granisetron and bemesetron

granisetron has been researched along with bemesetron in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's11 (84.62)18.2507
2000's2 (15.38)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1
Gandara, DR; Hesketh, PJ1
Chen, HI1
Futuro-Neto, HA; Pires, JG; Silva, SR1
Allison, K; Arnold, B; Greenshaw, AJ; Ivanová, S; Paetsch, PR; Paslawski, T1
Maksay, G1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Hensler, JG; Hodge, CW; Overstreet, DH1
Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD1
Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT1
Carr, AA; Hibert, MF; Hoffmann, R; Miller, RC1
Bermudez, J; Fake, CS; Joiner, GF; Joiner, KA; King, FD; Miner, WD; Sanger, GJ1
Bourguignon, JJ; Didier, B; Hoffmann, R; Rival, Y; Rybaltchenko, V; Wermuth, CG1

Other Studies

13 other study(ies) available for granisetron and bemesetron

ArticleYear
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
Evidence for the presynaptic action of 5-hydroxytryptamine and the involvement of purinergic innervation in the rabbit lower urinary tract.
    British journal of pharmacology, 1990, Volume: 101, Issue:1

    Topics: Adenosine Triphosphate; Animals; Atropine; Electric Stimulation; Female; Granisetron; In Vitro Techniques; Indazoles; Indoles; Male; Muscle Contraction; Muscle, Smooth; Purines; Rabbits; Serotonin; Serotonin Antagonists; Synapses; Tropanes; Tropisetron; Urethra; Urinary Tract

1990
Effects of 5-HT3 receptor antagonists on neuroleptic-induced catalepsy in mice.
    Neuropharmacology, 1995, Volume: 34, Issue:1

    Topics: Animals; Catalepsy; Granisetron; Haloperidol; Mice; Serotonin Antagonists; Time Factors; Tropanes

1995
5HT3 receptor antagonists do not block nicotine induced hyperactivity in rats.
    Psychopharmacology, 1995, Volume: 119, Issue:2

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Granisetron; Haloperidol; Indoles; Male; Motor Activity; Nicotine; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Time Factors; Tropanes; Tropisetron

1995
Bidirectional allosteric modulation of strychnine-sensitive glycine receptors by tropeines and 5-HT3 serotonin receptor ligands.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: Allosteric Regulation; Animals; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Glycine; Granisetron; Indoles; Ligands; Male; Medulla Oblongata; Ondansetron; Pons; Rats; Rats, Wistar; Receptors, Glycine; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Strychnine; Tropanes; Tropisetron; Tubocurarine

1998
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
Reduced 5-HT3 receptor binding and lower baseline plus maze anxiety in the alcohol-preferring inbred fawn-hooded rat.
    Pharmacology, biochemistry, and behavior, 2004, Volume: 77, Issue:2

    Topics: Alcohol Drinking; Animals; Anxiety; Autoradiography; Brain Chemistry; Cerebral Cortex; Granisetron; Image Processing, Computer-Assisted; Limbic System; Male; Radioligand Assay; Rats; Rats, Inbred ACI; Rats, Inbred Strains; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Species Specificity; Tropanes

2004
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction

1992
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes

1990
Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Binding Sites; Guinea Pigs; Mice; Protein Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1990
5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:7

    Topics: Animals; Antiemetics; Carboxylic Acids; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Indicators and Reagents; Indolizines; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Muscle Contraction; Muscle, Smooth; Pyrazoles; Rats; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

1990
5-HT3 antagonists derived from aminopyridazine-type muscarinic M1 agonists.
    Journal of medicinal chemistry, 1998, Jan-29, Volume: 41, Issue:3

    Topics: Animals; Brain Stem; Hippocampus; In Vitro Techniques; Models, Molecular; Muscarinic Agonists; Myocardium; Protein Conformation; Pyridazines; Rats; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists

1998