Page last updated: 2024-09-03

gr 65630 and indazoles

gr 65630 has been researched along with indazoles in 4 studies

Compound Research Comparison

Studies
(gr 65630)
Trials
(gr 65630)
Recent Studies (post-2010)
(gr 65630)
Studies
(indazoles)
Trials
(indazoles)
Recent Studies (post-2010) (indazoles)
57045,6095503,265

Protein Interaction Comparison

ProteinTaxonomygr 65630 (IC50)indazoles (IC50)
Chain A, Cell Division Protein Kinase 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, Cell Division Protein Kinase 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, Cell Division Protein Kinase 2Homo sapiens (human)185

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Airey, JE; Campbell, HF; Darkes, P; Fitzpatrick, LR; Klein, S; Neuenschwander, K; Pendley, CE; Powers, M; Schnapper, M; Youssefyeh, RD1
Fletcher, PW; Miller, K; Teitler, M; Weisberg, E1
Champaneria, S; Costall, B; Naylor, RJ; Robertson, DW1
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1

Other Studies

4 other study(ies) available for gr 65630 and indazoles

ArticleYear
Development of high-affinity 5-HT3 receptor antagonists. 1. Initial structure-activity relationship of novel benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Animals; Antiemetics; Benzamides; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Male; Metoclopramide; Molecular Structure; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting

1992
Membrane-bound and solubilized brain 5HT3 receptors: improved radioligand binding assays using bovine area postrema or rat cortex and the radioligands 3H-GR65630, 3H-BRL43694, and 3H-LY278584.
    Synapse (New York, N.Y.), 1992, Volume: 11, Issue:1

    Topics: Animals; Binding, Competitive; Brain Chemistry; Cattle; Cerebral Cortex; Chromatography, Gel; Granisetron; Imidazoles; Indazoles; Indoles; Membranes; Radioligand Assay; Rats; Receptors, Serotonin; Tropanes

1992
Identification and distribution of 5-HT3 recognition sites in the rat gastrointestinal tract.
    British journal of pharmacology, 1992, Volume: 106, Issue:3

    Topics: Affinity Labels; Animals; Digestive System; Female; Imidazoles; In Vitro Techniques; Indazoles; Indoles; Intestine, Small; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin Antagonists; Tissue Distribution; Tritium; Tropanes

1992
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991