go 6976 and wortmannin

go 6976 has been researched along with wortmannin in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (13.64)18.2507
2000's17 (77.27)29.6817
2010's2 (9.09)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
Bilter, GK; Dias, J; Huang, Z; Keon, BH; Lamerdin, J; MacDonald, ML; Michnick, SW; Minami, T; Owens, S; Shang, Z; Westwick, JK; Yu, H1
Giranda, VL; Johnson, EF; Luo, Y; Stewart, KD; Woods, KW1
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Alexander, JS; Kevil, CG; Mire, E; Payne, DK1
Shibuya, M; Takahashi, T; Ueno, H1
Barnes, PJ; Giembycz, MA; Hellewell, PG; Lindsay, MA; Lynch, OT1
Adlersberg, M; Gershon, MD; Hsiung, S; Liu, K; Sacktor, T; Tamir, H1
Fathallah, H; Giraud, F; Mazière, P; Sauvage, M1
Ishizawa, M; Ishizuka, T; Kajita, K; Kanoh, Y; Miura, A; Yasuda, K1
Altura, BM; Altura, BT; Wang, J; Yang, ZW; Zheng, T2
Chang, LC; Wang, JP1
Barnes, PJ; Giembycz, MA; Lindsay, MA; Lynch, OT1
Farnell, MB; Genovese, K; He, H; Kogut, MH1
Anel, A; Boyer, C; Buferne, M; Martínez-Lorenzo, MJ; Naval, J; Pardo, J; Schmitt-Verhulst, AM1
Altura, BM; Altura, BT; Li, J; Li, W; Liu, W1
Choi, HJ; Kim, CH; Park, YG1
Nakamura, J1
Churikov, D; Price, CM1
Boaglio, AC; Crocenzi, FA; Mottino, AD; Ochoa, JE; Pellegrino, JM; Roma, MG; Sánchez Pozzi, EJ; Vore, M; Zucchetti, AE1
Karam, M; Lassarre, C; Legay, C; Ricort, JM1

Other Studies

22 other study(ies) available for go 6976 and wortmannin

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Identifying off-target effects and hidden phenotypes of drugs in human cells.
    Nature chemical biology, 2006, Volume: 2, Issue:6

    Topics: Bacterial Proteins; Cell Line; Cell Proliferation; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Genetics; Humans; Luminescent Proteins; Molecular Structure; Phenotype; Recombinant Fusion Proteins; Signal Transduction; Structure-Activity Relationship

2006
Pharmacological and functional comparison of the polo-like kinase family: insight into inhibitor and substrate specificity.
    Biochemistry, 2007, Aug-21, Volume: 46, Issue:33

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Androstadienes; Binding Sites; Cell Cycle Proteins; Humans; Models, Molecular; Molecular Sequence Data; Peptide Library; Polo-Like Kinase 1; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Pteridines; Substrate Specificity; Wortmannin

2007
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Vascular permeability factor/vascular endothelial cell growth factor-mediated permeability occurs through disorganization of endothelial junctional proteins.
    The Journal of biological chemistry, 1998, Jun-12, Volume: 273, Issue:24

    Topics: Androstadienes; Antigens, CD; Cadherins; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cell Membrane Permeability; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Flavonoids; Histocytochemistry; Humans; Indoles; Lymphokines; Membrane Proteins; Muscle, Smooth, Vascular; Nitriles; Occludin; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Serum Albumin; Staurosporine; Tyrphostins; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin

1998
VEGF activates protein kinase C-dependent, but Ras-independent Raf-MEK-MAP kinase pathway for DNA synthesis in primary endothelial cells.
    Oncogene, 1999, Apr-01, Volume: 18, Issue:13

    Topics: 3T3 Cells; Adenoviridae; Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Chromones; DNA Replication; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genes, ras; Genetic Vectors; Indoles; Lymphokines; Maleimides; MAP Kinase Kinase Kinase 1; Mice; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Isoforms; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-raf; Proto-Oncogene Proteins p21(ras); Rats; Receptor Protein-Tyrosine Kinases; Receptors, Growth Factor; Receptors, Vascular Endothelial Growth Factor; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin

1999
'Outside-in' signalling mechanisms underlying CD11b/CD18-mediated NADPH oxidase activation in human adherent blood eosinophils.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: Androstadienes; Carbazoles; CD18 Antigens; Cell Adhesion; Cell Count; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Humans; Imidazoles; Indoles; Isoenzymes; Macrophage-1 Antigen; Maleimides; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Pyrazoles; Pyridines; Pyrimidines; Signal Transduction; src-Family Kinases; Superoxides; Tetradecanoylphorbol Acetate; Wortmannin

1999
Ca(2+)-evoked serotonin secretion by parafollicular cells: roles in signal transduction of phosphatidylinositol 3'-kinase, and the gamma and zeta isoforms of protein kinase C.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Feb-15, Volume: 20, Issue:4

    Topics: Androstadienes; Animals; Calcium; Calcium Channels; Carbazoles; Cell Membrane; Cells, Cultured; Cytosol; Enzyme Inhibitors; Indoles; Isoenzymes; Naphthalenes; Phosphatidylinositol 3-Kinases; Protein Kinase C; Serotonin; Sheep; Signal Transduction; Tetradecanoylphorbol Acetate; Thyroid Gland; Wortmannin

2000
Insulin stimulates NHE1 activity by sequential activation of phosphatidylinositol 3-kinase and protein kinase C zeta in human erythrocytes.
    European journal of biochemistry, 2000, Volume: 267, Issue:4

    Topics: Androstadienes; Biological Transport; Carbazoles; Enzyme Activation; Erythrocytes; Humans; Indoles; Insulin; Isoenzymes; Maleimides; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Phosphotyrosine; Precipitin Tests; Protein Binding; Protein Kinase C; Protein Kinase C-alpha; Signal Transduction; Sodium-Hydrogen Exchangers; Time Factors; Wortmannin

2000
The role of atypical and conventional PKC in dehydroepiandrosterone-induced glucose uptake and dexamethasone-induced insulin resistance.
    Biochemical and biophysical research communications, 2000, Oct-22, Volume: 277, Issue:2

    Topics: Adipocytes; Adjuvants, Immunologic; Androstadienes; Animals; Antimetabolites; Carbazoles; Cells, Cultured; Dehydroepiandrosterone; Deoxyglucose; Dexamethasone; Enzyme Activation; Enzyme Inhibitors; Genes, Dominant; Glucocorticoids; Glucose; Indoles; Insulin Antagonists; Insulin Resistance; Male; Myristic Acids; Phosphatidylinositol 3-Kinases; Precipitin Tests; Protein Kinase C; Rats; Time Factors; Transfection; Wortmannin

2000
Low [Mg(2+)](o) induces contraction and [Ca(2+)](i) rises in cerebral arteries: roles of ca(2+), PKC, and PI3.
    American journal of physiology. Heart and circulatory physiology, 2000, Volume: 279, Issue:6

    Topics: Androstadienes; Animals; Anticoagulants; Basilar Artery; Caffeine; Calcium; Carbazoles; Chromones; Dogs; Enzyme Inhibitors; Extracellular Space; Heparin; In Vitro Techniques; Indoles; Magnesium; Maleimides; Morpholines; Muscle, Smooth, Vascular; Phosphatidylinositol 3-Kinases; Phosphodiesterase Inhibitors; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Ryanodine; Signal Transduction; Thapsigargin; Vasoconstriction; Wortmannin

2000
Importance of PKC and PI3Ks in ethanol-induced contraction of cerebral arterial smooth muscle.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:5

    Topics: Androstadienes; Animals; Basilar Artery; Calcium; Carbazoles; Central Nervous System Depressants; Chromones; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethanol; Indoles; Male; Maleimides; Morpholines; Muscle, Smooth, Vascular; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Signal Transduction; Stroke; Vasoconstriction; Vasospasm, Intracranial; Wortmannin

2001
Signal transduction pathways for activation of extracellular signal-regulated kinase by arachidonic acid in rat neutrophils.
    Journal of leukocyte biology, 2001, Volume: 69, Issue:4

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Androstadienes; Animals; Arachidonic Acid; Arachidonic Acids; Butadienes; Calcium; Carbazoles; Chelating Agents; Chromones; Cyclooxygenase Inhibitors; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; GTP-Binding Protein alpha Subunits, Gi-Go; Heterotrimeric GTP-Binding Proteins; Indoles; Lipoxygenase Inhibitors; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Neutrophils; Nitriles; Pertussis Toxin; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Processing, Post-Translational; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Type C Phospholipases; Virulence Factors, Bordetella; Wortmannin

2001
Pharmacological comparison of LTB(4)-induced NADPH oxidase activation in adherent and non-adherent guinea-pig eosinophils.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Androstadienes; Animals; Antibodies; Carbazoles; CD18 Antigens; Cell Adhesion; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Enzyme Precursors; Eosinophils; Flavonoids; Guinea Pigs; Imidazoles; Indoles; Integrin beta1; Intracellular Signaling Peptides and Proteins; Leukotriene B4; Macrophage-1 Antigen; Male; Maleimides; Mitogen-Activated Protein Kinases; NADPH Oxidases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein-Tyrosine Kinases; Pyrazoles; Pyridines; Pyrimidines; Rats; src-Family Kinases; Stilbenes; Syk Kinase; Time Factors; Wortmannin

2001
Pharmacological analysis of signal transduction pathways required for oxidative burst in chicken heterophils stimulated by a Toll-like receptor 2 agonist.
    International immunopharmacology, 2003, Volume: 3, Issue:12

    Topics: Androstadienes; Animals; Animals, Newborn; Carbazoles; Chickens; Estrenes; Flavonoids; Indoles; Lipopolysaccharides; Male; Membrane Glycoproteins; Neutrophils; Nitriles; Pyrrolidinones; Receptors, Cell Surface; Respiratory Burst; Signal Transduction; Sulfones; Teichoic Acids; Toll-Like Receptor 2; Toll-Like Receptors; Wortmannin

2003
Differential implication of protein kinase C isoforms in cytotoxic T lymphocyte degranulation and TCR-induced Fas ligand expression.
    International immunology, 2003, Volume: 15, Issue:12

    Topics: Acetophenones; Androstadienes; Animals; Antibodies, Monoclonal; Benzopyrans; Carbazoles; Cell Degranulation; Cell Line; Chromones; Cycloheximide; Cytotoxicity, Immunologic; Dactinomycin; Fas Ligand Protein; Humans; Indoles; Ionomycin; Isoenzymes; Jurkat Cells; Luciferases; Lymphocyte Activation; Membrane Glycoproteins; Mice; Morpholines; Perforin; Phorbol Esters; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pore Forming Cytotoxic Proteins; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Protein Kinase C-theta; Receptor-CD3 Complex, Antigen, T-Cell; Receptors, Antigen, T-Cell; Signal Transduction; T-Lymphocytes, Cytotoxic; Transfection; Wortmannin

2003
Mechanisms of hydroxyl radical-induced contraction of rat aorta.
    European journal of pharmacology, 2004, Sep-19, Volume: 499, Issue:1-2

    Topics: Androstadienes; Animals; Aorta; Calcium; Carbazoles; Cells, Cultured; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Ferrous Compounds; Genistein; Hydrogen Peroxide; Hydroxyl Radical; In Vitro Techniques; Indoles; Male; Maleimides; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Phosphoinositide-3 Kinase Inhibitors; Proadifen; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Staurosporine; Vasoconstriction; Wortmannin

2004
Lactosylceramide alpha2,3-sialyltransferase is induced via a PKC/ERK/CREB-dependent pathway in K562 human leukemia cells.
    Molecules and cells, 2007, Apr-30, Volume: 23, Issue:2

    Topics: 5' Flanking Region; Androstadienes; Carbazoles; Cell Differentiation; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Humans; Indoles; K562 Cells; Megakaryocytes; Mutation; Neuraminidase; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Promoter Regions, Genetic; Protein Kinase C; Sialyltransferases; Signal Transduction; Tetradecanoylphorbol Acetate; Wortmannin

2007
Protein kinase C-dependent antilipolysis by insulin in rat adipocytes.
    Biochimica et biophysica acta, 2007, Volume: 1771, Issue:9

    Topics: Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Androstadienes; Angiotensin II; Animals; Carbazoles; Carcinogens; Dobutamine; Enzyme Activation; Enzyme Inhibitors; Glycerol; Imidazoles; Indoles; Insulin; Isoenzymes; Lipolysis; Male; Maleimides; Protein Kinase C; Rats; Receptor, Insulin; Tetradecanoylphorbol Acetate; Wortmannin

2007
Pot1 and cell cycle progression cooperate in telomere length regulation.
    Nature structural & molecular biology, 2008, Volume: 15, Issue:1

    Topics: Androstadienes; Ataxia Telangiectasia Mutated Proteins; Caffeine; Carbazoles; Cell Cycle; Cell Cycle Proteins; Cell Line; DNA-Binding Proteins; Enzyme Inhibitors; Flow Cytometry; G2 Phase; Humans; Indoles; Kinetics; Protein Serine-Threonine Kinases; S Phase; Shelterin Complex; Tamoxifen; Telomere; Telomere-Binding Proteins; Tumor Suppressor Proteins; Wortmannin

2008
Phosphoinositide 3-kinase/protein kinase B signaling pathway is involved in estradiol 17β-D-glucuronide-induced cholestasis: complementarity with classical protein kinase C.
    Hepatology (Baltimore, Md.), 2010, Volume: 52, Issue:4

    Topics: 1-Phosphatidylinositol 4-Kinase; Androstadienes; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Canaliculi; Biliary Tract; Carbazoles; Cholestasis; Colchicine; Endocytosis; Estradiol; Glutathione; In Vitro Techniques; Male; Microtubules; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Perfusion; Protein Kinase C; Proto-Oncogene Proteins c-akt; Rats; Rats, Wistar; Signal Transduction; Taurocholic Acid; Wortmannin

2010
Phosphatidylinositol 3-kinase and protein kinase D1 specifically cooperate to negatively regulate the insulin-like growth factor signaling pathway.
    Biochimica et biophysica acta, 2012, Volume: 1823, Issue:2

    Topics: Androstadienes; Carbazoles; Cell Line, Tumor; Enzyme Inhibitors; Epidermal Growth Factor; Extracellular Signal-Regulated MAP Kinases; Fibroblast Growth Factors; Humans; Indoles; Insulin Receptor Substrate Proteins; Maleimides; Phosphatidylinositol 3-Kinase; Protein Kinase C; Signal Transduction; Somatomedins; Wortmannin

2012