granisetron and metoclopramide

granisetron has been researched along with metoclopramide in 85 studies

Research

Studies (85)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's53 (62.35)18.2507
2000's18 (21.18)29.6817
2010's10 (11.76)24.3611
2020's4 (4.71)2.80

Authors

AuthorsStudies
Airey, JE; Campbell, HF; Darkes, P; Fitzpatrick, LR; Klein, S; Neuenschwander, K; Pendley, CE; Powers, M; Schnapper, M; Youssefyeh, RD1
Diehl, V1
Kaizer, L; Laberge, F; Latreille, J; O'Connell, G; Osoba, D; Pater, J; Stewart, D; Venner, P; Warr, D; Wilan, A1
Anderson, I; Cowen, P1
Gandara, DR; Hesketh, PJ1
King, GL1
Elliott, P; Wallis, DI1
Elliott, P; Seemungal, BM; Wallis, DI1
Chevallier, B2
Chen, PM; Chiou, TJ; Fan, FS; Hsieh, RK; Liu, JH; Wei, CH1
Heron, JF1
Collis, C; Cunningham, J; Cunningham, S; Gandhi, L; Hamon, MD; Prentice, HG1
Arioka, H; Eguchi, K; Karato, A; Kunikane, H; Nakashima, H; Nisio, M; Ohe, Y; Ohmatsu, H; Shinkai, T; Tamura, T1
Cedar, E; Cunningham, J; Goedhals, L; Heron, JF; Jordaan, JP1
Osoba, D; Pater, J; Rusthoven, J; Slamet, L; Warr, D; Zee, B1
Ang, PT; Khoo, KS; Tan, EH1
Fukuda, T; Haga, K; Inaba, K; Morimoto, Y; Setoguchi, M; Shoji, H1
Kirchner, V1
Kawashima, T; Miyata, K; Morita, N; Ohmata, T; Sakamoto, T; Wada, T1
Essien, E; Thut, PD; Wynn, RL1
Ohta, J; Taguchi, T; Tsukagoshi, S1
Snyman, JR; Sommers, DK; van Wyk, M1
Cannata, G; Gebbia, N; Gebbia, V; Testa, A; Tirrito, ML; Valenza, R1
Hojo, F; Kakinuma, R; Kodama, T; Kubota, K; Matsumoto, T; Nishiwaki, Y; Ohmatsu, H; Sekine, I; Yokozaki, M1
Asano, S; Ikeda, Y; Kimura, Y; Miyawaki, S; Oh, H; Okamoto, S; Onozawa, Y; Sakamaki, H; Takahashi, S; Tanosaki, R; Toyama, K1
Attia, M; Channa, AB; el Bakry, AK; el Gammal, K; el Gammal, M; Elhattab, YS; Jaroudi, R; Khoshim, MH; Naguib, M; Saddique, A1
Cubeddu, LX; Cupissol, D; Gralla, RJ; Homesley, HD; Kris, MG; Tyson, LB; Venkatraman, E1
Fujii, Y; Tanaka, H; Toyooka, H6
Chang, CS; Chen, LT; Chen, TP; Huang, SM; Lin, SF; Liu, TC; Wei, TC1
Cheng, X; Itamochi, H; Kigawa, J; Minagawa, Y; Okada, M; Terakawa, N1
Goto, K; Hojo, F; Kakinuma, R; Kodama, T; Kubota, K; Matsumoto, T; Miyamoto, T; Nishiwaki, Y; Ohmatsu, H; Sekine, I; Takafuji, J; Yokozaki, M1
Basurto, C; Ciccarese, G; Palladino, MA; Roila, F1
Fujii, Y; Saitoh, Y; Tanaka, H; Toyooka, H2
Fujii, Y; Tanaka, H2
Brown, RS; Brown, TK; Gaze, MN; Hoare, D1
Fujii, Y; Kobayashi, N; Tanaka, H1
Granisétron, PK; Mabro, M1
Endo, K; Ichimura, H; Inoue, S1
Khan, NA; Poisson, JP1
Boeckxstaens, GE; De Man, JG; De Winter, BY; Herman, AG; Moreels, TG; Peeters, TL; Pelckmans, PA; Schuurkes, JA1
Fujii, Y; Somekawa, Y; Tanaka, H1
Fujii, Y; Kawasaki, T; Tanaka, H2
Endo, K; Inoue, S; Suzuki, H1
Leelasiri, A; Mongkonsritragoon, W; Numbenjapon, T; Prayoonwiwat, W; Sriswasdi, C1
Aapro, MS; Bernhard, J; De Pree, C; Maibach, R; Sessa, C; Thuerlimann, B1
Endo, K; Inoue, S; Itou, H; Nakamura, R1
Caran, EM; Luisi, FA; Petrilli, AS; Tanaka, C1
Ito, Y; Tomono, H; Watanabe, T1
del Giglio, A; Lajolo, PP1
Ahlburg, P; Nielsen, JO1
Aćimović, M; Argirović, R; Dragićević, D; Filimonović, J; Krivić, B; Ladjević, N; Likić Ladjević, I1
Ezberci, M; Oksuz, H; Zencirci, B1
Du Bois, A1
Baraka, AS; Dabbous, AS; El-Khatib, MF; Jabbour-Khoury, SI; Khouzam, NE; Moussa, AA; Nasr, VG; Zbeidy, RA1
Bi, F; Cao, D; Gou, HF; Hou, M; Jiang, M; Luo, de Y; Qiu, M; Shen, Y; Wang, J; Xu, F; Yang, Y; Yi, C; Zang, J; Zhou, XJ1
Eksborg, S; Lönnqvist, PA; Öbrink, E; Oddby-Muhrbeck, E; Rotstein, S1
Abdul Kassim, MS; Keat, CH; Phua, G; Poh, WK; Sriraman, M1
Ghani, NA; Keat, CH1
Cázares-Delgadillo, J; Ganem-Rondero, A; Kalia, YN; Merino, V1
Abushouk, AI; Ahmed, H; Al Nahrawi, S; Attia, A; Awad, K; Elsherbeny, MY; Mustafa, SM1
Huss, IB; Ritchie, HE; Webster, WS1
Acosta-Reyes, J; Florez, ID; Niño-Serna, LF; Veroniki, AA1
Adib-Majlesi, M; Hajigholami, A; Moghaddas, A; Riechelmann, R; Sabzghabaee, AM1
Ebrahimian, M; Ghayebi, N; Kialashaki, M; Mirhashemi, SH; Oshidari, B; Shadidi-Asil, R; Zamani, A1
Abd-ElGawad, M; Abdelhay, HM; Abdelmonem, H; Abdelwadoud, GT; Ahmed, AE; Al-Dardery, NM; Alhosini, ANM; Kamel, MA; Mohamed, SW1
Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD1
Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT1
Carr, AA; Hibert, MF; Hoffmann, R; Miller, RC1
Bourguignon, JJ; Didier, B; Hoffmann, R; Rival, Y; Rybaltchenko, V; Wermuth, CG1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1

Reviews

11 review(s) available for granisetron and metoclopramide

ArticleYear
Inconsistency of prognostic factors for post-chemotherapy nausea and vomiting.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 1994, Volume: 2, Issue:3

    Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Doxorubicin; Female; Granisetron; Humans; Male; Methylprednisolone; Metoclopramide; Middle Aged; Nausea; Neoplasms; Prognosis; Randomized Controlled Trials as Topic; Serotonin Antagonists; Treatment Outcome; Vomiting

1994
Clinical studies to assess the economic impact of new therapies: pragmatic approaches to measuring costs.
    Anti-cancer drugs, 1993, Volume: 4 Suppl 3

    Topics: Antiemetics; Clinical Trials as Topic; Cost-Benefit Analysis; Costs and Cost Analysis; Drug Therapy, Combination; Granisetron; Humans; Metoclopramide; Ondansetron; Serotonin Antagonists

1993
[An outline of 5-HT3 receptor antagonists (2)--In clinical applications].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1993, Volume: 20, Issue:15

    Topics: Antineoplastic Agents; Granisetron; Humans; Metoclopramide; Nausea; Ondansetron; Serotonin Antagonists; Vomiting

1993
Are more antiemetic trials with a placebo necessary? Report of patient data from randomized trials of placebo antiemetics with cisplatin.
    Cancer, 1996, Nov-15, Volume: 78, Issue:10

    Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Cisplatin; Double-Blind Method; Female; Granisetron; Humans; Male; Metoclopramide; Middle Aged; Ondansetron; Placebos; Randomized Controlled Trials as Topic; Vomiting

1996
[Recent improvements in antiemetic therapy].
    Tumori, 1997, Volume: 83, Issue:2 Suppl

    Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Drug Therapy, Combination; Granisetron; Humans; Indoles; Metoclopramide; Nausea; Ondansetron; Phenothiazines; Serotonin Antagonists; Tropisetron; Vomiting

1997
[Prevention of postoperative nausea and vomiting].
    Ugeskrift for laeger, 2007, Aug-13, Volume: 169, Issue:33

    Topics: Antiemetics; Dexamethasone; Droperidol; Evidence-Based Medicine; Granisetron; Humans; Indoles; Metoclopramide; Postoperative Nausea and Vomiting; Quinolizines; Randomized Controlled Trials as Topic; Treatment Outcome

2007
[Management of chemotherapy-induced emesis: what is the standard after 20 years of clinical research].
    Medizinische Klinik (Munich, Germany : 1983), 1998, Volume: 93 Suppl 1

    Topics: Antineoplastic Combined Chemotherapy Protocols; Benchmarking; Dexamethasone; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Granisetron; Humans; Indoles; Metoclopramide; Nausea; Ondansetron; Premedication; Randomized Controlled Trials as Topic; Research; Serotonin 5-HT3 Receptor Antagonists; Tropisetron; Vomiting

1998
Dexamethasone combined with other antiemetics versus single antiemetics for prevention of postoperative nausea and vomiting after laparoscopic cholecystectomy: An updated systematic review and meta-analysis.
    International journal of surgery (London, England), 2016, Volume: 36, Issue:Pt A

    Topics: Antiemetics; Benzimidazoles; Cholecystectomy, Laparoscopic; Dexamethasone; Drug Therapy, Combination; Granisetron; Humans; Isoquinolines; Metoclopramide; Ondansetron; Palonosetron; Postoperative Nausea and Vomiting; Quinuclidines; Randomized Controlled Trials as Topic

2016
Antiemetics in Children With Acute Gastroenteritis: A Meta-analysis.
    Pediatrics, 2020, Volume: 145, Issue:4

    Topics: Acute Disease; Antiemetics; Child; Child, Preschool; Dexamethasone; Diarrhea; Dimenhydrinate; Domperidone; Fluid Therapy; Gastroenteritis; Granisetron; Hospitalization; Humans; Infant; Metoclopramide; Network Meta-Analysis; Ondansetron; Randomized Controlled Trials as Topic; Regression Analysis; Vomiting

2020
The efficacy and safety of metoclopramide in relieving acute migraine attacks compared with other anti-migraine drugs: a systematic review and network meta-analysis of randomized controlled trials.
    BMC neurology, 2023, Jun-08, Volume: 23, Issue:1

    Topics: Chlorpromazine; Granisetron; Headache; Humans; Ketorolac; Metoclopramide; Migraine Disorders; Nausea; Network Meta-Analysis; Prochlorperazine; Randomized Controlled Trials as Topic; Sumatriptan; Valproic Acid

2023
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

46 trial(s) available for granisetron and metoclopramide

ArticleYear
Fractionated chemotherapy--granisetron or conventional antiemetics? The Granisetron Study Group.
    European journal of cancer (Oxford, England : 1990), 1992, Volume: 28A Suppl 1

    Topics: Adult; Antiemetics; Antineoplastic Agents; Dexamethasone; Drug Administration Schedule; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Nausea; Pyrrolidines; Single-Blind Method; Vomiting

1992
A randomised, double-blind comparison of granisetron with high-dose metoclopramide, dexamethasone and diphenhydramine for cisplatin-induced emesis. An NCI Canada Clinical Trials Group Phase III Trial.
    European journal of cancer (Oxford, England : 1990), 1992, Volume: 29A, Issue:1

    Topics: Antiemetics; Cisplatin; Dexamethasone; Diphenhydramine; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Nausea; Vomiting

1992
Efficacy and safety of granisetron compared with high-dose metoclopramide plus dexamethasone in patients receiving high-dose cisplatin in a single-blind study. The Granisetron Study Group.
    European journal of cancer (Oxford, England : 1990), 1990, Volume: 26 Suppl 1

    Topics: Cisplatin; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Headache; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Neoplasms; Serotonin Antagonists; Single-Blind Method; Vomiting

1990
Comparison of intravenous granisetron with metoclopramide in the treatment of chemotherapy-induced emesis.
    Zhonghua yi xue za zhi = Chinese medical journal; Free China ed, 1995, Volume: 56, Issue:1

    Topics: Adult; Aged; Antiemetics; Cisplatin; Female; Granisetron; Humans; Injections, Intravenous; Male; Metoclopramide; Middle Aged; Serotonin Antagonists; Vomiting

1995
Single-agent oral granisetron for the prevention of acute cisplatin-induced emesis: a double-blind, randomized comparison with granisetron plus dexamethasone and high-dose metoclopramide plus dexamethasone.
    Seminars in oncology, 1995, Volume: 22, Issue:4 Suppl 10

    Topics: Acute Disease; Administration, Oral; Adult; Aged; Cisplatin; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Male; Metoclopramide; Middle Aged; Vomiting

1995
Granisetron in the prevention of irradiation-induced emesis.
    Bone marrow transplantation, 1995, Volume: 15, Issue:3

    Topics: Adult; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Follow-Up Studies; Granisetron; Humans; Lorazepam; Male; Metoclopramide; Vomiting; Whole-Body Irradiation

1995
A randomized cross-over study of high-dose metoclopramide plus dexamethasone versus granisetron plus dexamethasone in patients receiving chemotherapy with high-dose cisplatin.
    Japanese journal of cancer research : Gann, 1994, Volume: 85, Issue:11

    Topics: Adult; Aged; Cisplatin; Cross-Over Studies; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Humans; Lung Neoplasms; Male; Metoclopramide; Middle Aged; Multivariate Analysis; Nausea; Single-Blind Method; Vomiting

1994
Oral granisetron alone and in combination with dexamethasone: a double-blind randomized comparison against high-dose metoclopramide plus dexamethasone in prevention of cisplatin-induced emesis. The Granisetron Study Group.
    Annals of oncology : official journal of the European Society for Medical Oncology, 1994, Volume: 5, Issue:7

    Topics: Administration, Oral; Adult; Aged; Chi-Square Distribution; Cisplatin; Constipation; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Europe; Female; Granisetron; Headache; Humans; Male; Metoclopramide; Middle Aged; Nausea; Prognosis; South Africa; Vomiting

1994
Inconsistency of prognostic factors for post-chemotherapy nausea and vomiting.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 1994, Volume: 2, Issue:3

    Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Doxorubicin; Female; Granisetron; Humans; Male; Methylprednisolone; Metoclopramide; Middle Aged; Nausea; Neoplasms; Prognosis; Randomized Controlled Trials as Topic; Serotonin Antagonists; Treatment Outcome; Vomiting

1994
Control of emesis by intravenous granisetron in breast cancer patients treated with 5-FU, epirubicin and cyclophosphamide.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 1994, Volume: 2, Issue:3

    Topics: Administration, Oral; Adult; Aged; Breast Neoplasms; Constipation; Cyclophosphamide; Epirubicin; Female; Fluorouracil; Flushing; Granisetron; Headache; Humans; Injections, Intravenous; Metoclopramide; Middle Aged; Nausea; Tablets; Vomiting

1994
[Clinical effects of granisetron and methylprednisolone against nausea, vomiting and anorexia induced by cisplatin].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1993, Volume: 20, Issue:13

    Topics: Adult; Aged; Anorexia; Cisplatin; Domperidone; Drug Therapy, Combination; Female; Granisetron; Humans; Male; Methylprednisolone; Metoclopramide; Middle Aged; Mouth Neoplasms; Nausea; Vomiting

1993
Effect of metoclopramide, ondansetron and granisetron on aldosterone secretion in man.
    European journal of clinical pharmacology, 1993, Volume: 44, Issue:4

    Topics: Adult; Aldosterone; Granisetron; Humans; Indazoles; Male; Metoclopramide; Ondansetron; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Single-Blind Method

1993
The control of acute cisplatin-induced emesis--a comparative study of granisetron and a combination regimen of high-dose metoclopramide and dexamethasone. Granisetron Study Group.
    British journal of cancer, 1993, Volume: 68, Issue:1

    Topics: Blood Pressure; Cisplatin; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Nausea; Neoplasms; Pulse

1993
The antiemetic efficacy and safety of granisetron compared with metoclopramide plus dexamethasone in patients receiving fractionated chemotherapy over 5 days. The Granisetron Study Group.
    Journal of cancer research and clinical oncology, 1993, Volume: 119, Issue:9

    Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Drug Administration Schedule; Drug Therapy, Combination; Etoposide; Female; Granisetron; Humans; Ifosfamide; Indazoles; Male; Metoclopramide; Middle Aged; Vomiting

1993
Oral granisetron with or without methylprednisolone versus metoclopramide plus methylprednisolone in the management of delayed nausea and vomiting induced by cisplatin-based chemotherapy. A prospective randomized trial.
    Cancer, 1995, Nov-15, Volume: 76, Issue:10

    Topics: Administration, Oral; Adult; Aged; Antiemetics; Cisplatin; Drug Therapy, Combination; Female; Granisetron; Humans; Male; Methylprednisolone; Metoclopramide; Middle Aged; Nausea; Neoplasms; Prospective Studies; Vomiting

1995
A randomized cross-over trial of granisetron and dexamethasone versus granisetron alone: the role of dexamethasone on day 1 in the control of cisplatin-induced delayed emesis.
    Japanese journal of clinical oncology, 1996, Volume: 26, Issue:3

    Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Cisplatin; Cross-Over Studies; Dexamethasone; Drug Administration Schedule; Drug Therapy, Combination; Female; Granisetron; Humans; Lung Neoplasms; Male; Metoclopramide; Middle Aged; Single-Blind Method; Vomiting

1996
Granisetron in the prevention of vomiting induced by conditioning for stem cell transplantation: a prospective randomized study.
    Bone marrow transplantation, 1996, Volume: 17, Issue:5

    Topics: Adolescent; Adult; Antiemetics; Antineoplastic Agents; Female; Granisetron; Hematopoietic Stem Cell Transplantation; Humans; Male; Metoclopramide; Middle Aged; Prospective Studies; Safety; Serotonin Antagonists; Time Factors; Transplantation Conditioning; Vomiting; Whole-Body Irradiation

1996
Prophylactic antiemetic therapy with ondansetron, tropisetron, granisetron and metoclopramide in patients undergoing laparoscopic cholecystectomy: a randomized, double-blind comparison with placebo.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1996, Volume: 43, Issue:3

    Topics: Adult; Aged; Antiemetics; Cholecystectomy, Laparoscopic; Double-Blind Method; Female; Granisetron; Humans; Indoles; Male; Metoclopramide; Middle Aged; Nausea; Ondansetron; Postoperative Complications; Prospective Studies; Serotonin Antagonists; Tropisetron; Vomiting

1996
Antiemetic efficacy of granisetron and metoclopramide in children undergoing ophthalmic or ENT surgery.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1996, Volume: 43, Issue:11

    Topics: Adenoidectomy; Antiemetics; Child; Child, Preschool; Double-Blind Method; Granisetron; Humans; Metoclopramide; Ophthalmologic Surgical Procedures; Postoperative Complications; Tonsillectomy; Vomiting

1996
Combination effect of granisetron and methylprednisolone for preventing emesis induced by cytotoxic agents.
    Gynecologic and obstetric investigation, 1997, Volume: 43, Issue:3

    Topics: Adult; Aged; Antineoplastic Agents; Drug Therapy, Combination; Female; Granisetron; Humans; Hydroxyindoleacetic Acid; Methylprednisolone; Metoclopramide; Middle Aged; Ovarian Neoplasms; Vomiting

1997
Phase II study of high-dose dexamethasone-based association in acute and delayed high-dose cisplatin-induced emesis--JCOG study 9413.
    British journal of cancer, 1997, Volume: 76, Issue:1

    Topics: Antiemetics; Cisplatin; Dexamethasone; Female; Granisetron; Humans; Lung Neoplasms; Male; Metoclopramide; Middle Aged; Vomiting

1997
Prevention of PONV with granisetron, droperidol and metoclopramide in female patients with history of motion sickness.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1997, Volume: 44, Issue:8

    Topics: Adult; Antiemetics; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Metoclopramide; Middle Aged; Motion Sickness; Nausea; Postoperative Complications; Vomiting

1997
Prevention of nausea and vomiting in female patients undergoing breast surgery: a comparison with granisetron, droperidol, metoclopramide and placebo.
    Acta anaesthesiologica Scandinavica, 1998, Volume: 42, Issue:2

    Topics: Adult; Antiemetics; Breast Neoplasms; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Metoclopramide; Middle Aged; Nausea; Postoperative Complications; Vomiting

1998
Prevention of PONV with granisetron, droperidol or metoclopramide in patients with postoperative emesis.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1998, Volume: 45, Issue:2

    Topics: Adult; Double-Blind Method; Droperidol; Female; Gastrointestinal Agents; Granisetron; Humans; Metoclopramide; Middle Aged; Nausea; Postoperative Complications; Serotonin Antagonists; Vomiting

1998
Prophylactic therapy with granisetron in the prevention of vomiting after paediatric surgery. A randomized, double-blind comparison with droperidol and metoclopramide.
    Paediatric anaesthesia, 1998, Volume: 8, Issue:2

    Topics: Antiemetics; Child; Child, Preschool; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Intraoperative Period; Male; Metoclopramide; Postoperative Complications; Prospective Studies; Vomiting

1998
Anti-emetic efficacy of prophylactic granisetron, droperidol and metoclopramide in the prevention of nausea and vomiting after laparoscopic cholecystectomy: a randomized, double-blind, placebo-controlled trial.
    European journal of anaesthesiology, 1998, Volume: 15, Issue:2

    Topics: Adult; Aged; Antiemetics; Cholecystectomy, Laparoscopic; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Metoclopramide; Middle Aged; Nausea; Vomiting

1998
Prevention of postoperative nausea and vomiting in female patients during menstruation: comparison of droperidol, metoclopramide and granisetron.
    British journal of anaesthesia, 1998, Volume: 80, Issue:2

    Topics: Adult; Antiemetics; Double-Blind Method; Droperidol; Female; Granisetron; Gynecologic Surgical Procedures; Humans; Menstruation; Metoclopramide; Middle Aged; Nausea; Postoperative Complications; Vomiting

1998
Prevention of nausea and vomiting with granisetron, droperidol and metoclopramide during and after spinal anaesthesia for caesarean section: a randomized, double-blind, placebo-controlled trial.
    Acta anaesthesiologica Scandinavica, 1998, Volume: 42, Issue:8

    Topics: Adult; Anesthesia, Spinal; Antiemetics; Cesarean Section; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Metoclopramide; Placebos; Postoperative Nausea and Vomiting; Pregnancy

1998
Prophylactic anti-emetic therapy with granisetron, droperidol and metoclopramide in female patients undergoing middle ear surgery.
    Anaesthesia, 1998, Volume: 53, Issue:12

    Topics: Adult; Aged; Anesthesia, General; Antiemetics; Double-Blind Method; Droperidol; Ear, Middle; Female; Granisetron; Humans; Metoclopramide; Middle Aged; Postoperative Nausea and Vomiting

1998
Granisetron, droperidol, and metoclopramide for preventing postoperative nausea and vomiting after thyroidectomy.
    The Laryngoscope, 1999, Volume: 109, Issue:4

    Topics: Adult; Antiemetics; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Metoclopramide; Middle Aged; Nausea; Postoperative Complications; Prospective Studies; Thyroidectomy; Treatment Outcome; Vomiting

1999
[Comparative trial of oral granisetron and intravenous ondansetron in patients receiving chemotherapy for breast cancer. Study Group of Granisetron].
    Bulletin du cancer, 1999, Volume: 86, Issue:3

    Topics: Administration, Oral; Adult; Aged; Antiemetics; Breast Neoplasms; Drug Therapy, Combination; Female; Granisetron; Humans; Injections, Intravenous; Male; Metoclopramide; Middle Aged; Nausea; Ondansetron; Vomiting

1999
[Anti-emetic treatment for patients with non-small cell lung cancer after chemotherapy, usefulness of preventive combination of anti-emetic agents and importance of psychiatric aspect of patients].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1999, Volume: 26, Issue:6

    Topics: Adult; Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Non-Small-Cell Lung; Cisplatin; Drug Administration Schedule; Drug Therapy, Combination; Female; Granisetron; Humans; Lung Neoplasms; Male; Methylprednisolone; Metoclopramide; Middle Aged; Mitomycin; Personality; Vindesine; Vomiting, Anticipatory

1999
Granisetron, droperidol, and metoclopramide for the treatment of established postoperative nausea and vomiting in women undergoing gynecologic surgery.
    American journal of obstetrics and gynecology, 2000, Volume: 182, Issue:1 Pt 1

    Topics: Adult; Anesthesia, General; Antiemetics; Double-Blind Method; Droperidol; Female; Granisetron; Gynecologic Surgical Procedures; Humans; Metoclopramide; Middle Aged; Nausea; Postoperative Complications; Vomiting

2000
Randomized clinical trial of granisetron, droperidol and metoclopramide for the treatment of nausea and vomiting after laparoscopic cholecystectomy.
    The British journal of surgery, 2000, Volume: 87, Issue:3

    Topics: Adult; Antiemetics; Cholecystectomy, Laparoscopic; Droperidol; Female; Granisetron; Humans; Male; Metoclopramide; Middle Aged; Postoperative Nausea and Vomiting; Treatment Outcome

2000
[Anti-emetic treatment for patients with lung cancer after chemotherapy, and usefulness of prochlorperazine for psychiatric emesis].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2000, Volume: 27, Issue:3

    Topics: Aged; Antiemetics; Cisplatin; Drug Administration Schedule; Drug Evaluation; Drug Therapy, Combination; Female; Granisetron; Humans; Lung Neoplasms; Male; Methylprednisolone; Metoclopramide; Middle Aged; Prochlorperazine; Vomiting, Anticipatory

2000
Comparison of granisetron, droperidol, and metoclopramide for prevention of postoperative vomiting in children with a history of motion sickness undergoing tonsillectomy.
    Journal of pediatric surgery, 2001, Volume: 36, Issue:3

    Topics: Analysis of Variance; Antiemetics; Child, Preschool; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Infant; Injections, Intravenous; Intraoperative Care; Male; Metoclopramide; Motion Sickness; Postoperative Nausea and Vomiting; Prospective Studies; Statistics, Nonparametric; Tonsillectomy

2001
Comparative study of low-dose oral granisetron plus dexamethasone and high-dose metoclopramide plus dexamethasone in prevention of nausea and vomiting induced by CHOP-therapy in young patients with non-Hodgkin's lymphoma.
    Journal of the Medical Association of Thailand = Chotmaihet thangphaet, 2002, Volume: 85, Issue:11

    Topics: Administration, Oral; Adolescent; Adult; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Chi-Square Distribution; Cross-Over Studies; Cyclophosphamide; Dexamethasone; Dose-Response Relationship, Drug; Double-Blind Method; Doxorubicin; Drug Therapy, Combination; Female; Follow-Up Studies; Granisetron; Humans; Lymphoma, Non-Hodgkin; Male; Metoclopramide; Middle Aged; Nausea; Patient Satisfaction; Prednisone; Probability; Treatment Outcome; Vincristine; Vomiting

2002
A randomized double-blind trial to compare the clinical efficacy of granisetron with metoclopramide, both combined with dexamethasone in the prophylaxis of chemotherapy-induced delayed emesis.
    Annals of oncology : official journal of the European Society for Medical Oncology, 2003, Volume: 14, Issue:2

    Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Male; Metoclopramide; Middle Aged; Neoplasms; Vomiting

2003
A comparison of granisetron, droperidol, and metoclopramide in the treatment of established nausea and vomiting after breast surgery: a double-blind, randomized, controlled trial.
    Clinical therapeutics, 2003, Volume: 25, Issue:4

    Topics: Adult; Aged; Anesthesia, General; Antiemetics; Double-Blind Method; Droperidol; Female; Granisetron; Humans; Mastectomy; Metoclopramide; Middle Aged; Nausea; Prospective Studies; Treatment Outcome; Vomiting

2003
Contribution to the treatment of nausea and emesis induced by chemotherapy in children and adolescents with osteosarcoma.
    Sao Paulo medical journal = Revista paulista de medicina, 2006, Mar-02, Volume: 124, Issue:2

    Topics: Adolescent; Antiemetics; Antineoplastic Agents; Bone Neoplasms; Child; Dimenhydrinate; Female; Granisetron; Humans; Male; Metoclopramide; Nausea; Osteosarcoma; Prospective Studies; Vomiting

2006
Skipping day 2 antiemetic medications may improve chemotherapy induced delayed nausea and vomiting control: results of two pilot phase II trials.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 2007, Volume: 15, Issue:3

    Topics: Adolescent; Adult; Aged; Analysis of Variance; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Brazil; Dexamethasone; Drug Hypersensitivity; Female; Granisetron; Humans; Hypersensitivity, Delayed; Logistic Models; Male; Metoclopramide; Middle Aged; Nausea; Ondansetron; Pilot Projects; Quality of Life; Research Design; Serotonin Antagonists; Treatment Outcome; Vomiting

2007
Comparison of the effectiveness of metoclopramide, ondansetron, and granisetron on the prevention of nausea and vomiting after laparoscopic cholecystectomy.
    Journal of laparoendoscopic & advanced surgical techniques. Part A, 2007, Volume: 17, Issue:6

    Topics: Adult; Aged; Analysis of Variance; Antiemetics; Chi-Square Distribution; Cholecystectomy, Laparoscopic; Double-Blind Method; Female; Granisetron; Humans; Male; Metoclopramide; Middle Aged; Ondansetron; Postoperative Nausea and Vomiting; Treatment Outcome

2007
Dexamethasone with either granisetron or ondansetron for postoperative nausea and vomiting in laparoscopic surgery.
    Middle East journal of anaesthesiology, 2010, Volume: 20, Issue:4

    Topics: Adult; Antiemetics; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Laparoscopy; Male; Metoclopramide; Middle Aged; Ondansetron; Patient Satisfaction; Postoperative Nausea and Vomiting; Prospective Studies; Severity of Illness Index; Treatment Outcome

2010
Antiemetic activity of megestrol acetate in patients receiving chemotherapy.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 2011, Volume: 19, Issue:5

    Topics: Adult; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Cross-Over Studies; Drug Therapy, Combination; Female; Granisetron; Humans; Male; Megestrol; Metoclopramide; Middle Aged; Nausea; Neoplasms; Single-Blind Method; Treatment Outcome; Vomiting

2011
Can granisetron injection used as primary prophylaxis improve the control of nausea and vomiting with low- emetogenic chemotherapy?
    Asian Pacific journal of cancer prevention : APJCP, 2013, Volume: 14, Issue:1

    Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Humans; Logistic Models; Male; Metoclopramide; Middle Aged; Multivariate Analysis; Nausea; Neoplasms; Vomiting

2013
Effects of ondansetron, metoclopramide and granisetron on perioperative nausea and vomiting in patients undergone bariatric surgery: a randomized clinical trial.
    Surgical endoscopy, 2023, Volume: 37, Issue:6

    Topics: Antiemetics; Bariatric Surgery; Double-Blind Method; Granisetron; Humans; Metoclopramide; Ondansetron; Postoperative Nausea and Vomiting

2023

Other Studies

29 other study(ies) available for granisetron and metoclopramide

ArticleYear
Development of high-affinity 5-HT3 receptor antagonists. 1. Initial structure-activity relationship of novel benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Animals; Antiemetics; Benzamides; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Male; Metoclopramide; Molecular Structure; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting

1992
Neuroendocrine responses to L-tryptophan as an index of brain serotonin function: effect of weight loss.
    Advances in experimental medicine and biology, 1991, Volume: 294

    Topics: Adult; Biological Transport, Active; Brain Chemistry; Clomipramine; Depression; Diet, Reducing; Female; Granisetron; Growth Hormone; Humans; Hydroxyindoleacetic Acid; Indazoles; Infusions, Intravenous; Male; Metergoline; Metoclopramide; Neurosecretory Systems; Prolactin; Ritanserin; Serotonin; Sex Characteristics; Synaptic Transmission; Thyrotropin-Releasing Hormone; Tryptophan; Tryptophan Hydroxylase; Weight Loss

1991
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
Emesis and defecations induced by the 5-hydroxytryptamine (5-HT3) receptor antagonist zacopride in the ferret.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Administration, Oral; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Defecation; Dose-Response Relationship, Drug; Ferrets; Granisetron; Indazoles; Injections, Intravenous; Male; Metoclopramide; Pyrazoles; Serotonin; Serotonin Antagonists; Vagotomy; Vomiting

1990
Analysis of the actions of 5-hydroxytryptamine on the rabbit isolated vagus nerve.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:6

    Topics: Action Potentials; Animals; Biguanides; Citalopram; Electric Stimulation; Evoked Potentials; Female; gamma-Aminobutyric Acid; Granisetron; Indazoles; Male; Membrane Potentials; Metoclopramide; Motor Neurons; Rabbits; Serotonin; Vagus Nerve

1990
Antagonism of the effects of 5-hydroxytryptamine on the rabbit isolated vagus nerve by BRL 43694 and metoclopramide.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:6

    Topics: Action Potentials; Animals; Dimethylphenylpiperazinium Iodide; Female; gamma-Aminobutyric Acid; Granisetron; In Vitro Techniques; Indazoles; Kinetics; Male; Metoclopramide; Pyrazoles; Rabbits; Serotonin; Serotonin Antagonists; Vagus Nerve

1990
The effects of orally administered Y-25130, a selective serotonin3-receptor antagonist, on chemotherapeutic agent-induced emesis.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:3

    Topics: Administration, Oral; Animals; Antiemetics; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Cyclophosphamide; Dogs; Domperidone; Dose-Response Relationship, Drug; Doxorubicin; Female; Ferrets; Granisetron; Male; Metoclopramide; Ondansetron; Oxazines; Serotonin Antagonists; Vomiting

1993
The effects of different antiemetic agents on morphine-induced emesis in ferrets.
    European journal of pharmacology, 1993, Sep-07, Volume: 241, Issue:1

    Topics: Anesthesia; Animals; Antiemetics; Droperidol; Ferrets; Granisetron; Injections, Intravenous; Isoflurane; Male; Metoclopramide; Morphine; Naloxone; Ondansetron; Vomiting

1993
Comparison of intravenous granisetron with metoclopramide plus dexamethasone in the prevention of nausea and vomiting associated with emetogenic cytotoxic chemotherapy.
    The Kaohsiung journal of medical sciences, 1997, Volume: 13, Issue:2

    Topics: Adult; Aged; Antineoplastic Agents; Dexamethasone; Female; Granisetron; Humans; Injections, Intravenous; Male; Metoclopramide; Middle Aged; Nausea; Neoplasms; Vomiting

1997
An audit of antiemetic use with CMF chemotherapy.
    Clinical oncology (Royal College of Radiologists (Great Britain)), 1998, Volume: 10, Issue:5

    Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cyclophosphamide; Dexamethasone; Drug Therapy, Combination; Female; Fluorouracil; Granisetron; Humans; Medical Records; Methotrexate; Metoclopramide; Retrospective Studies; Serotonin Antagonists; Treatment Outcome; Vomiting

1998
5-HT3 receptor-channels coupled with Na+ influx in human T cells: role in T cell activation.
    Journal of neuroimmunology, 1999, Sep-01, Volume: 99, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Calcium Signaling; Cell Cycle; Enzyme Activation; Granisetron; Humans; Ion Channel Gating; Ion Transport; Jurkat Cells; Lymphocyte Activation; Metoclopramide; Neoplasm Proteins; Phytohemagglutinins; Piperazines; Protein Kinase C; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Ryanodine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium; Sodium Channels; T-Lymphocytes; Thapsigargin

1999
Effect of different prokinetic agents and a novel enterokinetic agent on postoperative ileus in rats.
    Gut, 1999, Volume: 45, Issue:5

    Topics: Animals; Cisapride; Dopamine Antagonists; Erythromycin; Gastrointestinal Agents; Granisetron; Intestinal Obstruction; Male; Metoclopramide; Postoperative Complications; Random Allocation; Rats; Rats, Wistar; Serotonin Antagonists

1999
[Relationship between neurotransmitter blood noradrenalin and nausea/emesis after chemotherapy for lung cancer].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2006, Volume: 33, Issue:7

    Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Catecholamines; Cisplatin; Docetaxel; Drug Administration Schedule; Drug Therapy, Combination; Granisetron; Humans; Lung Neoplasms; Methylprednisolone; Metoclopramide; Nausea; Neurotransmitter Agents; Norepinephrine; Serotonin; Taxoids; Vomiting, Anticipatory

2006
[Successful antiemetic treatment of TSUMURA Rikkunshi-to Extract Granules for ethical use in addition to other antiemetic agents in neoadjuvant chemotherapy for an advanced breast cancer patient].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2006, Volume: 33, Issue:8

    Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Chemotherapy, Adjuvant; Cyclophosphamide; Dexamethasone; Drug Administration Schedule; Drugs, Chinese Herbal; Epirubicin; Female; Fluorouracil; Granisetron; Humans; Lymph Nodes; Lymphatic Metastasis; Mastectomy, Segmental; Metoclopramide; Middle Aged

2006
[Comparison of granisetron and metoclopramide for prevention of nausea and vomiting following total cystectomy and ileal conduit].
    Acta chirurgica Iugoslavica, 2007, Volume: 54, Issue:2

    Topics: Antiemetics; Cystectomy; Granisetron; Humans; Metoclopramide; Middle Aged; Postoperative Nausea and Vomiting; Urinary Diversion

2007
Is there an association between PONV and chemotherapy-induced nausea and vomiting?
    Acta anaesthesiologica Scandinavica, 2013, Volume: 57, Issue:6

    Topics: Adult; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Betamethasone; Breast Neoplasms; Chemotherapy, Adjuvant; Combined Modality Therapy; Cyclophosphamide; Disease Resistance; Droperidol; Epirubicin; Female; Fluorouracil; Granisetron; Humans; Mastectomy; Methotrexate; Metoclopramide; Middle Aged; Models, Biological; Narcotics; Nausea; Ondansetron; Postoperative Nausea and Vomiting; Prospective Studies; Risk Factors; Vomiting

2013
Cost-effectiveness analysis of granisetron-based versus standard antiemetic regimens in low-emetogenic chemotherapy: a hospital-based perspective from Malaysia.
    Asian Pacific journal of cancer prevention : APJCP, 2013, Volume: 14, Issue:12

    Topics: Antiemetics; Antineoplastic Agents; Cost-Benefit Analysis; Dexamethasone; Drug Therapy, Combination; Follow-Up Studies; Granisetron; Humans; Malaysia; Metoclopramide; Nausea; Neoplasms; Prognosis; Retrospective Studies; Vomiting

2013
Controlled transdermal iontophoresis for poly-pharmacotherapy: Simultaneous delivery of granisetron, metoclopramide and dexamethasone sodium phosphate in vitro and in vivo.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2016, Mar-31, Volume: 85

    Topics: Administration, Cutaneous; Animals; Dexamethasone; Granisetron; Hydrolysis; Iontophoresis; Male; Metoclopramide; Polypharmacy; Rats; Rats, Wistar; Skin; Swine

2016
The effect of anti-emetic drugs on rat embryonic heart activity.
    Reproductive toxicology (Elmsford, N.Y.), 2019, Volume: 87

    Topics: Animals; Antiemetics; Bradycardia; Domperidone; Droperidol; Embryo, Mammalian; Granisetron; Heart; Heart Rate; Meclizine; Metoclopramide; Rats, Sprague-Dawley; Trifluoperazine

2019
Potential drug-drug Interactions in hospitalized cancer patients: A report from the Middle-East.
    Journal of oncology pharmacy practice : official publication of the International Society of Oncology Pharmacy Practitioners, 2021, Volume: 27, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Cross-Sectional Studies; Dopamine Antagonists; Drug Interactions; Female; Granisetron; Hospitals, University; Humans; Inpatients; Iran; Male; Metoclopramide; Middle Aged; Middle East; Neoplasms; Retrospective Studies; Serotonin Antagonists; Young Adult

2021
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction

1992
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes

1990
Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Binding Sites; Guinea Pigs; Mice; Protein Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1990
5-HT3 antagonists derived from aminopyridazine-type muscarinic M1 agonists.
    Journal of medicinal chemistry, 1998, Jan-29, Volume: 41, Issue:3

    Topics: Animals; Brain Stem; Hippocampus; In Vitro Techniques; Models, Molecular; Muscarinic Agonists; Myocardium; Protein Conformation; Pyridazines; Rats; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists

1998
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010