Page last updated: 2024-09-03

gyki 53655 and 2-amino-5-phosphonovalerate

gyki 53655 has been researched along with 2-amino-5-phosphonovalerate in 12 studies

Compound Research Comparison

Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010)
(gyki 53655)
Studies
(2-amino-5-phosphonovalerate)
Trials
(2-amino-5-phosphonovalerate)
Recent Studies (post-2010) (2-amino-5-phosphonovalerate)
1110224,3931539

Protein Interaction Comparison

ProteinTaxonomygyki 53655 (IC50)2-amino-5-phosphonovalerate (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.29

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (33.33)18.2507
2000's6 (50.00)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Banczerowski-Pelyhe, I; Csúcs, G; Tarnawa, I; Világi, I1
Collingridge, GL; Vignes, M1
Banczerowski-Pelyhe, I; Kocsis, P; Tarnawa, I; Világi, I1
Ben-Ari, Y; Chevassus-Au-Louis, N; Diabira, D; Gozlan, H; Hennou, S1
Lerma, J; López-García, JC; Rodríguez-Moreno, A1
Bleakman, D; Bortolotto, ZA; Collingridge, GL; Isaac, JT; Lauri, SE; Lodge, D; Ornstein, PL1
Heggelund, P; Kielland, A1
Ali, AB1
Clarke, VR; Collingridge, GL1
Breustedt, J; Schmitz, D1
Chen, T; Kaang, BK; Koga, K; Sim, SE; Wu, LJ; Zhuo, M1
Jiang, L; Kang, D; Kang, J1

Other Studies

12 other study(ies) available for gyki 53655 and 2-amino-5-phosphonovalerate

ArticleYear
An increased intensity of N-methyl-D-aspartate (NMDA) but not non-NMDA receptor activation may be responsible for the enhancement of excitatory processes in the neocortex of two-week-old rats: a brain slices study.
    Neuroscience letters, 1996, Jan-19, Volume: 203, Issue:2

    Topics: Action Potentials; Animals; Animals, Suckling; Benzodiazepines; Binding, Competitive; Cerebral Cortex; Electric Stimulation; Excitatory Amino Acid Antagonists; Organophosphonates; Pentanoic Acids; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Somatosensory Cortex; Synaptic Transmission; Valine

1996
The synaptic activation of kainate receptors.
    Nature, 1997, Jul-10, Volume: 388, Issue:6638

    Topics: 2-Amino-5-phosphonovalerate; Aminoquinolines; Animals; Benzodiazepines; Bicuculline; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; Hippocampus; In Vitro Techniques; Picrotoxin; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Synapses

1997
Effect of glutamate receptor antagonists on excitatory postsynaptic potentials in striatum.
    Brain research bulletin, 1998, Volume: 46, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Benzodiazepines; Corpus Striatum; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Male; Organ Culture Techniques; Rats; Rats, Inbred Strains; Receptors, Glutamate

1998
Late embryonic expression of AMPA receptor function in the CA1 region of the intact hippocampus in vitro.
    The European journal of neuroscience, 1999, Volume: 11, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Afferent Pathways; Aging; Animals; Animals, Newborn; Benzodiazepines; Bicuculline; Cations, Divalent; Electric Stimulation; Embryonic and Fetal Development; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; Hippocampus; Hypoxia; Lysine; Pyramidal Cells; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Synapses; Tetrodotoxin

1999
Two populations of kainate receptors with separate signaling mechanisms in hippocampal interneurons.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Feb-01, Volume: 97, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Bicuculline; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Indoles; Interneurons; Isoxazoles; Kainic Acid; Lidocaine; Maleimides; Naphthalenes; Nerve Tissue Proteins; Patch-Clamp Techniques; Propionates; Protein Kinase C; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Kainic Acid; Receptors, Presynaptic; Signal Transduction; Staurosporine; Virulence Factors, Bordetella

2000
A critical role of a facilitatory presynaptic kainate receptor in mossy fiber LTP.
    Neuron, 2001, Nov-20, Volume: 32, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Benzodiazepines; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Isoquinolines; Long-Term Potentiation; Mossy Fibers, Hippocampal; Rats; Receptors, Kainic Acid; Receptors, Presynaptic; Synapses; Synaptic Transmission

2001
AMPA receptor properties at the synapse between retinal afferents and thalamocortical cells in the dorsal lateral geniculate nucleus of the rat.
    Neuroscience letters, 2001, Volume: 316, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Geniculate Bodies; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA; Retinal Ganglion Cells; Synapses; Visual Cortex; Visual Pathways

2001
Involvement of post-synaptic kainate receptors during synaptic transmission between unitary connections in rat neocortex.
    The European journal of neuroscience, 2003, Volume: 17, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Dicarboxylic Acids; Drug Interactions; Electric Conductivity; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Membrane Potentials; Neocortex; Neural Pathways; Neurotransmitter Uptake Inhibitors; Patch-Clamp Techniques; Pyramidal Cells; Pyrrolidines; Rats; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission; Time Factors; Valine

2003
Characterisation of the effects of ATPA, a GLU(K5) kainate receptor agonist, on GABAergic synaptic transmission in the CA1 region of rat hippocampal slices.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: Animals; Benzodiazepines; Dose-Response Relationship, Drug; Drug Interactions; Electric Impedance; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agents; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Isoxazoles; Kainic Acid; Membrane Potentials; Neural Inhibition; Propionates; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission; Valine

2004
Assessing the role of GLUK5 and GLUK6 at hippocampal mossy fiber synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Nov-10, Volume: 24, Issue:45

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids, Dicarboxylic; Animals; Benzodiazepines; Cyclopropanes; Excitatory Postsynaptic Potentials; Gene Deletion; GluK2 Kainate Receptor; Glycine; Isoquinolines; Isoxazoles; Kainic Acid; Mice; Mice, Knockout; Mossy Fibers, Hippocampal; Neuronal Plasticity; Patch-Clamp Techniques; Potassium; Propionates; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Kainic Acid; Synaptic Transmission

2004
Kainate receptor-mediated synaptic transmissions in the adult rodent insular cortex.
    Journal of neurophysiology, 2012, Volume: 108, Issue:7

    Topics: 2-Amino-5-phosphonovalerate; Alanine; Animals; Benzodiazepines; Cerebral Cortex; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; GluK2 Kainate Receptor; Mice; Mice, Inbred C57BL; Mice, Knockout; Picrotoxin; Pyramidal Cells; Receptors, Kainic Acid; Synaptic Transmission; Thymine

2012
Potentiation of tonic GABAergic inhibition by activation of postsynaptic kainate receptors.
    Neuroscience, 2015, Jul-09, Volume: 298

    Topics: Action Potentials; Animals; Animals, Newborn; Benzodiazepines; Biophysics; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agents; GABAergic Neurons; Hippocampus; Humans; In Vitro Techniques; Kainic Acid; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Tetrodotoxin; Valine

2015