go 6976 has been researched along with tetradecanoylphorbol acetate in 112 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 25 (22.32) | 18.2507 |
2000's | 66 (58.93) | 29.6817 |
2010's | 19 (16.96) | 24.3611 |
2020's | 2 (1.79) | 2.80 |
Authors | Studies |
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Schächtele, C; Seifert, R; Wenzel-Seifert, K | 1 |
Dickens, G; Guroff, G; Lavarreda, M; Zheng, WH | 1 |
Harris, TE; Jones, PM; Persaud, SJ | 1 |
Goode, N; Keenan, C; Pears, C | 1 |
Houghton, PJ; Luo, W; Sharif, M; Sharif, TR | 1 |
Alameda, F; Batlle, E; de Herreros, AG; del Mont Llosas, M; Díaz, V; Domínguez, D; Loukili, N; Paciucci, R; Verdú, J | 1 |
Ikeda, K; Kawasaki, M; Kumakura, K; Misonou, H; Murakami, T; Ohara-Imaizumi, M; Wakai, T | 1 |
MacGlashan, DW; Miura, K | 1 |
Chik, CL; Ho, AK; Negishi, T; Ogiwara, T | 1 |
El-Mansoury, AM; Morgan, NG | 1 |
Solem, ML; Thomas, AP | 1 |
Alderton, JM; Bi, GQ; Steinhardt, RA; Togo, T | 1 |
Bissonnette, M; Brasitus, TA; Khare, S; Scaglione-Sewell, B; Sitrin, MD; Wali, RK | 1 |
Chaban, VV; Dirksen, ER; Woodruff, ML; Worley, CM | 1 |
Shibuya, M; Takahashi, T; Ueno, H | 1 |
Araki, E; Furukawa, N; Kaneko, K; Kishikawa, H; Matsumoto, K; Motoshima, H; Shichiri, M; Shirotani, T; Todaka, M; Tsuruzoe, K; Yoshizato, K | 1 |
Buchan, AM; Meloche, RM; Moore, ED; Ring, M; Scriven, DR; Smith, VC | 1 |
Baudier, J; Deloulme, JC; Delphin, C; Scotto, C | 1 |
Foster, DA; Frankel, P; Hornia, A; Joseph, T; Lu, Z; Sukezane, T; Zhong, M | 1 |
Inoue, T; Koono, M; Nabeshima, K; Shimao, Y | 1 |
Palmer, TM; Stiles, GL | 1 |
Altman, A; Genestier, L; Green, DR; Kasibhatla, S; Mahboubi, A; Villalba, M | 1 |
Barnes, PJ; Giembycz, MA; Hellewell, PG; Lindsay, MA; Lynch, OT | 1 |
Gear, AR; Polanowska-Grabowska, R | 1 |
Farokhzad, OC; Hrnjez, BJ; Matthews, JB; Song, JC | 1 |
Eckert, RL; Efimova, T | 1 |
Adlersberg, M; Gershon, MD; Hsiung, S; Liu, K; Sacktor, T; Tamir, H | 1 |
Kataoka, H; Kobayashi, H; Koono, M; Minami, S; Shiraishi, S; Wada, A; Yamamoto, R; Yanagita, T; Yokoo, H | 1 |
Kataoka, K; Nakamura, Y; Si, Q | 1 |
Chang, RC; Hong, JS; Jeohn, GH; Kim, WG; Mohney, RP; Wetsel, WC; Wilson, B | 1 |
Hong, JS; Jeohn, GH; Wetsel, WC; Wilson, B | 1 |
Häussermann, S; Marks, F; Rennecke, J; Richter, KH; Stempka, L; Stöhr, M; Strand, S | 1 |
Hunziker, IP; Keller, HU; Niggli, V; Sordat, B; Sroka, J | 1 |
Bruni, P; Cencetti, F; Donati, C; Meacci, E; Romiti, E | 1 |
Clarke, H; Ginanni, N; Laughlin, KV; Mullin, JM; Pettit, GR; Smith, JB | 1 |
Honda, S; Kohsaka, S; Kurihara, T; Nakajima, K; Tohyama, Y | 1 |
Shibuya, M; Takahashi, T | 1 |
Giardina, JB; Khalil, RA; Tanner, DJ | 1 |
Zawalich, KC; Zawalich, WS | 1 |
Braileanu, GT; Hu, J; Mirando, MA | 1 |
Chen, JS; Song, JG | 1 |
Crow, T; Neary, JT; Siddiqi, V; Xue-Bian, JJ | 1 |
Koo, EH; Lin, YH; McMahon, T; Messing, RO; Wang, D; Zhu, G | 1 |
Cruciani, V; Husøy, T; Mikalsen, SO | 1 |
Honda, S; Imai, Y; Kohsaka, S; Kurihara, T; Nakajima, K; Tohyama, Y | 1 |
Biswas, DK; Cruz, A; Dai, SC; Graner, E; Pardee, AB; Weiser, B | 1 |
Cidlowski, JA; Gómez-Angelats, M | 1 |
Hur, SY; Ki, IK; Kim, JW; Kim, TE; Kim, YW; Lee, JM; Namkoong, SE | 1 |
Albert, PR; Kushwaha, N; Penington, NJ; Wu, X | 1 |
Greenstein, S; Hendey, B; Zhu, CL | 1 |
Barritault, D; Crépin, M; Ledoux, D; Liu, JF; Liu, JM | 1 |
Auberger, P; Bottero, V; Busuttil, V; Frelin, C; Imbert, V; Peyron, JF; Ricci, JE | 1 |
Bollag, WB; Calle, RA; Jung, E | 1 |
Fährmann, M; Kaufhold, M; Rieg, T; Seidler, U | 1 |
González, MI; Kazanietz, MG; Robinson, MB | 1 |
Matthews, JB; Rangachari, PK; Song, JC | 1 |
Chen, YZ; Huang, XY; Qiu, J; Wang, CG | 1 |
Brown, MA; Hock, MB | 1 |
Ito, H; Kato, K; Kozawa, O; Niwa, M; Oiso, Y; Tokuda, H | 1 |
Chain, BM; Cho, JY; Katz, DR | 1 |
Abe-Dohmae, S; Hayashi, M; Ikeda, Y; Matsuo, M; Okuhira, K; Ueda, K; Yokoyama, S | 1 |
Chang, YY; Sun, SH; Wang, CM | 1 |
Dutta, S; Häussinger, D; Kubitz, R; Kühlkamp, T; Saha, N; vom Dahl, S; Wettstein, M | 1 |
Ding, L; Lang, W; Wang, H; Xiao, L | 1 |
Imamura, T; Ishisaki, A; Tsunobuchi, H | 1 |
Blois, JT; Chiles, TC; Mataraza, JM; Mecklenbraüker, I; Tarakhovsky, A | 1 |
Azuma, C; Hama-Inaba, H; Hayata, I; Kojima, S; Nakajima, T; Ohyama, H; Wang, B; Yukawa, O | 1 |
Chignell, CF; He, YY; Huang, JL | 1 |
Gylfe, E; Rask, L; Sakwe, AM | 1 |
Cruciani, V; Flørenes, VA; Jørgensen, K; Mikalsen, SO; Skrede, M; Slipicevic, A | 1 |
Chang, Q; Soper, BD; Tepperman, BL | 1 |
Bhoumik, A; Habelhah, H; López-Bergami, P; Ronai, Z; Wang, LH; Zhang, W | 1 |
Ikewaki, N; Inoko, H; Kulski, JK | 1 |
Gosens, R; Grootte Bromhaar, MM; Maarsingh, H; Meurs, H; Nelemans, SA; ten Damme, A; Zaagsma, J | 1 |
Hayashi, H; Kondo, T; Suzuki, S; Takagi, K; Ueyama, J; Wakusawa, S | 1 |
Li, F; Shi, J; Song, J; Wang, D; Zhou, Y | 1 |
Di Jeso, B; Elia, MG; Marsigliante, S; Muscella, A; Storelli, C; Treglia, AS; Ulianich, L | 1 |
Grybko, MJ; Pores-Fernando, AT; Wurth, GA; Zweifach, A | 1 |
Aronson, PS; Hassan, HA; Karniski, LP; Mentone, S; Rajendran, VM | 1 |
Fan, Y; Li, HL; Li, ZW; Teng, ZY; Wu, XW; Zhang, YN; Zhang, YQ | 1 |
Chou, CC; Hsu, CY; Yung, BY | 1 |
Choi, HJ; Kim, CH; Park, YG | 1 |
Bíró, T; Griger, Z; Kovács, I; Kovács, L; Páyer, E; Sipka, S; Tóth, BI | 1 |
Gergely, P; Kovács, I; Sipka, S; Szíjgyártó, Z; Szucs, K; Zákány, R | 1 |
Nakamura, J | 1 |
Abdullah, LH; Davis, CW; Ehre, C; Messing, RO; Nakayama, K; Nakayama, KI; Olsen, J; Zhu, Y | 1 |
Czerwinski, P; Förstermann, U; Hortmann, M; Li, H; Sohn, HY; Xu, H | 1 |
Hanai, Y; Kozawa, O; Matsushima-Nishiwaki, R; Minamitani, C; Otsuka, T; Takai, S; Tokuda, H | 1 |
Friis, MB; Lambert, IH; Vorum, KG | 1 |
Alexander, JS; Carpenter, AC | 1 |
Fujikake, T; Fujioka, K; Hanamoto, T; Ikeda, T; Ishizuka, T; Kajita, K; Mori, I; Morita, H; Nagano, I; Okada, H; Takahashi, Y; Uno, Y; Zhiliang, W | 1 |
Du, CL; Liu, XS; Qiao, LF; Xie, JG; Xie, M; Xu, YJ; Zhang, J; Zhang, ZX | 1 |
Arun, SN; Bollag, WB; Dodd, ME; Xie, D; Zhong, X | 1 |
Higuchi, C; Nakura, A; Yoshida, K; Yoshikawa, H | 1 |
Krafczyk, K; Lee, AC; Murray, M; Zhou, F; Zhu, L | 1 |
Adapala, RK; Bratz, IN; Meszaros, JG; Suzuki, M; Talasila, PK; Thodeti, CK; Zhang, DX | 1 |
Lai, R; Li, S; Lin, W; Tchantchou, F; Wen, J; Zhang, Y | 1 |
Bloehs, R; Joss, N; Karle, CA; Katus, HA; Scherer, D; Scholz, EP; Seyler, C; Thomas, D; Völkers, M; Welke, F; Zhang, W; Zitron, E | 1 |
Hu, JM; Ma, LT; Qin, SZ; Xu, GZ; Xu, ZX | 1 |
Gao, B; Ingram, AJ; Krepinsky, JC; Peng, F; Zhang, Y | 1 |
Chock, PB; Oubrahim, H; Wilson, BA; Wong, A | 1 |
Furue, MK; Hirata, M; Hirayama, N; Kawamura, S; Kinehara, M; Kohara, A; Matsumura, H; Mimura, S; Suga, M; Tateyama, D; Uchio-Yamada, K; Yanagihara, K | 1 |
Erdjument-Bromage, H; Gao, C; Guo, S; Kao, HY; Liu, Y; Miyagi, M; Su, YT; Tempst, P; Wang, A; Wang, B | 1 |
Chaudhari, S; Cunningham, JT; Ding, M; Ding, Y; He, S; Krishnamoorthy, R; Ma, R; Stankowska, D; Wang, Y; Yuan, J | 1 |
Brown, GC; Hornik, TC; Neniskyte, U | 1 |
Czerwinski, P; Förstermann, U; Li, H; Xia, N; Xu, H | 1 |
Brown, GC; Fricker, M; Neniskyte, U | 1 |
Arias-Montaño, JA; Escamilla-Sánchez, J; García-Hernández, U; Montejo-López, W; Rivera-Ramírez, N | 1 |
Choi, YJ; Clarke, CJ; Hannun, YA; Liu, M; Obeid, LM; Salama, MF | 1 |
Bertelsen, V; Dietrich, M; Malik, MS; Skeie, M; Stang, E | 1 |
Leng, TD; Li, J; Xiong, ZG; Yang, T; Zhang, L | 1 |
Karhu, ST; Ruskoaho, H; Talman, V | 1 |
112 other study(ies) available for go 6976 and tetradecanoylphorbol acetate
Article | Year |
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N-protein kinase C isoenzymes may be involved in the regulation of various neutrophil functions.
Topics: Carbazoles; Enzyme Activation; Humans; In Vitro Techniques; Indoles; Isoenzymes; Maleimides; Muramidase; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Protein Kinase C; Respiratory Burst; Superoxides; Tetradecanoylphorbol Acetate | 1994 |
Involvement of protein kinase C in nerve growth factor- and K-252a-stimulated calcium uptake into PC12 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Calcium; Calcium Channel Agonists; Carbazoles; Carcinogens; Enzyme Inhibitors; Indole Alkaloids; Indoles; Isoenzymes; Naphthalenes; Nerve Growth Factors; PC12 Cells; Phorbol Esters; Protein Kinase C; Protein Kinase C-alpha; Rats; Receptors, Nerve Growth Factor; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate | 1997 |
Gö 6976: an inhibitor of Ca2+/DAG-dependent protein kinase C isoforms in islets of Langerhans.
Topics: Animals; Calcium; Carbazoles; Cells, Cultured; Cricetinae; Diglycerides; Enzyme Inhibitors; Glucose; Indoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Isoenzymes; Kinetics; Pancreatic Neoplasms; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1997 |
Isoform specificity of activators and inhibitors of protein kinase C gamma and delta.
Topics: Acetophenones; Alkaloids; Benzophenanthridines; Benzopyrans; Bryostatins; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Indoles; Isoenzymes; Lactones; Macrolides; Maleimides; Naphthalenes; Phenanthridines; Protein Kinase C; Protein Kinase C-delta; Recombinant Proteins; Schizosaccharomyces; Sphingosine; Tetradecanoylphorbol Acetate; Transformation, Genetic | 1997 |
CGP 41251 and tamoxifen selectively inhibit mitogen-activated protein kinase activation and c-Fos phosphoprotein induction by substance P in human astrocytoma cells.
Topics: Astrocytoma; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Proto-Oncogene Proteins c-fos; Staurosporine; Substance P; Tamoxifen; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tyrosine | 1997 |
Protein kinase C-alpha activity inversely modulates invasion and growth of intestinal cells.
Topics: Animals; Cadherins; Carbazoles; Cell Adhesion; Cell Movement; Cell Size; Gene Expression Regulation, Neoplastic; Humans; Indoles; Maleimides; Mice; Mice, Nude; Mutagenesis, Site-Directed; Neoplasm Invasiveness; Neoplasms, Experimental; Protein Kinase C; Tetradecanoylphorbol Acetate; Transfection; Transplantation, Heterologous; Tumor Cells, Cultured; Urokinase-Type Plasminogen Activator | 1998 |
Protein kinase C controls the priming step of regulated exocytosis in adrenal chromaffin cells.
Topics: Adenosine Triphosphate; Adrenal Medulla; Animals; Antibodies; Calcium; Carbazoles; Catecholamines; Cattle; Cells, Cultured; Chromaffin Cells; Enzyme Inhibitors; Exocytosis; GAP-43 Protein; Indoles; Peptide Fragments; Protein Kinase C; Tetradecanoylphorbol Acetate | 1998 |
Expression of protein kinase C isozymes in human basophils: regulation by physiological and nonphysiological stimuli.
Topics: Antibodies, Anti-Idiotypic; Basophils; Biological Transport; Calcium; Carbazoles; Cell Membrane; Cells, Cultured; Enzyme Induction; Enzyme Inhibitors; Histamine Release; Humans; Indoles; Ionomycin; Ionophores; Isoenzymes; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; Naphthalenes; Protein Kinase C; Tetradecanoylphorbol Acetate | 1998 |
Differential effects of two protein kinase C inhibitors, calphostin C and Gö6976, on pineal cyclic nucleotide accumulation.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Carbazoles; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Indoles; Isoproterenol; Male; Naphthalenes; Nucleotides, Cyclic; Phosphodiesterase Inhibitors; Pineal Gland; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1998 |
Activation of protein kinase C modulates alpha2-adrenergic signalling in rat pancreatic islets.
Topics: Adrenergic alpha-Agonists; Animals; Carbazoles; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Glucose; GTP-Binding Proteins; In Vitro Techniques; Indoles; Insulin; Insulin Secretion; Islets of Langerhans; Male; Norepinephrine; Phosphorylation; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Signal Transduction; Substrate Specificity; Tetradecanoylphorbol Acetate | 1998 |
Modulation of cardiac Ca2+ channels by IGF1.
Topics: Animals; Calcium; Calcium Channels; Carbazoles; Cells, Cultured; Chromones; Cytosol; Enzyme Inhibitors; Heart; Humans; Indoles; Insulin-Like Growth Factor I; Isoquinolines; Kinetics; Male; Manganese; Morpholines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Sarcolemma; Sulfonamides; Tetradecanoylphorbol Acetate | 1998 |
The mechanism of facilitated cell membrane resealing.
Topics: 3T3 Cells; Animals; Brefeldin A; Calcium; Carbazoles; Cell Membrane; Cytochalasin D; Endocytosis; Enzyme Activation; Enzyme Inhibitors; Exocytosis; Fluorescent Dyes; Indoles; Maleimides; Mice; Protein Kinase C; Pyridinium Compounds; Quaternary Ammonium Compounds; Tetradecanoylphorbol Acetate | 1999 |
1,25-dihydroxyvitamin D3 and TPA activate phospholipase D in Caco-2 cells: role of PKC-alpha.
Topics: Caco-2 Cells; Calcitriol; Calcium; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Ionomycin; Isoenzymes; Kinetics; Maleimides; Phospholipase D; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Tetradecanoylphorbol Acetate | 1999 |
PKC role in mechanically induced Ca2+ waves and ATP-induced Ca2+ oscillations in airway epithelial cells.
Topics: Adenosine Triphosphate; Animals; Calcium; Carbazoles; Cell Membrane; Cells, Cultured; Diglycerides; Electric Stimulation; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Indoles; Kinetics; Maleimides; Oscillometry; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Trachea | 1999 |
VEGF activates protein kinase C-dependent, but Ras-independent Raf-MEK-MAP kinase pathway for DNA synthesis in primary endothelial cells.
Topics: 3T3 Cells; Adenoviridae; Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Chromones; DNA Replication; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genes, ras; Genetic Vectors; Indoles; Lymphokines; Maleimides; MAP Kinase Kinase Kinase 1; Mice; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Isoforms; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-raf; Proto-Oncogene Proteins p21(ras); Rats; Receptor Protein-Tyrosine Kinases; Receptors, Growth Factor; Receptors, Vascular Endothelial Growth Factor; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin | 1999 |
Possible involvement of atypical protein kinase C (PKC) in glucose-sensitive expression of the human insulin gene: DNA-binding activity and transcriptional activity of pancreatic and duodenal homeobox gene-1 (PDX-1) are enhanced via calphostin C-sensitive
Topics: Animals; Carbazoles; Cell Line; DNA; Enzyme Inhibitors; Gene Expression; Glucose; Homeodomain Proteins; Humans; Indoles; Insulin; Islets of Langerhans; Mice; Naphthalenes; Phosphoric Monoester Hydrolases; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Trans-Activators; Transcription, Genetic; Transfection | 1999 |
The role of protein kinase C isozymes in bombesin-stimulated gastrin release from human antral gastrin cells.
Topics: Adult; Biological Transport; Bombesin; Carbazoles; Female; Gastrin-Secreting Cells; Gastrins; Humans; Image Processing, Computer-Assisted; Immunohistochemistry; Indoles; Isoenzymes; Male; Maleimides; Naphthalenes; Protein Kinase C; Pyloric Antrum; Tetradecanoylphorbol Acetate | 1999 |
Concerted regulation of wild-type p53 nuclear accumulation and activation by S100B and calcium-dependent protein kinase C.
Topics: Animals; Biological Transport; Calcium Signaling; Calcium-Binding Proteins; Carbazoles; Cell Nucleus; G1 Phase; Indoles; Mice; Nerve Growth Factors; Protein Kinase C; Rats; S100 Calcium Binding Protein beta Subunit; S100 Proteins; Tetradecanoylphorbol Acetate; Tumor Suppressor Protein p53 | 1999 |
Antagonistic effects of protein kinase C alpha and delta on both transformation and phospholipase D activity mediated by the epidermal growth factor receptor.
Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; Cell Transformation, Neoplastic; Cells, Cultured; Crosses, Genetic; Epidermal Growth Factor; ErbB Receptors; Indoles; Isoenzymes; Models, Genetic; Mutagenesis, Insertional; Phospholipase D; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Rats; Recombinant Proteins; Tetradecanoylphorbol Acetate | 1999 |
TPA-enhanced motility and invasion in a highly metastatic variant (L-10) of human rectal adenocarcinoma cell line RCM-1: selective role of PKC-alpha and its inhibition by a combination of PDBu-induced PKC downregulation and antisense oligonucleotides trea
Topics: Adenocarcinoma; Base Sequence; Carbazoles; Down-Regulation; Humans; Indoles; Isoenzymes; Naphthalenes; Neoplasm Invasiveness; Neoplasm Metastasis; Oligonucleotides, Antisense; Phorbol 12,13-Dibutyrate; Phorbol Esters; Protein Kinase C; Protein Kinase C-alpha; Rectal Neoplasms; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1999 |
Stimulation of A(2A) adenosine receptor phosphorylation by protein kinase C activation: evidence for regulation by multiple protein kinase C isoforms.
Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; CHO Cells; Consensus Sequence; Cricetinae; Cyclic AMP; Dogs; Endothelin-1; Enzyme Activation; Enzyme Inhibitors; Glioma; Indoles; Isoenzymes; Maleimides; Mutagenesis, Site-Directed; Phosphorylation; Protein Kinase C; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Signal Transduction; Tetradecanoylphorbol Acetate; Triazines; Triazoles; Tumor Cells, Cultured | 1999 |
Protein kinase ctheta cooperates with calcineurin to induce Fas ligand expression during activation-induced T cell death.
Topics: Acetophenones; Animals; Apoptosis; Benzopyrans; Binding Sites; Calcineurin; Carbazoles; DNA-Binding Proteins; Drug Interactions; Fas Ligand Protein; Gene Expression Regulation; Humans; Indoles; Ionomycin; Isoenzymes; Jurkat Cells; Membrane Glycoproteins; Mice; Mutation; NFATC Transcription Factors; Nuclear Proteins; Promoter Regions, Genetic; Protein Kinase C; Protein Kinase C-theta; Signal Transduction; T-Lymphocytes; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Transcription Factors | 1999 |
'Outside-in' signalling mechanisms underlying CD11b/CD18-mediated NADPH oxidase activation in human adherent blood eosinophils.
Topics: Androstadienes; Carbazoles; CD18 Antigens; Cell Adhesion; Cell Count; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Humans; Imidazoles; Indoles; Isoenzymes; Macrophage-1 Antigen; Maleimides; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Pyrazoles; Pyridines; Pyrimidines; Signal Transduction; src-Family Kinases; Superoxides; Tetradecanoylphorbol Acetate; Wortmannin | 1999 |
Activation of protein kinase C is required for the stable attachment of adherent platelets to collagen but is not needed for the initial rapid adhesion under flow conditions.
Topics: Animals; Antibodies; Blood Flow Velocity; Blood Platelets; Blood Proteins; Carbazoles; Carcinogens; Cell Adhesion Molecules; Collagen; Enzyme Inhibitors; Enzyme Precursors; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Indoles; Integrins; Intracellular Signaling Peptides and Proteins; Maleimides; Phosphoproteins; Phosphorylation; Platelet Adhesiveness; Protein Conformation; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Receptors, Collagen; Skin; Stimulation, Chemical; Syk Kinase; Tetradecanoylphorbol Acetate; Tyrosine | 1999 |
PKC-epsilon regulates basolateral endocytosis in human T84 intestinal epithelia: role of F-actin and MARCKS.
Topics: Acetophenones; Acetylcholine; Actin Cytoskeleton; Actins; Amino Acid Sequence; Benzopyrans; Biological Transport; Carbachol; Carbazoles; Carcinogens; Cell Membrane; Cell Polarity; Cells, Cultured; Cholinergic Agonists; Cross-Linking Reagents; Cytochalasin D; Diglycerides; Endocytosis; Enzyme Inhibitors; Epithelial Cells; Humans; Indoles; Intestines; Intracellular Signaling Peptides and Proteins; Isoenzymes; Maleimides; Membrane Proteins; Molecular Sequence Data; Myristoylated Alanine-Rich C Kinase Substrate; Nucleic Acid Synthesis Inhibitors; Pinocytosis; Protein Kinase C; Protein Kinase C-epsilon; Proteins; Tetradecanoylphorbol Acetate | 1999 |
Regulation of human involucrin promoter activity by novel protein kinase C isoforms.
Topics: Acetophenones; Benzopyrans; Carbazoles; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Genes, Dominant; Humans; Indoles; Isoenzymes; Keratinocytes; Luciferases; Plasmids; Promoter Regions, Genetic; Protein Isoforms; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Protein Precursors; Proto-Oncogene Proteins c-fos; Tetradecanoylphorbol Acetate; Transfection | 2000 |
Ca(2+)-evoked serotonin secretion by parafollicular cells: roles in signal transduction of phosphatidylinositol 3'-kinase, and the gamma and zeta isoforms of protein kinase C.
Topics: Androstadienes; Animals; Calcium; Calcium Channels; Carbazoles; Cell Membrane; Cells, Cultured; Cytosol; Enzyme Inhibitors; Indoles; Isoenzymes; Naphthalenes; Phosphatidylinositol 3-Kinases; Protein Kinase C; Serotonin; Sheep; Signal Transduction; Tetradecanoylphorbol Acetate; Thyroid Gland; Wortmannin | 2000 |
Protein kinase C-alpha and -epsilon down-regulate cell surface sodium channels via differential mechanisms in adrenal chromaffin cells.
Topics: Adrenal Glands; Animals; Brefeldin A; Carbazoles; Carcinogens; Cattle; Cells, Cultured; Chromaffin Cells; Down-Regulation; Enzyme Inhibitors; Gene Expression Regulation; Immunoblotting; Indoles; Isoenzymes; Phorbol Esters; Protein Binding; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Protein Synthesis Inhibitors; RNA, Messenger; Saxitoxin; Sodium Channels; Tetradecanoylphorbol Acetate; Tetrodotoxin; Tritium | 2000 |
Differential regulation of microglial NO production by protein kinase C inhibitors.
Topics: Animals; Carbazoles; Drug Synergism; Enzyme Induction; Enzyme Inhibitors; Indoles; Isoquinolines; Lipopolysaccharides; Microglia; Nerve Tissue Proteins; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Protein Isoforms; Protein Kinase C; Pyrroles; Rats; Signal Transduction; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 2001 |
Post-transcriptional inhibition of lipopolysaccharide-induced expression of inducible nitric oxide synthase by Gö6976 in murine microglia.
Topics: Animals; Brain; Carbazoles; Cells, Cultured; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Indoles; Kinetics; Lipopolysaccharides; Mice; Neuroglia; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Protein Kinase C; Protein Kinase Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA Processing, Post-Transcriptional; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic | 2000 |
The indolocarbazole Gö6976 protects neurons from lipopolysaccharide/interferon-gamma-induced cytotoxicity in murine neuron/glia co-cultures.
Topics: Animals; Animals, Newborn; Carbazoles; Cell Survival; Coculture Techniques; Gene Expression Regulation; Indoles; Interferon-gamma; Interleukin-1; Lipopolysaccharides; Mice; Microtubule-Associated Proteins; Neural Cell Adhesion Molecules; Neuroglia; Neurons; Neuroprotective Agents; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Protein Kinase C; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2000 |
Biphasic effect of protein kinase C activators on spontaneous and glucocorticoid-induced apoptosis in primary mouse thymocytes.
Topics: Animals; Apoptosis; Bryostatins; Carbazoles; Cells, Cultured; DNA Fragmentation; Down-Regulation; Enzyme Activation; Female; Fluocinolone Acetonide; Glucocorticoids; Immunoblotting; Indoles; Isoenzymes; Lactones; Macrolides; Mice; Protein Kinase C; Tetradecanoylphorbol Acetate; Thymus Gland | 2000 |
Protein kinase C isoforms involved in regulation of cell shape and locomotion of human fibrosarcoma HT1080 cells.
Topics: Carbazoles; Cell Membrane; Cell Movement; Cell Size; Cytosol; Enzyme Inhibitors; Fibrosarcoma; Humans; Indoles; Isoenzymes; Kinetics; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured | 2000 |
Permissive role of protein kinase C alpha but not protein kinase C delta in sphingosine 1-phosphate-induced Rho A activation in C2C12 myoblasts.
Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; Cell Fractionation; Cell Line; Cell Membrane; Endoplasmic Reticulum; Endosomes; Enzyme Inhibitors; Golgi Apparatus; Indoles; Isoenzymes; Lysophospholipids; Maleimides; Mice; Muscle, Skeletal; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Transport; rhoA GTP-Binding Protein; Sphingosine; Tetradecanoylphorbol Acetate | 2000 |
The transient increase of tight junction permeability induced by bryostatin 1 correlates with rapid downregulation of protein kinase C-alpha.
Topics: Animals; Biological Transport; Bryostatins; Carbazoles; Cell Line; Cell Membrane Permeability; Cysteine Endopeptidases; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Indoles; Isoenzymes; Kinetics; Lactones; Leupeptins; Macrolides; Mannitol; Membrane Potentials; Multienzyme Complexes; Polyethylene Glycols; Proteasome Endopeptidase Complex; Protein Kinase C; Protein Kinase C-alpha; Tetradecanoylphorbol Acetate; Tight Junctions | 2000 |
Ceramide-enhanced urokinase-type plasminogen activator (uPA) release is mediated by protein kinase C in cultured microglia.
Topics: Animals; Carbazoles; Carcinogens; Cells, Cultured; Diglycerides; Enzyme Activation; Enzyme Inhibitors; Hydrolysis; Indoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Maleimides; MAP Kinase Kinase 4; Microglia; Mitogen-Activated Protein Kinase Kinases; NF-kappa B; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Kinase C-epsilon; Rats; Receptor, Nerve Growth Factor; Signal Transduction; Sphingomyelin Phosphodiesterase; Sphingomyelins; Sphingosine; Tetradecanoylphorbol Acetate; Urokinase-Type Plasminogen Activator | 2000 |
The overexpression of PKCdelta is involved in vascular endothelial growth factor-resistant apoptosis in cultured primary sinusoidal endothelial cells.
Topics: Acetophenones; Animals; Apoptosis; Benzopyrans; Carbazoles; Cells, Cultured; Dose-Response Relationship, Drug; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Humans; Indoles; Isoenzymes; Lymphokines; Protein Kinase C; Protein Kinase C-delta; Rats; Recombinant Proteins; Tetradecanoylphorbol Acetate; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2001 |
Oxidized-LDL enhances coronary vasoconstriction by increasing the activity of protein kinase C isoforms alpha and epsilon.
Topics: Animals; Blotting, Western; Calcium; Calcium Channel Blockers; Carbazoles; Coronary Vessels; Enzyme Activation; Enzyme Inhibitors; Fura-2; In Vitro Techniques; Indoles; Isoenzymes; Isometric Contraction; Lipoproteins, LDL; Male; Maleimides; Muscle, Smooth, Vascular; Potassium Chloride; Protein Kinase C; Serotonin; Subcellular Fractions; Swine; Tetradecanoylphorbol Acetate; Vasoconstriction; Verapamil | 2001 |
Effects of protein kinase C inhibitors on insulin secretory responses from rodent pancreatic islets.
Topics: Animals; Carbachol; Carbazoles; Cholinergic Agonists; Colforsin; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Glucose; Indoles; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mice; Potassium; Protein Kinase C; Rats; Rats, Sprague-Dawley; Staurosporine; Tetradecanoylphorbol Acetate | 2001 |
Oxytocin stimulates prostaglandin F2alpha secretion from porcine endometrial cells through activation of calcium-dependent protein kinase C.
Topics: Animals; Calcium; Carbazoles; Dinoprost; Drug Synergism; Endometrium; Enzyme Activation; Enzyme Inhibitors; Female; Indoles; Inositol Phosphates; L-Lactate Dehydrogenase; Male; Oxytocin; Protein Kinase C; Swine; Tetradecanoylphorbol Acetate; Thapsigargin | 2001 |
Bradykinin induces protein kinase C-dependent activation of phospholipase D in A-431 cells.
Topics: Acetophenones; Benzopyrans; Bradykinin; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Humans; Immunoblotting; Indoles; Isoenzymes; Kinetics; Maleimides; Phospholipase D; Phospholipids; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Serotonin activation of the ERK pathway in Hermissenda: contribution of calcium-dependent protein kinase C.
Topics: Animals; Calcium; Carbazoles; Chelating Agents; Conditioning, Classical; Egtazic Acid; Enzyme Inhibitors; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Mollusca; Phosphorylation; Serotonin; Tetradecanoylphorbol Acetate | 2001 |
Protein kinase C epsilon suppresses Abeta production and promotes activation of alpha-secretase.
Topics: Alzheimer Disease; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Carbazoles; CHO Cells; Cricetinae; Down-Regulation; Endopeptidases; Enzyme Activation; Humans; Indoles; Isoenzymes; Maleimides; Protein Kinase C; Protein Kinase C-epsilon; Protein Processing, Post-Translational; Recombinant Proteins; Tetradecanoylphorbol Acetate | 2001 |
Pharmacological evidence for system-dependent involvement of protein kinase C isoenzymes in phorbol ester-suppressed gap junctional communication.
Topics: Carbazoles; Cell Communication; Cells, Cultured; Connexin 43; Dose-Response Relationship, Drug; Gap Junctions; Indoles; Isoenzymes; Maleimides; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate | 2001 |
Neurotrophin secretion from cultured microglia.
Topics: Animals; Antibodies; Brain-Derived Neurotrophic Factor; Carbazoles; Carcinogens; Cells, Cultured; Cerebral Cortex; Culture Media, Conditioned; Diglycerides; Enzyme Inhibitors; Indoles; Isoenzymes; Lipopolysaccharides; Maleimides; Microglia; Nerve Growth Factor; Nerve Growth Factors; Neurotrophin 3; Protein Kinase C; Protein Kinase C-alpha; Rats; Tetradecanoylphorbol Acetate | 2001 |
The nuclear factor kappa B (NF-kappa B): a potential therapeutic target for estrogen receptor negative breast cancers.
Topics: Animals; Base Sequence; Breast Neoplasms; Carbazoles; Cell Division; Cyclin D1; DNA Primers; Enzyme Inhibitors; Female; Humans; I-kappa B Kinase; Indoles; Mammary Neoplasms, Experimental; Mice; Mice, Inbred A; Mutation; NF-kappa B; Protein Kinase C; Protein Serine-Threonine Kinases; Receptors, Estrogen; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 2001 |
Protein kinase C regulates FADD recruitment and death-inducing signaling complex formation in Fas/CD95-induced apoptosis.
Topics: Adaptor Proteins, Signal Transducing; Animals; Antineoplastic Agents; Apoptosis; Blotting, Western; Bryostatins; Carbazoles; Carcinogens; Carrier Proteins; Caspase 3; Caspase 8; Caspase 9; Caspases; Cell Separation; Cytosol; Enzyme Inhibitors; fas Receptor; Fas-Associated Death Domain Protein; Flow Cytometry; Humans; Indoles; Jurkat Cells; Lactones; Macrolides; Mitogens; Precipitin Tests; Protein Binding; Protein Kinase C; Protein Transport; Signal Transduction; Subcellular Fractions; Tetradecanoylphorbol Acetate | 2001 |
Protein kinase C modulates telomerase activity in human cervical cancer cells.
Topics: Alternative Splicing; Carbazoles; Catalytic Domain; Enzyme Inhibitors; Female; HeLa Cells; Humans; Indoles; Maleimides; Protein Kinase C; RNA, Messenger; Telomerase; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Uterine Cervical Neoplasms | 2001 |
A critical protein kinase C phosphorylation site on the 5-HT(1A) receptor controlling coupling to N-type calcium channels.
Topics: Animals; Binding Sites; Calcium Channels; Calcium Channels, N-Type; Carbazoles; Cells, Cultured; Dose-Response Relationship, Drug; Enkephalin, Leucine-2-Alanine; Enzyme Inhibitors; Guanosine 5'-O-(3-Thiotriphosphate); Hybrid Cells; Indoles; Mice; Mutation; Osmolar Concentration; Phosphorylation; Protein Kinase C; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Tetradecanoylphorbol Acetate | 2002 |
Fas activation opposes PMA-stimulated changes in the localization of PKCdelta: a mechanism for reducing neutrophil adhesion to endothelial cells.
Topics: Acetophenones; Benzopyrans; Carbazoles; Cell Adhesion; Cell Membrane; Cells, Cultured; Endothelium; Enzyme Inhibitors; fas Receptor; Humans; Indoles; Isoenzymes; Kinetics; Neutrophils; Protein Kinase C; Protein Kinase C-delta; Protein Transport; Tetradecanoylphorbol Acetate | 2002 |
FGF-2 and TPA induce matrix metalloproteinase-9 secretion in MCF-7 cells through PKC activation of the Ras/ERK pathway.
Topics: Acetophenones; Benzopyrans; Carbazoles; Collagenases; Enzyme Inhibitors; Fibroblast Growth Factor 2; Genes, Dominant; Humans; Indoles; Maleimides; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Matrix Metalloproteinase 9; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Models, Biological; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-raf; ras Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 2002 |
Blocking NF-kappaB activation in Jurkat leukemic T cells converts the survival agent and tumor promoter PMA into an apoptotic effector.
Topics: Apoptosis; Carbazoles; Caspase 8; Caspase 9; Caspases; DNA-Binding Proteins; Enzyme Activation; Enzyme Inhibitors; Fas Ligand Protein; fas Receptor; Gene Expression Regulation, Leukemic; Humans; I-kappa B Proteins; Indoles; Isoenzymes; Jurkat Cells; Maleimides; Membrane Glycoproteins; Neoplasm Proteins; NF-kappa B; NF-KappaB Inhibitor alpha; Protein Kinase C; Recombinant Fusion Proteins; Sequence Deletion; Tetradecanoylphorbol Acetate | 2002 |
Mechanism of angiotensin II-induced phospholipase D activation in bovine adrenal glomerulosa cells.
Topics: 1-Butanol; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aldosterone; Angiotensin II; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Carbazoles; Cattle; Cells, Cultured; Diglycerides; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Indoles; Ionomycin; Nitrendipine; Phospholipase D; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Zona Glomerulosa | 2002 |
Different actions of protein kinase C isoforms alpha and epsilon on gastric acid secretion.
Topics: Animals; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbazoles; Cells, Cultured; Enzyme Activators; Gastric Acid; In Vitro Techniques; Indoles; Male; Parietal Cells, Gastric; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Rabbits; Tetradecanoylphorbol Acetate | 2002 |
Regulation of the neuronal glutamate transporter excitatory amino acid carrier-1 (EAAC1) by different protein kinase C subtypes.
Topics: Amino Acid Transport System X-AG; Animals; Bryostatins; Carbazoles; Carcinogens; Carrier Proteins; Cells, Cultured; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Transporter 3; Female; Glutamate Plasma Membrane Transport Proteins; Indoles; Lactones; Macrolides; Neurons; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Symporters; Tetradecanoylphorbol Acetate | 2002 |
Opposing effects of PKCalpha and PKCepsilon on basolateral membrane dynamics in intestinal epithelia.
Topics: Actins; Calcium; Carbazoles; Carcinogens; Cell Membrane; Cell Polarity; Cells, Cultured; Cytoskeleton; Drug Interactions; Endocytosis; Enzyme Inhibitors; Epithelial Cells; Humans; Indoles; Intestinal Mucosa; Isoenzymes; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate; Thapsigargin | 2002 |
Nongenomic mechanism of glucocorticoid inhibition of bradykinin-induced calcium influx in PC12 cells: possible involvement of protein kinase C.
Topics: Animals; Bradykinin; Calcium; Calcium Channel Blockers; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Glucocorticoids; GTP-Binding Proteins; Indoles; omega-Conotoxins; PC12 Cells; Pertussis Toxin; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Thapsigargin | 2003 |
Nuclear factor of activated T cells 2 transactivation in mast cells: a novel isoform-specific transactivation domain confers unique FcepsilonRI responsiveness.
Topics: Acetophenones; Amino Acid Sequence; Animals; Base Sequence; Benzopyrans; Binding Sites; Carbazoles; Cell Line; DNA; DNA-Binding Proteins; Enzyme Inhibitors; In Vitro Techniques; Indoles; Ionomycin; Mast Cells; Mice; Molecular Sequence Data; Mutagenesis, Site-Directed; NFATC Transcription Factors; Nuclear Proteins; Protein Isoforms; Protein Kinase C; Protein Kinase C-delta; Protein Structure, Tertiary; Receptors, IgE; Recombinant Proteins; Tetradecanoylphorbol Acetate; Transcription Factors; Transcriptional Activation; Two-Hybrid System Techniques | 2003 |
Involvement of stress-activated protein kinase/c-Jun N-terminal kinase in endothelin-1-induced heat shock protein 27 in osteoblasts.
Topics: Animals; Anthracenes; Blotting, Northern; Blotting, Western; Carbazoles; Endothelin-1; Enzyme Activators; Enzyme Inhibitors; Gene Expression Regulation; Heat-Shock Proteins; Immunoenzyme Techniques; Indoles; JNK Mitogen-Activated Protein Kinases; MAP Kinase Kinase 4; Mice; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Molecular Chaperones; Naphthalenes; Neoplasm Proteins; Osteoblasts; p38 Mitogen-Activated Protein Kinases; RNA, Messenger; Tetradecanoylphorbol Acetate | 2003 |
Staurosporine induces rapid homotypic intercellular adhesion of U937 cells via multiple kinase activation.
Topics: Acetophenones; Adenosine Triphosphate; Benzopyrans; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; CD18 Antigens; Cell Aggregation; Cycloheximide; Cytoskeleton; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genistein; Humans; Imidazoles; Indoles; Integrin beta1; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinases; Naphthalenes; Phosphorylation; Phosphotransferases; Protein Kinase C; Protein-Tyrosine Kinases; Pyridines; Staurosporine; Temperature; Tetradecanoylphorbol Acetate; Time Factors; Tyrosine; U937 Cells | 2003 |
Human ABCA7 supports apolipoprotein-mediated release of cellular cholesterol and phospholipid to generate high density lipoprotein.
Topics: Apolipoprotein A-I; Apolipoproteins; ATP Binding Cassette Transporter 1; ATP-Binding Cassette Transporters; Bucladesine; Carbazoles; Cell Line; Cholesterol; Cloning, Molecular; Cysteine Proteinase Inhibitors; DNA, Complementary; Enzyme Inhibitors; Humans; Indoles; Kinetics; Leupeptins; Lipoproteins, HDL; Phospholipids; Recombinant Proteins; Tetradecanoylphorbol Acetate; Transfection | 2004 |
Activation of P2X7 purinoceptor-stimulated TGF-beta 1 mRNA expression involves PKC/MAPK signalling pathway in a rat brain-derived type-2 astrocyte cell line, RBA-2.
Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Astrocytes; Blotting, Northern; Blotting, Western; Brain; Carbazoles; Cell Line; Dose-Response Relationship, Drug; Flavonoids; Gene Expression; Indoles; Kinetics; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X4; Receptors, Purinergic P2X7; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetradecanoylphorbol Acetate; Transforming Growth Factor beta; Transforming Growth Factor beta1 | 2003 |
Ca2+-dependent protein kinase C isoforms induce cholestasis in rat liver.
Topics: Animals; Bacterial Proteins; Bile; Biological Transport; Blotting, Western; Calcium; Carbazoles; Cell Line; Cell Membrane; Cells, Cultured; Cholestasis; Cloning, Molecular; Densitometry; Detergents; Dose-Response Relationship, Drug; Enzyme Activation; Hepatocytes; Humans; Indoles; Liver; Luminescent Proteins; Male; Maleimides; Microscopy, Confocal; Models, Biological; Perfusion; Phorbol Esters; Polymerase Chain Reaction; Protein Isoforms; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Protein Transport; Rats; Rats, Wistar; Signal Transduction; Taurocholic Acid; Tetradecanoylphorbol Acetate; Time Factors; Transfection | 2004 |
Cooperation between PKC-alpha and PKC-epsilon in the regulation of JNK activation in human lung cancer cells.
Topics: Animals; Carbazoles; Carcinoma, Non-Small-Cell Lung; Carcinoma, Small Cell; Cell Membrane; Cytoplasm; Humans; Indoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Lung Neoplasms; Maleimides; Mice; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; rac1 GTP-Binding Protein; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2004 |
Expressions of inhibitory Smads, Smad6 and Smad7, are differentially regulated by TPA in human lung fibroblast cells.
Topics: Blotting, Western; Butadienes; Carbazoles; Cells, Cultured; DNA-Binding Proteins; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Humans; Indoles; Luciferases; Lung; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; NF-kappa B; Nitriles; Phosphorylation; Promoter Regions, Genetic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Smad6 Protein; Smad7 Protein; Tetradecanoylphorbol Acetate; Time Factors; Trans-Activators; Transfection; Transforming Growth Factor beta; Transforming Growth Factor beta1; Up-Regulation | 2004 |
B cell receptor-induced cAMP-response element-binding protein activation in B lymphocytes requires novel protein kinase Cdelta.
Topics: Acetamides; Acetophenones; Animals; B-Lymphocytes; Benzopyrans; Binding Sites; Blotting, Western; Bryostatins; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cell Division; Cross-Linking Reagents; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Indoles; Lactones; Macrolides; Mice; Mice, Inbred BALB C; Mice, Inbred CBA; Mitogens; Phosphorylation; Promoter Regions, Genetic; Protein Isoforms; Protein Kinase C; Protein Kinase C-delta; Protein Structure, Tertiary; Pyrans; Receptors, Antigen, B-Cell; Ribosomal Protein S6 Kinases, 90-kDa; Serine; Signal Transduction; Spiro Compounds; Tetradecanoylphorbol Acetate; Time Factors | 2004 |
Involvement of protein kinase C-related anti-apoptosis signaling in radiation-induced apoptosis in murine thymic lymphoma(3SBH5) cells.
Topics: Alkaloids; Animals; Apoptosis; Benzophenanthridines; Carbazoles; Cell Line, Tumor; Dose-Response Relationship, Radiation; Indoles; Lymphoma; Mice; Phenanthridines; Protein Kinase C; Radiation Dosage; Radiation Tolerance; Signal Transduction; Tetradecanoylphorbol Acetate | 2004 |
Delayed and sustained activation of extracellular signal-regulated kinase in human keratinocytes by UVA: implications in carcinogenesis.
Topics: Animals; Apoptosis; Blotting, Western; Calcium; Carbazoles; Caspase 3; Caspases; Cell Line; Cell Line, Tumor; Cell Membrane; Cell Survival; Cell Transformation, Neoplastic; Chelating Agents; COS Cells; Cytosol; Dose-Response Relationship, Radiation; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; ErbB Receptors; Estrenes; Flow Cytometry; Genes, Dominant; Golgi Apparatus; Humans; Indoles; Keratinocytes; Mitogen-Activated Protein Kinase 3; Models, Biological; Neoplasms; Plasmids; Protein Kinase C; Pyrrolidinones; ras Proteins; Skin Neoplasms; Subcellular Fractions; Tetradecanoylphorbol Acetate; Time Factors; Transfection; Ultraviolet Rays | 2004 |
Protein kinase C modulates agonist-sensitive release of Ca2+ from internal stores in HEK293 cells overexpressing the calcium sensing receptor.
Topics: Calcium; Carbazoles; Cations; Cell Line; Culture Media, Serum-Free; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Humans; Immunoblotting; Indoles; Maleimides; Neomycin; Protein Isoforms; Protein Kinase C; Protein Kinase C-epsilon; Receptors, Calcium-Sensing; Signal Transduction; Subcellular Fractions; Tetradecanoylphorbol Acetate; Time Factors | 2005 |
Phorbol ester phorbol-12-myristate-13-acetate promotes anchorage-independent growth and survival of melanomas through MEK-independent activation of ERK1/2.
Topics: Anoikis; Apoptosis; Butadienes; Carbazoles; Cell Adhesion; Cell Culture Techniques; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cell Survival; Disease Progression; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Immunoblotting; Indoles; Melanocytes; Melanoma; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Nitriles; Oligonucleotides, Antisense; Protein Kinase C; Protein Kinase C-alpha; Signal Transduction; Tetradecanoylphorbol Acetate; Time Factors; Transfection | 2005 |
Effect of protein kinase C activation on intracellular Ca2+ signaling and integrity of intestinal epithelial cells.
Topics: Acetophenones; Animals; Benzopyrans; Calcium; Calcium Channel Blockers; Calcium Signaling; Carbazoles; Cell Line; Cell Survival; Chelating Agents; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Indoles; Intestinal Mucosa; Intracellular Space; Maleimides; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate; Verapamil | 2005 |
RACK1 mediates activation of JNK by protein kinase C [corrected].
Topics: Animals; Anisomycin; Antibodies, Phospho-Specific; Apoptosis; Binding Sites; Carbazoles; Catalysis; Cell Line; Cell Line, Tumor; Cytoplasm; Enzyme Inhibitors; Gene Deletion; GTP-Binding Proteins; Humans; Indoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; MAP Kinase Kinase 4; MAP Kinase Kinase 7; MAP Kinase Kinase Kinase 1; Mice; Mice, Nude; Mitogen-Activated Protein Kinase 8; Mitogen-Activated Protein Kinase 9; Models, Biological; Neoplasm Proteins; Phosphopeptides; Phosphorylation; Protein Binding; Protein Kinase C; Protein Kinase C beta; Receptors for Activated C Kinase; Receptors, Cell Surface; RNA, Small Interfering; Serine; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Tumor Necrosis Factor-alpha; Ultraviolet Rays | 2005 |
Regulation of CD93 cell surface expression by protein kinase C isoenzymes.
Topics: Acetophenones; Benzopyrans; Benzoquinones; Carbazoles; Down-Regulation; Endothelial Cells; Flow Cytometry; Humans; Immunoenzyme Techniques; Indoles; Interferon-gamma; Interleukin-8; Isoenzymes; Isoquinolines; Lactams, Macrocyclic; Membrane Glycoproteins; Monocytes; Protein Kinase C; Protein Kinase Inhibitors; Quinones; Receptors, Complement; Rifabutin; Sulfonamides; Tetradecanoylphorbol Acetate; U937 Cells; Up-Regulation | 2006 |
Bradykinin augments EGF-induced airway smooth muscle proliferation by activation of conventional protein kinase C isoenzymes.
Topics: Animals; Bradykinin; Carbazoles; Cattle; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Indoles; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocytes, Smooth Muscle; Protein Kinase C; Receptor, Bradykinin B2; Tetradecanoylphorbol Acetate; Thymidine; Trachea; Tritium | 2006 |
Protein kinase Cbeta isoform down-regulates the expression of MDR3 P-glycoprotein in human Chang liver cells.
Topics: ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Transporters; Carbazoles; Cells, Cultured; Down-Regulation; Humans; Indoles; Isoenzymes; Liver; Maleimides; Protein Kinase C; Protein Kinase C beta; Tetradecanoylphorbol Acetate | 2006 |
Different roles of protein kinase C-betaI and -delta in the regulation of adipocyte differentiation.
Topics: 3T3-L1 Cells; Acetophenones; Adipocytes; Adipogenesis; Animals; Benzopyrans; Carbazoles; Cell Differentiation; Cell Membrane; Cell Proliferation; Chromans; Cytosol; Epidermal Growth Factor; Gene Expression; Genes, Dominant; Indoles; Mice; Mutant Proteins; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-delta; Protein Transport; Tetradecanoylphorbol Acetate; Thiazolidinediones; Transforming Growth Factor beta; Troglitazone | 2006 |
The sarcoplasmic-endoplasmic reticulum Ca2+ ATPase 2b regulates the Ca2+ transients elicited by P2Y2 activation in PC Cl3 thyroid cells.
Topics: Adenosine Triphosphate; Animals; Barium; Biological Transport, Active; Calcium; Carbazoles; Cell Line; Enzyme Activation; Indoles; Maleimides; Manganese; Microscopy, Fluorescence; Protein Kinase C; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Tetradecanoylphorbol Acetate; Thapsigargin; Thyroid Gland; Uridine Triphosphate | 2006 |
Protein kinase C activity is required for cytotoxic T cell lytic granule exocytosis, but the theta isoform does not play a preferential role.
Topics: Acetophenones; Benzopyrans; Calcium; Carbazoles; Cell Line, Tumor; Cell Membrane; Cytotoxicity, Immunologic; Exocytosis; Humans; Indoles; Mutation; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase Inhibitors; Structure-Activity Relationship; T-Lymphocytes, Cytotoxic; Tetradecanoylphorbol Acetate | 2007 |
Regulation of anion exchanger Slc26a6 by protein kinase C.
Topics: Acetophenones; Animals; Anion Transport Proteins; Antiporters; Benzopyrans; Biological Transport, Active; Carbazoles; Cell Membrane; Chlorides; Cytoplasm; Enzyme Activation; Female; Formates; In Vitro Techniques; Indoles; Maleimides; Mice; Oocytes; Oxalates; Protein Kinase C-delta; Protein Transport; Sulfate Transporters; Tetradecanoylphorbol Acetate; Xenopus | 2007 |
[Phosphorylation of PKCdelta participates in the toxicity of 6-hydroxydopamine on dopaminergic neuroblastoma cell].
Topics: Acetophenones; Benzopyrans; Blotting, Western; Carbazoles; Cell Line, Tumor; Cell Survival; Dopamine; Enzyme Activators; Humans; Indoles; Maleimides; Neuroblastoma; Oxidopamine; Phosphorylation; Protein Kinase C-delta; Signal Transduction; Tetradecanoylphorbol Acetate | 2006 |
Involvement of nPKC-MAPK pathway in the decrease of nucleophosmin/B23 during megakaryocytic differentiation of human myelogenous leukemia K562 cells.
Topics: Carbazoles; Cell Differentiation; Cell Line, Tumor; Humans; Indoles; K562 Cells; Leukemia, Myeloid; Maleimides; Megakaryocytes; Mitogen-Activated Protein Kinases; Nuclear Proteins; Nucleolin; Nucleophosmin; Phosphoproteins; Proteasome Endopeptidase Complex; Proteasome Inhibitors; Protein Kinase C; RNA-Binding Proteins; Tetradecanoylphorbol Acetate | 2007 |
Lactosylceramide alpha2,3-sialyltransferase is induced via a PKC/ERK/CREB-dependent pathway in K562 human leukemia cells.
Topics: 5' Flanking Region; Androstadienes; Carbazoles; Cell Differentiation; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Humans; Indoles; K562 Cells; Megakaryocytes; Mutation; Neuraminidase; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Promoter Regions, Genetic; Protein Kinase C; Sialyltransferases; Signal Transduction; Tetradecanoylphorbol Acetate; Wortmannin | 2007 |
Protein kinase C-beta and -delta isoenzymes promote arachidonic acid production and proliferation of MonoMac-6 cells.
Topics: Arachidonic Acid; Blotting, Western; Carbazoles; Cell Line; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flow Cytometry; Gene Expression; Green Fluorescent Proteins; Humans; Indoles; Isoenzymes; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-delta; Reverse Transcriptase Polymerase Chain Reaction; RNA Interference; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Transfection | 2007 |
The role of protein kinase C isoenzymes in the regulation of calcineurin activity in human peripheral blood mononuclear cells.
Topics: Adaptor Proteins, Signal Transducing; Base Sequence; Calcimycin; Calcineurin; Calcineurin Inhibitors; Carbazoles; DNA Primers; Enzyme Activation; Humans; In Vitro Techniques; Indoles; Ionophores; Isoenzymes; Leukocytes, Mononuclear; Maleimides; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate | 2007 |
Protein kinase C-dependent antilipolysis by insulin in rat adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Androstadienes; Angiotensin II; Animals; Carbazoles; Carcinogens; Dobutamine; Enzyme Activation; Enzyme Inhibitors; Glycerol; Imidazoles; Indoles; Insulin; Isoenzymes; Lipolysis; Male; Maleimides; Protein Kinase C; Rats; Receptor, Insulin; Tetradecanoylphorbol Acetate; Wortmannin | 2007 |
nPKCepsilon, a P2Y2-R downstream effector in regulated mucin secretion from airway goblet cells.
Topics: Adenosine Triphosphate; Animals; Carbazoles; Cell Line; Dose-Response Relationship, Drug; Goblet Cells; Indoles; Maleimides; Mice; Mice, Inbred C57BL; Mice, Knockout; Mucins; Mutation; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase Inhibitors; Protein Transport; Purinergic P2 Receptor Agonists; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Trachea; Transfection | 2007 |
Protein kinase C alpha promotes angiogenic activity of human endothelial cells via induction of vascular endothelial growth factor.
Topics: Angiogenesis Inducing Agents; Autocrine Communication; Blotting, Western; Carbazoles; Cell Line; Cell Shape; Cells, Cultured; Endothelial Cells; Enzyme Activation; Fibroblast Growth Factor 2; Humans; Neovascularization, Physiologic; Polymerase Chain Reaction; Protein Kinase C-alpha; Protein Kinase Inhibitors; Receptors, Vascular Endothelial Growth Factor; RNA Interference; RNA, Messenger; RNA, Small Interfering; Stem Cells; Tetradecanoylphorbol Acetate; Time Factors; Up-Regulation; Vascular Endothelial Growth Factor A | 2008 |
P70 S6 kinase negatively regulates fibroblast growth factor 2-stimulated interleukin-6 synthesis in osteoblasts: function at a point downstream from protein kinase C.
Topics: Animals; Carbazoles; Cells, Cultured; Fibroblast Growth Factor 2; Indoles; Interleukin-6; Maleimides; Mice; Osteoblasts; Phosphorylation; Protein Kinase C; Ribosomal Protein S6 Kinases, 70-kDa; Sirolimus; Tetradecanoylphorbol Acetate | 2008 |
Volume-sensitive NADPH oxidase activity and taurine efflux in NIH3T3 mouse fibroblasts.
Topics: Adenosine Triphosphate; Animals; Arachidonic Acid; Benzophenanthridines; Calcium; Carbazoles; Cell Size; Cytochrome b Group; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; Fibroblasts; Hypotonic Solutions; Lysophospholipids; Mice; NADPH Oxidase 4; NADPH Oxidases; NIH 3T3 Cells; Onium Compounds; Osmotic Pressure; Phosphoproteins; Protein Kinase C; rac1 GTP-Binding Protein; Reactive Oxygen Species; RNA Interference; Taurine; Tetradecanoylphorbol Acetate; Time Factors; Transfection | 2008 |
Endothelial PKC delta activation attenuates neutrophil transendothelial migration.
Topics: Antineoplastic Agents; Bryostatins; Carbazoles; Carcinogens; Cell Movement; Cells, Cultured; Endothelium, Vascular; Enzyme Inhibitors; Focal Adhesion Kinase 1; Humans; Leukotriene B4; Neutrophils; Paxillin; Protein Kinase C-delta; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha; Vinculin | 2008 |
Effects of phorbol ester-sensitive PKC (c/nPKC) activation on the production of adiponectin in 3T3-L1 adipocytes.
Topics: 3T3-L1 Cells; Adipocytes; Adiponectin; Angiotensin II; Animals; Benzimidazoles; Biphenyl Compounds; Carbazoles; Chromones; Enzyme Activation; Gene Expression; Glucose; Insulin; Mice; Morpholines; NF-kappa B; PPAR gamma; Protein Kinase C; Tetradecanoylphorbol Acetate; Tetrazoles; Tumor Necrosis Factor-alpha | 2009 |
Up-regulation of cyclin D1 expression in asthma serum-sensitized human airway smooth muscle promotes proliferation via protein kinase C alpha.
Topics: Adult; Asthma; Bronchi; Carbazoles; Cell Proliferation; Cells, Cultured; Cyclin D1; Female; Humans; Isoenzymes; Male; Middle Aged; Myocytes, Smooth Muscle; Protein Kinase C-alpha; Serum; Tetradecanoylphorbol Acetate; Up-Regulation; Young Adult | 2010 |
The potential use of protein kinase D inhibitors for prevention/treatment of epidermal tumors.
Topics: Animals; Anticarcinogenic Agents; Carbazoles; Cell Differentiation; Cell Proliferation; Cells, Cultured; Epidermis; Isoquinolines; Keratinocytes; Mice; Protein Kinase C; Protein Kinase Inhibitors; Resveratrol; Skin Neoplasms; Stilbenes; Sulfonamides; Tetradecanoylphorbol Acetate | 2010 |
PKCα suppresses osteoblastic differentiation.
Topics: Adenoviridae; Animals; Carbazoles; Cell Differentiation; Enzyme Activation; Gene Knockdown Techniques; Mice; Osteoblasts; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Tetradecanoylphorbol Acetate | 2011 |
Protein kinase C regulates the internalization and function of the human organic anion transporting polypeptide 1A2.
Topics: Animals; Biotinylation; Carbazoles; Chlorocebus aethiops; COS Cells; Enzyme Inhibitors; Genetic Vectors; Humans; Organic Anion Transporters; Phagocytosis; Plasmids; Protein Kinase C; Tetradecanoylphorbol Acetate | 2011 |
PKCα mediates acetylcholine-induced activation of TRPV4-dependent calcium influx in endothelial cells.
Topics: Acetylcholine; Animals; Calcium Signaling; Carbazoles; Cells, Cultured; Endothelial Cells; Enzyme Activation; Male; Mesenteric Arteries; Mice; Mice, Inbred C57BL; Mice, Knockout; Mutation; Nitric Oxide Synthase Type III; Phosphorylation; Protein Kinase C-alpha; Protein Kinase Inhibitors; Tetradecanoylphorbol Acetate; Time Factors; Transfection; TRPV Cation Channels; Vasodilation; Vasodilator Agents | 2011 |
Protein kinase C mediates peroxynitrite toxicity to oligodendrocytes.
Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; Cells, Cultured; Chlorides; Enzyme Activation; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Indoles; Isoenzymes; Maleimides; Molsidomine; Oligodendroglia; Peroxynitrous Acid; Protein Kinase C; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Signal Transduction; Tetradecanoylphorbol Acetate; Zinc Compounds | 2011 |
Central role of PKCα in isoenzyme-selective regulation of cardiac transient outward current Ito and Kv4.3 channels.
Topics: Animals; Carbazoles; Enzyme Inhibitors; Female; Isoenzymes; Membrane Potentials; Myocytes, Cardiac; Oocytes; Patch-Clamp Techniques; Plasmids; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Rats; Recombinant Proteins; Shal Potassium Channels; Signal Transduction; Substrate Specificity; Tetradecanoylphorbol Acetate; Transfection; Xenopus | 2011 |
Enhancement of axonal regeneration of retinal ganglion cells in adult rats by etomidate: involvement of protein kinase C.
Topics: Anesthetics, Intravenous; Animals; Axons; Axotomy; Carbazoles; Cell Count; Cell Survival; Enzyme Inhibitors; Etomidate; Female; Injections, Intraperitoneal; Nerve Regeneration; Optic Nerve; Peripheral Nerves; Protein Kinase C; Rats; Rats, Sprague-Dawley; Retinal Ganglion Cells; Tetradecanoylphorbol Acetate | 2011 |
High glucose-induced RhoA activation requires caveolae and PKCβ1-mediated ROS generation.
Topics: Acetophenones; Acetylcysteine; Animals; Carbazoles; Caveolae; Cyclodextrins; Diabetic Nephropathies; Enzyme Activation; Filipin; Glucose; Indoles; Maleimides; Mesangial Cells; Mice; Mice, Knockout; NADPH Oxidases; Protein Kinase C; Protein Kinase C beta; Rats; Reactive Oxygen Species; rhoA GTP-Binding Protein; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Transforming Growth Factor beta1 | 2012 |
Mammalian target of rapamycin complex 1 (mTORC1) plays a role in Pasteurella multocida toxin (PMT)-induced protein synthesis and proliferation in Swiss 3T3 cells.
Topics: 3T3 Cells; Adenosine Triphosphate; Animals; Bacterial Proteins; Bacterial Toxins; Carbazoles; Cell Movement; GTP-Binding Protein alpha Subunits, Gq-G11; Mechanistic Target of Rapamycin Complex 1; Methionine; Mice; Models, Biological; Multiprotein Complexes; Phospholipase C beta; Phosphorylation; Protein Kinase C; Receptor Protein-Tyrosine Kinases; Ribosomal Protein S6; Signal Transduction; Tetradecanoylphorbol Acetate; TOR Serine-Threonine Kinases; Wound Healing | 2013 |
Protein kinase C regulates human pluripotent stem cell self-renewal.
Topics: Activins; Alkaline Phosphatase; Blotting, Western; Carbazoles; Cell Line; Cell Proliferation; Chromones; Extracellular Signal-Regulated MAP Kinases; Fibroblast Growth Factor 2; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Immunohistochemistry; Indoles; Maleimides; Morpholines; Phosphatidylinositol 3-Kinases; Phosphorylation; Pluripotent Stem Cells; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Proto-Oncogene Proteins c-akt; RNA Interference; Signal Transduction; Tetradecanoylphorbol Acetate | 2013 |
Monoubiquitination of filamin B regulates vascular endothelial growth factor-mediated trafficking of histone deacetylase 7.
Topics: Amino Acid Sequence; Carbazoles; Cell Line, Tumor; Cell Movement; Contractile Proteins; Endothelial Cells; Filamins; HeLa Cells; Histone Deacetylases; Humans; Indoles; Maleimides; Matrix Metalloproteinase 10; Microfilament Proteins; Neovascularization, Physiologic; Nuclear Receptor Subfamily 4, Group A, Member 1; Protein Kinase C; Protein Structure, Tertiary; Protein Transport; RNA Interference; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Ubiquitin; Ubiquitination; Vascular Endothelial Growth Factors | 2013 |
Nuclear factor κB mediates suppression of canonical transient receptor potential 6 expression by reactive oxygen species and protein kinase C in kidney cells.
Topics: Carbazoles; Carcinogens; Cell Line; Enzyme Inhibitors; Gene Expression Regulation; Gene Knockdown Techniques; Histone Deacetylase 2; Histone Deacetylase Inhibitors; Humans; Hydrogen Peroxide; Hydroxamic Acids; Kidney; NF-kappa B p50 Subunit; Oxidants; Protein Kinase C; Response Elements; Tetradecanoylphorbol Acetate; Transcription Factor RelA; Transcription, Genetic; TRPC Cation Channels; TRPC6 Cation Channel | 2013 |
Inflammation induces multinucleation of Microglia via PKC inhibition of cytokinesis, generating highly phagocytic multinucleated giant cells.
Topics: alpha-Synuclein; Amyloid beta-Peptides; Animals; Carbazoles; Cell Fusion; Cell Line; Cell Nucleus; Cytokinesis; Female; Giant Cells; Inflammation; Interferon-gamma; Interleukin-4; Lipopolysaccharides; Male; Mice; Microglia; PC12 Cells; Phagocytosis; Primary Cell Culture; Protein Kinase C; Protein Kinase Inhibitors; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2014 |
Downregulation of BDNF Expression by PKC and by TNF-α in Human Endothelial Cells.
Topics: Acetophenones; Benzopyrans; Brain-Derived Neurotrophic Factor; Carbazoles; Down-Regulation; Endothelial Cells; Endothelium, Vascular; Human Umbilical Vein Endothelial Cells; Humans; Indoles; Maleimides; Neovascularization, Physiologic; Nerve Tissue Proteins; Peptides, Cyclic; Phorbol Esters; Protein Kinase C; Receptor, trkB; Receptors, Nerve Growth Factor; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2015 |
Amyloid β induces microglia to phagocytose neurons via activation of protein kinase Cs and NADPH oxidase.
Topics: Amyloid beta-Peptides; Carbazoles; Carcinogens; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Maleimides; Microglia; NADPH Oxidases; Neurons; Phagocytosis; Protein Kinase C; Tetradecanoylphorbol Acetate | 2016 |
Heterologous, PKC-Mediated Desensitization of Human Histamine H3 Receptors Expressed in CHO-K1 Cells.
Topics: Adenosine Triphosphate; Animals; Carbazoles; Cell Membrane; CHO Cells; Colforsin; Cricetulus; Humans; Indoles; Phosphorylation; Protein Kinase C; Receptors, Histamine H3; Signal Transduction; Tetradecanoylphorbol Acetate | 2016 |
Co-ordinated activation of classical and novel PKC isoforms is required for PMA-induced mTORC1 activation.
Topics: Adenosine Triphosphatases; Carbazoles; Endocytosis; Endosomes; Enzyme Activation; HEK293 Cells; HeLa Cells; Humans; Lysosomes; Mechanistic Target of Rapamycin Complex 1; Multiprotein Complexes; Phospholipase D; Phosphorylation; Protein Isoforms; Protein Kinase C; RNA Interference; Signal Transduction; Tetradecanoylphorbol Acetate; TOR Serine-Threonine Kinases | 2017 |
Protein kinase C regulates ErbB3 turnover.
Topics: Carbazoles; Cell Membrane; Endocytosis; Enzyme Activation; Humans; Lysosomes; MCF-7 Cells; Neuregulin-1; Phosphorylation; Phosphotyrosine; Protein Kinase C-delta; Protein Kinase Inhibitors; Protein Stability; Protein Transport; Proteolysis; Receptor, ErbB-3; Tetradecanoylphorbol Acetate; Ubiquitination | 2019 |
Protein Kinase C Regulates ASIC1a Protein Expression and Channel Function via NF-kB Signaling Pathway.
Topics: Acid Sensing Ion Channels; Animals; Carbazoles; Cell Line; Cerebral Cortex; Mice; Naphthalenes; Neurons; Neurotoxicity Syndromes; NF-kappa B; Proteasome Endopeptidase Complex; Protein Biosynthesis; Protein Kinase C; Proteolysis; Signal Transduction; Tetradecanoylphorbol Acetate; Time Factors; Ubiquitin | 2020 |
Distinct Regulation of Cardiac Fibroblast Proliferation and Transdifferentiation by Classical and Novel Protein Kinase C Isoforms: Possible Implications for New Antifibrotic Therapies.
Topics: Actins; Animals; Carbazoles; Cell Adhesion Molecules; Cell Proliferation; Cell Transdifferentiation; Cells, Cultured; Female; Fibroblasts; Fibrosis; Humans; Indoles; Maleimides; Mice; Myocardium; Myofibroblasts; Primary Cell Culture; Protein Kinase C; Tetradecanoylphorbol Acetate | 2021 |