gr 73632 has been researched along with neurokinin a in 22 studies
Studies (gr 73632) | Trials (gr 73632) | Recent Studies (post-2010) (gr 73632) | Studies (neurokinin a) | Trials (neurokinin a) | Recent Studies (post-2010) (neurokinin a) |
---|---|---|---|---|---|
77 | 1 | 9 | 1,765 | 34 | 91 |
Protein | Taxonomy | gr 73632 (IC50) | neurokinin a (IC50) |
---|---|---|---|
Substance-K receptor | Homo sapiens (human) | 0.0017 | |
Neuromedin-K receptor | Homo sapiens (human) | 0.045 | |
Substance-K receptor | Mesocricetus auratus (golden hamster) | 0.001 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 17 (77.27) | 18.2507 |
2000's | 4 (18.18) | 29.6817 |
2010's | 1 (4.55) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Clark, D; Elliott, PJ; Hagan, RM; Overton, P | 1 |
Ball, DI; Coleman, RA; Sheldrick, RL | 1 |
Hall, JM; Mitchell, D; Morton, IK | 1 |
Elliott, PJ; Hagan, RM; Mason, GS; Stephens-Smith, M | 1 |
Beresford, IJ; Deal, MJ; Hagan, RM; Ireland, SJ; Jordan, CC; Ward, P | 1 |
Hall, JM; Morton, IK | 1 |
Bristow, LJ; Young, L | 1 |
Buéno, L; Julia, V; Morteau, O | 1 |
Beattie, DT; Connor, HE; Feniuk, W; Stubbs, CM | 1 |
Dray, A; Maggi, CA; Nagy, I; Urban, L; Woolf, CJ | 1 |
Barker, R; Dunnett, S; Fawcett, J | 1 |
Dalforno, G; Gaviraghi, G; Hagan, RM; Palea, S; Pietra, C; Trist, DG | 1 |
Beattie, DT; Connor, HE; McNeil, DK | 1 |
Honda, K; Kamiya, H; Nakayama, Y; Saigo, A; Saito, R; Takano, Y | 1 |
Beresford, IJ; Hagan, RM; Hawcock, AB; Marshall, FH | 1 |
Burkholder, TP; Kehne, JH; Knippenberg, RW; Kudlacz, EM; McCloskey, TC; Shatzer, SA | 1 |
Cody, C; Jones, RS; Maubach, KA | 1 |
Holzer, P; Shahbazian, A | 1 |
Greenwood-Van Meerveld, B; Venkova, K | 1 |
Adolfsson, R; Ahlstedt, I; de Verdier, J; Drmota, T; Engberg, S; Johansson, A; Jussila, R; Kristensson, E; Leffler, A; Lindström, E; Novén, A; Påhlman, I; Sigfridsson, K; Sundqvist, M; von Mentzer, B | 1 |
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T | 1 |
Navarro, VM; Ohkura, S; Okamura, H; Wakabayashi, Y; Yamamura, T | 1 |
22 other study(ies) available for gr 73632 and neurokinin a
Article | Year |
---|---|
Neurokinin agonists differentially affect A9 and A10 dopamine cells in the rat.
Topics: Animals; Dopamine; Neurokinin A; Neurons; Peptide Fragments; Rats; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Substantia Nigra; Tegmentum Mesencephali | 1992 |
Characterisation of the neurokinin receptors mediating contraction of isolated tracheal preparations from a variety of species.
Topics: Animals; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Neurokinin B; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Neurotransmitter; Substance P; Swine; Trachea | 1990 |
Neurokinin receptors in the rabbit iris sphincter characterised by novel agonist ligands.
Topics: Animals; In Vitro Techniques; Iris; Kinetics; Ligands; Male; Neurokinin A; Peptide Fragments; Rabbits; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P | 1991 |
Behavioural and biochemical responses following activation of midbrain dopamine pathways by receptor selective neurokinin agonists.
Topics: Amino Acid Sequence; Animals; Chromatography, High Pressure Liquid; Dopamine; Haloperidol; Limbic System; Male; Mesencephalon; Molecular Sequence Data; Motor Activity; Neural Pathways; Neurokinin A; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Substantia Nigra; Tegmentum Mesencephali | 1991 |
Receptor-selective, peptidase-resistant agonists at neurokinin NK-1 and NK-2 receptors: new tools for investigating neurokinin function.
Topics: Administration, Cutaneous; Amino Acid Sequence; Animals; Bronchoconstriction; Capillary Permeability; Chromatography, High Pressure Liquid; Guinea Pigs; Male; Molecular Sequence Data; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Trachea | 1991 |
Novel ligands confirm NK-1 receptor-mediated modulation of neurotransmission in the guinea pig vas deferens preparation.
Topics: Animals; Electric Stimulation; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Synaptic Transmission; Vas Deferens | 1991 |
Chromodacryorrhea and repetitive hind paw tapping: models of peripheral and central tachykinin NK1 receptor activation in gerbils.
Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Synergism; Gerbillinae; Harderian Gland; Indoles; Injections, Intravenous; Injections, Intraventricular; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Substance P | 1994 |
Involvement of neurokinin 1 and 2 receptors in viscerosensitive response to rectal distension in rats.
Topics: Abdomen; Animals; Benzamides; Biphenyl Compounds; Colon; Colonic Diseases, Functional; Gastrointestinal Motility; Hypnotics and Sedatives; Indoles; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Rectum; Substance P; Tachykinins | 1994 |
Neurokinin-induced changes in pial artery diameter in the anaesthetized guinea-pig.
Topics: Animals; Arteries; Calcitonin Gene-Related Peptide; Guinea Pigs; Male; Neurokinin A; Peptide Fragments; Physalaemin; Pia Mater; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Vasodilation | 1993 |
The role of neurokinin and N-methyl-D-aspartate receptors in synaptic transmission from capsaicin-sensitive primary afferents in the rat spinal cord in vitro.
Topics: 2-Amino-5-phosphonovalerate; Afferent Pathways; Animals; Biphenyl Compounds; Capsaicin; Ganglia, Spinal; In Vitro Techniques; Membrane Potentials; N-Methylaspartate; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Spinal Cord; Substance P; Synapses; Synaptic Transmission | 1993 |
A selective tachykinin receptor agonist promotes differentiation but not survival of rat chromaffin cells in vitro.
Topics: Adrenal Glands; Animals; Cell Differentiation; Cell Survival; Chromaffin System; Fluorescent Antibody Technique; Hexamethonium Compounds; Immunohistochemistry; In Vitro Techniques; Nerve Growth Factors; Neurites; Neurokinin A; Peptide Fragments; Phenotype; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tyrosine 3-Monooxygenase | 1993 |
Further studies on the effects of selective neurokinin agonists upon the activation of micturition reflex in rats. Evidence for a dual NK-1 receptor mediated excitatory and inhibitory activity.
Topics: Animals; Dose-Response Relationship, Drug; Injections, Intra-Arterial; Injections, Intraventricular; Male; Neurokinin A; Peptide Fragments; Physalaemin; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Reflex; Substance P; Urinary Bladder; Urination | 1993 |
The influence of neurokinins and calcitonin gene-related peptide on cerebral blood flow in anaesthetized guinea-pigs.
Topics: Anesthesia; Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Cerebrovascular Circulation; Guinea Pigs; Kinetics; Male; Neurokinin A; Peptide Fragments; Substance P | 1993 |
Role of NK-1 receptor in central cardiovascular regulation in rats: studies on a novel non-peptide antagonist, CP-96,345, of substance P NK-1 receptor.
Topics: Animals; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Heart Rate; Hypnotics and Sedatives; Injections, Intraventricular; Male; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Receptors, Neurokinin-1; Substance P; Tachykinins; Vas Deferens | 1993 |
Temperature and agonist dependency of tachykinin NK1 receptor antagonist potencies in rat isolated superior cervical ganglion.
Topics: Animals; In Vitro Techniques; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Receptors, Neurokinin-1; Substance P; Superior Cervical Ganglion; Temperature; Tetrodotoxin | 1995 |
The peripheral NK-1/NK-2 receptor antagonist MDL 105,172A inhibits tachykinin-mediated respiratory effects in guinea-pigs.
Topics: Animals; Behavior, Animal; Capillary Permeability; Gerbillinae; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Male; Morpholines; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Plethysmography, Whole Body; Radioligand Assay; Receptors, Neurokinin-2; Respiratory Mechanics; Substance P; Tachykinins | 1997 |
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins | 1998 |
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin | 2000 |
Effects of TAK-637 on NK(1) receptor-mediated mechanisms regulating colonic secretion.
Topics: Animals; Capsaicin; Colforsin; Colon; Electric Stimulation; Electrophysiology; Guinea Pigs; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Male; Naphthyridines; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Statistics, Nonparametric; Substance P; Tetrodotoxin | 2004 |
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists.
Topics: Animals; Autoradiography; Behavior, Animal; Brain; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Foot; Gerbillinae; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P | 2007 |
Neurokinin receptor modulation of respiratory activity in the rabbit.
Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy | 2008 |
Effects of intravenous administration of neurokinin receptor subtype-selective agonists on gonadotropin-releasing hormone pulse generator activity and luteinizing hormone secretion in goats.
Topics: Animals; Estradiol; Female; Goats; Gonadotropin-Releasing Hormone; Infusions, Intravenous; Kisspeptins; Ligands; Luteinizing Hormone; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Signal Transduction; Substance P; Time Factors | 2015 |