gyki 52466 and 2-amino-5-phosphonovalerate

gyki 52466 has been researched along with 2-amino-5-phosphonovalerate in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's11 (55.00)18.2507
2000's7 (35.00)29.6817
2010's2 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Payne, RS; Rigor, BM; Schurr, A1
Mennerick, S; Zorumski, CF1
Croucher, MJ; Patel, DR; Sturt, NJ1
Crunelli, V; Guyon, A; Leresche, N; Soltesz, I; Turner, JP1
Hauber, W; Waldenmeier, MT1
Müller, W; Parsons, C; Rammes, G; Swandulla, D1
Block, F; Schwarz, M1
Schmidt, WJ; Tzschentke, TM1
Jaw, SP; Nguyen, M; Vuong, QT1
Conrad, P; Schacher, S; Wu, F1
Kullmann, DM; Melyan, Z; Min, MY1
Ciotti, MT; Eusebi, F; Giovannelli, A; Limatola, C; Mercanti, D; Miledi, R; Ragozzino, D; Santoni, A; Vacca, F1
Kalfin, R; Kiss, JP; Lazarova, M; Milenov, K; Raichev, P; Rakovska, A1
Banczerowski-Pelyhe, I; Détári, L; Dóczi, J; Gulyás-Kovács, A; Tarnawa, I; Világi, I1
Farkas, S; Kocsis, P; Szombathelyi, Z; Tarnawa, I1
Choi, JH; Chun, SW; Kim, MS; Park, BR1
Avshalumov, MV; Patel, JC; Rice, ME1
Bakos, M; Borbély, S; Czégé, D; Dobó, E; Mihály, A; Molnár, E; Szucs, B; Világi, I; Vincze, A1
Borbély, S; Czégé, D; Dobó, E; Mihály, A; Molnár, E; Világi, I1
Folbergrová, J; Haugvicová, R; Kubová, H; Mareš, P1

Other Studies

20 other study(ies) available for gyki 52466 and 2-amino-5-phosphonovalerate

ArticleYear
Protection by MK-801 against hypoxia-, excitotoxin-, and depolarization-induced neuronal damage in vitro.
    Neurochemistry international, 1995, Volume: 26, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Anti-Anxiety Agents; Benzodiazepines; Diltiazem; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Kynurenic Acid; Membrane Potentials; Neurons; Nifedipine; Pipecolic Acids; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1995
Presynaptic influence on the time course of fast excitatory synaptic currents in cultured hippocampal cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Kinetics; Magnesium; Neurons; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Time Factors

1995
Modulation of D-[2,3 3H]aspartate release from rat forebrain slices by non-NMDA receptor agonists and antagonists.
    Biochemical Society transactions, 1995, Volume: 23, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Aspartic Acid; Benzodiazepines; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; In Vitro Techniques; Kainic Acid; Kinetics; Kynurenic Acid; Male; Prosencephalon; Quinoxalines; Rats; Rats, Wistar; Tritium

1995
Sensory input and burst firing output of rat and cat thalamocortical cells: the role of NMDA and non-NMDA receptors.
    The Journal of physiology, 1994, Oct-15, Volume: 480 ( Pt 2)

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Benzodiazepines; Calcium; Cats; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; Female; Geniculate Bodies; In Vitro Techniques; Male; Membrane Potentials; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Synaptic Transmission

1994
The AMPA receptor antagonist GYKI 52466 reverses the anti-cataleptic effects of the competitive NMDA receptor antagonist CGP 37849.
    European journal of pharmacology, 1994, May-02, Volume: 256, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Catalepsy; Drug Interactions; Haloperidol; Injections, Intraperitoneal; Male; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

1994
Modulation of fast excitatory synaptic transmission by cyclothiazide and GYKI 52466 in the rat hippocampus.
    Neuroscience letters, 1994, Jul-04, Volume: 175, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Binding Sites; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Organophosphorus Compounds; Picrotoxin; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

1994
The depressant effect of GYKI 52466 on spinal reflex transmission in rats is mediated via non-NMDA and benzodiazepine receptors.
    European journal of pharmacology, 1994, Apr-21, Volume: 256, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; H-Reflex; Injections, Spinal; Male; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex; Synaptic Transmission

1994
Morphine-induced catalepsy is augmented by NMDA receptor antagonists, but is partially attenuated by an AMPA receptor antagonist.
    European journal of pharmacology, 1996, Jan-11, Volume: 295, Issue:2-3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Benzodiazepines; Catalepsy; Dizocilpine Maleate; Male; Morphine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Time Factors

1996
Effects of glutamate receptor antagonists on posthypoxic myoclonus in rats.
    Brain research bulletin, 1996, Volume: 40, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Hypoxia, Brain; Male; Myoclonus; Quinoxalines; Rats; Rats, Sprague-Dawley

1996
Changes in functional glutamate receptors on a postsynaptic neuron accompany formation and maturation of an identified synapse.
    Journal of neurobiology, 1999, Volume: 39, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Aplysia; Axons; Benzodiazepines; Cells, Cultured; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Neurons, Afferent; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Synapses

1999
Synaptically released glutamate reduces gamma-aminobutyric acid (GABA)ergic inhibition in the hippocampus via kainate receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, Aug-17, Volume: 96, Issue:17

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Guinea Pigs; Hippocampus; Kynurenic Acid; Receptors, AMPA; Receptors, Kainic Acid; Seizures

1999
The chemokine growth-related gene product beta protects rat cerebellar granule cells from apoptotic cell death through alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, May-23, Volume: 97, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Apoptosis; Benzodiazepines; Cerebellar Cortex; Chemokines, CXC; Chemotactic Factors; DNA, Complementary; Gene Expression Regulation; Growth Substances; Intercellular Signaling Peptides and Proteins; Interleukin-8; Ion Channel Gating; Nerve Tissue Proteins; Neuroprotective Agents; Oligodeoxyribonucleotides, Antisense; Potassium; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2000
Somatostatin stimulates striatal acetylcholine release by glutamatergic receptors: an in vivo microdialysis study.
    Neurochemistry international, 2002, Volume: 40, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Anti-Anxiety Agents; Benzodiazepines; Corpus Striatum; Excitatory Amino Acid Antagonists; Male; Microdialysis; Quinoxalines; Rats; Rats, Wistar; Receptors, Glutamate; Somatostatin; Tetrodotoxin

2002
Comparison of spontaneous and evoked epileptiform activity in three in vitro epilepsy models.
    Brain research, 2002, Aug-02, Volume: 945, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 4-Aminopyridine; Animals; Anti-Anxiety Agents; Benzodiazepines; Bicuculline; Convulsants; Electric Stimulation; Electrophysiology; Epilepsy; Excitatory Amino Acid Antagonists; Female; Magnesium Deficiency; Male; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Somatosensory Cortex

2002
Participation of AMPA- and NMDA-type excitatory amino acid receptors in the spinal reflex transmission, in rat.
    Brain research bulletin, 2003, Apr-15, Volume: 60, Issue:1-2

    Topics: Action Potentials; Animals; Animals, Newborn; Anti-Anxiety Agents; Benzodiazepines; Dizocilpine Maleate; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; In Vitro Techniques; Magnesium; Models, Neurological; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Reflex, Monosynaptic; Spinal Cord; Synapses; Time Factors; Valine

2003
Characterization of spontaneous synaptic transmission in rat medial vestibular nucleus.
    Neuroreport, 2003, Aug-06, Volume: 14, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; Animals; Benzodiazepines; Bicuculline; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA-A Receptor Antagonists; Glycine Agents; In Vitro Techniques; Kinetics; N-Methylaspartate; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Strychnine; Synaptic Transmission; Vestibular Nuclei

2003
AMPA receptor-dependent H2O2 generation in striatal medium spiny neurons but not dopamine axons: one source of a retrograde signal that can inhibit dopamine release.
    Journal of neurophysiology, 2008, Volume: 100, Issue:3

    Topics: Analysis of Variance; Animals; Axons; Benzodiazepines; Catalase; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Electric Stimulation; Excitatory Amino Acid Antagonists; Guinea Pigs; Hydrogen Peroxide; In Vitro Techniques; Male; Neural Pathways; Neurons; Patch-Clamp Techniques; Receptors, AMPA; Thiomalates; Tyrosine 3-Monooxygenase; Valine

2008
Modification of ionotropic glutamate receptor-mediated processes in the rat hippocampus following repeated, brief seizures.
    Neuroscience, 2009, Mar-03, Volume: 159, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 4-Aminopyridine; Action Potentials; Animals; Benzodiazepines; Biophysics; Calcium; Cobalt; Electric Stimulation; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Hippocampus; In Vitro Techniques; Male; Neurons; Protein Subunits; Rats; Rats, Wistar; Receptors, Glutamate; Seizures; Synaptic Transmission

2009
Repeated application of 4-aminopyridine provoke an increase in entorhinal cortex excitability and rearrange AMPA and kainate receptors.
    Neurotoxicity research, 2015, Volume: 27, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 4-Aminopyridine; Animals; Benzodiazepines; Entorhinal Cortex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kainic Acid; Male; Protein Subunits; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Seizures

2015
Do stereoisomers of homocysteic acid exhibit different convulsant action in immature rats?
    Physiological research, 2019, 12-20, Volume: 68, Issue:Suppl 3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Benzodiazepines; Dizocilpine Maleate; Homocysteine; Male; Quinoxalines; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Seizures; Stereoisomerism

2019