Page last updated: 2024-09-02

gr 127935 and oxadiazoles

gr 127935 has been researched along with oxadiazoles in 193 studies

Research

Studies (193)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's92 (47.67)18.2507
2000's80 (41.45)29.6817
2010's20 (10.36)24.3611
2020's1 (0.52)2.80

Authors

AuthorsStudies
Hill, RG; Longmore, J; Razzaque, Z1
Feniuk, W; Skingle, M; Sleight, AJ1
Bristow, LJ; Cunningham, JR; Hogg, JE; Hutson, PH; Longmore, J; Murray, F; Pearce, D; Razzaque, Z; Saywell, K; Tricklebank, MD1
Colpaert, FC; Pauwels, PJ2
Craven, R; Grahame-Smith, D; Newberry, N1
Davidson, C; Stamford, JA3
Maura, G; Raiteri, M1
Kalkman, HO; Neumann, V1
Palmier, C; Pauwels, PJ1
Bobirnac, I; Schoeffter, P1
Crick, H; Manuel, NA; Wallis, DI1
Beattie, DT; Connor, HE; Walsh, DM1
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM3
Terrón, JA5
Burton, M; Jones, BJ; Middlemiss, DN; Mulholland, K; Price, GW; Roberts, C; Watson, J1
Beattie, DT; Connor, HE; Feniuk, W; Scopes, DI; Skingle, M; Starkey, SJ; Tyers, MB1
Colpaert, FC; Palmier, C; Pauwels, PJ; Wurch, T1
Clarke, T; Rollema, H; Schulz, DW; Sprouse, JS1
Fernández, AG; O'Neill, MF; Palacios, JM1
Bonnafous, R; John, GW; Valentin, JP1
Centurión, D; Sánchez-López, A; Villalón, CM1
Burton, MJ; Jones, BJ; Middlemiss, DN; Price, GW; Watson, JM1
Macor, JE; Mansbach, RS; Rovetti, CC1
Bertolino, F; Fauré, P; John, GW; Valentin, JP; Vieu, S1
Cistarelli, L; Gobert, A; Millan, MJ; Rivet, JM1
Millan, MJ; Perrin-Monneyron, S1
Centurión, D; Luján-Estrada, M; Sánchez-López, A; Terrón, JA; Villalón, CM1
Apaydin, S; De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM1
Curtis, MJ; Ellwood, AJ2
Hållbus, M; Magnusson, O; Magnusson, T1
Cutrer, FM; Moskowitz, MA; Waeber, C; Yu, XJ1
Hen, R; Lucas, JJ; Segu, L1
Centurión, D; Terrón, JA; Villalón, CM1
Gartside, SE; Sharp, T; Umbers, V1
Bulcäo, C; Cunha, M; De Castro-e-Silva, E; De Oliveira, IR; Fregoneze, JB; Luz, CP; Marinho, A; Nascimento, TA; Sarmento, C; Soares, T1
Gaster, L; Hagan, JJ; Hatcher, JP; Jeffrey, P; Middlemiss, DN; Slade, PD1
Goadsby, PJ; Knight, Y1
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM1
Hong, E; Meneses, A; Terrón, JA1
Audinot, V; Cistarelli, L; Gobert, A; Millan, MJ; Newman-Tancredi, A; Rivet, JM1
Gleason, SD; Shannon, HE1
Blaney, FE; Davies, S; Duckworth, DM; Gaster, LM; Hagan, JJ; Ham, P; Hatcher, J; Jenkins, S; Jennings, AJ; Joiner, GF; Jones, BJ; King, FD; Middlemiss, DN; Mulholland, KR; Price, GW; Riley, G; Roberts, C; Routledge, C; Selkirk, J; Slade, PD; Wyman, PA1
Goadsby, PJ; Hoskin, KL1
Belden, M; Carvey, PM; Goetz, CG; Pappert, EJ; Stebbins, GT1
Belenguer, A; Middlemiss, DN; Roberts, C; Routledge, C1
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM; Willems, EW1
John, GW; Le Grand, B; Vié, B1
Artigas, F; Bel, N; Fernández, AG; Hervás, I; Palacios, JM1
Dando, SB; Jordan, D; Ramage, AG; Skinner, MR1
Koob, GF; Parsons, LH; Weiss, F1
Pauwels, PJ1
Aguerre, S; Chaouloff, F; Mormede, P1
Branchek, TA; Zgombick, JM1
Beer, MS; Heald, MA; McAllister, G; Stanton, JA1
Nielsen, CK1
John, GW; Le Grand, B; Panissié, A; Pauwels, PJ1
Carvey, PM; Goetz, CG; Leurgans, S; Ling, ZD; Pappert, EJ; Raman, R; Vu, TQ1
Grailhe, R; Hen, R; Moskowitz, MA; Waeber, C; Yu, XJ1
Gaster, LM; Hagan, JJ; Ham, P; Joiner, GF; King, FD; Middlemiss, DN; Mulholland, KR; Price, GW; Roberts, C; Routledge, C; Selkirk, J; Slade, PD; Wyman, PA1
Centurión, D; Rabelo, G; Sánchez-López, A; Villalón, CM1
Barton, CL; Hutson, PH1
Harrison, AA; Koob, GF; Markou, A; Parsons, LH1
Chaouloff, F; Courvoisier, H; Moisan, MP; Mormède, P1
Hållbus, M; Larsson, LG; Magnusson, O; Magnusson, T; Ross, SB; Stenfors, C; Yu, H1
Beer, MS; Heald, MA; Hill, RG; Longmore, J; Maskell, L; Pickard, JD; Razzaque, Z1
Centurión, D; De Vries, P; Rabelo, G; Sánchez-López, A; Saxena, P; Villalón, CM1
Marcoli, M; Maura, G; Munari, C; Raiteri, M; Ruelle, A1
De Visser, PA; De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM1
Ayata, G; Cutrer, FM; Moskowitz, MA; Waeber, C; Yu, XJ1
Bankson, MG; Cunningham, KA; McCreary, AC1
Cohen, ML; Hemrick-Luecke, SH; Schenck, KW1
Fanelli, E; Grignaschi, G; Samanin, R; Scagnol, I1
Li, XF; Lovren, F; Lytton, J; Triggle, C1
De Vries, P; Heiligers, JP; Saxena, PR; Trion, M; Villalón, CM; Willems, EW1
Dawson, LA; Geiger, A; Nguyen, HQ1
Belknap, JK; Hain, HS; Mogil, JS1
Bischoff, A; Diener, H; Fetscher, C; Limmroth, V; Michel, MC; Wermelskirchen, D1
Faccidomo, S; Fish, EW; Miczek, KA1
Matsumoto, M; Miyamoto, A; Mori, K; Togashi, H; Ueno, K; Yoshioka, M1
Adrien, J; Chastanet, M; Evrard, A; Hamon, M; Hen, R; Laporte, AM1
Ferrari, MD; Maassen Van Den Brink, A; Roon, KI; Saxena, PR1
Dunn, AJ; Swiergiel, AH1
Knobelman, DA; Kung, HF; Lucki, I1
Fillion, G; Hong, E; Meneses, A; Orozco, G1
Dawson, LA; Nguyen, HQ1
Heisler, LK; Tecott, LH1
Lutz, EA; Shannon, HE1
Dulawa, SC; Geyer, MA; Hen, R; Scearce-Levie, KA1
Chen, J; Purdy, RE; Yildiz, O1
O'Neill, MF; Tomkins, DM1
Bosker, FJ; Cremers, TI; de Boer, P; den Boer, JA; Liao, Y; Westerink, BH; Wikström, HV1
John, GW; Le Grand, B; Panissié, A; Pauwels, PJ; Perez, M1
Boers, PM; Donaldson, C; Lambert, GA; Zagami, AS1
Beaufour, C; Evrard, A; Fabre, V; Hamon, M; Hanoun, N; Lanfumey, L; Lesch, KP; Martres, MP; Murphy, DL; Rioux, A1
Centurión, D; De Vries, P; Ortiz, MI; Sánchez-López, A; Saxena, PR; Villalón, CM1
Dremencov, E; Garcia, F; Gur, E; Lerer, B; Newman, ME; Van de Kar, LD2
Davidson, C; Hopwood, SE; McLaughlin, DP; Stamford, JA1
Dremencov, E; Gur, E; Lerer, B; Newman, ME2
Clarke, RW; Jenkins, S; Richardson, B1
Cordi, AA; Ragonnet, C; Vayssettes-Courchay, C; Verbeuren, TJ1
Bourin, M; Gardier, AM; Hen, R; Jacquot, C; Malagié, I; Trillat, AC1
Castanon, N; Hen, R; Lucas, JJ; Rocha, B; Scearce-Levie, K1
Conway, MW; O'Neill, MF1
Centurión, D; Sánchez-López, A; Saxena, PR; Villalón, CM1
Centurión, D; De Vries, P; Sánchez-López, A; Saxena, PR; Villalón, CM1
Akita, H; Inoue, N; Ishida, T; Kawashima, S; Miwa, Y; Sakoda, T; Shimokawa, Y; Shiomi, M; Ueyama, T; Yokoyama, M1
Filip, M; Papla, I; Przegalinski, E; Siwanowicz, J1
Bourin, M; Colombel, MC; David, D; Gardier, AM; Hascoët, M; Hen, R; Jacquot, C; Jolliet, P; Malagié, I; Trillat, AC1
Flieger, M; Pertz, HH; Schöning, C1
Honda, M; Ono, H1
Cooper, J; Greenslade, RG; Mitchell, SN1
Hicks, MN; Keegan, A; MacLean, MR; Morecroft, I; Smillie, D1
Bankson, MG; Cunningham, KA1
Dremencov, E; Gur, E; Lerer, B; Newman, ME; Van De Kar, LD1
Lin, D; Parsons, LH1
Clifton, PG; Dourish, CT; Hewitt, KN; Lee, MD1
Azampanah, A; Fletcher, PJ; Korth, KM1
De Vries, P; Heiligers, JP; John, GW; Kapoor, K; Saxena, PR; Tom, B; Willems, EW1
Baker, GB; Fletcher, PJ; Korth, KM; Robinson, SR1
de Groote, L; Klompmakers, AA; Olivier, B; Westenberg, HG1
Colpaert, FC; John, GW; Le Grand, B; Letienne, R; Perez, M; Verscheure, Y1
Crema, A; Crema, F; De Ponti, F; Frigo, G; Moro, E; Nardelli, G1
Adnot, S; Eddahibi, S; Hamon, M; Marcos, E; Nosjean, A; Pham, MH; Raffestin, B1
Avraham, Y; Berry, EM; Dremencov, E; Gur, E; Newman, ME1
Beauverie, P; Bourin, M; David, DJ; Douvier, E; Durier, S; Gardier, AM; Gruwez, B; Hen, R; Jacquot, C; Jego, G; Poisson, N; Przybylski, C1
Arulmani, U; Centurión, D; Sánchez-Lopez, A; Saxena, PR; Vázquez, E; Villalón, CM2
Donaldson, C; Hoskin, KL; Lambert, GA; Zagami, AS1
Folz, RJ; Liu, JQ1
Buhot, MC; Cazala, P; David, V; Ichaye, M; Segu, L1
Chojnacka-Wójcik, E; Kłodzińska, A; Stachowicz, K; Tatarczyńska, E2
Clarke, RW; Harris, J; Jackson, E; Lo, WC; Merriman, A1
Clifton, PG; Dourish, CT; Kennett, GA; Lee, MD; Somerville, EM1
Jähnichen, S; Pertz, HH; Radtke, OA1
Day, RM; Fanburg, BL; Liu, Y; Suzuki, YJ1
Honda, M; Imaida, K; Ono, H; Tanabe, M1
Castro, ME; Mostany, R; Pazos, A1
Bockaert, J; Compan, V; Conductier, G; Crosson, C; Hen, R1
Chojnacka-Wójcik, E; Kłodzińska, A; Tatarczyńska, E1
Greenshaw, A; Hayes, D; Mosher, T1
Bosker, FJ; Cremers, TI; den Boer, JA; Jongsma, ME; Westerink, BH1
Blanchet, JC; John, GW; Le Grand, B; Létienne, R; Sole, E1
Clarke, KL; Dawson, LA; Hagan, JJ; Langmead, CJ; Price, GW; Scott, C; Smith, PW; Starr, KR; Watson, J; Wyman, P1
Benini, Q; De Almeida, RM; Miczek, KA; Rosa, MM; Saft, DM; Santos, DM1
Aubel, B; Bourgoin, S; Farré, A; Hamon, M; Kayser, V1
Bloemarts, E; Groenink, L; Olivier, B; Oosting, RS; van den Bergh, FS1
Komada, T; Yano, S1
Centurión, D; Gupta, S; Mehrotra, S; Saxena, PR; VandenBrink, AM; Villalón, CM1
Bannai, M; Faccidomo, S; Fish, EW; Miczek, KA1
Martínez-García, E; Sánchez-Maldonado, C; Terrón, JA2
Fink, H; Rex, A; Voigt, JP; Wicke, KM1
Chen, ZQ; Cheng, HW; Dennis, RL1
Inoue, T; Koyama, T; Muraki, I1
Guptarak, J; Hiegel, C; Maswood, N; Uphouse, L1
Bourin, M; Chenu, F; David, DJ; Gardier, AM; Le Maître, E; Leroux-Nicollet, I1
Ansorge, M; Dulawa, SC; Geyer, MA; Gingrich, JA; Hen, R; Holick Pierz, KA; Masten, VL; Shanahan, NA; Waeber, C1
Graham, DA; Greenshaw, AJ; Hayes, DJ1
García-Iglesias, B; Martínez-García, E; Terrón, JA1
Centurión, D; Cobos-Puc, LE; González-Hernández, A; Lozano-Cuenca, J; Muñoz-Islas, E; Pertz, HH; Sánchez-López, A; Villalón, CM1
Carson, RE; Ding, YS; Frost, JJ; Huang, Y; McCarthy, T; Nabulsi, N; Ropchan, J; Weinzimmer, D1
Jiang, Z; Shang, J; Wang, W; Zhang, H; Zhang, L1
Abman, SH; Delaney, C; Gien, J; Grover, TR; Roe, G1
Cheng, HW; Dennis, RL1
Altamirano-Espinoza, AH; González-Hernández, A; MaassenVanDenBrink, A; Manrique-Maldonado, G; Marichal-Cancino, BA; Ruiz-Salinas, II; Villalón, CM1
Khatri, N; Lin, RC; Paul, IA; Simpson, KL1
Beaudet, G; Bouet, V; Boulouard, M; Dauphin, F; Freret, T; Gusmao-Montaigne, A; Nee, G; Paizanis, E1
Jamshidi-Mehr, M; Khakpai, F; Nasehi, M; Zarrindast, MR1
Anguiano-Robledo, L; Lacivita, E; Leopoldo, M; López-Sánchez, P; Sánchez-Maldonado, C; Terrón, JA1
Avila-Rojas, SH; Barragán-Iglesias, P; Granados-Soto, V; Pineda-Farias, JB; Salinas-Abarca, AB; Velázquez-Lagunas, I1
Cai, J; Chen, Z; Ji, G; Ji, Q; Li, Q; Liu, X; Song, H; Sui, H; Xu, H; Xu, Y; Zhou, L; Zhou, X1
Haeri-Rohani, SA; Najar, F; Nasehi, M; Zarrindast, MR1
Kawatani, M; Koyama, Y; Matsumoto-Miyai, K; Shimada, S; Shinzawa, E; Yamada, E; Yoshizumi, M1
Aronsen, D; Bukholt, N; Foote, J; Highgate, Q; Schenk, S; Van de Wetering, R; Webster, J1
Bojanowska, E; Drobnik, J; Juszczak, M; Wierucka-Rybak, M; Wolak, M1
Babapour, V; Keramati-Nojedehsadat, M; Oryan, S; Zarrindast, MR1
Afshari, K; Daneshpazhooh, M; Dehpour, AR; Foroutan, A; Haddadi, NS; Ostadhadi, S; Shakiba, S1
González-Hernández, A; Lozano-Cuenca, J; MaassenVanDenBrink, A; Marichal-Cancino, BA; Villalón, CM1
Abbaszadeh-Kasbi, A; Afshari, K; Amirlak, B; Dehdashtian, A; Dehpour, AR; Haddadi, NS; Jazaeri, F; Sheikhi, M; Tavangar, SM; Zarifeh Jazaeri, S1
Abdollahi, A; Dehpour, AR; Gharishvandi, F; Mohammad Jafari, R; Pasalar, P; Shafaroodi, H1

Reviews

2 review(s) available for gr 127935 and oxadiazoles

ArticleYear
GR127935: a potent and selective 5-HT1D receptor antagonist.
    Behavioural brain research, 1996, Volume: 73, Issue:1-2

    Topics: Animals; Behavior, Animal; Dogs; Guinea Pigs; Humans; Oxadiazoles; Piperazines; Rats; Receptors, Serotonin; Serotonin Antagonists

1996
Control of dorsal raphé 5-HT function by multiple 5-HT(1) autoreceptors: parallel purposes or pointless plurality?
    Trends in neurosciences, 2000, Volume: 23, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Second-Generation; Autoreceptors; Dimerization; Guinea Pigs; Humans; Ion Channels; Ion Transport; Mice; Nerve Tissue Proteins; Neurons; Oxadiazoles; Piperazines; Protein Isoforms; Pyridines; Pyrimidines; Raphe Nuclei; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Second Messenger Systems; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Spiperone; Sumatriptan

2000

Other Studies

191 other study(ies) available for gr 127935 and oxadiazoles

ArticleYear
Differences in the effects of ketanserin and GR127935 on 5-HT-receptor mediated responses in rabbit saphenous vein and guinea-pig jugular vein.
    European journal of pharmacology, 1995, Sep-05, Volume: 283, Issue:1-3

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Jugular Veins; Ketanserin; Male; Myenteric Plexus; Nifedipine; Oxadiazoles; Piperazines; Rabbits; Saphenous Vein; Serotonin; Serotonin Antagonists; Sumatriptan

1995
Effects of the 5-HT1D receptor antagonist GR127935 on extracellular levels of 5-HT in the guinea-pig frontal cortex as measured by microdialysis.
    Neuropharmacology, 1995, Volume: 34, Issue:4

    Topics: Animals; Frontal Lobe; Guinea Pigs; Male; Microdialysis; Neurons; Oxadiazoles; Piperazines; Serotonin; Serotonin Antagonists; Tetrodotoxin

1995
The effects of GR127935, a putative 5-HT1D receptor antagonist, on brain 5-HT metabolism, extracellular 5-HT concentration and behaviour in the guinea pig.
    Neuropharmacology, 1995, Volume: 34, Issue:4

    Topics: Animals; Biogenic Monoamines; Brain; Dyskinesia, Drug-Induced; Electric Stimulation; Fluoxetine; Guinea Pigs; Humans; In Vitro Techniques; Male; Methiothepin; Oxadiazoles; Paroxetine; Piperazines; Raphe Nuclei; Serotonin Antagonists; Synaptic Transmission; Tryptophan

1995
The 5-HT1D receptor antagonist GR 127,935 is an agonist at cloned human 5-HT1D alpha receptor sites.
    Neuropharmacology, 1995, Volume: 34, Issue:2

    Topics: Animals; Cells, Cultured; Cloning, Molecular; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Oxadiazoles; Piperazines; Rats; Receptors, Serotonin; Serotonin Antagonists

1995
WAY-100635 and GR127935: effects on 5-hydroxytryptamine-containing neurones.
    European journal of pharmacology, 1994, Dec-12, Volume: 271, Issue:1

    Topics: Action Potentials; Animals; Guinea Pigs; In Vitro Techniques; Male; Mesencephalon; Neurons; Oxadiazoles; Piperazines; Pyridines; Raphe Nuclei; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1994
The effect of paroxetine on 5-HT efflux in the rat dorsal raphe nucleus is potentiated by both 5-HT1A and 5-HT1B/D receptor antagonists.
    Neuroscience letters, 1995, Mar-16, Volume: 188, Issue:1

    Topics: Animals; Electric Stimulation; Male; Methiothepin; Oxadiazoles; Paroxetine; Piperazines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Time Factors

1995
Serotonin 5-HT1D and 5-HT1A receptors respectively mediate inhibition of glutamate release and inhibition of cyclic GMP production in rat cerebellum in vitro.
    Journal of neurochemistry, 1996, Volume: 66, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Afferent Pathways; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cerebellum; Cyclic GMP; Glutamic Acid; Male; N-Methylaspartate; Oxadiazoles; Piperazines; Potassium; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Agents; Signal Transduction; Sumatriptan; Synapses; Synaptic Transmission

1996
Evidence for a 5-HT1D receptor-mediated hypothermic effect of the alpha 1-adrenoceptor agonist, SDZ NVI-085, in guinea-pigs.
    European journal of pharmacology, 1995, Oct-24, Volume: 285, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Body Temperature; Bridged-Ring Compounds; Clonidine; Guinea Pigs; In Vitro Techniques; Male; Oxadiazoles; Oxazines; Piperazines; Prazosin; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Functional effects of the 5-HT1D receptor antagonist GR 127,935 at human 5-HT1D alpha, 5-HT1D beta, 5-HT1A and opossum 5-HT1B receptors.
    European journal of pharmacology, 1995, Jul-18, Volume: 290, Issue:2

    Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; HeLa Cells; Humans; Methiothepin; Opossums; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Transfection

1995
5-Hydroxytryptamine 5-HT1D receptors mediating inhibition of cyclic AMP accumulation in Madin-Darby canine kidney (MDCK) cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprostadil; Animals; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Epithelial Cells; Epithelium; Ketanserin; Kidney Cortex; Methiothepin; Oxadiazoles; Pertussis Toxin; Piperazines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Virulence Factors, Bordetella; Yohimbine

1995
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan

1995
The activity of 5-HT1D receptor ligands at cloned human 5-HT1D alpha and 5-HT1D beta receptors.
    European journal of pharmacology, 1995, Dec-04, Volume: 287, Issue:1

    Topics: Cyclic AMP; HeLa Cells; Humans; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

1995
Blockade of porcine carotid vascular response to sumatriptan by GR 127935, a selective 5-HT1D receptor antagonist.
    British journal of pharmacology, 1996, Volume: 118, Issue:1

    Topics: Animals; Arteriovenous Anastomosis; Blood Flow Velocity; Blood Pressure; Carotid Artery, Common; Heart Rate; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Sumatriptan; Swine

1996
GR127935 is a potent antagonist of the 5-HT1-like receptor mediating contraction in the canine coronary artery.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Coronary Vessels; Dogs; Drug Interactions; Ketanserin; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction

1996
Selective antagonism of human 5-HT1D and 5-HT1B receptor-mediated responses in stably transfected C6-glial cells by ketanserin and GR 127,935.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Drug Interactions; Humans; Ketanserin; Neuroglia; Oxadiazoles; Piperazines; Rats; Serotonin Antagonists; Transfection

1996
Species differences in 5-HT autoreceptors.
    Behavioural brain research, 1996, Volume: 73, Issue:1-2

    Topics: Animals; Central Nervous System; Guinea Pigs; Humans; Mice; Oxadiazoles; Piperazines; Rabbits; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Swine

1996
The relaxant 5-HT receptor in the dog coronary artery smooth muscle: pharmacological resemblance to the cloned 5-ht7 receptor subtype.
    British journal of pharmacology, 1996, Volume: 118, Issue:6

    Topics: Animals; Antipsychotic Agents; Cloning, Molecular; Coronary Vessels; Dinoprost; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Promotion of cell growth by stimulation of cloned human 5-HT1D receptor sites in transfected C6-glial cells is highly sensitive to intrinsic activity at 5-HT1D receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:2

    Topics: Animals; Cell Division; Cyclic AMP; Humans; Metergoline; Neuroglia; Oxadiazoles; Piperazines; Rats; Receptors, Serotonin; Serotonin; Thymidine; Transfection

1996
Combined administration of a 5-hydroxytryptamine (5-HT)1D antagonist and a 5-HT reuptake inhibitor synergistically increases 5-HT release in guinea pig hypothalamus in vivo.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: 1-Naphthylamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Drug Synergism; Guinea Pigs; Hydroxyindoleacetic Acid; Hypothalamus; Indoles; Kinetics; Neurons; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Sertraline

1996
GR 127935 blocks the locomotor and antidepressant-like effects of RU 24969 and the action of antidepressants in the mouse tail suspension test.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Indoles; Locomotion; Male; Mice; Mice, Inbred Strains; Oxadiazoles; Piperazines; Serotonin Antagonists; Serotonin Receptor Agonists; Tail

1996
Influence of the endothelium and nitric oxide on the contractile responses evoked by 5-HT1D receptor agonists in the rabbit isolated saphenous vein.
    British journal of pharmacology, 1996, Volume: 119, Issue:1

    Topics: Animals; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

1996
Typical and atypical antipsychotic drugs are potent antagonists of the relaxant 5-hydroxytryptamine receptor in the smooth muscle of canine coronary artery.
    Proceedings of the Western Pharmacology Society, 1996, Volume: 39

    Topics: Animals; Antipsychotic Agents; Clozapine; Coronary Vessels; Dogs; In Vitro Techniques; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoconstriction; Vasodilation

1996
Operational characteristics of the 5-HT1-like receptors mediating external carotid vasoconstriction in vagosympathectomized dogs. Close resemblance to the 5-HT1D receptor subtype.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:5

    Topics: Analysis of Variance; Animals; Blood Pressure; Carotid Artery, Common; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Male; Methysergide; Oxadiazoles; Piperazines; Receptors, Serotonin; Regional Blood Flow; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction

1996
GR127935 acts as a partial agonist at recombinant human 5-HT1D alpha and 5-HT1D beta receptors.
    European journal of pharmacology, 1996, Oct-31, Volume: 314, Issue:3

    Topics: Adenylyl Cyclases; Alkylating Agents; Animals; CHO Cells; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Logistic Models; Oxadiazoles; Piperazines; Quinolines; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists

1996
CP-135,807, a selective 5-HT1D agonist: effects in drug discrimination and punishment procedures in the pigeon.
    Psychopharmacology, 1996, Volume: 128, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Columbidae; Conditioning, Operant; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Indoles; Male; Oxadiazoles; Piperazines; Punishment; Pyridines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Differential involvement of serotonin 2A/C and thromboxane A2/prostanoid receptors in high- vs. low-shear rate arterial thrombosis in rabbits.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Arteriovenous Shunt, Surgical; Aspirin; Blood Pressure; Bridged Bicyclo Compounds, Heterocyclic; Carotid Arteries; Carotid Stenosis; Endothelium, Vascular; Fatty Acids, Unsaturated; Heart Rate; Hemodynamics; Hydrazines; Jugular Veins; Ketanserin; Male; Oxadiazoles; Piperazines; Platelet Aggregation; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Prostaglandin; Receptors, Serotonin; Receptors, Thromboxane; Ritanserin; Serotonin Antagonists; Stress, Mechanical

1997
Potentiation of the fluoxetine-induced increase in dialysate levels of serotonin (5-HT) in the frontal cortex of freely moving rats by combined blockade of 5-HT1A and 5-HT1B receptors with WAY 100,635 and GR 127,935.
    Journal of neurochemistry, 1997, Volume: 68, Issue:3

    Topics: Animals; Drug Synergism; Fluoxetine; Frontal Lobe; Male; Microdialysis; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

1997
5-HT1B/D antagonists potentiate paroxetine's effect on 5-HT efflux in the lateral geniculate nucleus: in vitro voltammetric data.
    Biochemical Society transactions, 1997, Volume: 25, Issue:1

    Topics: Animals; Electrochemistry; Geniculate Bodies; Male; Methiothepin; Oxadiazoles; Paroxetine; Piperazines; Propanolamines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1997
Potentiation of fluoxetine-induced penile erections by combined blockade of 5-HT1A and 5-HT1B receptors.
    European journal of pharmacology, 1997, Mar-05, Volume: 321, Issue:3

    Topics: Animals; Antidepressive Agents, Second-Generation; Drug Synergism; Fluoxetine; Male; Oxadiazoles; Penile Erection; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists

1997
Mediation of 5-HT-induced external carotid vasodilatation in GR 127935-pretreated vagosympathectomized dogs by the putative 5-HT7 receptor.
    British journal of pharmacology, 1997, Volume: 120, Issue:7

    Topics: 5-Methoxytryptamine; Acetylcholine; Animals; Carotid Arteries; Dogs; Hemodynamics; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasodilation

1997
Interactions of GR127935, a 5-HT(1B/D) receptor ligand, with functional 5-HT receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:4

    Topics: Animals; Cats; Dose-Response Relationship, Drug; Male; Oxadiazoles; Piperazines; Rabbits; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Sumatriptan

1997
Mechanism of actions of sumatriptan on coronary flow before and after endothelial dysfunction in guinea-pig isolated heart.
    British journal of pharmacology, 1997, Volume: 120, Issue:6

    Topics: Animals; Coronary Circulation; Coronary Vessels; Endothelium, Vascular; Enzyme Inhibitors; Ergolines; Guinea Pigs; Heart; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Piperazines; Saponins; Serotonin Receptor Agonists; Sumatriptan; Vasoconstrictor Agents

1997
Influence of 5-HT1B/1D receptors on dopamine release in the guinea pig nucleus accumbens: a microdialysis study.
    Neuroscience letters, 1997, Mar-28, Volume: 225, Issue:1

    Topics: Analysis of Variance; Animals; Dopamine; Guinea Pigs; Male; Microdialysis; Nucleus Accumbens; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

1997
The 5-HT1D receptor antagonist GR-127,935 prevents inhibitory effects of sumatriptan but not CP-122,288 and 5-CT on neurogenic plasma extravasation within guinea pig dura mater.
    Neuropharmacology, 1997, Volume: 36, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Dura Mater; Electric Stimulation; Female; Guinea Pigs; Male; Oxadiazoles; Pertussis Toxin; Piperazines; Prosencephalon; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Trigeminal Nerve; Virulence Factors, Bordetella

1997
5-Hydroxytryptamine1B receptors modulate the effect of cocaine on c-fos expression: converging evidence using 5-hydroxytryptamine1B knockout mice and the 5-hydroxytryptamine1B/1D antagonist GR127935.
    Molecular pharmacology, 1997, Volume: 51, Issue:5

    Topics: Animals; Cocaine; Corpus Striatum; Gene Expression Regulation; Genes, fos; Indoles; Mice; Mice, Knockout; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
GR127935 antagonizes the 5-HT1-like receptor-mediated external carotid vasoconstriction in vagosympathectomized dogs.
    Annals of the New York Academy of Sciences, 1997, May-30, Volume: 812

    Topics: Animals; Dogs; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Sympathectomy; Vagotomy; Vasoconstriction

1997
Effect of a selective 5-HT reuptake inhibitor in combination with 5-HT1A and 5-HT1B receptor antagonists on extracellular 5-HT in rat frontal cortex in vivo.
    British journal of pharmacology, 1997, Volume: 121, Issue:5

    Topics: Animals; Electrophysiology; Extracellular Space; Male; Microdialysis; Neurons; Oxadiazoles; Paroxetine; Piperazines; Prefrontal Cortex; Pyridines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Stereotaxic Techniques

1997
Nature of 5-HT1-like receptors mediating depressor responses in vagosympathectomized rats; close resemblance to the cloned 5-ht7 receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 5-Methoxytryptamine; Adrenergic beta-Agonists; Animals; Blood Pressure; Clozapine; Ergolines; Heart Rate; Isoproterenol; Lisuride; Male; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy

1997
Synergism of 5-HT 1B/D antagonists with paroxetine on serotonin efflux in rat ventral lateral geniculate nucleus slices.
    Brain research bulletin, 1997, Volume: 43, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Drug Synergism; Geniculate Bodies; Male; Oxadiazoles; Paroxetine; Piperazines; Propanolamines; Rats; Rats, Wistar; Serotonin

1997
Effect of third ventricle administration of L-694,247, a selective 5-HT1D receptor agonist, on water intake in rats.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 57, Issue:4

    Topics: Adrenergic beta-Agonists; Angiotensin II; Animals; Carbachol; Drinking; Injections, Intraventricular; Isoproterenol; Male; Microinjections; Muscarinic Agonists; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tryptamines; Water Deprivation

1997
Stimulation of 5-HT1B receptors causes hypothermia in the guinea pig.
    European journal of pharmacology, 1997, Jul-23, Volume: 331, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Body Temperature; Dose-Response Relationship, Drug; Guinea Pigs; Hypothermia; Indoles; Male; Oxadiazoles; Piperazines; Piperidones; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds

1997
Involvement of 5-HT(1B/1D) and 5-HT2A receptors in 5-HT-induced contraction of endothelium-denuded rabbit epicardial coronary arteries.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Coronary Vessels; Endothelium, Vascular; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Oxadiazoles; Pericardium; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstrictor Agents

1997
Inhibition of trigeminal neurones after intravenous administration of naratriptan through an action at 5-hydroxy-tryptamine (5-HT(1B/1D)) receptors.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Animals; Cats; Craniotomy; Electric Stimulation; Evoked Potentials, Somatosensory; Indoles; Injections, Intravenous; Neurons; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trigeminal Nucleus, Spinal; Tryptamines

1997
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents

1997
Effects of the 5-HT receptor antagonists GR127935 (5-HT1B/1D) and MDL100907 (5-HT2A) in the consolidation of learning.
    Behavioural brain research, 1997, Volume: 89, Issue:1-2

    Topics: Animals; Conditioning, Operant; Drug Interactions; Fluorobenzenes; Learning; Male; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
Simultaneous quantification of serotonin, dopamine and noradrenaline levels in single frontal cortex dialysates of freely-moving rats reveals a complex pattern of reciprocal auto- and heteroreceptor-mediated control of release.
    Neuroscience, 1998, Volume: 84, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Dopamine; Dopamine Agonists; Frontal Lobe; Guanabenz; Guinea Pigs; Homeostasis; Idazoxan; Imidazoles; Indoles; Isoindoles; Male; Medetomidine; Models, Neurological; Motor Activity; Norepinephrine; Oxadiazoles; Piperazines; Prazosin; Raclopride; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Serotonin

1998
Meta-chlorophenylpiperazine induced changes in locomotor activity are mediated by 5-HT1 as well as 5-HT2C receptors in mice.
    European journal of pharmacology, 1998, Jan-12, Volume: 341, Issue:2-3

    Topics: Animals; Dose-Response Relationship, Drug; Ergolines; Male; Mice; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists

1998
The selective 5-HT1B receptor inverse agonist 1'-methyl-5-[[2'-methyl-4'-(5-methyl-1,2, 4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) potently blocks terminal 5-HT autoreceptor function b
    Journal of medicinal chemistry, 1998, Apr-09, Volume: 41, Issue:8

    Topics: Animals; Aspartic Acid; Autoreceptors; CHO Cells; Cricetinae; Frontal Lobe; Guinea Pigs; Humans; Hypothermia; In Vitro Techniques; Indoles; Male; Models, Molecular; Oxadiazoles; Piperazines; Piperidones; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Structure-Activity Relationship; Swine

1998
Characterization of 5-HT receptors mediating constriction of porcine carotid arteriovenous anastomoses; involvement of 5-HT1B/1D and novel receptors.
    British journal of pharmacology, 1998, Volume: 123, Issue:8

    Topics: Animals; Arteriovenous Anastomosis; Carotid Arteries; Ergot Alkaloids; Hemodynamics; Ketanserin; Oxadiazoles; Oxygen; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Swine; Vasoconstriction

1998
Serotonin inhibits trigeminal nucleus activity evoked by craniovascular stimulation through a 5HT1B/1D receptor: a central action in migraine?
    Annals of neurology, 1998, Volume: 43, Issue:6

    Topics: Animals; Cats; Electric Stimulation; Electrophysiology; Membrane Potentials; Migraine Disorders; Neural Inhibition; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Trigeminal Nucleus, Spinal

1998
5-Hydroxytryptophan-induced myoclonus in guinea pigs: mediation through 5-HT1/2 receptor subtypes.
    European journal of pharmacology, 1998, Apr-17, Volume: 347, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Guinea Pigs; Male; Methiothepin; Myoclonus; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Substrate Specificity

1998
Differential effects of 5-HT1B/1D receptor antagonists in dorsal and median raphe innervated brain regions.
    European journal of pharmacology, 1998, Apr-10, Volume: 346, Issue:2-3

    Topics: Animals; Antidepressive Agents, Second-Generation; Brain; Cerebral Cortex; Chromatography, High Pressure Liquid; Dentate Gyrus; Electrochemistry; Extracellular Space; Guinea Pigs; Male; Microdialysis; Neostriatum; Oxadiazoles; Paroxetine; Piperazines; Piperidones; Raphe Nuclei; Serotonin Antagonists; Spiro Compounds

1998
The antimigraine agent alniditan selectively constricts porcine carotid arteriovenous anastomoses via 5-HT1B/1D receptors.
    European journal of pharmacology, 1998, Jun-19, Volume: 351, Issue:2

    Topics: Analgesics; Animals; Arteriovenous Anastomosis; Benzopyrans; Carotid Arteries; Hemodynamics; Humans; Jugular Veins; Male; Migraine Disorders; Oxadiazoles; Oxygen; Piperazines; Propylamines; Pyrimidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swine; Vasoconstrictor Agents

1998
Effects of sumatriptan on coronary flow and left ventricular function in the isolated perfused guinea pig heart.
    Journal of cardiovascular pharmacology, 1998, Volume: 32, Issue:3

    Topics: Animals; Coronary Circulation; Diastole; Dihydroergotamine; Endothelium, Vascular; Guinea Pigs; In Vitro Techniques; NG-Nitroarginine Methyl Ester; Oxadiazoles; Oxazoles; Oxazolidinones; Perfusion; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Ventricular Function, Left

1998
In vivo control of 5-hydroxytryptamine release by terminal autoreceptors in rat brain areas differentially innervated by the dorsal and median raphe nuclei.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:3

    Topics: Animals; Autoreceptors; Brain; Chromatography, High Pressure Liquid; Hydroxyindoleacetic Acid; Male; Methiothepin; Microdialysis; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

1998
Modulation of the vagal bradycardia evoked by stimulation of upper airway receptors by central 5-HT1 receptors in anaesthetized rabbits.
    British journal of pharmacology, 1998, Volume: 125, Issue:2

    Topics: Anesthesia; Animals; Aortic Bodies; Bradycardia; Buspirone; Ligands; Male; Oxadiazoles; Piperazines; Pyridines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reflex; Serotonin Antagonists; Serotonin Receptor Agonists; Smoke

1998
Serotonin1B receptor stimulation enhances cocaine reinforcement.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Dec-01, Volume: 18, Issue:23

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Indoles; Injections, Intraventricular; Male; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Antagonists; Serotonin Receptor Agonists

1998
Na(+)-dependent metabolic coupling upon 5-HT1B receptor activation by sumatriptan and related agonists.
    Receptors & channels, 1998, Volume: 5, Issue:6

    Topics: Animals; CHO Cells; Cricetinae; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Sodium; Sumatriptan; Vasoconstrictor Agents

1998
GR 127935 and (+)-WAY 100135 do not affect TFMPP-induced inhibition of 5-HT synthesis in the midbrain and hippocampus of Wistar-Kyoto rats.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Hippocampus; Idazoxan; Ketanserin; Male; Mesencephalon; Mianserin; Nerve Endings; Oxadiazoles; Piperazines; Rats; Rats, Inbred WKY; Rats, Wistar; Reserpine; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Tryptophan Hydroxylase

1998
Antagonism of the relaxant 5-HT receptor in the dog basilar artery by the high-affinity 5-HT7 receptor ligand, LY215840.
    Proceedings of the Western Pharmacology Society, 1998, Volume: 41

    Topics: Animals; Basilar Artery; Dinoprost; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Lysergic Acid; Muscle Relaxation; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1998
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:5

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella

1998
Pharmacological characterisation of a cloned dog 5-HT1B receptor cell line.
    European journal of pharmacology, 1998, Oct-30, Volume: 360, Issue:1

    Topics: Animals; Binding, Competitive; CHO Cells; Clone Cells; Cricetinae; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Methiothepin; Oxadiazoles; Piperazines; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Fusion Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfur Radioisotopes; Tritium

1998
Head and whole-body jerking in guinea pigs are differentially modulated by 5-HT1A, 5-HT1B/1D and 5-HT2A receptor antagonists.
    European journal of pharmacology, 1998, Nov-20, Volume: 361, Issue:2-3

    Topics: 5-Hydroxytryptophan; Animals; Benzazepines; Guinea Pigs; Head Movements; Male; Methoxydimethyltryptamines; Myoclonus; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists

1998
Activation of recombinant h 5-HT1B and h 5-HT1D receptors stably expressed in C6 glioma cells produces increases in Ca2+-dependent K+ current.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:6

    Topics: Animals; Calcium; Cyclic AMP; Dose-Response Relationship, Drug; Glioma; Oxadiazoles; Piperazines; Potassium; Potassium Channels; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Sumatriptan; Tumor Cells, Cultured

1998
Animal model of posthypoxic myoclonus: effects of serotonergic antagonists.
    Neurology, 1999, Jan-01, Volume: 52, Issue:1

    Topics: Acoustic Stimulation; Animals; Brain Chemistry; Disease Models, Animal; Dose-Response Relationship, Drug; Ergolines; Heart Arrest; Hypoxia; Hypoxia, Brain; Male; Methiothepin; Myoclonus; Oxadiazoles; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists

1999
Putative 5-ht5 receptors: localization in the mouse CNS and lack of effect in the inhibition of dural protein extravasation.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Binding Sites; Blood Proteins; Brain; Crosses, Genetic; Female; Lysergic Acid Diethylamide; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Organ Specificity; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Trigeminal Ganglion; Tritium

1998
The selective 5-HT1B receptor inverse agonist SB-224289, potently blocks terminal 5-HT autoreceptor function both in vitro and in vivo.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: Animals; Body Temperature Regulation; Cerebral Cortex; CHO Cells; Cricetinae; Dentate Gyrus; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; Oxadiazoles; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Spiro Compounds; Sumatriptan; Transfection

1998
Pharmacological profile of the prejunctional 5-HT1 receptors mediating inhibition of sympathetic vasopressor outflow in the pithed rat.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Central Nervous System; Oxadiazoles; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathetic Nervous System

1998
Evidence for the putative 5-HT7 receptor mediating direct relaxation to 5-hydroxytryptamine in canine cerebral blood vessels.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 5-Hydroxytryptophan; Animals; Basilar Artery; Cerebral Arteries; Cerebrovascular Circulation; Dinoprost; Dogs; In Vitro Techniques; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoconstriction; Vasodilation

1998
Inhibition of hippocampal 5-HT synthesis by fluoxetine and paroxetine: evidence for the involvement of both 5-HT1A and 5-HT1B/D autoreceptors.
    Synapse (New York, N.Y.), 1999, Volume: 31, Issue:1

    Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Enzyme Inhibitors; Fluoxetine; Hippocampus; Hydrazines; Male; Oxadiazoles; Paroxetine; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
RU 24969, a 5-HT1A/1B agonist, elevates brain stimulation reward thresholds: an effect reversed by GR 127935, a 5-HT1B/1D antagonist.
    Psychopharmacology, 1999, Volume: 141, Issue:3

    Topics: Animals; Brain; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electric Stimulation; Indoles; Male; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reward; Self Stimulation; Serotonin Antagonists; Serotonin Receptor Agonists

1999
GR 127935 reduces basal locomotor activity and prevents RU 24969-, but not D-amphetamine-induced hyperlocomotion, in the Wistar-Kyoto hyperactive (WKHA) rat.
    Psychopharmacology, 1999, Volume: 141, Issue:3

    Topics: Animals; Central Nervous System Stimulants; Dextroamphetamine; Dose-Response Relationship, Drug; Indoles; Male; Motor Activity; Oxadiazoles; Piperazines; Rats; Rats, Inbred WKY; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Synergism between 5-HT1B/1D and 5-HT1A receptor antagonists on turnover and release of 5-HT in guinea-pig brain in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:2

    Topics: Animals; Brain; Drug Synergism; Guinea Pigs; Hydroxyindoleacetic Acid; Male; Microdialysis; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Synaptic Transmission

1999
Vasoconstriction in human isolated middle meningeal arteries: determining the contribution of 5-HT1B- and 5-HT1F-receptor activation.
    British journal of clinical pharmacology, 1999, Volume: 47, Issue:1

    Topics: Animals; Benzamides; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; Humans; In Vitro Techniques; Meningeal Arteries; Oxadiazoles; Piperazines; Pyridines; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction

1999
Canine external carotid vasoconstriction to methysergide, ergotamine and dihydroergotamine: role of 5-HT1B/1D receptors and alpha2-adrenoceptors.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Flow Velocity; Carotid Arteries; Clonidine; Dihydroergotamine; Dogs; Ergotamine; Female; Hemodynamics; Male; Methysergide; Oxadiazoles; Phenylephrine; Piperazines; Prazosin; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents; Yohimbine

1999
Pharmacological diversity between native human 5-HT1B and 5-HT1D receptors sited on different neurons and involved in different functions.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adult; Aged; Binding Sites; Biphenyl Compounds; Cerebral Cortex; Female; Glutamic Acid; Humans; Male; Middle Aged; Neurons; Oxadiazoles; Piperazines; Piperidones; Potassium Chloride; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiro Compounds; Synaptosomes; Tritium

1999
Changes in systemic and regional haemodynamics during 5-HT7 receptor-mediated depressor responses in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adrenal Glands; Animals; Blood Pressure; Cardiac Output; Heart Rate; Hemodynamics; Kidney; Lisuride; Lung; Male; Muscle, Skeletal; Oxadiazoles; Pancreas; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism; Stroke Volume; Vascular Capacitance

1999
Effects of PNU-109,291, a selective 5-HT1D receptor agonist, on electrically induced dural plasma extravasation and capsaicin-evoked c-fos immunoreactivity within trigeminal nucleus caudalis.
    Neuropharmacology, 1999, Volume: 38, Issue:7

    Topics: Animals; Benzopyrans; Binding, Competitive; Blood Pressure; Blood Proteins; Capsaicin; Dura Mater; Electric Stimulation; Guinea Pigs; Male; Oxadiazoles; Piperazines; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trigeminal Nuclei

1999
Pharmacological studies of the acute and chronic effects of (+)-3, 4-methylenedioxymethamphetamine on locomotor activity: role of 5-hydroxytryptamine(1A) and 5-hydroxytryptamine(1B/1D) receptors.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Behavior, Animal; Drug Administration Schedule; Frontal Lobe; Indoles; Male; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Chloride

1999
5-Hydroxytryptamine(1A) receptor activation enhances norepinephrine release from nerves in the rabbit saphenous vein.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic Fibers; Animals; Electric Stimulation; Ergolines; Male; Muscle Contraction; Norepinephrine; Oxadiazoles; Piperazines; Pyridines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Saphenous Vein; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Synaptic Transmission

1999
Studies on the role of serotonin receptor subtypes in the effect of sibutramine in various feeding paradigms in rats.
    British journal of pharmacology, 1999, Volume: 127, Issue:5

    Topics: Animals; Appetite Depressants; Cyclobutanes; Dose-Response Relationship, Drug; Eating; Male; Neuropeptide Y; Oxadiazoles; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin

1999
Functional characterization and m-RNA expression of 5-HT receptors mediating contraction in human umbilical artery.
    British journal of pharmacology, 1999, Volume: 127, Issue:5

    Topics: Humans; Ketanserin; Oxadiazoles; Piperazines; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Sumatriptan; Umbilical Arteries; Vasoconstriction

1999
Pharmacological evidence that alpha1-and alpha2-adrenoceptors mediate vasoconstriction of carotid arteriovenous anastomoses in anaesthetized pigs.
    British journal of pharmacology, 1999, Volume: 127, Issue:5

    Topics: Anesthesia; Animals; Arteriovenous Anastomosis; Azepines; Carotid Arteries; Hemodynamics; Migraine Disorders; Oxadiazoles; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Sumatriptan; Swine; Vasoconstriction

1999
Effects of venlafaxine on extracellular concentrations of 5-HT and noradrenaline in the rat frontal cortex: augmentation via 5-HT1A receptor antagonism.
    Neuropharmacology, 1999, Volume: 38, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Cyclohexanols; Dose-Response Relationship, Drug; Idazoxan; Male; Norepinephrine; Oxadiazoles; Piperazines; Prazosin; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Venlafaxine Hydrochloride

1999
Pharmacogenetic evidence for the involvement of 5-hydroxytryptamine (Serotonin)-1B receptors in the mediation of morphine antinociceptive sensitivity.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics; Animals; Dose-Response Relationship, Drug; Drug Interactions; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Morphine; Oxadiazoles; Piperazines; Receptors, Serotonin; Sensitivity and Specificity; Serotonin Antagonists; Species Specificity; Time Factors

1999
Effects of alniditan on neurogenic oedema in the rat dura mater and on contraction of rat basilar artery.
    European journal of pharmacology, 1999, Oct-08, Volume: 382, Issue:2

    Topics: Animals; Basilar Artery; Benzopyrans; Brain Edema; Capillary Permeability; Dose-Response Relationship, Drug; Dura Mater; Extravasation of Diagnostic and Therapeutic Materials; In Vitro Techniques; Ketanserin; Male; Oxadiazoles; Piperazines; Propylamines; Pyrimidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Agents; Serotonin Antagonists; Substance P; Sumatriptan; Vasoconstriction; Vasoconstrictor Agents

1999
Aggression heightened by alcohol or social instigation in mice: reduction by the 5-HT(1B) receptor agonist CP-94,253.
    Psychopharmacology, 1999, Volume: 146, Issue:4

    Topics: Aggression; Animals; Behavior, Animal; Central Nervous System Depressants; Ethanol; Male; Mice; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Characterization of endogenous serotonin-mediated regulation of dopamine release in the rat prefrontal cortex.
    European journal of pharmacology, 1999, Oct-21, Volume: 383, Issue:1

    Topics: Animals; Dopamine; Dose-Response Relationship, Drug; Electric Stimulation; Fluoxetine; Male; Microdialysis; Oligonucleotides, Antisense; Oxadiazoles; Piperazines; Prefrontal Cortex; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Time Factors

1999
5-HT1A and 5-HT1B receptors control the firing of serotoninergic neurons in the dorsal raphe nucleus of the mouse: studies in 5-HT1B knock-out mice.
    The European journal of neuroscience, 1999, Volume: 11, Issue:11

    Topics: Animals; Autoradiography; Brain; Citalopram; Electric Stimulation; Evoked Potentials; Membrane Potentials; Mice; Mice, Knockout; Neurons; Oxadiazoles; Piperazines; Pyridines; Radioligand Assay; Raphe Nuclei; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

1999
Bovine isolated middle cerebral artery contractions to antimigraine drugs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:5

    Topics: Animals; Cattle; In Vitro Techniques; Ketanserin; Middle Cerebral Artery; Muscle Contraction; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstrictor Agents

1999
Lack of evidence for a role of serotonin in interleukin-1-induced hypophagia.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 65, Issue:3

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Eating; Interleukin-1; Ketanserin; Lipopolysaccharides; Male; Mice; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiro Compounds; Sulfonamides

2000
Regulation of extracellular concentrations of 5-hydroxytryptamine (5-HT) in mouse striatum by 5-HT(1A) and 5-HT(1B) receptors.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:3

    Topics: Animals; Autoreceptors; Corpus Striatum; Fenfluramine; Fluoxetine; Male; Mice; Microdialysis; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Tetrahydronaphthalenes

2000
Effect of 5-HT-moduline, an endogenous peptide, in associative learning.
    Proceedings of the Western Pharmacology Society, 1999, Volume: 42

    Topics: Animals; Association Learning; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Neuropeptides; Oligopeptides; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
The role of 5-HT(1A) and 5-HT(1B/1D) receptors on the modulation of acute fluoxetine-induced changes in extracellular 5-HT: the mechanism of action of (+/-)pindolol.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: Animals; Autoreceptors; Drug Synergism; Extracellular Space; Fluoxetine; Male; Microdialysis; Oxadiazoles; Pindolol; Piperazines; Propanolamines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

2000
A paradoxical locomotor response in serotonin 5-HT(2C) receptor mutant mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Apr-15, Volume: 20, Issue:8

    Topics: Animals; Drug Interactions; Indoles; Male; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Motor Activity; Mutation; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Yohimbine produces antinociception in the formalin test in rats: involvement of serotonin(1A) receptors.
    Psychopharmacology, 2000, Volume: 149, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Benzofurans; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Ergolines; Formaldehyde; Male; Nociceptors; Oxadiazoles; Pain; Pain Measurement; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors; Yohimbine

2000
Serotonin releasers increase prepulse inhibition in serotonin 1B knockout mice.
    Psychopharmacology, 2000, Volume: 149, Issue:3

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Mice; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reflex, Startle; Serotonin; Serotonin Agents; Serotonin Antagonists

2000
Phenylephrine precontraction increases the sensitivity of rabbit femoral artery to serotonin by enabling 5-HT1-like receptors.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Femoral Artery; In Vitro Techniques; Oxadiazoles; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Specific Pathogen-Free Organisms; Sumatriptan; Vasoconstriction

2000
Effect of 5-HT(1B) receptor ligands on self-administration of ethanol in an operant procedure in rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:1

    Topics: Alcohol Drinking; Animals; Conditioning, Operant; Ethanol; Indoles; Male; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration

2000
Augmentation with a 5-HT(1A), but not a 5-HT(1B) receptor antagonist critically depends on the dose of citalopram.
    European journal of pharmacology, 2000, May-26, Volume: 397, Issue:1

    Topics: Animals; Autoreceptors; Citalopram; Dose-Response Relationship, Drug; Drug Synergism; Hippocampus; Injections, Subcutaneous; Male; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Agents; Time Factors

2000
Zolmitriptan stimulates a Ca(2+)-dependent K(+) current in C6 glioma cells stably expressing recombinant human 5-HT(1B) receptors.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: Animals; Calcium; Dose-Response Relationship, Drug; Humans; Membrane Potentials; Oxadiazoles; Oxazoles; Oxazolidinones; Peptides; Piperazines; Potassium Channels; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Fusion Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Tetraethylammonium; Tryptamines; Tumor Cells, Cultured

2000
5-HT(1A) and 5-HT(1B/1D) receptors are involved in the modulation of the trigeminovascular system of the cat: a microiontophoretic study.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Benzopyrans; Cats; Electric Stimulation; Iontophoresis; Oxadiazoles; Piperazines; Propylamines; Pyridines; Pyrimidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Trigeminal Caudal Nucleus

2000
Altered expression and functions of serotonin 5-HT1A and 5-HT1B receptors in knock-out mice lacking the 5-HT transporter.
    The European journal of neuroscience, 2000, Volume: 12, Issue:7

    Topics: Animals; Autoreceptors; Binding, Competitive; Brain Chemistry; Carrier Proteins; Citalopram; Dipeptides; Down-Regulation; Gene Expression; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Hydroxyindoleacetic Acid; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Nerve Tissue Proteins; Oxadiazoles; Piperazines; Pyridines; Pyrimidines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; RNA, Messenger; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Spiro Compounds; Substantia Nigra; Sulfur Radioisotopes; Synaptic Transmission; Tritium

2000
Mediation of 5-HT-induced internal carotid vasodilatation in GR127935- and ritanserin-pretreated dogs by 5-HT7 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 362, Issue:2

    Topics: Animals; Carotid Arteries; Dogs; Female; Hemodynamics; In Vitro Techniques; Male; Oxadiazoles; Piperazines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sympathectomy; Vagotomy; Vasodilation

2000
Chronic clomipramine alters presynaptic 5-HT(1B) and postsynaptic 5-HT(1A) receptor sensitivity in rat hypothalamus and hippocampus, respectively.
    Neuropharmacology, 2000, Volume: 39, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Tricyclic; Clomipramine; Corticosterone; Cyclic AMP; Hippocampus; Hypothalamus; Male; Microdialysis; Oxadiazoles; Piperazines; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Presynaptic; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists

2000
Chronic repetitive transcranial magnetic stimulation induces subsensitivity of presynaptic serotonergic autoreceptor activity in rat brain.
    Neuroreport, 2000, Sep-11, Volume: 11, Issue:13

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Depression; Male; Microdialysis; Oxadiazoles; Piperazines; Prefrontal Cortex; Presynaptic Terminals; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Transcranial Magnetic Stimulation

2000
Effects of a selective 5-HT(1B/1D) receptor agonist on spinal and trigeminal reflexes in the anaesthetized rabbit.
    British journal of pharmacology, 2000, Volume: 131, Issue:5

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Female; Heart Rate; Male; Oxadiazoles; Pain; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reflex; Serotonin Receptor Agonists; Spinal Cord; Trigeminal Caudal Nucleus

2000
In vivo analysis of adrenergic and serotoninergic constrictions of the rabbit saphenous vein.
    European journal of pharmacology, 2000, Nov-24, Volume: 408, Issue:3

    Topics: Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthesia; Animals; Benzazepines; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Indoles; Injections, Intravenous; Isoindoles; Oxadiazoles; Peripheral Nervous System; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Agents; Serotonin Receptor Agonists; Sumatriptan; Tetrahydronaphthalenes; Time Factors; Ultrasonography, Doppler; Vasoconstrictor Agents

2000
Functional effects of corticosterone on 5-HT(1A) and 5-HT(1B) receptor activity in rat brain: in vivo microdialysis studies.
    European journal of pharmacology, 2001, Jan-05, Volume: 411, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Inflammatory Agents; Brain; Colforsin; Corticosterone; Cyclic AMP; Hippocampus; Hypothalamus; Male; Microdialysis; Oxadiazoles; Piperazines; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2001
5-HT1B Autoreceptors limit the effects of selective serotonin re-uptake inhibitors in mouse hippocampus and frontal cortex.
    Journal of neurochemistry, 2001, Volume: 76, Issue:3

    Topics: Animals; Antidepressive Agents, Second-Generation; Autoreceptors; Drug Combinations; Frontal Lobe; Hippocampus; Male; Mice; Mice, Knockout; Microdialysis; Oxadiazoles; Paroxetine; Piperazines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reference Values; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

2001
Modulation of the effects of cocaine by 5-HT1B receptors: a comparison of knockouts and antagonists.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 67, Issue:3

    Topics: Animals; Cocaine; Corpus Striatum; Dopamine Uptake Inhibitors; Male; Mice; Mice, Knockout; Motor Activity; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Antagonists

2000
Role of 5-HT(1A) and 5-HT(1B) receptors in the mediation of behavior in the forced swim test in mice.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 24, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Tricyclic; Behavior, Animal; Dose-Response Relationship, Drug; Female; Imipramine; Indoles; Mice; Mice, Inbred Strains; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Pyridines; Reaction Time; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2001
Unravelling the pharmacological profile of the canine external carotid vasodilator '5-HT1-like' receptors: coexistence of sympatho-inhibitory 5-HT1B and postjunctional 5-HT7 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:1

    Topics: 5-Methoxytryptamine; Acetylcholine; Animals; Biphenyl Compounds; Blood Flow Velocity; Blood Pressure; Carotid Artery, External; Chromans; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Hemodynamics; Male; Neuromuscular Junction; Oxadiazoles; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sumatriptan; Sympathetic Nervous System; Vasodilation

2001
The GR127935-sensitive 5-HT(1) receptors mediating canine internal carotid vasoconstriction: resemblance to the 5-HT(1B), but not to the 5-HT(1D) or 5-ht(1F), receptor subtype.
    British journal of pharmacology, 2001, Volume: 132, Issue:5

    Topics: Animals; Blood Pressure; Carotid Artery, Internal; Dogs; Female; Heart Rate; Male; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT1F; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoconstriction

2001
Serotonin-induced hypercontraction through 5-hydroxytryptamine 1B receptors in atherosclerotic rabbit coronary arteries.
    Circulation, 2001, Mar-06, Volume: 103, Issue:9

    Topics: Animals; Arteriosclerosis; Calcium; Coronary Vessels; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Oxadiazoles; Phenylephrine; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction

2001
Effect of serotonin (5-HT)1B receptor ligands on cocaine sensitization in rats.
    Behavioural pharmacology, 2001, Volume: 12, Issue:2

    Topics: Animals; Cocaine-Related Disorders; Discrimination Learning; Drug Interactions; Drug Tolerance; Male; Motivation; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2001
[5-HT1B serotonin receptors and antidepressant effects of selective serotonin reuptake inhibitors ].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 2001, Volume: 324, Issue:5

    Topics: Animals; Antidepressive Agents; Drug Synergism; Frontal Lobe; Hippocampus; Male; Mice; Mice, Knockout; Microdialysis; Oxadiazoles; Paroxetine; Piperazines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

2001
Complex interaction of ergovaline with 5-HT2A, 5-HT1B/1D, and alpha1 receptors in isolated arteries of rat and guinea pig.
    Journal of animal science, 2001, Volume: 79, Issue:8

    Topics: Animals; Arteries; Ergotamines; Guinea Pigs; Iliac Artery; Ketanserin; Norepinephrine; Oxadiazoles; Piperazines; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Vasoconstriction

2001
No involvement of 5-HT(7) or 5-HT(1D) receptors in the (R)-8-OH-DPAT-induced depression of the monosynaptic reflex in spinalized rats.
    European journal of pharmacology, 2001, Sep-14, Volume: 427, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Clozapine; Decerebrate State; Dose-Response Relationship, Drug; Ergolines; Indoles; Male; Methiothepin; Oxadiazoles; Phenols; Piperazines; Pyridines; Rats; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Time Factors

2001
LY393558, a 5-hydroxytryptamine reuptake inhibitor and 5-HT(1B/1D) receptor antagonist: effects on extracellular levels of 5-hydroxytryptamine in the guinea pig and rat.
    European journal of pharmacology, 2001, Nov-30, Volume: 432, Issue:1

    Topics: Administration, Oral; Animals; Cyclic S-Oxides; Dose-Response Relationship, Drug; Extracellular Space; Female; Fenfluramine; Fluoxetine; Frontal Lobe; Guinea Pigs; Hypothalamus; Injections, Intraperitoneal; Male; Oxadiazoles; Paroxetine; Piperazines; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Tetrodotoxin; Thiadiazines; Time Factors

2001
Contribution of the 5-HT(1B) receptor to hypoxia-induced pulmonary hypertension: converging evidence using 5-HT(1B)-receptor knockout mice and the 5-HT(1B/1D)-receptor antagonist GR127935.
    Circulation research, 2001, Dec-07, Volume: 89, Issue:12

    Topics: Animals; Atmosphere Exposure Chambers; Blood Pressure; Chronic Disease; Heart Rate; Heart Ventricles; Hypertension, Pulmonary; Hypoxia; In Vitro Techniques; Lung; Male; Mice; Mice, Inbred Strains; Mice, Knockout; Organ Size; Oxadiazoles; Piperazines; Pulmonary Artery; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoconstrictor Agents; Vasodilator Agents; Ventricular Dysfunction, Right

2001
Pharmacological studies of the acute effects of (+)-3,4-methylenedioxymethamphetamine on locomotor activity: role of 5-HT(1B/1D) and 5-HT(2) receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 26, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Fluorobenzenes; Hallucinogens; Indoles; Male; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Oxadiazoles; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists

2002
Effects of chronically administered venlafaxine on 5-HT receptor activity in rat hippocampus and hypothalamus.
    European journal of pharmacology, 2002, Feb-01, Volume: 436, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Corticosterone; Cyclohexanols; Hippocampus; Hypothalamus; Male; Oxadiazoles; Oxytocin; Piperazines; Rats; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Venlafaxine Hydrochloride

2002
Anxiogenic-like effect of serotonin(1B) receptor stimulation in the rat elevated plus-maze.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 71, Issue:4

    Topics: Animals; Anxiety; Behavior, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Serotonin 2C receptor agonists and the behavioural satiety sequence in mice.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 71, Issue:4

    Topics: Aminopyridines; Animals; Diet; Dose-Response Relationship, Drug; Ethylamines; Feeding Behavior; Indoles; Mice; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Satiety Response; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Activation of 5-HT(1B) receptors in the nucleus accumbens reduces self-administration of amphetamine on a progressive ratio schedule.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 71, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Amphetamines; Animals; Central Nervous System Stimulants; Conditioning, Operant; Dose-Response Relationship, Drug; Food; Male; Nucleus Accumbens; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reinforcement Schedule; Self Administration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Effects of donitriptan on carotid haemodynamics and cardiac output distribution in anaesthetized pigs.
    Cephalalgia : an international journal of headache, 2002, Volume: 22, Issue:1

    Topics: Animals; Blood Flow Velocity; Blood Pressure; Brain; Cardiac Output; Carotid Arteries; Dose-Response Relationship, Drug; Heart Rate; Nitriles; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Regional Blood Flow; Serotonin Antagonists; Serotonin Receptor Agonists; Swine; Tryptamines; Vascular Resistance

2002
Multiple 5-HT receptors are involved in the effects of acute MDMA treatment: studies on locomotor activity and responding for conditioned reinforcement.
    Psychopharmacology, 2002, Volume: 162, Issue:3

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Ethylamines; Indoles; Ketanserin; Male; Motor Activity; Oxadiazoles; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors

2002
Functional effects of chronic electroconvulsive shock on serotonergic 5-HT(1A) and 5-HT(1B) receptor activity in rat hippocampus and hypothalamus.
    Brain research, 2002, Oct-11, Volume: 952, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cyclic AMP; Electroshock; Extracellular Space; Hippocampus; Hypothalamus; Male; Oxadiazoles; Piperazines; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission

2002
An evaluation of the effect of NAS-181, a new selective 5-HT(1B) receptor antagonist, on extracellular 5-HT levels in rat frontal cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:2

    Topics: Animals; Benzopyrans; Dose-Response Relationship, Drug; Extracellular Fluid; Extracellular Space; Fluvoxamine; Frontal Lobe; Male; Microdialysis; Morpholines; Oxadiazoles; Piperazines; Piperidones; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Spiro Compounds; Time Factors

2003
Donitriptan selectively decreases jugular venous oxygen saturation in the anesthetized pig: further insights into its mechanism of action relevant to headache relief.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:2

    Topics: Anesthesia; Animals; Blood Gas Analysis; Carbon Dioxide; Carotid Arteries; Electrocardiography; Headache; Hemodynamics; Hemoglobins; Jugular Veins; Male; Nitriles; Oxadiazoles; Oxygen; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swine; Tryptamines; Vascular Resistance; Vasoconstriction

2003
Role of 5-HT1B/D receptors in canine gastric accommodation: effect of sumatriptan and 5-HT1B/D receptor antagonists.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:1

    Topics: Animals; Atropine; Benzamides; Bethanechol; Biphenyl Compounds; Dogs; Enzyme Inhibitors; Female; Gastric Emptying; NG-Nitroarginine Methyl Ester; Oxadiazoles; Parasympatholytics; Parasympathomimetics; Piperazines; Pressure; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Sumatriptan; Vagus Nerve

2003
Serotonin transporter inhibitors protect against hypoxic pulmonary hypertension.
    American journal of respiratory and critical care medicine, 2003, Aug-15, Volume: 168, Issue:4

    Topics: Analysis of Variance; Animals; Carrier Proteins; Chronic Disease; Citalopram; Disease Models, Animal; Fluoxetine; Hypertension, Pulmonary; Hypertrophy, Right Ventricular; Hypoxia; Ketanserin; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Muscle, Smooth, Vascular; Nerve Tissue Proteins; Oxadiazoles; Piperazines; Pulmonary Artery; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Statistics, Nonparametric

2003
The differential effects of food restriction on 5-HT1A and 5-HT1B receptor mediated control of serotonergic transmission in the hippocampus and hypothalamus of rats.
    Nutritional neuroscience, 2003, Volume: 6, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Weight; Female; Hippocampus; Hypothalamus; Oxadiazoles; Piperazines; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003
Effects of chronic paroxetine treatment on dialysate serotonin in 5-HT1B receptor knockout mice.
    Journal of neurochemistry, 2003, Volume: 86, Issue:1

    Topics: Animals; Brain Chemistry; Carrier Proteins; Chromatography, High Pressure Liquid; Dialysis Solutions; Drug Administration Routes; Extracellular Space; Hippocampus; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Microdialysis; Nerve Tissue Proteins; Oxadiazoles; Paroxetine; Piperazines; Prefrontal Cortex; Pyridines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Time

2003
Pharmacological profile of the 5-HT-induced inhibition of cardioaccelerator sympathetic outflow in pithed rats: correlation with 5-HT1 and putative 5-ht5A/5B receptors.
    British journal of pharmacology, 2003, Volume: 140, Issue:4

    Topics: Animals; Autonomic Fibers, Preganglionic; Blood Pressure; Decerebrate State; Desipramine; Disease Models, Animal; Drug Therapy, Combination; Electric Stimulation; Ergotamine; Infusions, Intravenous; Injections, Intravenous; Male; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sympathetic Nervous System; Tachycardia

2003
Further characterization of the 5-HT1 receptors mediating cardiac sympatho-inhibition in pithed rats: pharmacological correlation with the 5-HT1B and 5-HT1D subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 369, Issue:2

    Topics: Animals; Biphenyl Compounds; Decerebrate State; Male; Norepinephrine; Oxadiazoles; Piperazines; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Sympathomimetics; Tachycardia

2004
The 5-hydroxytryptamine1B/1D/1F receptor agonists eletriptan and naratriptan inhibit trigeminovascular input to the nucleus tractus solitarius in the cat.
    Brain research, 2004, Feb-13, Volume: 998, Issue:1

    Topics: Action Potentials; Animals; Cats; Drug Interactions; Electric Stimulation; Indoles; Maximum Tolerated Dose; Neural Inhibition; Oxadiazoles; Piperazines; Piperidines; Pyrrolidines; Reaction Time; Receptor, Serotonin, 5-HT1F; Receptors, Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Trigeminal Nuclei; Tryptamines

2004
Extracellular superoxide enhances 5-HT-induced murine pulmonary artery vasoconstriction.
    American journal of physiology. Lung cellular and molecular physiology, 2004, Volume: 287, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Antioxidants; Endothelium, Vascular; Extracellular Fluid; Humans; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Nitric Oxide; Oxadiazoles; Oxidants; Piperazines; Pulmonary Artery; Serotonin; Serotonin Antagonists; Superoxides; Vasoconstriction; Vasoconstrictor Agents

2004
Rewarding effects elicited by cocaine microinjections into the ventral tegmental area of C57BL/6 mice: involvement of dopamine D1 and serotonin1B receptors.
    Psychopharmacology, 2004, Volume: 174, Issue:3

    Topics: Analysis of Variance; Anesthetics, Local; Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Mice, Inbred C57BL; Microinjections; Oxadiazoles; Piperazines; Reaction Time; Receptor, Serotonin, 5-HT1B; Receptors, Dopamine D1; Reward; Self Administration; Serotonin Antagonists; Spatial Behavior; Ventral Tegmental Area

2004
Effect of combined administration of 5-HT1A or 5-HT1B/1D receptor antagonists and antidepressants in the forced swimming test.
    European journal of pharmacology, 2004, Mar-08, Volume: 487, Issue:1-3

    Topics: Adrenergic Uptake Inhibitors; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Citalopram; Depression; Desipramine; Imipramine; Male; Moclobemide; Monoamine Oxidase Inhibitors; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Swimming

2004
5-HT receptors involved in opioid-activated descending inhibition of spinal withdrawal reflexes in the decerebrated rabbit.
    Pain, 2004, Volume: 109, Issue:1-2

    Topics: Afferent Pathways; Analgesics, Opioid; Analysis of Variance; Animals; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Female; Fentanyl; Indoles; Injections, Intraventricular; Male; Muscle, Skeletal; Neural Inhibition; Oxadiazoles; Piperazines; Quinolines; Rabbits; Reaction Time; Receptors, Serotonin; Reflex; Serotonin Antagonists; Spinal Cord; Tropisetron

2004
Tonic regulation of satiety by 5-HT receptors in the mouse: converging evidence from behavioural and c-fos immunoreactivity studies?
    The European journal of neuroscience, 2004, Volume: 19, Issue:11

    Topics: Animals; Behavior, Animal; Body Weight; Brain; Dose-Response Relationship, Drug; Drug Interactions; Eating; Feeding Behavior; Gene Expression Regulation; Immunohistochemistry; Mice; Mice, Knockout; Oxadiazoles; Piperazines; Piperidones; Proto-Oncogene Proteins c-fos; Pyridines; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Time Factors

2004
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines

2004
Rho kinase-induced nuclear translocation of ERK1/ERK2 in smooth muscle cell mitogenesis caused by serotonin.
    Circulation research, 2004, Sep-17, Volume: 95, Issue:6

    Topics: Active Transport, Cell Nucleus; Amides; Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Division; Cells, Cultured; Cytochalasin D; Enzyme Activation; Intracellular Signaling Peptides and Proteins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Myosin-Light-Chain Phosphatase; Oxadiazoles; Phosphoproteins; Phosphorylation; Piperazines; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein Subunits; Protein Transport; Pulmonary Artery; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Recombinant Fusion Proteins; rho-Associated Kinases; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Signal Transduction; Thiazoles; Thiazolidines; Transcription Factors

2004
Endogenously released 5-hydroxytryptamine depresses the spinal monosynaptic reflex via 5-HT1D receptors.
    European journal of pharmacology, 2004, Oct-25, Volume: 503, Issue:1-3

    Topics: Animals; Biphenyl Compounds; Clorgyline; Decerebrate State; Male; Monoamine Oxidase Inhibitors; Oxadiazoles; p-Chloroamphetamine; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1D; Reflex, Monosynaptic; Serotonin; Serotonin Agents; Serotonin Antagonists; Spinal Cord

2004
Effects of a selective 5-HT1B receptor agonist and antagonists in animal models of anxiety and depression.
    Behavioural pharmacology, 2004, Volume: 15, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Anxiety; Behavior, Animal; Benzamides; Conflict, Psychological; Depressive Disorder; Diazepam; Electroshock; Exploratory Behavior; Imipramine; Male; Mice; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Reaction Time; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2004
Autoradiographic characterisation of [35S]GTPgammaS binding stimulation mediated by 5-HT1B receptor in postmortem human brain.
    Neuropharmacology, 2005, Volume: 48, Issue:1

    Topics: Aged; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain; Dipeptides; Drug Interactions; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidones; Postmortem Changes; Protein Binding; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfur Isotopes

2005
3,4-N-methlenedioxymethamphetamine-induced hypophagia is maintained in 5-HT1B receptor knockout mice, but suppressed by the 5-HT2C receptor antagonist RS102221.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:6

    Topics: Animals; Body Weight; Eating; Hallucinogens; Kinetics; Male; Mice; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Spiro Compounds; Starvation; Sulfonamides

2005
The anxiolytic-like effect of 5-HT1B receptor ligands in rats: a possible mechanism of action.
    The Journal of pharmacy and pharmacology, 2005, Volume: 57, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzamides; Conflict, Psychological; Diazepam; Disease Models, Animal; Drinking Behavior; Drug Administration Schedule; Electroshock; Flumazenil; Men; Neurons; Oxadiazoles; p-Chloroamphetamine; Piperazines; Poland; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Water

2005
Differential effects of 5-HT2C receptor ligands on place conditioning and locomotor activity in rats.
    European journal of pharmacology, 2005, May-16, Volume: 515, Issue:1-3

    Topics: Aminopyridines; Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Indoles; Ligands; Male; Motor Activity; Oxadiazoles; Piperazines; Pyrazines; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Time Factors

2005
The effect of chronic selective serotonin reuptake inhibitor treatment on serotonin 1B receptor sensitivity and HPA axis activity.
    Progress in neuro-psychopharmacology & biological psychiatry, 2005, Volume: 29, Issue:5

    Topics: Adrenocorticotropic Hormone; Animals; Brain; Catecholamines; Citalopram; Corticosterone; Extracellular Space; Hippocampus; Hypothalamo-Hypophyseal System; Male; Microdialysis; Oxadiazoles; Piperazines; Piperidones; Prefrontal Cortex; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Presynaptic; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Spiro Compounds

2005
Donitriptan decreases jugular venous oxygen saturation in rats in the absence of cranial vasoconstriction: an overlooked mechanism of antimigraine action?
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 315, Issue:2

    Topics: Animals; Blood Gas Analysis; Cerebrovascular Circulation; Hemodynamics; Jugular Veins; Male; Migraine Disorders; Nitriles; Oxadiazoles; Oxygen; Piperazines; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tryptamines; Vasoconstriction

2005
SB-616234-A (1-[6-(cis-3,5-dimethylpiperazin-1-yl)-2,3-dihydro-5-methoxyindol-1-yl]-1-[2'methyl-4'-(5-methyl-1,2,3-oxadiazol-3-yl)biphenyl-4-yl]methanone hydrochloride): a novel, potent and selective 5-HT1B receptor antagonist.
    Neuropharmacology, 2006, Volume: 50, Issue:8

    Topics: Analysis of Variance; Animals; Binding, Competitive; Cerebral Cortex; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; In Vitro Techniques; Indoles; Membrane Potentials; Neurons; Oxadiazoles; Patch-Clamp Techniques; Piperazines; Protein Binding; Rats; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Sulfur Isotopes; Tritium

2006
5-HT(1B) receptors, ventral orbitofrontal cortex, and aggressive behavior in mice.
    Psychopharmacology, 2006, Volume: 185, Issue:4

    Topics: Aggression; Animals; Behavior, Animal; Data Interpretation, Statistical; Dose-Response Relationship, Drug; Limbic System; Male; Mice; Microinjections; Oxadiazoles; Piperazines; Prefrontal Cortex; Pyridines; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists

2006
Evidence for adenosine- and serotonin-mediated antihyperalgesic effects of cizolirtine in rats suffering from diabetic neuropathy.
    Neuropharmacology, 2007, Volume: 52, Issue:2

    Topics: Adenosine; Analgesics; Animals; Area Under Curve; Caffeine; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Hyperalgesia; Male; Oxadiazoles; Pain Measurement; Pain Threshold; Piperazines; Psychomotor Performance; Pyrazoles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Vocalization, Animal

2007
Delay aversion: effects of 7-OH-DPAT, 5-HT1A/1B-receptor stimulation and D-cycloserine.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 85, Issue:4

    Topics: Animals; Central Nervous System Stimulants; Cycloserine; Dextroamphetamine; Impulsive Behavior; Male; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Dopamine D3; Receptors, N-Methyl-D-Aspartate; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Tetrahydronaphthalenes

2006
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:3

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin

2007
A61603-induced contractions of the porcine meningeal artery are mediated by alpha1- and alpha2-adrenoceptors.
    Basic & clinical pharmacology & toxicology, 2007, Volume: 100, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Alkaloids; Animals; Benzophenanthridines; Colforsin; Dose-Response Relationship, Drug; Female; Forecasting; Imidazoles; In Vitro Techniques; Meningeal Arteries; Methiothepin; Norepinephrine; Oxadiazoles; Phenylephrine; Piperazines; Potassium Chloride; Prazosin; Protein Kinase C; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Swine; Tetrahydronaphthalenes; Vasoconstriction; Yohimbine

2007
Anti-aggressive effects of agonists at 5-HT1B receptors in the dorsal raphe nucleus of mice.
    Psychopharmacology, 2007, Volume: 193, Issue:2

    Topics: Aggression; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Male; Mice; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Raphe Nuclei; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists

2007
Pharmacological evidence that 5-HT(1B/1D) receptors mediate hypotension in anesthetized rats.
    European journal of pharmacology, 2007, Dec-08, Volume: 576, Issue:1-3

    Topics: Anesthesia; Animals; Blood Pressure; Hypotension; Male; Oxadiazoles; Phenols; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2007
In vivo/ex vivo and behavioural study on central effects of 5-HT1B/1D and 5-HT1A antagonists in guinea pigs.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 88, Issue:3

    Topics: Animals; Behavior, Animal; Brain Chemistry; Depression; Female; Guinea Pigs; Hydroxyindoleacetic Acid; Microdialysis; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin; Serotonin Antagonists; Swimming

2008
Serotonergic mediation of aggression in high and low aggressive chicken strains.
    Poultry science, 2008, Volume: 87, Issue:4

    Topics: Agonistic Behavior; Animals; Body Weight; Chickens; Dopamine; Epinephrine; Female; Norepinephrine; Oxadiazoles; Piperazines; Random Allocation; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Selection, Genetic; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists

2008
Effect of co-administration of the selective 5-HT1A receptor antagonist WAY 100,635 and selective 5-HT1B/1D receptor antagonist GR 127,935 on anxiolytic effect of citalopram in conditioned fear stress in the rat.
    European journal of pharmacology, 2008, May-31, Volume: 586, Issue:1-3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Citalopram; Conditioning, Psychological; Data Interpretation, Statistical; Fear; Male; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Stress, Psychological; Synaptic Transmission

2008
Progesterone reduces the effect of the serotonin 1B/1D receptor antagonist, GR 127935, on lordosis behavior.
    Hormones and behavior, 2009, Volume: 55, Issue:1

    Topics: Analysis of Variance; Animals; Catheterization; Estradiol; Estrogens; Female; Ovariectomy; Oxadiazoles; Piperazines; Posture; Progesterone; Rats; Rats, Inbred F344; Restraint, Physical; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus

2009
Serotonin1B heteroreceptor activation induces an antidepressant-like effect in mice with an alteration of the serotonergic system.
    Journal of psychiatry & neuroscience : JPN, 2008, Volume: 33, Issue:6

    Topics: 5,7-Dihydroxytryptamine; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Behavior, Animal; Citalopram; Dopamine; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Chronic reductions in serotonin transporter function prevent 5-HT1B-induced behavioral effects in mice.
    Biological psychiatry, 2009, Mar-01, Volume: 65, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Female; Fluoxetine; Globus Pallidus; Indoles; Mice; Mice, Inbred BALB C; Mice, Knockout; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Reflex, Startle; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Plasma Membrane Transport Proteins; Substantia Nigra

2009
Effects of systemic 5-HT(1B) receptor compounds on ventral tegmental area intracranial self-stimulation thresholds in rats.
    European journal of pharmacology, 2009, Feb-14, Volume: 604, Issue:1-3

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Reward; Self Stimulation; Sensory Thresholds; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Ventral Tegmental Area

2009
Effect of central serotonin depletion on 5-HT receptor-mediated vasomotor responses in the middle meningeal artery of anaesthetized rats.
    Autonomic & autacoid pharmacology, 2009, Volume: 29, Issue:1-2

    Topics: 5,7-Dihydroxytryptamine; Anesthesia; Animals; Blood Pressure; Cerebrovascular Circulation; Dopamine; Heart Rate; Male; Meningeal Arteries; Meninges; Norepinephrine; Oxadiazoles; Paraventricular Hypothalamic Nucleus; Phenols; Piperazines; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Vasodilation

2009
Pharmacological profile of the inhibition by dihydroergotamine and methysergide on the cardioaccelerator sympathetic outflow in pithed rats.
    European journal of pharmacology, 2009, Jun-10, Volume: 612, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Blood Pressure; Decerebrate State; Dihydroergotamine; Dose-Response Relationship, Drug; Drug Combinations; Electric Stimulation; Heart Rate; Hemodynamics; Male; Methysergide; Norepinephrine; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, alpha-2; Serotonin Antagonists; Sympathetic Nervous System; Tachycardia; Yohimbine

2009
High-resolution imaging of brain 5-HT 1B receptors in the rhesus monkey using [11C]P943.
    Nuclear medicine and biology, 2010, Volume: 37, Issue:2

    Topics: Animals; Brain; Carbon Radioisotopes; Macaca mulatta; Magnetic Resonance Imaging; Oxadiazoles; Piperazines; Positron-Emission Tomography; Pyrrolidinones; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Antagonists; Substrate Specificity

2010
Differential involvement of 5-HT(1A) and 5-HT(1B/1D) receptors in human interferon-alpha-induced immobility in the mouse forced swimming test.
    Arzneimittel-Forschung, 2010, Volume: 60, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Depression; Fluoxetine; Interferon-alpha; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2010
Pulmonary vascular effects of serotonin and selective serotonin reuptake inhibitors in the late-gestation ovine fetus.
    American journal of physiology. Lung cellular and molecular physiology, 2011, Volume: 301, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Dose-Response Relationship, Drug; Female; Fetus; Fluoxetine; Hemodynamics; Hypertension, Pulmonary; Hysterotomy; Indoles; Ketanserin; Lung; Oxadiazoles; Piperazines; Pregnancy; Pulmonary Artery; Pyridines; Receptors, Serotonin; rho-Associated Kinases; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Sertraline; Sheep; Vascular Resistance

2011
Effects of selective serotonin antagonism on central neurotransmission.
    Poultry science, 2012, Volume: 91, Issue:4

    Topics: Aggression; Animals; Chickens; Chromatography, High Pressure Liquid; Female; Hypothalamus; Oxadiazoles; Piperazines; Random Allocation; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Selection, Genetic; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Species Specificity; Synaptic Transmission

2012
5-HT7 receptor-mediated meningeal dilatation induced by 5-carboxamidotryptamine in rats is not altered by 5-HT depletion and chronic corticosterone treatment.
    Proceedings of the Western Pharmacology Society, 2011, Volume: 54

    Topics: Animals; Brain; Corticosterone; Male; Meningeal Arteries; Oxadiazoles; Phenols; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Sulfonamides; Vasodilation

2011
Intrathecal dihydroergotamine inhibits capsaicin-induced vasodilatation in the canine external carotid circulation via GR127935- and rauwolscine-sensitive receptors.
    European journal of pharmacology, 2012, Oct-05, Volume: 692, Issue:1-3

    Topics: Acetylcholine; Animals; Blood Circulation; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Arteries; Dihydroergotamine; Dogs; Dose-Response Relationship, Drug; Hemodynamics; Injections, Spinal; Male; Oxadiazoles; Piperazines; Propylene Glycol; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Antagonists; Vasodilation; Vasodilator Agents; Yohimbine

2012
Lasting neurobehavioral abnormalities in rats after neonatal activation of serotonin 1A and 1B receptors: possible mechanisms for serotonin dysfunction in autistic spectrum disorders.
    Psychopharmacology, 2014, Volume: 231, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Brain; Citalopram; Exploratory Behavior; Female; Freezing Reaction, Cataleptic; Locomotion; Male; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Social Behavior

2014
Modulation of 5-HT7 receptor: effect on object recognition performances in mice.
    Psychopharmacology, 2014, Volume: 231, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Male; Memory, Episodic; Mice; Oxadiazoles; Phenols; Piperazines; Receptors, Serotonin; Recognition, Psychology; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2014
Possible involvement of CA1 5-HT1B/1D and 5-HT2A/2B/2C receptors in harmaline-induced amnesia.
    Pharmacology, biochemistry, and behavior, 2014, Volume: 125

    Topics: Amnesia; Animals; CA1 Region, Hippocampal; Central Nervous System Stimulants; Cinanserin; Harmaline; Male; Memory; Mice, Inbred Strains; Oxadiazoles; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists

2014
GR-127935-sensitive mechanism mediating hypotension in anesthetized rats: are 5-HT5B receptors involved?
    Journal of cardiovascular pharmacology, 2015, Volume: 65, Issue:4

    Topics: Animals; Biphenyl Compounds; Blood Pressure; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ergotamine; Hypotension; Oxadiazoles; Piperazines; Piperidones; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds

2015
Role of spinal 5-HT5A, and 5-HT1A/1B/1D, receptors in neuropathic pain induced by spinal nerve ligation in rats.
    Brain research, 2015, Oct-05, Volume: 1622

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Female; Ganglia, Spinal; Hyperalgesia; Lumbar Vertebrae; Methiothepin; Neuralgia; Oxadiazoles; Piperazines; Pyridines; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Spinal Nerves; Touch

2015
5-hydroxytryptamine receptor (5-HT1DR) promotes colorectal cancer metastasis by regulating Axin1/β-catenin/MMP-7 signaling pathway.
    Oncotarget, 2015, Sep-22, Volume: 6, Issue:28

    Topics: Animals; Axin Protein; beta Catenin; Blotting, Western; Cell Line, Tumor; Cell Movement; Colorectal Neoplasms; Female; Gene Expression Regulation, Neoplastic; HCT116 Cells; HT29 Cells; Humans; Immunohistochemistry; Male; Matrix Metalloproteinase 7; Mice, Nude; Middle Aged; Neoplasm Metastasis; Oxadiazoles; Piperazines; Receptor, Serotonin, 5-HT1D; Reverse Transcriptase Polymerase Chain Reaction; Serotonin Antagonists; Signal Transduction; Tumor Burden; Xenograft Model Antitumor Assays

2015
The involvement of medial septum 5-HT1 and 5-HT2 receptors on ACPA-induced memory consolidation deficit: possible role of TRPC3, TRPC6 and TRPV2.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:11

    Topics: Animals; Arachidonic Acids; Avoidance Learning; Cinanserin; Imidazoles; Male; Memory Consolidation; Memory Disorders; Oxadiazoles; Piperazines; Pyridines; Rats; Septal Nuclei; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; TRPC Cation Channels

2015
Serotonergic regulation of distention-induced ATP release from the urothelium.
    American journal of physiology. Renal physiology, 2016, 04-01, Volume: 310, Issue:7

    Topics: Adenosine Triphosphate; Animals; Citalopram; Dioxanes; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin, 5-HT4; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Urinary Bladder; Urothelium

2016
Serotonin antagonists fail to alter MDMA self-administration in rats.
    Pharmacology, biochemistry, and behavior, 2016, Volume: 148

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Drug-Seeking Behavior; Extinction, Psychological; Ketanserin; Male; N-Methyl-3,4-methylenedioxyamphetamine; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Self Administration; Serotonin Antagonists

2016
The inhibitory effect of combination treatment with leptin and cannabinoid CB1 receptor agonist on food intake and body weight gain is mediated by serotonin 1B and 2C receptors.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2016, Volume: 67, Issue:3

    Topics: Aminopyridines; Animals; Cannabinoid Receptor Agonists; Drug Synergism; Eating; Indoles; Leptin; Male; Oxadiazoles; Piperazines; Piperidines; Pyrazoles; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Weight Gain

2016
Activation and Deactivation of 5-HT1 Receptor of Accumbens Shell Area does not Alter ACPA-induced Aversive Memory Deficit in Male Rat.
    Archives of Iranian medicine, 2017, Volume: 20, Issue:3

    Topics: Animals; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Exploratory Behavior; Male; Maze Learning; Memory; Memory Disorders; Microinjections; Nucleus Accumbens; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists

2017
Attenuation of serotonin-induced itch by sumatriptan: possible involvement of endogenous opioids.
    Archives of dermatological research, 2018, Volume: 310, Issue:2

    Topics: Animals; Disease Models, Animal; Drug Therapy, Combination; Humans; Injections, Intradermal; Male; Mice; Naltrexone; Narcotic Antagonists; Opioid Peptides; Oxadiazoles; Piperazines; Pruritus; Quaternary Ammonium Compounds; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Sumatriptan

2018
Functional Characterization of the Prejunctional Receptors Mediating the Inhibition by Ergotamine of the Rat Perivascular Sensory Peptidergic Drive.
    ACS chemical neuroscience, 2019, 07-17, Volume: 10, Issue:7

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Autonomic Nervous System; Blood Pressure; Calcitonin Gene-Related Peptide; Dopamine Antagonists; Electric Stimulation; Ergotamine; Haloperidol; Heart Rate; Male; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Yohimbine

2019
Sumatriptan Increases Skin Flap Survival through Activation of 5-Hydroxytryptamine 1b/1d Receptors in Rats: The Mediating Role of the Nitric Oxide Pathway.
    Plastic and reconstructive surgery, 2019, Volume: 144, Issue:1

    Topics: Animals; Graft Survival; Male; Nitric Oxide; Oxadiazoles; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Skin Transplantation; Sumatriptan; Surgical Flaps; Vasodilator Agents

2019
Involvement of 5-HT1B/1D receptors in the inflammatory response and oxidative stress in intestinal ischemia/reperfusion in rats.
    European journal of pharmacology, 2020, Sep-05, Volume: 882

    Topics: Animals; Calcitonin Gene-Related Peptide; Ileum; Inflammation; Intestinal Mucosa; Male; Mesenteric Ischemia; Oxadiazoles; Oxidative Stress; Piperazines; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Reperfusion Injury; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Sumatriptan

2020