gr 127935 and piperidines
gr 127935 has been researched along with piperidines in 12 studies
Research
Studies (12)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (25.00) | 18.2507 |
2000's | 7 (58.33) | 29.6817 |
2010's | 2 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Goadsby, PJ; Knight, Y | 1 |
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM | 1 |
Hong, E; Meneses, A; Terrón, JA | 1 |
Conway, MW; O'Neill, MF | 1 |
Bankson, MG; Cunningham, KA | 1 |
Baker, GB; Fletcher, PJ; Korth, KM; Robinson, SR | 1 |
Donaldson, C; Hoskin, KL; Lambert, GA; Zagami, AS | 1 |
Jähnichen, S; Pertz, HH; Radtke, OA | 1 |
Komada, T; Yano, S | 1 |
Bourin, M; Chenu, F; David, DJ; Gardier, AM; Le Maître, E; Leroux-Nicollet, I | 1 |
Kawatani, M; Koyama, Y; Matsumoto-Miyai, K; Shimada, S; Shinzawa, E; Yamada, E; Yoshizumi, M | 1 |
Bojanowska, E; Drobnik, J; Juszczak, M; Wierucka-Rybak, M; Wolak, M | 1 |
Other Studies
12 other study(ies) available for gr 127935 and piperidines
Article | Year |
---|---|
Inhibition of trigeminal neurones after intravenous administration of naratriptan through an action at 5-hydroxy-tryptamine (5-HT(1B/1D)) receptors.
Topics: Animals; Cats; Craniotomy; Electric Stimulation; Evoked Potentials, Somatosensory; Indoles; Injections, Intravenous; Neurons; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trigeminal Nucleus, Spinal; Tryptamines | 1997 |
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents | 1997 |
Effects of the 5-HT receptor antagonists GR127935 (5-HT1B/1D) and MDL100907 (5-HT2A) in the consolidation of learning.
Topics: Animals; Conditioning, Operant; Drug Interactions; Fluorobenzenes; Learning; Male; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1997 |
Role of 5-HT(1A) and 5-HT(1B) receptors in the mediation of behavior in the forced swim test in mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Tricyclic; Behavior, Animal; Dose-Response Relationship, Drug; Female; Imipramine; Indoles; Mice; Mice, Inbred Strains; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Pyridines; Reaction Time; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming | 2001 |
Pharmacological studies of the acute effects of (+)-3,4-methylenedioxymethamphetamine on locomotor activity: role of 5-HT(1B/1D) and 5-HT(2) receptors.
Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Fluorobenzenes; Hallucinogens; Indoles; Male; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Oxadiazoles; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists | 2002 |
Multiple 5-HT receptors are involved in the effects of acute MDMA treatment: studies on locomotor activity and responding for conditioned reinforcement.
Topics: 3,4-Methylenedioxyamphetamine; Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Ethylamines; Indoles; Ketanserin; Male; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2002 |
The 5-hydroxytryptamine1B/1D/1F receptor agonists eletriptan and naratriptan inhibit trigeminovascular input to the nucleus tractus solitarius in the cat.
Topics: Action Potentials; Animals; Cats; Drug Interactions; Electric Stimulation; Indoles; Maximum Tolerated Dose; Neural Inhibition; Oxadiazoles; Piperazines; Piperidines; Pyrrolidines; Reaction Time; Receptor, Serotonin, 5-HT1F; Receptors, Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Trigeminal Nuclei; Tryptamines | 2004 |
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines | 2004 |
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin | 2007 |
Serotonin1B heteroreceptor activation induces an antidepressant-like effect in mice with an alteration of the serotonergic system.
Topics: 5,7-Dihydroxytryptamine; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Behavior, Animal; Citalopram; Dopamine; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
Serotonergic regulation of distention-induced ATP release from the urothelium.
Topics: Adenosine Triphosphate; Animals; Citalopram; Dioxanes; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin, 5-HT4; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Urinary Bladder; Urothelium | 2016 |
The inhibitory effect of combination treatment with leptin and cannabinoid CB1 receptor agonist on food intake and body weight gain is mediated by serotonin 1B and 2C receptors.
Topics: Aminopyridines; Animals; Cannabinoid Receptor Agonists; Drug Synergism; Eating; Indoles; Leptin; Male; Oxadiazoles; Piperazines; Piperidines; Pyrazoles; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Weight Gain | 2016 |