gsk1210151a and quinoline

gsk1210151a has been researched along with quinoline* in 1 studies

Other Studies

1 other study(ies) available for gsk1210151a and quinoline

Article	Year
From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151. Bioorganic & medicinal chemistry letters, 2012, Apr-15, Volume: 22, Issue:8 The discovery, synthesis and biological evaluation of a novel series of 7-isoxazoloquinolines is described. Several analogs are shown to increase ApoA1 expression within the nanomolar range in the human hepatic cell line HepG2. Topics: Animals; Anti-Inflammatory Agents; Apolipoprotein A-I; Drug Discovery; Hep G2 Cells; Heterocyclic Compounds, 4 or More Rings; Histone Acetyltransferases; Histone Chaperones; Humans; Inhibitory Concentration 50; Mice; Mice, Inbred BALB C; Nerve Tissue Proteins; Nuclear Proteins; Quinolines; Rats; Structure-Activity Relationship; Up-Regulation	2012

Article

Year

From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151.

Bioorganic & medicinal chemistry letters, 2012, Apr-15, Volume: 22, Issue:8

The discovery, synthesis and biological evaluation of a novel series of 7-isoxazoloquinolines is described. Several analogs are shown to increase ApoA1 expression within the nanomolar range in the human hepatic cell line HepG2.

Topics: Animals; Anti-Inflammatory Agents; Apolipoprotein A-I; Drug Discovery; Hep G2 Cells; Heterocyclic Compounds, 4 or More Rings; Histone Acetyltransferases; Histone Chaperones; Humans; Inhibitory Concentration 50; Mice; Mice, Inbred BALB C; Nerve Tissue Proteins; Nuclear Proteins; Quinolines; Rats; Structure-Activity Relationship; Up-Regulation

2012