granisetron and fomesafen

granisetron has been researched along with fomesafen in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (76.92)18.2507
2000's3 (23.08)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Choudry, NB; Fuller, RW; Lavender, EA; McEwan, JR; Williams, AJ1
Moss, HE; Sanger, GJ1
Buéno, L; Gué, M; Junien, JL1
Daniels, S; Eglen, RM; Fontana, DJ; Khabbaz, M; Kilfoil, T; Lee, CH; Wong, EH1
Ichikawa, S; Ishii, A; Karasawa, A; Kishibayashi, N; Yokoyama, T1
Bueno, L; Camman, F; Delvaux, M; Fioramonti, J; Frexinos, J; Louvel, D; Staumont, G1
Kawakita, T; Kuroita, T; Sakamori, M1
Inaba, K; Kanzaki, K; Kawakita, T; Kuroita, T; Marubayashi, N; Sano, M1
Futuro-Neto, HA; Pires, JG; Ramage, AG; Silva, SR1
Björnsson, ES; Chey, WD; Hasler, WL; Hooper, FG; Ladabaum, U; Owyang, C; Woods, ML1
Alonso-Cires, L; Innerárity, A; Labeaga, L; López-Tudanca, PL; Mosquera, R; Orjales, A; Tapia, I1
Machado, BH; Weissheimer, KV1
Bernard, JF; Hamon, M; Laguzzi, R; Mandjee, N; Netzer, F; Sévoz-Couche, C; Verberne, AJ1

Trials

2 trial(s) available for granisetron and fomesafen

ArticleYear
Human responses to inhaled capsaicin are not inhibited by granisetron.
    British journal of clinical pharmacology, 1991, Volume: 31, Issue:3

    Topics: Administration, Inhalation; Adult; Airway Resistance; Capsaicin; Cough; Granisetron; Humans; Indazoles; Male; Reflex; Serotonin Antagonists

1991
Intracolonic injection of glycerol: a model for abdominal pain in irritable bowel syndrome?
    Gastroenterology, 1996, Volume: 110, Issue:2

    Topics: Abdominal Pain; Adult; Aged; Colon; Colonic Diseases, Functional; Electromyography; Female; Gastrointestinal Agents; Gastrointestinal Motility; Glycerol; Granisetron; Humans; Injections; Male; Middle Aged; Models, Biological; Muscle Contraction; Muscle, Smooth; Octreotide; Parasympatholytics; Phloroglucinol; Reflex; Reproducibility of Results; Serotonin Antagonists

1996

Other Studies

11 other study(ies) available for granisetron and fomesafen

ArticleYear
The effects of granisetron, ICS 205-930 and ondansetron on the visceral pain reflex induced by duodenal distension.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Blood Pressure; Duodenum; Granisetron; Imidazoles; Indazoles; Indoles; Male; Morphine; Muscle Contraction; Muscle, Smooth; Ondansetron; Pain; Pyrazoles; Rats; Rats, Inbred Strains; Reflex; Serotonin Antagonists; Stomach; Tropisetron; Vagotomy

1990
The kappa agonist fedotozine modulates colonic distention-induced inhibition of gastric motility and emptying in dogs.
    Gastroenterology, 1994, Volume: 107, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzyl Compounds; Bretylium Compounds; Catheterization; Colon; Dogs; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Gastric Emptying; Gastrointestinal Motility; Granisetron; Hexamethonium; Male; Naltrexone; Narcotic Antagonists; Propylamines; Pyrrolidines; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reflex; Stomach

1994
Comparison of potencies of 5-HT3 receptor antagonists at inhibiting aversive behavior to illumination and the von Bezold-Jarisch reflex in the mouse.
    Neuropharmacology, 1994, Volume: 33, Issue:2

    Topics: Animals; Behavior, Animal; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Granisetron; Heart Rate; Lighting; Mice; Motor Activity; Ondansetron; Reflex; Serotonin Antagonists; Stereoisomerism

1994
Pharmacological properties of KF18259, a novel 5-HT3-receptor antagonist, in rats: inhibition of the distal colonic function.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:4

    Topics: Animals; Benzimidazoles; Cisplatin; Colon; Defecation; Gastric Emptying; Gastrointestinal Motility; Granisetron; Male; Ondansetron; Quinolines; Rats; Rats, Sprague-Dawley; Reflex; Serotonin; Serotonin Antagonists

1993
Design and synthesis of 6-chloro-3,4-dihydro-4-methyl-2H-1,4-benzoxazine-8-carboxamide derivatives as potent serotonin-3 (5-HT3) receptor antagonists.
    Chemical & pharmaceutical bulletin, 1996, Volume: 44, Issue:4

    Topics: Animals; Benzamides; Binding, Competitive; Blood Pressure; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Granisetron; Heart Rate; In Vitro Techniques; Male; Oxazines; Rats; Receptors, Serotonin; Reflex; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

1996
Benzoxazines. II. Synthesis, conformational analysis, and structure--activity relationships of 3,4-dihydro-2H-1,4-benzoxazine-8-carboxamide derivatives as potent and long-acting serotonin-3 (5-HT3) receptor antagonists.
    Chemical & pharmaceutical bulletin, 1996, Volume: 44, Issue:11

    Topics: Amides; Animals; Brain Chemistry; Granisetron; Hemodynamics; Magnetic Resonance Spectroscopy; Male; Molecular Conformation; Oxazines; Rats; Rats, Wistar; Receptors, Serotonin; Reflex; Serotonin Antagonists; Structure-Activity Relationship

1996
Evidence that 5-HT3 receptors in the nucleus tractus solitarius and other brainstem areas modulate the vagal bradycardia evoked by activation of the von Bezold-Jarisch reflex in the anesthetized rat.
    Brain research, 1998, Apr-27, Volume: 791, Issue:1-2

    Topics: Anesthetics; Animals; Biguanides; Bradycardia; Brain Stem; Cisterna Magna; Granisetron; Injections; Male; Rats; Rats, Wistar; Receptors, Serotonin; Reflex; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Vagus Nerve

1998
Differential 5-HT3 mediation of human gastrocolonic response and colonic peristaltic reflex.
    The American journal of physiology, 1998, Volume: 275, Issue:3

    Topics: Adult; Colon; Dilatation; Double-Blind Method; Duodenum; Female; Granisetron; Humans; Male; Mechanoreceptors; Middle Aged; Muscle Tonus; Muscle, Smooth; Peristalsis; Pressure; Pyloric Antrum; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Reflex; Stomach

1998
Synthesis and pharmacological characterization of a new benzoxazole derivative as a potent 5-HT3 receptor agonist.
    Bioorganic & medicinal chemistry, 2003, Jul-03, Volume: 11, Issue:13

    Topics: Animals; Benzoxazoles; Dose-Response Relationship, Drug; Drug Antagonism; Granisetron; Radioligand Assay; Rats; Rats, Wistar; Reflex; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tachyphylaxis

2003
Inhibitory modulation of chemoreflex bradycardia by stimulation of the nucleus raphe obscurus is mediated by 5-HT3 receptors in the NTS of awake rats.
    Autonomic neuroscience : basic & clinical, 2007, Mar-30, Volume: 132, Issue:1-2

    Topics: Animals; Blood Pressure; Bradycardia; Chemoreceptor Cells; Consciousness; Glutamic Acid; Granisetron; Heart; Heart Rate; Injections, Intraventricular; Male; Microinjections; Neural Pathways; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Reflex; Serotonin Antagonists; Solitary Nucleus

2007
Inhibition of the bradycardic component of the von Bezold-Jarisch reflex and carotid chemoreceptor reflex by periaqueductal gray stimulation: involvement of medullary receptors.
    The European journal of neuroscience, 2009, Volume: 29, Issue:10

    Topics: Animals; Bicuculline; Biguanides; Bradycardia; Carotid Arteries; Chemoreceptor Cells; GABA Antagonists; Granisetron; Immunohistochemistry; Male; Microinjections; Parasympathetic Nervous System; Periaqueductal Gray; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Neurokinin-1; Receptors, Serotonin, 5-HT3; Reflex; Serotonin Agents; Solitary Nucleus; Sympathetic Nervous System; Tetrazoles

2009