Page last updated: 2024-09-02

gr 127935 and piperidines

gr 127935 has been researched along with piperidines in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (25.00)18.2507
2000's7 (58.33)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Goadsby, PJ; Knight, Y1
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM1
Hong, E; Meneses, A; Terrón, JA1
Conway, MW; O'Neill, MF1
Bankson, MG; Cunningham, KA1
Baker, GB; Fletcher, PJ; Korth, KM; Robinson, SR1
Donaldson, C; Hoskin, KL; Lambert, GA; Zagami, AS1
Jähnichen, S; Pertz, HH; Radtke, OA1
Komada, T; Yano, S1
Bourin, M; Chenu, F; David, DJ; Gardier, AM; Le Maître, E; Leroux-Nicollet, I1
Kawatani, M; Koyama, Y; Matsumoto-Miyai, K; Shimada, S; Shinzawa, E; Yamada, E; Yoshizumi, M1
Bojanowska, E; Drobnik, J; Juszczak, M; Wierucka-Rybak, M; Wolak, M1

Other Studies

12 other study(ies) available for gr 127935 and piperidines

ArticleYear
Inhibition of trigeminal neurones after intravenous administration of naratriptan through an action at 5-hydroxy-tryptamine (5-HT(1B/1D)) receptors.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Animals; Cats; Craniotomy; Electric Stimulation; Evoked Potentials, Somatosensory; Indoles; Injections, Intravenous; Neurons; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trigeminal Nucleus, Spinal; Tryptamines

1997
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents

1997
Effects of the 5-HT receptor antagonists GR127935 (5-HT1B/1D) and MDL100907 (5-HT2A) in the consolidation of learning.
    Behavioural brain research, 1997, Volume: 89, Issue:1-2

    Topics: Animals; Conditioning, Operant; Drug Interactions; Fluorobenzenes; Learning; Male; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
Role of 5-HT(1A) and 5-HT(1B) receptors in the mediation of behavior in the forced swim test in mice.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 24, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Tricyclic; Behavior, Animal; Dose-Response Relationship, Drug; Female; Imipramine; Indoles; Mice; Mice, Inbred Strains; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Pyridines; Reaction Time; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2001
Pharmacological studies of the acute effects of (+)-3,4-methylenedioxymethamphetamine on locomotor activity: role of 5-HT(1B/1D) and 5-HT(2) receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 26, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Fluorobenzenes; Hallucinogens; Indoles; Male; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Oxadiazoles; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists

2002
Multiple 5-HT receptors are involved in the effects of acute MDMA treatment: studies on locomotor activity and responding for conditioned reinforcement.
    Psychopharmacology, 2002, Volume: 162, Issue:3

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Ethylamines; Indoles; Ketanserin; Male; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors

2002
The 5-hydroxytryptamine1B/1D/1F receptor agonists eletriptan and naratriptan inhibit trigeminovascular input to the nucleus tractus solitarius in the cat.
    Brain research, 2004, Feb-13, Volume: 998, Issue:1

    Topics: Action Potentials; Animals; Cats; Drug Interactions; Electric Stimulation; Indoles; Maximum Tolerated Dose; Neural Inhibition; Oxadiazoles; Piperazines; Piperidines; Pyrrolidines; Reaction Time; Receptor, Serotonin, 5-HT1F; Receptors, Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Trigeminal Nuclei; Tryptamines

2004
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines

2004
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:3

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin

2007
Serotonin1B heteroreceptor activation induces an antidepressant-like effect in mice with an alteration of the serotonergic system.
    Journal of psychiatry & neuroscience : JPN, 2008, Volume: 33, Issue:6

    Topics: 5,7-Dihydroxytryptamine; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Behavior, Animal; Citalopram; Dopamine; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Serotonergic regulation of distention-induced ATP release from the urothelium.
    American journal of physiology. Renal physiology, 2016, 04-01, Volume: 310, Issue:7

    Topics: Adenosine Triphosphate; Animals; Citalopram; Dioxanes; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin, 5-HT4; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Urinary Bladder; Urothelium

2016
The inhibitory effect of combination treatment with leptin and cannabinoid CB1 receptor agonist on food intake and body weight gain is mediated by serotonin 1B and 2C receptors.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2016, Volume: 67, Issue:3

    Topics: Aminopyridines; Animals; Cannabinoid Receptor Agonists; Drug Synergism; Eating; Indoles; Leptin; Male; Oxadiazoles; Piperazines; Piperidines; Pyrazoles; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Weight Gain

2016
chemdatabank.com