Compounds > gyki 52466

gyki 52466 and ly 303070

gyki 52466 has been researched along with ly 303070 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cagnotto, A; Colleoni, S; Diana, V; Grasso, S; Lazzaro, J; Mennini, T; Micale, N; Pellicanò, A; Postorino, G; Zappalà, M1
Csillik-Perczel, V; Harsing, LG; Ling, I; Sólyom, S1
Niu, L; Sheng, Z; Wang, C1
Niu, L; Wang, C; Wu, A1

Other Studies

4 other study(ies) available for gyki 52466 and ly 303070

ArticleYear
Structure-activity study of 2,3-benzodiazepin-4-ones noncompetitive AMPAR antagonists: identification of the 1-(4-amino-3-methylphenyl)-3,5-dihydro-7,8-ethylenedioxy-4H-2,3-benzodiazepin-4-one as neuroprotective agent.
    Bioorganic & medicinal chemistry, 2008, Mar-01, Volume: 16, Issue:5

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Calcium; Cells, Cultured; Hippocampus; Inhibitory Concentration 50; Kainic Acid; Ligands; Mice; Molecular Structure; Neurons; Neuroprotective Agents; Protein Binding; Receptors, AMPA; Structure-Activity Relationship

2008
Negative allosteric modulators of AMPA-preferring receptors inhibit [(3)H]GABA release in rat striatum.
    Neurochemistry international, 2000, Volume: 37, Issue:1

    Topics: Allosteric Site; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Corpus Striatum; Drug Synergism; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Receptors, AMPA

2000
Mechanism of inhibition of the GluA2 AMPA receptor channel opening: consequences of adding an N-3 methylcarbamoyl group to the diazepine ring of 2,3-benzodiazepine derivatives.
    Biochemistry, 2011, Aug-23, Volume: 50, Issue:33

    Topics: Benzodiazepines; Cells, Cultured; Humans; Ion Channel Gating; Kidney; Kinetics; Lasers; Photolysis; Protein Binding; Receptors, AMPA; Structure-Activity Relationship

2011
Mechanism of inhibition of the GluA1 AMPA receptor channel opening by the 2,3-benzodiazepine compound GYKI 52466 and a N-methyl-carbamoyl derivative.
    Biochemistry, 2014, May-13, Volume: 53, Issue:18

    Topics: Animals; Benzodiazepines; HEK293 Cells; Humans; Ion Channel Gating; Rats; Receptors, AMPA

2014