Page last updated: 2024-09-03

glycerophosphoinositol 4,5-bisphosphate and oxotremorine

glycerophosphoinositol 4,5-bisphosphate has been researched along with oxotremorine in 12 studies

Compound Research Comparison

Studies
(glycerophosphoinositol 4,5-bisphosphate)
Trials
(glycerophosphoinositol 4,5-bisphosphate)
Recent Studies (post-2010)
(glycerophosphoinositol 4,5-bisphosphate)
Studies
(oxotremorine)
Trials
(oxotremorine)
Recent Studies (post-2010) (oxotremorine)
3,38131,0431,930699

Protein Interaction Comparison

ProteinTaxonomyglycerophosphoinositol 4,5-bisphosphate (IC50)oxotremorine (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.4
Muscarinic acetylcholine receptor M4Homo sapiens (human)5
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)2.321
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Homo sapiens (human)8
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.5012

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19901 (8.33)18.7374
1990's4 (33.33)18.2507
2000's6 (50.00)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Joseph, JA; Kowatch, MA; Maki, T; Roth, GS1
Alger, BE; McCarren, M; Pitler, TA1
Ferrari-DiLeo, G; Flynn, DD; Mash, DC1
Ebihara, T; Saffen, D1
Fisher, SK; Linseman, DA; McEwen, EL; Sorensen, SD1
Abogadie, FC; Brown, DA; Filippov, AK; Hughes, S; Marsh, SJ; Tatulian, L; Winks, JS1
Hilgemann, DW; Hille, B; Hirdes, W; Horowitz, LF; Mackie, K; Suh, BC1
Gamper, N; Hilgemann, DW; Li, Y; Shapiro, MS1
Hille, B; Inoue, T; Meyer, T; Suh, BC1
Billups, B; Billups, D; Challiss, RA; Nahorski, SR1
Hancock, J; Hobson, SA; Kelly, E; Marrion, NV; Mason, A; Oldfield, S; Randall, AD; Wynick, D1
Hille, B; Leal, K; Suh, BC1

Other Studies

12 other study(ies) available for glycerophosphoinositol 4,5-bisphosphate and oxotremorine

ArticleYear
Selective cross-activation/inhibition of second messenger systems and the reduction of age-related deficits in the muscarinic control of dopamine release from perifused rat striata.
    Brain research, 1990, Dec-24, Volume: 537, Issue:1-2

    Topics: Aging; Animals; Arachidonic Acid; Arachidonic Acids; Biotransformation; Carbachol; Corpus Striatum; Dopamine; In Vitro Techniques; Inosine Triphosphate; Male; Neomycin; Oxotremorine; Perfusion; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Second Messenger Systems; Type C Phospholipases

1990
Calcium-dependent pirenzepine-sensitive muscarinic response in the rat hippocampal slice.
    Neuroscience letters, 1988, Aug-31, Volume: 91, Issue:2

    Topics: Animals; Calcium; Carbachol; Hippocampus; In Vitro Techniques; Membrane Potentials; Oxotremorine; Parasympathomimetics; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Pirenzepine; Rats; Receptors, Muscarinic

1988
Attenuation of muscarinic receptor-G-protein interaction in Alzheimer disease.
    Molecular and chemical neuropathology, 1995, Volume: 24, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Carbachol; Cerebral Cortex; Choline O-Acetyltransferase; Female; Frontal Lobe; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Humans; Male; Middle Aged; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Pirenzepine; Receptors, Muscarinic; Reference Values; Regression Analysis; Synaptic Membranes; Synaptosomes

1995
Muscarinic acetylcholine receptor-mediated induction of zif268 mRNA in PC12D cells requires protein kinase C and the influx of extracellular calcium.
    Journal of neurochemistry, 1997, Volume: 68, Issue:3

    Topics: Animals; Calcium; Carbachol; DNA-Binding Proteins; Early Growth Response Protein 1; Extracellular Space; Immediate-Early Proteins; Muscarinic Agonists; Oxotremorine; PC12 Cells; Phosphatidylinositol 4,5-Diphosphate; Protein Kinase C; Rats; Receptors, Muscarinic; RNA, Messenger; Transcription Factors

1997
Agonist-induced endocytosis of muscarinic cholinergic receptors: relationship to stimulated phosphoinositide turnover.
    Journal of neurochemistry, 1997, Volume: 68, Issue:4

    Topics: Blotting, Western; Diglycerides; Endocytosis; Glioma; Humans; Isoenzymes; Lipid Metabolism; Muscarinic Agonists; Neuroblastoma; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Receptors, Muscarinic; Subcellular Fractions; Substrate Specificity; Tumor Cells, Cultured; Type C Phospholipases

1997
Relationship between membrane phosphatidylinositol-4,5-bisphosphate and receptor-mediated inhibition of native neuronal M channels.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Mar-30, Volume: 25, Issue:13

    Topics: Animals; Animals, Newborn; Bradykinin; Calcium; Calcium-Binding Proteins; Cell Membrane; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Estrenes; Female; Fluorescent Dyes; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Gene Expression; Green Fluorescent Proteins; Immunohistochemistry; Isoenzymes; Male; Microscopy, Confocal; Muscarinic Agonists; Mutation; Neural Inhibition; Neuronal Calcium-Sensor Proteins; Neurons; Neuropeptides; Oxotremorine; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphodiesterase Inhibitors; Phospholipase C delta; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Superior Cervical Ganglion; Transfection; Type C Phospholipases

2005
Phospholipase C in living cells: activation, inhibition, Ca2+ requirement, and regulation of M current.
    The Journal of general physiology, 2005, Volume: 126, Issue:3

    Topics: Alkylation; Animals; Calcium; CHO Cells; Cricetinae; Enzyme Activation; Estrenes; Ethylmaleimide; Humans; Inositol Phosphates; KCNQ Potassium Channels; KCNQ1 Potassium Channel; Membrane Potentials; Muscarinic Agonists; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Diacylglycerol-Lyase; Phospholipid Ethers; Potassium Channels, Voltage-Gated; Protein Kinase C; Pyrrolidinones; Receptor, Muscarinic M1; Sulfonamides; Time Factors; Transfection

2005
Regulation of Kv7 (KCNQ) K+ channel open probability by phosphatidylinositol 4,5-bisphosphate.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Oct-26, Volume: 25, Issue:43

    Topics: Animals; Carbachol; CHO Cells; Cholinergic Agonists; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Electric Stimulation; Extracellular Space; Green Fluorescent Proteins; Humans; Ion Channel Gating; KCNQ Potassium Channels; Membrane Potentials; Muscarinic Agonists; Oncogene Protein v-akt; Oxotremorine; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phospholipase C gamma; Phosphotransferases (Alcohol Group Acceptor); Probability; src-Family Kinases; Structure-Activity Relationship; Transfection

2005
Rapid chemically induced changes of PtdIns(4,5)P2 gate KCNQ ion channels.
    Science (New York, N.Y.), 2006, Dec-01, Volume: 314, Issue:5804

    Topics: Animals; Calcium; Cell Line; Cell Membrane; Diglycerides; Dimerization; Humans; Inositol Polyphosphate 5-Phosphatases; Ion Channel Gating; KCNQ Potassium Channels; KCNQ2 Potassium Channel; KCNQ3 Potassium Channel; Mice; NIH 3T3 Cells; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Phosphoric Monoester Hydrolases; Phosphorylation; Recombinant Fusion Proteins; Second Messenger Systems; Sirolimus

2006
Modulation of Gq-protein-coupled inositol trisphosphate and Ca2+ signaling by the membrane potential.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Sep-27, Volume: 26, Issue:39

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium Signaling; Cell Line; Cell Line, Tumor; Cells, Cultured; Cerebellum; CHO Cells; Cricetinae; Cricetulus; Humans; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isoenzymes; Kidney; Membrane Potentials; Microscopy, Fluorescence; Neuroblastoma; Neuronal Plasticity; Neurons; Nifedipine; Oxotremorine; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phospholipase C delta; Photolysis; Rats; Receptor, Muscarinic M3; Recombinant Fusion Proteins; Thapsigargin; Transfection; Type C Phospholipases

2006
Receptor-mediated suppression of potassium currents requires colocalization within lipid rafts.
    Molecular pharmacology, 2009, Volume: 76, Issue:6

    Topics: Animals; Blotting, Western; Calcium; Carbachol; Cell Line; Cholinergic Agents; Ganglia, Spinal; Humans; KCNQ2 Potassium Channel; KCNQ3 Potassium Channel; Membrane Microdomains; Membrane Potentials; Mice; Muscarine; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Potassium Channel Blockers; Potassium Channels; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Receptors, Muscarinic

2009
Modulation of high-voltage activated Ca(2+) channels by membrane phosphatidylinositol 4,5-bisphosphate.
    Neuron, 2010, Jul-29, Volume: 67, Issue:2

    Topics: Adenosine Triphosphate; Barium; Biophysics; Calcium; Calcium Channels, L-Type; Cell Line, Transformed; Chelating Agents; Egtazic Acid; Electric Stimulation; Fluorescence Resonance Energy Transfer; Green Fluorescent Proteins; Humans; Immunosuppressive Agents; Ion Channel Gating; Membrane Potentials; Muscarinic Agonists; Oxotremorine; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphoric Monoester Hydrolases; Sirolimus; Time Factors; Transfection

2010