Page last updated: 2024-09-03

gr 73632 and neurokinin a

gr 73632 has been researched along with neurokinin a in 22 studies

Compound Research Comparison

Studies
(gr 73632)
Trials
(gr 73632)
Recent Studies (post-2010)
(gr 73632)
Studies
(neurokinin a)
Trials
(neurokinin a)
Recent Studies (post-2010) (neurokinin a)
77191,7653491

Protein Interaction Comparison

ProteinTaxonomygr 73632 (IC50)neurokinin a (IC50)
Substance-K receptorHomo sapiens (human)0.0017
Neuromedin-K receptorHomo sapiens (human)0.045
Substance-K receptorMesocricetus auratus (golden hamster)0.001

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's17 (77.27)18.2507
2000's4 (18.18)29.6817
2010's1 (4.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clark, D; Elliott, PJ; Hagan, RM; Overton, P1
Ball, DI; Coleman, RA; Sheldrick, RL1
Hall, JM; Mitchell, D; Morton, IK1
Elliott, PJ; Hagan, RM; Mason, GS; Stephens-Smith, M1
Beresford, IJ; Deal, MJ; Hagan, RM; Ireland, SJ; Jordan, CC; Ward, P1
Hall, JM; Morton, IK1
Bristow, LJ; Young, L1
Buéno, L; Julia, V; Morteau, O1
Beattie, DT; Connor, HE; Feniuk, W; Stubbs, CM1
Dray, A; Maggi, CA; Nagy, I; Urban, L; Woolf, CJ1
Barker, R; Dunnett, S; Fawcett, J1
Dalforno, G; Gaviraghi, G; Hagan, RM; Palea, S; Pietra, C; Trist, DG1
Beattie, DT; Connor, HE; McNeil, DK1
Honda, K; Kamiya, H; Nakayama, Y; Saigo, A; Saito, R; Takano, Y1
Beresford, IJ; Hagan, RM; Hawcock, AB; Marshall, FH1
Burkholder, TP; Kehne, JH; Knippenberg, RW; Kudlacz, EM; McCloskey, TC; Shatzer, SA1
Cody, C; Jones, RS; Maubach, KA1
Holzer, P; Shahbazian, A1
Greenwood-Van Meerveld, B; Venkova, K1
Adolfsson, R; Ahlstedt, I; de Verdier, J; Drmota, T; Engberg, S; Johansson, A; Jussila, R; Kristensson, E; Leffler, A; Lindström, E; Novén, A; Påhlman, I; Sigfridsson, K; Sundqvist, M; von Mentzer, B1
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T1
Navarro, VM; Ohkura, S; Okamura, H; Wakabayashi, Y; Yamamura, T1

Other Studies

22 other study(ies) available for gr 73632 and neurokinin a

ArticleYear
Neurokinin agonists differentially affect A9 and A10 dopamine cells in the rat.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: Animals; Dopamine; Neurokinin A; Neurons; Peptide Fragments; Rats; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Substantia Nigra; Tegmentum Mesencephali

1992
Characterisation of the neurokinin receptors mediating contraction of isolated tracheal preparations from a variety of species.
    Agents and actions. Supplements, 1990, Volume: 31

    Topics: Animals; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Neurokinin B; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Neurotransmitter; Substance P; Swine; Trachea

1990
Neurokinin receptors in the rabbit iris sphincter characterised by novel agonist ligands.
    European journal of pharmacology, 1991, Jun-18, Volume: 199, Issue:1

    Topics: Animals; In Vitro Techniques; Iris; Kinetics; Ligands; Male; Neurokinin A; Peptide Fragments; Rabbits; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P

1991
Behavioural and biochemical responses following activation of midbrain dopamine pathways by receptor selective neurokinin agonists.
    Neuropeptides, 1991, Volume: 19, Issue:2

    Topics: Amino Acid Sequence; Animals; Chromatography, High Pressure Liquid; Dopamine; Haloperidol; Limbic System; Male; Mesencephalon; Molecular Sequence Data; Motor Activity; Neural Pathways; Neurokinin A; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Substantia Nigra; Tegmentum Mesencephali

1991
Receptor-selective, peptidase-resistant agonists at neurokinin NK-1 and NK-2 receptors: new tools for investigating neurokinin function.
    Neuropeptides, 1991, Volume: 19, Issue:2

    Topics: Administration, Cutaneous; Amino Acid Sequence; Animals; Bronchoconstriction; Capillary Permeability; Chromatography, High Pressure Liquid; Guinea Pigs; Male; Molecular Sequence Data; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Trachea

1991
Novel ligands confirm NK-1 receptor-mediated modulation of neurotransmission in the guinea pig vas deferens preparation.
    Annals of the New York Academy of Sciences, 1991, Volume: 632

    Topics: Animals; Electric Stimulation; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Synaptic Transmission; Vas Deferens

1991
Chromodacryorrhea and repetitive hind paw tapping: models of peripheral and central tachykinin NK1 receptor activation in gerbils.
    European journal of pharmacology, 1994, Mar-03, Volume: 253, Issue:3

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Synergism; Gerbillinae; Harderian Gland; Indoles; Injections, Intravenous; Injections, Intraventricular; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Substance P

1994
Involvement of neurokinin 1 and 2 receptors in viscerosensitive response to rectal distension in rats.
    Gastroenterology, 1994, Volume: 107, Issue:1

    Topics: Abdomen; Animals; Benzamides; Biphenyl Compounds; Colon; Colonic Diseases, Functional; Gastrointestinal Motility; Hypnotics and Sedatives; Indoles; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Rectum; Substance P; Tachykinins

1994
Neurokinin-induced changes in pial artery diameter in the anaesthetized guinea-pig.
    British journal of pharmacology, 1993, Volume: 108, Issue:1

    Topics: Animals; Arteries; Calcitonin Gene-Related Peptide; Guinea Pigs; Male; Neurokinin A; Peptide Fragments; Physalaemin; Pia Mater; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Vasodilation

1993
The role of neurokinin and N-methyl-D-aspartate receptors in synaptic transmission from capsaicin-sensitive primary afferents in the rat spinal cord in vitro.
    Neuroscience, 1993, Volume: 52, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Afferent Pathways; Animals; Biphenyl Compounds; Capsaicin; Ganglia, Spinal; In Vitro Techniques; Membrane Potentials; N-Methylaspartate; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Spinal Cord; Substance P; Synapses; Synaptic Transmission

1993
A selective tachykinin receptor agonist promotes differentiation but not survival of rat chromaffin cells in vitro.
    Experimental brain research, 1993, Volume: 92, Issue:3

    Topics: Adrenal Glands; Animals; Cell Differentiation; Cell Survival; Chromaffin System; Fluorescent Antibody Technique; Hexamethonium Compounds; Immunohistochemistry; In Vitro Techniques; Nerve Growth Factors; Neurites; Neurokinin A; Peptide Fragments; Phenotype; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tyrosine 3-Monooxygenase

1993
Further studies on the effects of selective neurokinin agonists upon the activation of micturition reflex in rats. Evidence for a dual NK-1 receptor mediated excitatory and inhibitory activity.
    Neuropeptides, 1993, Volume: 24, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Injections, Intra-Arterial; Injections, Intraventricular; Male; Neurokinin A; Peptide Fragments; Physalaemin; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Reflex; Substance P; Urinary Bladder; Urination

1993
The influence of neurokinins and calcitonin gene-related peptide on cerebral blood flow in anaesthetized guinea-pigs.
    Neuropeptides, 1993, Volume: 24, Issue:6

    Topics: Anesthesia; Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Cerebrovascular Circulation; Guinea Pigs; Kinetics; Male; Neurokinin A; Peptide Fragments; Substance P

1993
Role of NK-1 receptor in central cardiovascular regulation in rats: studies on a novel non-peptide antagonist, CP-96,345, of substance P NK-1 receptor.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Heart Rate; Hypnotics and Sedatives; Injections, Intraventricular; Male; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Receptors, Neurokinin-1; Substance P; Tachykinins; Vas Deferens

1993
Temperature and agonist dependency of tachykinin NK1 receptor antagonist potencies in rat isolated superior cervical ganglion.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Animals; In Vitro Techniques; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Receptors, Neurokinin-1; Substance P; Superior Cervical Ganglion; Temperature; Tetrodotoxin

1995
The peripheral NK-1/NK-2 receptor antagonist MDL 105,172A inhibits tachykinin-mediated respiratory effects in guinea-pigs.
    Journal of autonomic pharmacology, 1997, Volume: 17, Issue:2

    Topics: Animals; Behavior, Animal; Capillary Permeability; Gerbillinae; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Male; Morpholines; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Plethysmography, Whole Body; Radioligand Assay; Receptors, Neurokinin-2; Respiratory Mechanics; Substance P; Tachykinins

1997
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
    Neuroscience, 1998, Volume: 83, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins

1998
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:2

    Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin

2000
Effects of TAK-637 on NK(1) receptor-mediated mechanisms regulating colonic secretion.
    Toxicology and applied pharmacology, 2004, Apr-15, Volume: 196, Issue:2

    Topics: Animals; Capsaicin; Colforsin; Colon; Electric Stimulation; Electrophysiology; Guinea Pigs; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Male; Naphthyridines; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Statistics, Nonparametric; Substance P; Tetrodotoxin

2004
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists.
    European journal of pharmacology, 2007, Dec-22, Volume: 577, Issue:1-3

    Topics: Animals; Autoradiography; Behavior, Animal; Brain; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Foot; Gerbillinae; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

2007
Neurokinin receptor modulation of respiratory activity in the rabbit.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy

2008
Effects of intravenous administration of neurokinin receptor subtype-selective agonists on gonadotropin-releasing hormone pulse generator activity and luteinizing hormone secretion in goats.
    The Journal of reproduction and development, 2015, Volume: 61, Issue:1

    Topics: Animals; Estradiol; Female; Goats; Gonadotropin-Releasing Hormone; Infusions, Intravenous; Kisspeptins; Ligands; Luteinizing Hormone; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Signal Transduction; Substance P; Time Factors

2015