Page last updated: 2024-09-04

gw420867x and quinidine

gw420867x has been researched along with quinidine in 1 studies

Compound Research Comparison

Studies
(gw420867x)
Trials
(gw420867x)
Recent Studies (post-2010)
(gw420867x)
Studies
(quinidine)
Trials
(quinidine)
Recent Studies (post-2010) (quinidine)
17526,608387594

Protein Interaction Comparison

ProteinTaxonomygw420867x (IC50)quinidine (IC50)
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)6.4
CholinesteraseHomo sapiens (human)1.23
ATP-dependent translocase ABCB1Mus musculus (house mouse)10
ATP-dependent translocase ABCB1Homo sapiens (human)3.32
Cytochrome P450 2D26Rattus norvegicus (Norway rat)2.8
Cytochrome P450 2D6Homo sapiens (human)0.3532
Potassium voltage-gated channel subfamily A member 5Homo sapiens (human)7.3
CholinesteraseEquus caballus (horse)7.37
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)6.4
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.7882
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)6.4
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)6.4
Sodium channel protein type 5 subunit alphaHomo sapiens (human)6.9
Potassium voltage-gated channel subfamily D member 2Rattus norvegicus (Norway rat)2.2

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Huang, L; Humphreys, JE; Morgan, JB; Polli, JW; Serabjit-Singh, CS; Webster, LO; Wring, SA1

Other Studies

1 other study(ies) available for gw420867x and quinidine

ArticleYear
Rational use of in vitro P-glycoprotein assays in drug discovery.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:2

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Chromatography, Liquid; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; Mass Spectrometry; Pharmacology; Spodoptera

2001