycine; Isoquinolines; Isoxazoles; Kainic Acid; Mice; Mice, Knockout; Mossy Fibers, Hippocampal; Neuronal Plasticity; Patch-Clamp Techniques; Potassium; Propionates; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission

2004
Kainate receptor-mediated synaptic transmission in the adult anterior cingulate cortex.
    Journal of neurophysiology, 2005, Volume: 94, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GluK2 Kainate Receptor; Gyrus Cinguli; In Vitro Techniques; Isoxazoles; Kainic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Patch-Clamp Techniques; Propionates; Receptors, Kainic Acid; Synaptic Transmission

2005
Use of [3H]fluorowillardiine to study properties of AMPA receptor allosteric modulators.
    Brain research, 2006, Mar-03, Volume: 1076, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alanine; Allosteric Site; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Membranes; Peptides, Cyclic; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tritium

2006
Fast regulation of axonal growth cone motility by electrical activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Jul-18, Volume: 27, Issue:29

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Animals, Newborn; Axons; Benzodiazepines; Calcium; Cell Movement; Cells, Cultured; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Growth Cones; Hippocampus; Kainic Acid; Mice; Mice, Knockout; Neurons; Receptors, Glutamate; Tetrodotoxin

2007
TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists.
    Science (New York, N.Y.), 2007, Nov-02, Volume: 318, Issue:5851

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Binding, Competitive; Cell Line; Cerebellum; Crystallography, X-Ray; Drug Partial Agonism; Hippocampus; Humans; In Vitro Techniques; Interneurons; Mice; Models, Molecular; Patch-Clamp Techniques; Protein Conformation; Protein Subunits; Pyramidal Cells; Quinoxalines; Receptors, AMPA; Structure-Activity Relationship; Synaptic Transmission; Trichlormethiazide

2007
Nonlinear interactions between excitatory and inhibitory retinal synapses control visual output.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Oct-19, Volume: 31, Issue:42

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Mice; Neural Inhibition; Nonlinear Dynamics; Patch-Clamp Techniques; Phosphinic Acids; Photic Stimulation; Presynaptic Terminals; Pyridines; Retina; Retinal Bipolar Cells; Retinal Ganglion Cells; Synapses; Synaptic Transmission

2011
Functional properties of spontaneous excitatory currents and encoding of light/dark transitions in horizontal cells of the mouse retina.
    The European journal of neuroscience, 2015, Volume: 42, Issue:9

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Dendrites; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; Glutamic Acid; Mice; Mice, Transgenic; Neural Pathways; Photic Stimulation; Receptors, AMPA; Receptors, Kainic Acid; Retinal Cone Photoreceptor Cells; Retinal Horizontal Cells

2015
TARP mediation of accelerated and more regular locus coeruleus network bursting in neonatal rat brain slices.
    Neuropharmacology, 2019, Volume: 148

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Benzodiazepines; Calcium; Kynurenic Acid; Locus Coeruleus; Membrane Potentials; Neurons; Rats; Receptors, AMPA; Tetrodotoxin

2019