gyki 52466 has been researched along with cyclothiazide in 31 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 19 (61.29) | 18.2507 |
2000's | 11 (35.48) | 29.6817 |
2010's | 1 (3.23) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chaudhary, A; Johansen, TH; Verdoorn, TA | 1 |
Burnett, JP; May, PC; Mayne, NG; Sharp, RL; Snyder, YM | 1 |
Fattman, CL; Hoyt, KR; Rajdev, S; Reynolds, IJ | 1 |
Balázs, R; Hack, N | 1 |
Camici, O; Corazzi, L; Fallarino, F; Fioretti, MC; Genazzani, AA; L'Episcopo, MR; Nicoletti, F; Silla, S | 1 |
Huettner, JE; Wilding, TJ | 1 |
Mennerick, S; Zorumski, CF | 1 |
Burnett, JP; Mayne, NG; Sharp, RL | 1 |
Müller, W; Parsons, C; Rammes, G; Swandulla, D | 1 |
Olney, JW; Price, MT; Yamada, KA; Zorumski, CF | 1 |
Arai, A; Kessler, M; Lynch, G; Quan, A | 1 |
Turetsky, DM; Yamada, KA | 1 |
Collingridge, GL; Hartmann, S; Parsons, CG; Rammes, G; Swandulla, D | 1 |
Ballyk, BA; Bath, CP; Bleakman, D; Bufton, HR; Kamboj, RK; Lodge, D; Palmer, AJ; Schoepp, DD; Sharpe, EF; Tarnawa, I; Woolley, ML | 1 |
Croucher, MJ; Patel, DR | 1 |
Fontana, G; Gemignani, A; Marchese, S; Raiteri, M | 1 |
Gao, F; Maguire, G; Maple, B; Wu, SM; Yang, JH | 1 |
Donevan, SD; Rogawski, MA | 1 |
Beart, PM; Cheung, NS; Giardina, SF; John, CA; Pascoe, CJ | 1 |
Kohda, K; Wang, Y; Yuzaki, M | 1 |
Csillik-Perczel, V; Harsing, LG; Ling, I; Sólyom, S | 1 |
Durkin, JP; Gendron, TF; MacLean, S; Mealing, G; Morley, P; Small, DL; Tremblay, R | 1 |
Arai, AC; Kessler, M; Lynch, G; Rogers, G | 1 |
Croucher, MJ; Patel, DR; Young, AM | 1 |
Scriabine, A | 1 |
Frye, GD; Hsiao, SH | 1 |
Bennett, SA; Cheung, EC; Cregan, SP; Ferguson, KL; McIntosh, WC; Melanson-Drapeau, L; Park, DS; Slack, RS; Vanderluit, JL | 1 |
Arai, AC; Kessler, M; Suzuki, E | 1 |
Cadetti, L; Thoreson, WB; Tranchina, D | 1 |
Kardos, J; Lasztóczi, B | 1 |
Barygin, OI | 1 |
31 other study(ies) available for gyki 52466 and cyclothiazide
Article | Year |
---|---|
Interactions among GYKI-52466, cyclothiazide, and aniracetam at recombinant AMPA and kainate receptors.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Humans; Pyrrolidinones; Receptors, AMPA; Receptors, Kainic Acid; Recombinant Proteins; Xenopus laevis | 1995 |
Cyclothiazide potentiates agonist responses at human AMPA/kainate receptors expressed in oocytes.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cloning, Molecular; Humans; Kainic Acid; Oocytes; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Xenopus laevis | 1994 |
Cyclothiazide modulates AMPA receptor-mediated increases in intracellular free Ca2+ and Mg2+ in cultured neurons from rat brain.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Drug Synergism; Glutamic Acid; Kainic Acid; Magnesium; Neurons; Prosencephalon; Rats; Receptors, AMPA | 1995 |
Properties of AMPA receptors expressed in rat cerebellar granule cell cultures: Ca2+ influx studies.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Calcium Radioisotopes; Cell Survival; Cells, Cultured; Cerebellum; Cobalt; Concanavalin A; Excitatory Amino Acids; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Wheat Germ Agglutinins | 1995 |
[3H]aniracetam binds to specific recognition sites in brain membranes.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Brain; Cells, Cultured; Cerebellum; Glutamic Acid; Male; Membranes; Phorbol 12,13-Dibutyrate; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tritium | 1995 |
Differential antagonism of alpha-amino-3-hydroxy-5-methyl-4- isoxazolepropionic acid-preferring and kainate-preferring receptors by 2,3-benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding, Competitive; Cerebral Cortex; Concanavalin A; Electrophysiology; Ganglia, Spinal; Kainic Acid; Membrane Potentials; Neurons; Rats; Rats, Inbred Strains; Receptors, AMPA; Receptors, Kainic Acid; Substrate Specificity | 1995 |
Presynaptic influence on the time course of fast excitatory synaptic currents in cultured hippocampal cells.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Kinetics; Magnesium; Neurons; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Time Factors | 1995 |
Cyclothiazide differentially modulates human metabotropic glutamate receptors linked to phosphoinositide hydrolysis stimulation in oocytes.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Diuretics; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Antagonists; Humans; Hydrolysis; Oocytes; Phosphatidylinositols; Receptors, Metabotropic Glutamate; Sodium Chloride Symporter Inhibitors; Xenopus laevis | 1994 |
Modulation of fast excitatory synaptic transmission by cyclothiazide and GYKI 52466 in the rat hippocampus.
Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Organophosphorus Compounds; Picrotoxin; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission | 1994 |
A benzodiazepine recognition site associated with the non-NMDA glutamate receptor.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Binding, Competitive; Cells, Cultured; Chick Embryo; Electric Conductivity; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Nerve Degeneration; Neurons; Quisqualic Acid; Rats; Receptors, Glutamate; Retina | 1993 |
Effect of cyclothiazide on binding properties of AMPA-type glutamate receptors: lack of competition between cyclothiazide and GYKI 52466.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Binding, Competitive; Excitatory Amino Acid Antagonists; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tritium | 1996 |
Allosteric interactions between cyclothiazide and AMPA/kainate receptor antagonists.
Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Drug Interactions; Electrophysiology; Excitatory Amino Acid Antagonists; Hippocampus; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid | 1996 |
Interactions of 2,3-benzodiazepines and cyclothiazide at AMPA receptors: patch clamp recordings in cultured neurones and area CA1 in hippocampal slices.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Dose-Response Relationship, Drug; Hippocampus; In Vitro Techniques; Patch-Clamp Techniques; Rats; Receptors, AMPA; Superior Colliculi | 1996 |
Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: stereospecificity and selectivity profiles.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Cerebellum; Cerebral Cortex; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Humans; Kidney; Membrane Potentials; Molecular Structure; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Spinal Cord; Structure-Activity Relationship; Transfection | 1996 |
Evidence for a role of presynaptic AMPA receptors in the control of neuronal glutamate release in the rat forebrain.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Aspartic Acid; Benzodiazepines; Benzothiadiazines; Binding, Competitive; Calcium; Electric Stimulation; Excitatory Amino Acid Antagonists; Glutamic Acid; Male; Neurons; Presynaptic Terminals; Prosencephalon; Rats; Rats, Wistar; Receptors, AMPA; Tetrodotoxin | 1997 |
Neuropeptide Y release from cultured hippocampal neurons: stimulation by glutamate acting at N-methyl-D-aspartate and AMPA receptors.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antibody Specificity; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Chromatography, High Pressure Liquid; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Kainic Acid; Magnesium; Neurons; Neuropeptide Y; Quinoxalines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tetrodotoxin | 1997 |
Postsynaptic responses of horizontal cells in the tiger salamander retina are mediated by AMPA-preferring receptors.
Topics: Ambystoma; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Concanavalin A; Dark Adaptation; Electrophysiology; Excitatory Amino Acid Antagonists; Fluorescent Dyes; Glutamic Acid; Isoquinolines; Membrane Potentials; Patch-Clamp Techniques; Photic Stimulation; Photoreceptor Cells; Receptors, AMPA; Synapses | 1998 |
Allosteric regulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionate receptors by thiocyanate and cyclothiazide at a common modulatory site distinct from that of 2,3-benzodiazepines.
Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Ion Channel Gating; Kainic Acid; Membrane Potentials; N-Methylaspartate; Neurons; Oocytes; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Thiocyanates; Xenopus | 1998 |
Cyclothiazide and GYKI 52466 modulate AMPA receptor-mediated apoptosis in cortical neuronal cultures.
Topics: Animals; Anti-Anxiety Agents; Apoptosis; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Glutamic Acid; Mice; Neocortex; Neurons; Neuroprotective Agents; Receptors, AMPA | 1999 |
Mutation of a glutamate receptor motif reveals its role in gating and delta2 receptor channel properties.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Conserved Sequence; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Humans; Ion Channel Gating; Kainic Acid; Kidney; Mice; Mice, Neurologic Mutants; Molecular Sequence Data; Mutagenesis; Neuromuscular Depolarizing Agents; Patch-Clamp Techniques; Purkinje Cells; Quinoxalines; Receptors, Glutamate; Transfection | 2000 |
Negative allosteric modulators of AMPA-preferring receptors inhibit [(3)H]GABA release in rat striatum.
Topics: Allosteric Site; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Corpus Striatum; Drug Synergism; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Receptors, AMPA | 2000 |
Pharmacological and molecular characterization of glutamate receptors in the MIN6 pancreatic beta-cell line.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Biological Transport; Calcium; Cell Survival; DNA Primers; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Islets of Langerhans; Kainic Acid; Protein Kinase C; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spider Venoms; Tumor Cells, Cultured | 2000 |
Effects of the potent ampakine CX614 on hippocampal and recombinant AMPA receptors: interactions with cyclothiazide and GYKI 52466.
Topics: Alanine; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cells, Cultured; Diuretics; Drug Interactions; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; Humans; In Vitro Techniques; Male; Oxazines; Pyrimidinones; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Sodium Chloride Symporter Inhibitors; Tritium; Uracil | 2000 |
Presynaptic alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate receptor-mediated stimulation of glutamate and GABA release in the rat striatum in vivo: a dual-label microdialysis study.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carbon Radioisotopes; Corpus Striatum; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Kynurenic Acid; Male; Microdialysis; Nootropic Agents; Potassium; Presynaptic Terminals; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Tritium | 2001 |
The Neurobiology and Neuropharmacology of Alzheimer's Disease. The ASPET - Ray Fuller Symposium. New Orleans, LA, USA, April 19-20, 2002.
Topics: Alzheimer Disease; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Humans; Neurobiology; Neuropharmacology; Neuroprotective Agents; Oxazines | 2002 |
AMPA receptors on developing medial septum/diagonal band neurons are sensitive to early postnatal binge-like ethanol exposure.
Topics: Alcohol-Induced Disorders, Nervous System; Alcoholic Intoxication; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Blotting, Western; Cells, Cultured; Central Nervous System Depressants; Diagonal Band of Broca; Ethanol; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Kainic Acid; Male; Membrane Potentials; Models, Animal; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, AMPA | 2003 |
Apoptosis-inducing factor is a key factor in neuronal cell death propagated by BAX-dependent and BAX-independent mechanisms.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Apoptosis; Apoptosis Inducing Factor; Apoptotic Protease-Activating Factor 1; bcl-2-Associated X Protein; Benzodiazepines; Benzothiadiazines; Camptothecin; Caspase Inhibitors; Cells, Cultured; Cerebellum; Cerebral Cortex; Convulsants; Dizocilpine Maleate; Drug Resistance; Flavoproteins; Glutamic Acid; Glycine; Hippocampus; Kainic Acid; Male; Membrane Proteins; Mice; Mice, Knockout; Mice, Mutant Strains; N-Methylaspartate; Neurons; Neurotoxins; Proteins; Proto-Oncogene Proteins c-bcl-2; Recombinant Fusion Proteins; Seizures | 2005 |
C-terminal truncation affects kinetic properties of GluR1 receptors.
Topics: Amino Acid Sequence; Benzodiazepines; Benzothiadiazines; Cell Line; Diuretics; Excitatory Amino Acid Antagonists; Glutamic Acid; Humans; Kidney; Kinetics; Ligands; Molecular Sequence Data; Mutagenesis; Protein Binding; Protein Structure, Tertiary; Receptors, AMPA; Structure-Activity Relationship | 2005 |
A comparison of release kinetics and glutamate receptor properties in shaping rod-cone differences in EPSC kinetics in the salamander retina.
Topics: Animals; Benzodiazepines; Benzothiadiazines; Calcium; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Kinetics; Models, Biological; Neurotransmitter Agents; Quinoxalines; Receptors, AMPA; Receptors, Glutamate; Retinal Bipolar Cells; Retinal Cone Photoreceptor Cells; Retinal Horizontal Cells; Retinal Rod Photoreceptor Cells; Synaptic Transmission; Synaptic Vesicles; Urodela | 2005 |
Cyclothiazide prolongs low [Mg2+]-induced seizure-like events.
Topics: 4-Aminopyridine; Animals; Benzodiazepines; Benzothiadiazines; Diuretics; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Magnesium Deficiency; Male; Potassium Channel Blockers; Pyramidal Cells; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Presynaptic; Seizures | 2006 |
Inhibition of calcium-permeable and calcium-impermeable AMPA receptors by perampanel in rat brain neurons.
Topics: Animals; Anticonvulsants; Benzodiazepines; Benzothiadiazines; Binding Sites; Brain; CA1 Region, Hippocampal; Calcium; Corpus Striatum; Drug Interactions; Glutamic Acid; Interneurons; Kainic Acid; Neurons; Nitriles; Pyramidal Cells; Pyridones; Rats, Wistar; Receptors, AMPA | 2016 |