Page last updated: 2024-09-03

gr 65630 and spiperone

gr 65630 has been researched along with spiperone in 2 studies

Compound Research Comparison

Studies
(gr 65630)
Trials
(gr 65630)
Recent Studies (post-2010)
(gr 65630)
Studies
(spiperone)
Trials
(spiperone)
Recent Studies (post-2010) (spiperone)
57042,9441385

Protein Interaction Comparison

ProteinTaxonomygr 65630 (IC50)spiperone (IC50)
Bile salt export pumpHomo sapiens (human)10
D(2) dopamine receptorHomo sapiens (human)0.0008
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.097
D(4) dopamine receptorHomo sapiens (human)0.0005
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.097
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.097
D(3) dopamine receptorHomo sapiens (human)0.0635
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.097
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0001
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.955

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Seyfried, CA; Tobler, P1
Hirokawa, Y; Kato, S; Morie, T; Yamazaki, H; Yoshida, N1

Other Studies

2 other study(ies) available for gr 65630 and spiperone

ArticleYear
Total versus unspecific binding: standardization and optimization of receptor-ligand binding assays.
    Drug metabolism and drug interactions, 1991, Volume: 9, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Filtration; Imidazoles; Indoles; Ketanserin; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1991
A novel series of N-(hexahydro-1,4-diazepin-6-yl) and N-(hexahydroazepin- 3-yl)benzamides with high affinity for 5-HT3 and dopamine D2 receptors.
    Bioorganic & medicinal chemistry letters, 1998, Mar-17, Volume: 8, Issue:6

    Topics: Animals; Benzamides; Binding Sites; Cerebral Cortex; Corpus Striatum; Domperidone; Dopamine Antagonists; Imidazoles; Indoles; Ligands; Metoclopramide; Models, Chemical; Ondansetron; Rats; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Spiperone; Stereoisomerism

1998