Compounds > gyki 52466

gyki 52466 and cfm 2

gyki 52466 has been researched along with cfm 2 in 13 studies

Research

Studies (13)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	4 (30.77)	18.2507
2000's	9 (69.23)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Chapman, AG; Chimirri, A; Constanti, A; De Sarro, A; De Sarro, G; Gitto, R; Giusti, P; Grasso, S; Libri, V; Quartarone, S; Zappalà, M	1
Cai, SX; Carter, RB; Ilyin, VI; Keana, JF; Konkoy, CS; Vanover, KE; Wang, Y; Weber, E; Woodward, RM	1
Chimirri, A; Constanti, A; De Sarro, A; De Sarro, G; Gitto, R; Libri, V; Quartarone, S; Zappalà, M	1
De Sarro, A; De Sarro, G; Gitto, R; Grasso, S; Micale, N; Quartarone, S; Zappalà, M	1
Bevacqua, F; Chimirri, A; De Sarro, A; De Sarro, G; Gitto, R; Quartarone, S; Rizzo, M; Zappalà, M	1
Barreca, ML; Chimirri, A; Constanti, A; De Luca, L; De Sarro, G; Ferreri, G; Gitto, R; Quartarone, S; Russo, E	1
Chimirri, A; De Sarro, A; De Sarro, G; Ferreri, G; Gitto, R; Orlando, V; Quartarone, S; Russo, E	1
Barreca, ML; Chimirri, A; Costantino, G; De Luca, L; Gitto, R; Macchiarulo, A; Pellicciari, R	1
Caruso, R; Chimirri, A; Citraro, R; De Luca, L; De Sarro, G; Gitto, R; Pagano, B; Russo, E	1
Barreca, ML; Caruso, R; Chimirri, A; De Sarro, G; Ferreri, G; Gitto, R; Orlando, V; Quartarone, S; Russo, E	1
Kandefer-Szerszeń, M; Majdan, M; Parada-Turska, J; Rzeski, W; Turski, WA	1
Brocke, K; Gratopp, A; Ikonomidou, C; Pohl, EE; Rzeski, W; Sifringer, M; Stepulak, A; Turski, L	1
Guan, X; Guan, Y; Park, JS; Raja, SN; Shih, MH; Tao, YX; Xu, JT; Yaster, M	1

Other Studies

13 other study(ies) available for gyki 52466 and cfm 2

Article	Year
1-Aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones: novel AMPA receptor antagonists. Journal of medicinal chemistry, 1997, Apr-11, Volume: 40, Issue:8 Topics: Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Benzodiazepinones; Convulsants; Mice; Mice, Inbred DBA; Pentylenetetrazole; Pyrrolidinones; Receptors, AMPA; Seizures	1997
Synthesis of 7,8-(methylenedioxy)-1-phenyl-3,5-dihydro-4H-2, 3-benzodiazepin-4-ones as novel and potent noncompetitive AMPA receptor antagonists. Journal of medicinal chemistry, 1998, Jul-02, Volume: 41, Issue:14 Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepines; Cerebral Cortex; Electroshock; Excitatory Amino Acid Antagonists; Male; Membrane Potentials; Mice; Oocytes; Rats; Receptors, AMPA; RNA, Messenger; Seizures; Xenopus laevis	1998
3,5-Dihydro-4H-2,3-benzodiazepine-4-thiones: a new class of AMPA receptor antagonists. Journal of medicinal chemistry, 1998, Aug-27, Volume: 41, Issue:18 Topics: Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Benzodiazepines; Convulsants; Electroshock; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Motor Activity; Olfactory Pathways; Patch-Clamp Techniques; Pentylenetetrazole; Pyrrolidinones; Rats; Receptors, AMPA; Seizures; Structure-Activity Relationship; Thiones	1998
7,8-Methylenedioxy-4H-2,3-benzodiazepin-4-ones as novel AMPA receptor antagonists. Bioorganic & medicinal chemistry letters, 1998, Apr-21, Volume: 8, Issue:8 Topics: Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Excitatory Amino Acid Antagonists; Indicators and Reagents; Mice; Mice, Inbred DBA; Molecular Structure; Motor Activity; Receptors, AMPA; Seizures; Structure-Activity Relationship	1998
Synthesis and evaluation of pharmacological and pharmacokinetic properties of 11H-[1,2,4]triazolo[4,5-c][2,3]benzodiazepin-3(2H)-ones. Journal of medicinal chemistry, 2000, Dec-14, Volume: 43, Issue:25 Topics: Acoustic Stimulation; Allosteric Regulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Benzodiazepines; Chromatography, High Pressure Liquid; Electroshock; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred DBA; Motor Activity; Pentylenetetrazole; Pyrrolidinones; Receptors, AMPA; Seizures; Structure-Activity Relationship	2000
Discovery of a novel and highly potent noncompetitive AMPA receptor antagonist. Journal of medicinal chemistry, 2003, Jan-02, Volume: 46, Issue:1 Topics: Acoustic Stimulation; Animals; Anticonvulsants; Excitatory Amino Acid Antagonists; Isoquinolines; Ligands; Mice; Mice, Inbred DBA; Receptors, AMPA; Seizures; Structure-Activity Relationship; Tetrahydroisoquinolines	2003
Synthesis and evaluation of pharmacological properties of novel annelated 2,3-benzodiazepine derivatives. Journal of medicinal chemistry, 2003, Aug-14, Volume: 46, Issue:17 Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Benzodiazepines; Disease Models, Animal; Epilepsy; Excitatory Amino Acid Agonists; In Vitro Techniques; Magnetic Resonance Spectroscopy; Mice; Mice, Inbred DBA; Neurons; Olfactory Pathways; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Structure-Activity Relationship; Triazoles	2003
QSAR study of anticonvulsant negative allosteric modulators of the AMPA receptor. Journal of medicinal chemistry, 2004, Mar-25, Volume: 47, Issue:7 Topics: Allosteric Regulation; Anticonvulsants; Benzodiazepines; Excitatory Amino Acid Antagonists; Isoquinolines; Linear Models; Models, Biological; Phthalazines; Quantitative Structure-Activity Relationship; Receptors, AMPA	2004
Novel potent anticonvulsant agent containing a tetrahydroisoquinoline skeleton. Journal of medicinal chemistry, 2006, Sep-07, Volume: 49, Issue:18 Topics: Acoustic Stimulation; Animals; Anticonvulsants; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred DBA; Olfactory Pathways; Piperidines; Rats; Rats, Wistar; Receptors, AMPA; Seizures; Structure-Activity Relationship; Tetrahydroisoquinolines	2006
Synthesis and anticonvulsant properties of tetrahydroisoquinoline derivatives. Farmaco (Societa chimica italiana : 1989), 2004, Volume: 59, Issue:1 Topics: Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Drug Evaluation, Preclinical; Excitatory Amino Acid Antagonists; Female; Male; Mice; Mice, Inbred DBA; Models, Molecular; Molecular Structure; Receptors, AMPA; Seizures; Structure-Activity Relationship; Tetrahydroisoquinolines	2004
Effect of glutamate receptor antagonists and antirheumatic drugs on proliferation of synoviocytes in vitro. European journal of pharmacology, 2006, Mar-27, Volume: 535, Issue:1-3 Topics: Animals; Antirheumatic Agents; Benzodiazepines; Benzodiazepinones; Celecoxib; Cell Line; Cell Proliferation; Cell Survival; Diclofenac; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Inhibitory Concentration 50; Methotrexate; Naproxen; Pyrazoles; Quinoxalines; Sulfasalazine; Sulfonamides; Synovial Membrane	2006
AMPA antagonists inhibit the extracellular signal regulated kinase pathway and suppress lung cancer growth. Cancer biology & therapy, 2007, Volume: 6, Issue:12 Topics: Adenocarcinoma; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Antineoplastic Agents; Benzodiazepines; Benzodiazepinones; Cell Cycle; Cell Line, Tumor; Drug Screening Assays, Antitumor; Enzyme Activation; Excitatory Amino Acid Antagonists; Gene Expression Regulation, Neoplastic; Humans; Lung Neoplasms; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Neoplasm Proteins; Phosphorylation; Protein Processing, Post-Translational; Receptors, AMPA; Signal Transduction	2007
Role of spinal cord alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors in complete Freund's adjuvant-induced inflammatory pain. Molecular pain, 2008, Dec-30, Volume: 4 Topics: Adjuvants, Immunologic; Animals; Benzodiazepines; Benzodiazepinones; Cell Membrane; Cytosol; Freund's Adjuvant; Inflammation; Male; Pain; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Spinal Cord; Thermosensing	2008