glyburide and tolbutamide

glyburide has been researched along with tolbutamide in 416 studies

Research

Studies (416)

TimeframeStudies, this research(%)All Research%
pre-1990196 (47.12)18.7374
1990's121 (29.09)18.2507
2000's63 (15.14)29.6817
2010's35 (8.41)24.3611
2020's1 (0.24)2.80

Authors

AuthorsStudies
Dietrich, H; Lehmann, C; Märki, F; Schweizer, EH1
Aguilar-Bryan, L; Bryan, J; Clement, JP; Gonoi, T; Gonzalez, G; Inagaki, N; Inazawa, J; Namba, N; Seino, S1
Higashiguchi, O; Horio, Y; Isomoto, S; Kondo, C; Kurachi, Y; Matsumoto, S; Matsuzawa, Y; Yamada, M1
Hashimoto, Y; Inui, K; Saito, H; Uwai, Y1
Topliss, JG; Yoshida, F1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Abe, T; Itoh, T; Kato, Y; Kusuhara, H; Meier, PJ; Shitara, Y; Sugiyama, D; Sugiyama, Y1
Koyabu, N; Murakami, H; Ohtani, H; Satoh, H; Sawada, Y; Tsujimoto, M; Yamashita, F1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Buttar, D; Colclough, N; Gerhardt, S; MacFaul, PA; Maskos, K; Phillips, SD; Plowright, A; Steinbacher, S; Steuber, H; Tam, K; Whittamore, P1
Barber, J; Dawson, S; Kenna, JG; Paul, N; Stahl, S1
Caradonna, NP; Hallifax, D; Houston, JB; Turlizzi, E; Zanelli, U1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Melander, A; Wåhlin-Boll, E2
Codina, J; Herrera, E; Lasuncion, MA1
Balant, L1
Alemany, M; Herrera, E; Remesar, X1
Bickel, M; Geisen, K; Schleyerbach, R1
Alemany, M; Codina, J; Herrera, E; Palou, A1
Alemany, M; Herrera, E; Palou, A1
Castoldi, D; Tofanetti, O1
Hasselblatt, A; Joost, HG1
Efendic, S; Lundberg, JM; Uvnäs, B; Uvnäs-Wallensten, K1
Bottermann, P; Lüders, L; Zilker, T1
Gotfredsen, CF1
Haslbeck, M1
Macchi, IA; Zeytinoğlu, FN1
Cerasi, E; Grill, V1
Handler, JS; Keiser, HR; Zusman, RM1
Brooker, G; Linden, J1
Grill, V1
Foy, JM; Lucas, PD1
Christensen, LK; Hansen, JM1
Bloom, A; Bulpitt, CJ; Shaw, KM1
Jorgensen, KD2
Di Saverio, S; Roncaia, R; Torri, A; Zanni, A1
Balant, L; Fabre, J; Loutan, L; Samimi, H; Tillolès, M1
Pfeiffer, EF; Schatz, H; Steinle, D1
Hausmann, L; Kaffarnik, H; Schumann, G1
Kamenisch, W; Laube, H; Pfeiffer, EF; Schatz, H; Sieradzki, J1
Greenstein, S; Kashyap, RP; Walfish, PG1
Hoder, A; Losert, W; Scholz, C1
Hassalacher, Ch; Lang, PD; Vollmar, J; Wahl, P1
Bennett, MA; Fitzgerald, MG; Malins, JM; Pentecost, BL; Soler, NG1
Blumenbach, L; Gerhards, E; Gutsche, H; Klein, W; Loge, O; Losert, W; Schillinger, E; Speck, U; Vetter, H; Wendt, H1
Krause, U; Puchinger, H; Wacker, A2
Willms, B1
Nierle, C; Pfeiffer, EF; Schatz, H1
Baumeister, G; Stahl, M; Wagner, H1
O'Connor, C; Pascual Leone, A; Valdés, M1
Andreev, D; Pampulov, L1
Baumeister, G; Stahl, M; Wagner, H; Zierden, E1
Müller, WE; Wollert, U1
Brown, KF; Crooks, MJ2
Alric, R; Loubatières, AL; Loubatieres-Mariani, MM; Ribes, G; Sorial, G; Tarasco, A1
Alric, R; Lignon, F; Loubatières, A; Manteghetti, M; Puech, R1
Balabolkin, MI; Danilova, TI; Ol'shanskaia, AA; Timofeev, AV; Zhuleva, LIu1
Ambrosi, F; Cristallini, S; Filipponi, P; Gregorio, F; Pedetti, M; Santeusanio, F1
de Hemptinne, A; Vanheel, B1
Auchampach, JA; Cavero, I; Gross, GJ; Maruyama, M1
Ferguson, PW; Judd, RL; Kunjathoor, VV; Medon, PJ; Pillai, UA1
Kozlowski, RZ; Nye, PC; Robertson, BE1
Buscema, M; Caltabiano, V; Forte, F; Purrello, F; Rabuazzo, AM; Vetri, M; Vigneri, R; Vinci, C1
Henderson, G; Hicks, GA1
Antunes, CM; Barbosa, RM; Rosario, LM; Santos, RM; Silva, AM1
Findlay, I3
Haddad, GG; Jiang, C; Xia, Y1
Bernardi, H; Fosset, M; Lazdunski, M1
Aguilar-Bryan, L; Bryan, J; Nelson, DA1
Katsumata, K; Katsumata, Y3
Aoki, M; Inoue, H; Kaku, K; Kaneko, T; Matsuda, M1
Cooper, GJ; Moore, CX1
Bosco, D; Chanson, M; Giordano, E; Meda, P; Soria, B1
Harrower, AD1
Fu, SX; Li, YS; Yang, XP; Zhang, HL1
Ammälä, C; Arkhammar, P; Berggren, PO; Bokvist, K; Larsson, O; Rorsman, P; Wåhlander, K1
Cooper, DR; Farese, RV; Ishizuka, T; Standaert, ML1
Collier, BH; D'Souza, MJ; Pollock, SH; Reichbaum, MI1
Nishikawa, M; Sato, Y; Shinkai, H; Sukegawa, E1
Buscema, M; Gatta, C; Gullo, D; Purrello, F; Rabuazzo, AM; Vetri, M; Vigneri, R; Vinci, C1
Ashcroft, SJ; Berggren, PO; Hubbard, P; Niki, I; Welsh, M1
Lamp, ST; Venkatesh, N; Weiss, JN1
Kanno, M; Nakaya, H; Takeda, Y; Tohse, N1
Chang, CC; Hong, SJ1
Garrino, MG; Henquin, JC1
Aranyi, Z; Ballagi-Pordány, G; Koltai, MZ; Köszeghy, A; Pogátsa, G1
Pilsudski, R; Rougier, O; Tourneur, Y1
Boutagy, JS; Shenfield, GM; Webb, C1
Cooper, DR; Farese, RV; Nair, G; Pollet, RJ; Standaert, M; Vila, MC; Watson, JE1
Antoine, MH; Berkenboom, G; Fang, ZY; Fontaine, J; Herchuelz, A; Hermann, M; Lebrun, P1
Krnjević, K1
Dash, RJ; Khandekar, S; Sethi, BK1
Ashford, ML; Boden, PR; Treherne, JM1
Gasser, RN; Vaughan-Jones, RD1
Angus, JA; Cocks, TM; King, SJ1
Ashford, ML; Cook, DL; Hales, CN; Sturgess, NC1
Abrahamsson, H; Berggren, PO; Rorsman, P1
Ohno-Shosaku, T; Rorsman, P; Trube, G1
Rosario, LM1
Castle, NA; Haylett, DG1
Lenzen, S; Männer, K; Panten, U; Trube, G; Zünkler, BJ1
Wilson, C1
Pfeifer, MA; Rothschild, AH; Rothschild, MA1
Anderson, EG; Grigg, JJ1
Brayden, JE; Davies, NW; Huang, Y; Nelson, MT; Quayle, JM; Standen, NB1
Faivre, JF; Findlay, I1
Sanguinetti, MC; Siegl, PK; Wolleben, CD1
Falke, LC; Gee, WM; Gillis, KD; Hammoud, A; McDaniel, ML; Misler, S1
Ashcroft, FM; Ashcroft, SJ; Kelly, RP; Niki, I1
Bartosiewicz, W; Czyzyk, A; Lao, B; Orłowska, K; Szczepanik, Z1
van Koetsveld, PM; Verschoor, L; Weber, RF; Weeks, L; Wolffenbuttel, BH1
Herchuelz, A; Lebrun, P; Malaisse, WJ1
Inaba, M; Inoue, A; Morii, H; Nishizawa, Y; Okuno, S1
Gepts, W; Gorus, FK; In't Veld, PA; Pipeleers, DG; Schuit, FC1
Anselmi, E; D'Ocon, MP; Ivora, MD; Villar, A1
Blas, SD; Davis, FB; Davis, PJ; Mylotte, KM; Warnick, PR1
Berg, M; Boyd, AE; Gaines, KL; Nelson, TY; Rajan, AS1
Anselmi, E; D'Ocon, MP; Villar, A1
Patel, TB1
Anselmi, E; D'Ocon, MP; Ivorra, MD; Villar, A1
Kimura, S; Mine, T; Ogata, E; Ohsawa, H1
Kar, RN; Mukherjee, B; Mukherjee, SK1
Cook, GA1
Kaku, K; Kaneko, T; Matsuda, M1
Dyson, J; Patel, TB; Rashed, HM; Waller, FM1
Pollet, RJ; Rogers, BJ; Standaert, ML1
Anselmi, E; Ivorra, MD; Villar, A1
Boyd, AE; Gaines, KL; Hamilton, S1
Morita, K; Murakumo, Y; Nakanishi, A; Oka, M; Teraoka, K1
Patel, TB; Rashed, HM; White, CW1
Ashford, ML; Carrington, CA; Hales, CN; Kozlowski, RZ; Sturgess, NC1
Matsuyama, E; Nakahara, Y; Tamura, T1
Malaisse, WJ; Malaisse-Lagae, F; Mathias, PC; Sener, A1
Boyajy, LD; Hanson, RL; Isaacson, CM1
Colombo, R; Pinelli, A; Tofanetti, O; Trivulzio, S; Zecca, L1
Balkányi, I; Dévai, J; Kiss, V; Koltai, MZ; Pogátsa, G1
Hatao, K; Kaku, K; Kaneko, T; Matsuda, M; Tsuchiya, M1
Ravina, A1
Reinwein, D1
Beyer, J; Cordes, U; Haupt, E; Kutschera, J; Schöffling, K1
Hellman, B; Sehlin, J; Täljedal, IB2
Beyer, J; Cordes, U; Haupt, E; Köberich, W; Rosak, C; Schöffling, K1
Bartelt, KM; Beyer, J; Haupt, E; Rosak, C; Schöffling, K1
Gey, KF; Lorch, E; Sommer, P1
Beyer, J; Cordes, U; Schöffling, K; Sell, G1
Beyer, J; Gather, W; Schöffling, K1
Beyer, J; Haupt, E; Köberich, W; Rosak, C; Schöffling, K1
Beyer, J; Cordes, U; Haupt, E; Köberich, W; Schöffling, K2
Ashcroft, SJ; Randle, PJ; Weerasinghe, LC1
Jackson, WP; Keller, P; Van Mieghem, W1
Foy, JM; Standing, VF1
Pfeiffer, EF; Raptis, S; Rothenbuchner, G1
Bosboom, RS; Bouman, PR; Zweens, J1
Daweke, H; Fähndrich, W; Liebermeister, H; Schmitt, H1
Stowers, JM1
Botros, M; Ghareeb, A; Ghoneim, K; Selim, R; Wahba, N1
Addah, SA; Crockford, PM; Powell, P1
Beyer, J; Cordes, U; Haupt, E; Schöffling, K; Sell, G2
de Baere, H; de Leeuw, I; Decraene, P; Lemmens, P; Verhaegen, H1
Beyer, J; Haupt, E; Schöffling, K2
Hsu, PL; Luzzi, LA; Ma, JK1
Beyer, J; Happ, J; Haupt, E; Jungmann, E; Scherer, U; Schöffling, K1
Ide, T; Kajinuma, H; Kuzuya, TT1
Dunbar, JC; Foà, PP1
Loubatières, A; Loubatières-Mariani, MM1
Okajima, J1
Kar, BC; Panda, NC; Parija, CR; Tej, SC; Tripathy, BB1
Täljedal, IB1
Pfeiffer, EF; Raptis, S; Schröder, KE1
Hellman, B1
Hasselblatt, A; Panten, U; Poser, W; Schönborn, J1
Mughini, L; Polosa, P1
Heine, P; Kewitz, H; Schnapperelle, U1
Beringer, A1
Althoff, PH; Beyer, J; Fröhlich, A; Happ, J; Nest, E; Schöffling, K1
Bavel'skii, ZE; Kuts, LG; Lazaris, YA1
Beyer, J; Haupt, E; Rosak, C; Schöffling, K1
Aziz, MT; Einen, MA; el-Ebrashy, N; Higazi, AM; Mashaly, M1
Leupold, H1
Loubatiéres, A; Mariani, MM1
Chapal, J; Loubathières, A; Mariani, MM; Ribes, G1
Heine, P; Kewitz, H; Wiegboldt, KA1
Adadevoh, BK; Bolodeoku, JO1
Jeanrenaud, B; Kanazawa, Y; Lambert, AE; Orci, L; Renold, AE1
Howell, SL; Montague, W1
Lundquist, I1
Ebert, R; Hillebrandt, O; Schwabe, U1
Bird, GW; Eeles, GH; Litchfield, JA; Rahman, M; Wingham, J1
Kewitz, H1
Parodi, FA1
Pfeiffer, EF; Raptis, S1
Mitra, D; Mutalik, GS; Nayak, NJ; Oak, VR1
Cacciari, E; Cicognani, A; Collina, A; Pirazzoli, P; Tassoni, P1
Dörfler, H; Wolfram, G; Zöllner, N1
Cheah, JS1
Bloom, A1
Hinz, M; Maier, V; Nierle, C; Pfeiffer, EF; Schatz, H1
Love, AH; Teale, JD1
Beyer, J; Haupt, E; Köberich, W; Schöffling, K3
Tjioe, TO; Wacker, A1
Beyer, J; Ewald, W; Haupt, E; Mehnert, H; Nemeth, N; Schöffling, K; Wicklmayr, M1
Loubatières, A1
Sigroth, K; Steen, B; Svanborg, A1
Marble, A1
Hasslacher, C; Wahl, P1
Creutzfeldt, W; Scheler, F; Wigger, W1
Chandra, P; Wacker, A; Wacker, D1
Madsen, SN; Persson, I1
Bürkle, PA; Federlin, K; Hemm, G; Huber, V1
Consiglio, D; Hopps, V; Mantia, G1
Bänder, A1
Müller, R1
Schöffling, K1
Brauch, K; Haslbeck, M; Hepp, KD; Mehnert, H1
Brunetti, P; Filipponi, P; Marcelli, M; Nicoletti, I; Pacifici, R; Santeusanio, F1
Kanatsuka, A; Kumagai, A; Makino, H; Osegawa, M1
Abdel-Hamid, M; Ammon, HP; Enz, G; Rao, PG1
Altszuler, N; Cherksey, B1
Kimura, M; Suzuki, J1
Deleers, M; Lebrun, P; Malaisse, WJ1
Norlund, L; Sehlin, J1
Matthews, EK; Shotton, PA1
Gylfe, E; Hellman, B; Sehlin, J; Täljedal, B1
Tattersall, RB1
Whitney, JE; Yelich, MR1
Loubatieres-Mariani, MM1
Melander, A; Sartor, G; Scherstén, B; Wåhlin-Boll, E2
Feldman, JM; Skillman, TG1
Lisch, HJ; Sailer, S1
Lohmann, D; Verlohren, HJ1
Gonnermann, B; Gustson, D; Schatz, H1
Annamala, PT; Augusti, KT1
Pados, G1
Appel, S; Hitzenberger, G; Kalafsky, G; Kallay, Z; Kutz, K; Rüfenacht, T; Tetzloff, W1
Dubinsky, WP; Mayorga-Wark, O; Schultz, SG1
Broadway, NM; Saggerson, ED1
Adogu, AA; Ashford, ML; Hales, CN; Khan, RN; Ozanne, SE1
Lacey, MG; Stanford, IM1
Do, ML; Halterman, TJ; Howe, BB; Kau, ST; Li, JH; McConville, MW; Trivedi, S; Yochim, CL; Zografos, P1
Chudziak, F; Dickel, C; Moshiri, A; Panten, U; Schwanstecher, C; Schwanstecher, M1
Erdemli, G; Krnjević, K2
Krishnaiah, YS; Satyanarayana, S; Visweswaram, D1
Ballanyi, K; Richter, DW; Trapp, S1
Cahill, AL; Perlman, RL1
Ashford, ML; Hales, CN; Lee, K; Ozanne, SE1
Auchampach, JA; Gross, GJ; Pieper, GM; Yao, Z1
Bachmann, C; Chudziak, F; Löser, S; Panten, U; Schwanstecher, M1
Ashford, ML; Hales, CN; Lee, K; Ozanne, SE; Rowe, IC1
Elliott, BD; Johnson, R; Langer, O; Prihoda, T; Schenker, S1
Godfraind, JM; Krnjević, K1
Baró, I; Berthon, B; Escande, D; Hongre, AS1
Kruseman, AC; Menheere, PP; Müller, PG; Nijst, L; Sels, JP; Wolffenbuttel, BH1
Comtois, A; Kong, M; Light, P; Renaud, JM1
Buettger, C; Epstein, AJ; Hang, TL; Matschinsky, FM; Ronner, P1
Freedman, JE; Greif, GJ; Lin, YJ1
Fox, AP; Kelly, JS; Penington, NJ1
Ashcroft, SJ; Niki, I1
Nakaya, H1
Finta, EP; Fischer, HD; Harms, L; Illes, P; Sevcik, J1
Cohen, RA; Cowan, CL; Najibi, S; Palacino, JJ1
Krnjević, K; Zhu, PJ1
Arkhammar, P; Berggren, PO; Bokvist, K; Hallberg, A; Nilsson, T; Rorsman, P; Sjöholm, A; Welsh, M; Welsh, N1
Ben-Ari, Y; Crépel, V; Krnjević, K1
Frey, G; Hanke, W; Schlue, WR1
Broillet, MC; Horisberger, JD1
Katsumata, K; Katsumata, Y; Ozawa, T1
Van Wagoner, DR1
Elford, BC; Horner, HA; Kirk, K; Spillett, DJ1
Ammälä, C; Berggren, PO; Bertorello, AM; Bokvist, K; Chibalin, A; Deeney, JT; Eliasson, L; Flatt, PR; Gäbel, J; Gromada, J; Larsson, O; Lindström, P; Renström, E; Rhodes, CJ; Rorsman, P1
Gross, AS; Rieutord, A; Shenfield, GM; Stupans, I1
Hara, T; Hotta, N; Koh, N; Nakamura, J; Sakakibara, F; Takeuchi, N1
Bischoff, AM; Pierrefiche, O; Richter, DW1
Garcia-Barrado, MJ; Gilon, P; Henquin, JC; Jonas, JC1
Bijlstra, PJ; Lutterman, JA; Russel, FG; Smits, P; Thien, T1
Ballanyi, K; Brockhaus, J; Doutheil, J1
Howes, LG; Lykos, D; Sundaresan, P1
Selvaag, E1
Gagliardino, JJ; García, ME; Rossi, PF1
Abenhaim, L; Monette, J; van Staa, T1
Brownhill, V; Lee, K; Richardson, PJ1
Akaike, N; Ishibashi, H; Koyama, S; Murai, Y1
Fullerton, DA; McIntyre, RC; Meldrum, DR; Sheridan, BC1
Koyama, H; Mori, S; Nakajima, K; Sugioka, N; Uno, A1
Luo, M; O'Brien, RC1
Kitagawa, T; Nitadori, Y; Owada, M1
Bernardi, G; Federici, M; Guatteo, E; Knöpfel, T; Mercuri, NB; Siniscalchi, A1
Kikuchi, M; Niki, I; Oka, Y; Sakurada, M; Tsukuda, K1
Haller, M; Langohr, K; Mironov, SL; Richter, DW1
Chan, TY1
Dixon, AK; Freeman, TC; Lee, K; Richardson, PJ1
Ashcroft, FM; Gribble, FM; Seino, S; Tucker, SJ1
Ashcroft, SJ; Johnson, G; Tian, YA1
Aguilar-Bryan, L; Babenko, AP; Bryan, J; Gonzalez, G1
Benington, S; Best, L1
Bernardi, G; Calabresi, P; Centonze, D; Marfia, GA; Pisani, A1
Ikeda, T; Ochi, H1
Chagneau, C; De Gottardi, A; Fléjou, JF; Fouassier, L; Housset, C; Lahaye, P; Lebrec, D; Moreau, R; Reichen, J; Rona, JP; Tazi, KA1
Furukawa, N; Ohta, T; Wakitani, K; Yonemori, F1
Bataille, D; Blache, P; Gros, L; Salazar, G; Virsolvy, A1
Anello, M; Henquin, JC; Sato, Y1
Barg, S; Berggren, PO; Bertorello, A; Bokvist, K; Braun, M; Eliasson, L; Holmes, WE; Köhler, M; Renström, E; Rorsman, P; Thévenod, F1
Golanov, EV; Reis, DJ1
Jones, RB; Simpson, AE1
Ashcroft, FM; Ashcroft, SJ; Ashfield, R; Gribble, FM1
Brismar, T; Hyllienmark, L1
Carpenter, E; Peers, C; Roberts, ML; Taylor, SC1
Anello, M; Gilon, P; Henquin, JC1
Nadal, A; Quesada, I; Soria, B1
Aguilar-Bryan, L; Bryan, J1
Dallaporta, M; Orsini, JC; Perrin, J1
Bernardi, G; Giacomini, P; Marinelli, S; Mercuri, NB1
Brioni, JD; Gopalakrishnan, M; Molinari, EJ; Monteggia, LM; Roch, JM; Scott, VE; Shieh, CC; Sullivan, JP; Whiteaker, KL1
Callingham, BA; Crosbie, AE; Latimer, RD; Ritchie, AJ; Vuylsteke, A1
Bloom, SR; Ghatei, MA; Kulkarni, RN; Smith, DM; Wang, RM; Wang, ZL1
Galli Kienle, M; Magni, F; Marazzini, L; Monti, L; Pereira, S1
Ashford, ML; Campbell, CM; Kinsella, JM; McKay, NG1
Mohan, RM; Paterson, DJ1
de Smet, PA; Fischer, HR1
Dijkman, HB; Engbersen, R; Kramers, C; Moons, MM; Russel, FG; Smits, P; Wouterse, AC1
Almond, SC; Paterson, DJ1
Carlen, PL; Pahapill, PA; Pelletier, MR; Pennefather, PS1
Ball, AJ; Flatt, PR; McClenaghan, NH1
Kang, YY; Kim, JA; Lee, YS1
Bae, YH; Kim, SW; Park, KH1
Bielfeld-Ackermann, A; Konstas, AA; Korbmacher, C1
Duarte, ID; Soares, AC1
Gonoi, T; Ichikawa, K; Kusama, H; Seino, S; Shibasaki, T; Sunaga, Y; Yano, H1
Bisaccia, F; Gasbarro, AR; Lograno, MD; Ostuni, A; Tamburro, AM1
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI; Rosas, R; Torres-López, JE; Vidal-Cantú, GC2
Alves, D; Duarte, I1
Ashcroft, SJ; Mikhailov, MV; Mikhailova, EA1
Clapp, LH; Wilson, AJ1
Argüelles, CF; Granados-Soto, V; Ortiz, MI1
Giblin, JP; Quinn, K; Tinker, A1
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI2
Brockmöller, J; Gerloff, T; Kirchheiner, J; Meisel, C; Mrozikiewicz, PM; Niewinski, P; Roots, I1
Dugravot, S; Grolleau, F; Hue, B; Huignard, J; Lapied, B; Macherel, D; Rochetaing, A; Stankiewicz, M1
Chen, M; Dong, Y; Simard, JM1
Berggren, PO; Corkey, BE; Hamilton, JA; Kamp, F; Kizilbash, N1
Alves, DP; Duarte, ID; Leite, R; Tatsuo, MA1
Ball, AJ; Flatt, PR; McClenaghan, NH; McCluskey, JT1
Alves, DP; Amarante, LH; Duarte, ID1
Bae, JH; Cho, CH; Han, J; Jang, BC; Kim, SP; Kim, SS; Lee, HY; Lim, JG; Park, JW; Park, MJ; Song, DK; Suh, SI; Yun, JE1
Borelli, F; Costa, ZS; Jacobsen, M; Jacobus, AP; Loss, ES; Wassermann, GF1
Dao, C; Koster, JC; Nichols, CG; Remedi, MS1
Avshalumov, MV; Bao, L; Rice, ME1
Han, ES; Kim, YJ; Ko, HH; Lee, CS1
Acevedo, JJ; Darszon, A; de la Vega-Beltrán, JL; Felix, R; Mendoza-Lujambio, I; Treviño, CL1
Castañeda-Hernández, G; Castro-Olguín, J; Ortiz, MI; Peña-Samaniego, N1
Conte Camerino, D; Desai, RR; George, AL; Lundquist, AL; Mele, A; Tricarico, D1
Granados-Soto, V; Medina-Tato, DA; Ortiz, MI; Palma-Martínez, J; Sarmiento-Heredia, D1
Ashcroft, FM; Clark, PM; Codner, E; Ellard, S; Flanagan, SE; Flechtner, I; Hattersley, AT; Holst, JJ; Iotova, V; Klimes, I; Larkin, B; Malecki, MT; Njølstad, PR; Pearson, ER; Polak, M; Robert, JJ; Shield, J; Slingerland, AS; Søvik, O1
Kaku, K; Katsura, M; Matsuda, M; Ohkuma, S; Shigeto, M1
Brito, GA; Cunha, FQ; Ferreira, SH; Lotufo, CM; Ribeiro, RA; Sachs, D; Vale, ML1
Duarte, ID; Reis, GM1
Brennan, L; Flatt, PR; Hewage, C; Malthouse, JP; McClenaghan, NH; Newsholme, P1
Coetzee, WA; Ghiu, I; Gutstein, DE; Hendricks-Munoz, KD; Kontogeorgis, A; Malester, B; Tong, X; Xu, J1
Antunes, CM; Baldeiras, IE; Barbosa, RM; Rosário, LM; Santos, RM; Silva, AM; Tomé, AR1
Iwasaki, M; Katoh, M; Miki, T; Minami, K; Seino, S; Shibasaki, T; Sunaga, Y; Takahashi, H; Yokoi, N; Zhang, CL1
Chen, SR; Li, DP; Pan, HL1
Breschi, MC; Calderone, V; Cecchetti, V; Martelli, A; Sabatini, S; Testai, L1
Bailey, CJ; Flatt, PR; Irwin, N; McClenaghan, NH; McKinney, JM1
Cheng, X; Gribenko, AV; Tsalkova, T1
Andersson, C; Gislason, GH; Hansen, PR; Jørgensen, CH; Køber, L; Mérie, C; Norgaard, ML; Olesen, JB; Schmiegelow, M; Sørensen, R; Torp-Pedersen, C; Vaag, A; Weeke, P1
Chung, KK; Freestone, PS; Lipski, J1
Abdelmoneim, AS; Brocks, DR; Hasenbank, SE; Light, PE; Seubert, JM; Simpson, SH1
Cannone, G; Carbonara, G; Cippone, V; Conte Camerino, D; Fracchiolla, G; Laghezza, A; Loiodice, F; Mele, A; Rolland, JF; Tortorella, P; Tricarico, D1
Ishii, I; Itoh, N; Kimura, H; Kimura, T; Kimura, Y; Naito, Y; Niki, I; Taniguchi, S; Umeki, T; Yamamoto, H1
Cui, G; McCarty, NA; Song, B; Turki, HW1
Fatehi, M; Lang, VY; Light, PE1
Ahmadi, A; Khalili, M; Nahri-Niknafs, B; Roudsari, EM; Seyedhoseyni, S1
Bond, R; Choisy, SC; El Haou, S; Hancox, JC; James, AF; Khaliulin, I; Kim, SJ; Lin, H; Milnes, JT; Suleiman, MS; Zhang, H1
Bo, S; Castiglione, A; Cavallo-Perin, P; Ciccone, G; Durazzo, M; Gentile, L; Ghigo, E1
Friščić, T; Mottillo, C; Štrukil, V; Tan, D1
Jung, JS; Kim, CH; Kim, SJ; Kim, SS; Lim, SM; Park, SH; Sim, YB; Suh, HW1
Andersson, C; Fosbøl, EL; Gislason, G; Køber, L; Mogensen, UM; Scheller, NM; Schramm, TK; Torp-Pedersen, C; Vaag, A1
Eliassi, A; Fahanik-Babaei, J; Ghasemi, M; Saghiri, R; Salari, S; Sauve, R1
Henquin, JC; Nenquin, M1
Brown, J; Crowther, CA; Hughes, B; Martis, R; Rowan, J1
Bashir, K; Chang, C; Chen, G; Fu, Q; Ge, Y; Guo, P; Jing, W; Luo, Z; Shu, H; Xu, X1
Barella, LF; Chen, W; Cheng, X; Cui, Y; Gurevich, VV; Mei, FC; Rossi, M; Wess, J; Zhu, L1
Jannetto, PJ; Langman, LJ1

Reviews

19 review(s) available for glyburide and tolbutamide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
["First" and "second" generation sulfonylureas: distinction or difference? (author's transl)].
    Diabete & metabolisme, 1978, Volume: 4, Issue:2

    Topics: Animals; Chlorpropamide; Dose-Response Relationship, Drug; Glipizide; Glyburide; Half-Life; Humans; Hypoglycemic Agents; Kinetics; Structure-Activity Relationship; Sulfonylurea Compounds; Tolbutamide

1978
[New aspects of therapy with oral antidiabetic agents].
    Wiener medizinische Wochenschrift (1946), 1979, Dec-30, Volume: 199, Issue:24

    Topics: Acidosis; Biguanides; Blood Proteins; Chlorpropamide; Diabetes Mellitus; Diabetic Nephropathies; Drug Interactions; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Protein Binding; Sulfonamides; Sulfonylurea Compounds; Tolbutamide

1979
Drug interactions with oral sulphonylurea hypoglycaemic drugs.
    Drugs, 1977, Volume: 13, Issue:1

    Topics: Allopurinol; Analgesics; Anticoagulants; Chloramphenicol; Chlorpropamide; Disulfiram; Drug Interactions; Ethanol; Glyburide; Humans; Hypoglycemic Agents; Hypolipidemic Agents; Kinetics; Monoamine Oxidase Inhibitors; Novobiocin; Phenylbutazone; Phenytoin; Probenecid; Propranolol; Rifampin; Sulfonamides; Sulfonylurea Compounds; Tolbutamide

1977
Oral treatment in diabetes.
    Clinics in endocrinology and metabolism, 1972, Volume: 1, Issue:3

    Topics: Acetohexamide; Acidosis; Administration, Oral; Animals; Biguanides; Cardiovascular Diseases; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Glyburide; Humans; Hypoglycemia; Liver; Obesity; Structure-Activity Relationship; Sulfonylurea Compounds; Tolazamide; Tolbutamide

1972
[Central role of the pancreas in the mechanism of action of hypoglycemic sulfonamides and their consequences in the therapy and prevention of diabetes].
    Revista clinica espanola, 1970, Jun-15, Volume: 117, Issue:5

    Topics: Animals; Diabetes Mellitus; Glyburide; Growth; Growth Hormone; Humans; Hypoglycemic Agents; Pancreas; Rats; Sulfonamides; Tolbutamide

1970
Glibenclamide, a new sulphonylurea: whither oral hypoglycaemic agents?
    Drugs, 1971, Volume: 1, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Blood Glucose; Carbohydrates; Child; Coronary Disease; Diabetes Complications; Diabetes Mellitus; Diet, Diabetic; Fatty Acids; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Sulfonylurea Compounds; Tolbutamide

1971
The pharmacology and metabolism of oral antidiabetic drugs.
    Australian and New Zealand journal of medicine, 1971, Volume: 1

    Topics: Administration, Oral; Adrenal Glands; Animals; Blood Glucose; Chemical Phenomena; Chemistry; Dogs; Glyburide; Guinea Pigs; Humans; Hypoglycemic Agents; In Vitro Techniques; Insulin; Islets of Langerhans; Mice; Rabbits; Rats; Semicarbazides; Sulfonamides; Sulfonylurea Compounds; Tolbutamide

1971
Interaction of sulfonylurea with the pancreatic B-cell.
    Experientia, 1984, Oct-15, Volume: 40, Issue:10

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Adenosine Triphosphate; Amino Acids; Animals; Calcimycin; Calcium; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Fatty Acids; Glucose; Glyburide; Humans; Islets of Langerhans; Lasalocid; Membrane Potentials; NADP; Phenylbutazone; Rubidium; Serum Albumin; Sulfonylurea Compounds; Time Factors; Tolbutamide

1984
[25 years of diabetic treatment by oral hypoglycemic agents: successes and failures].
    Journees annuelles de diabetologie de l'Hotel-Dieu, 1984

    Topics: Aged; Aging; Blood Glucose; Cardiovascular Diseases; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diet, Reducing; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Middle Aged; Phenformin; Sulfonylurea Compounds; Tolbutamide

1984
[Potential role of ATP-sensitive K+ channels in ischemia- and reperfusion-induced arrhythmias].
    Kokyu to junkan. Respiration & circulation, 1993, Volume: 41, Issue:6

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Arrhythmias, Cardiac; Benzopyrans; Cromakalim; Glyburide; Guanidines; Humans; Myocardial Ischemia; Myocardial Reperfusion Injury; Myocardium; Niacinamide; Nicorandil; Pinacidil; Potassium; Potassium Channels; Pyrroles; Tolbutamide

1993
Cardiovascular effects of sulphonylurea derivatives.
    Diabetes research and clinical practice, 1996, Volume: 31 Suppl

    Topics: Adenosine Triphosphate; Animals; Cardiovascular System; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemic Agents; Potassium Channels; Sulfonylurea Compounds; Tolbutamide

1996
Cardiovascular effects of oral hypoglycaemic drugs.
    Clinical and experimental pharmacology & physiology, 1996, Volume: 23, Issue:3

    Topics: Biguanides; Diabetes Mellitus, Type 2; Glyburide; Heart; Hemodynamics; Humans; Hypoglycemic Agents; Lipoproteins; Metformin; Myocardial Contraction; Potassium Channel Blockers; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide

1996
Anti-diabetic drugs as a cause of hypoglycaemia among acute medical admissions in Hong Kong and Singapore--relationship to the prescribing patterns in diabetic patients.
    Singapore medical journal, 1998, Volume: 39, Issue:4

    Topics: Acute Disease; Age Factors; Aged; China; Diabetes Mellitus; Drug Prescriptions; Drug Utilization; Glyburide; Hong Kong; Humans; Hypoglycemia; Hypoglycemic Agents; Middle Aged; Patient Admission; Practice Patterns, Physicians'; Prevalence; Risk Factors; Singapore; Tolbutamide

1998
Sulfonylurea receptors: ABC transporters that regulate ATP-sensitive K(+) channels.
    Biochimica et biophysica acta, 1999, Dec-06, Volume: 1461, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; ATP-Binding Cassette Transporters; Benzamides; Cell Line; Cytoplasm; Electrochemistry; Endoplasmic Reticulum; Glyburide; Humans; Magnesium; Models, Molecular; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

1999
[Timing of administration of sulfonyl urea derivatives].
    Nederlands tijdschrift voor geneeskunde, 2000, Jun-17, Volume: 144, Issue:25

    Topics: Biological Availability; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Drug Administration Schedule; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Tolbutamide

2000
Implications of pharmacogenetics for individualizing drug treatment and for study design.
    Journal of molecular medicine (Berlin, Germany), 2003, Volume: 81, Issue:3

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Clinical Trials as Topic; Cytochrome P-450 Enzyme System; Genotype; Glyburide; Humans; Hypoglycemic Agents; Pharmaceutical Preparations; Pharmacogenetics; Tolbutamide

2003
Variations in tissue selectivity amongst insulin secretagogues: a systematic review.
    Diabetes, obesity & metabolism, 2012, Volume: 14, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Cardiovascular Diseases; Cricetinae; Cyclohexanes; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Ischemic Preconditioning, Myocardial; Isoindoles; Mice; Muscle, Smooth, Vascular; Myocytes, Cardiac; Nateglinide; Phenylalanine; Piperidines; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Risk Factors; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2012
Oral anti-diabetic pharmacological therapies for the treatment of women with gestational diabetes.
    The Cochrane database of systematic reviews, 2017, 01-25, Volume: 1

    Topics: Acarbose; Administration, Oral; Diabetes, Gestational; Female; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Metformin; Pregnancy; Randomized Controlled Trials as Topic; Tolbutamide

2017

Trials

18 trial(s) available for glyburide and tolbutamide

ArticleYear
[Clinical investigations of the effect of tolbutamide and glibenclamide on pancreatic glucagon secretion (author's transl)].
    Klinische Wochenschrift, 1975, Jun-15, Volume: 53, Issue:12

    Topics: Adult; Arginine; Blood Glucose; Glucagon; Glyburide; Humans; Insulin; Male; Pancreas; Tolbutamide

1975
[Therapeutic effect of glibenclamide contrasted with other oral antidiabetic agents].
    Vutreshni bolesti, 1975, Volume: 14, Issue:3

    Topics: Administration, Oral; Adult; Biguanides; Chlorpropamide; Chronic Disease; Clinical Trials as Topic; Diabetes Mellitus; Drug Evaluation; Drug Therapy, Combination; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Tolbutamide

1975
Efficacy of gliclazide in comparison with other sulphonylureas in the treatment of NIDDM.
    Diabetes research and clinical practice, 1991, Volume: 14 Suppl 2

    Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Diet, Diabetic; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Tolbutamide

1991
A randomized crossover study of sulphonylurea and insulin treatment in patients with type 2 diabetes poorly controlled on dietary therapy.
    Diabetic medicine : a journal of the British Diabetic Association, 1989, Volume: 6, Issue:6

    Topics: Blood Glucose; C-Peptide; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Diet, Diabetic; Fasting; Female; Glyburide; Glycated Hemoglobin; Humans; Insulin; Islets of Langerhans; Male; Middle Aged; Random Allocation; Tolbutamide

1989
[The influence of various sulphonylurea derivatives on the oral glucose-tolerance tests in healthy subjects and obese and maturity-onset diabetics (author's transl)].
    Deutsche medizinische Wochenschrift (1946), 1974, Mar-01, Volume: 99, Issue:9

    Topics: Administration, Oral; Adult; Blood Glucose; Diabetes Mellitus; Glucose; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Obesity; Statistics as Topic; Stimulation, Chemical; Sulfonylurea Compounds; Time Factors; Tolbutamide

1974
Dose-response relationships of tolbutamide and glibenclamide in diabetes mellitus.
    European journal of clinical pharmacology, 1974, Aug-23, Volume: 7, Issue:5

    Topics: Adult; Aged; Blood Glucose; Clinical Trials as Topic; Colorimetry; Diabetes Mellitus; Dose-Response Relationship, Drug; Female; Glyburide; Humans; Injections; Insulin; Male; Middle Aged; Obesity; Radioimmunoassay; Time Factors; Tolbutamide

1974
[Blood sugar, serum insulin, nonesterified fatty acids and somatotropin in daily profile in adult diabetics under monotherapy with various sulfonylureas].
    Arzneimittel-Forschung, 1974, Volume: 24, Issue:8

    Topics: Blood Glucose; Body Weight; Diabetes Mellitus; Diet, Diabetic; Fatty Acids, Nonesterified; Glyburide; Glycosuria; Growth Hormone; Humans; Insulin; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1974
The effect of oral sulphonylureas on blood glucose and insulin.
    Ghana medical journal, 1973, Volume: 12, Issue:4

    Topics: Administration, Oral; Adult; Blood Glucose; Body Height; Body Weight; Clinical Trials as Topic; Female; Glyburide; Humans; Insulin; Male; Placebos; Sulfonylurea Compounds; Tolbutamide

1973
Controlled extension of oral antidiabetic therapy on former insulin dependent diabetics by means of the combined i.v. glibenclamide-glucose-response-test.
    Diabetologia, 1972, Volume: 8, Issue:1

    Topics: Administration, Oral; Adult; Age Factors; Aged; Clinical Trials as Topic; Diabetes Mellitus; Drug Combinations; Drug Resistance; Female; Glucose; Glyburide; Hemochromatosis; Humans; Hypoglycemic Agents; Injections, Intravenous; Insulin; Insulin Antibodies; Male; Methods; Middle Aged; Prognosis; Sulfonylurea Compounds; Tolbutamide

1972
[Clinical testing of a sulphonylurea derivative, glibornuride].
    Deutsche medizinische Wochenschrift (1946), 1972, Jul-21, Volume: 97, Issue:29

    Topics: Adult; Aged; Biguanides; Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus; Diet Therapy; Female; Glyburide; Glycosuria; Humans; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1972
A clinical evaluation of glibenclamide (HB 419, "Daonil") a new antidiabetic sulphonylurea.
    Singapore medical journal, 1972, Volume: 13, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Aged; Alcohol Drinking; Clinical Trials as Topic; Diabetes Mellitus; Female; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemia; Insulin; Male; Middle Aged; Pyrimidines; Sulfonylurea Compounds; Tolbutamide

1972
Oral substitutes for insulin: modern appraisal of their action and indications.
    Israel journal of medical sciences, 1972, Volume: 8, Issue:6

    Topics: Adolescent; Adult; Aged; Animals; Blood Glucose; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diet, Diabetic; Dogs; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemic Agents; Insulin; Middle Aged; Phenformin; Placebos; Rats; Sulfonamides; Tolbutamide

1972
[Therapy of diabetes in adults using Glibornurid. Results and clinical studies].
    Deutsche medizinische Wochenschrift (1946), 1973, May-04, Volume: 98, Issue:18

    Topics: Aged; Blood Glucose; Body Weight; Camphanes; Clinical Trials as Topic; Diabetes Mellitus; Drug Hypersensitivity; Female; Glyburide; Glycosuria; Humans; Hypoglycemic Agents; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1973
[Clinical testing of a sulfonylurea preparation (glibenclamide)].
    Lakartidningen, 1969, Nov-05, Volume: 66, Issue:45

    Topics: Adult; Aged; Chlorpropamide; Clinical Trials as Topic; Diabetes Mellitus; Diet Therapy; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Tolbutamide

1969
The clinical evaluation of an oral antidiabetic drug.
    Australian and New Zealand journal of medicine, 1971, Volume: 1

    Topics: Administration, Oral; Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus; Glyburide; Humans; Insulin; Lipids; Sulfonylurea Compounds; Tolbutamide

1971
Lack of interaction between fluvastatin and oral hypoglycemic agents in healthy subjects and in patients with non-insulin-dependent diabetes mellitus.
    The American journal of cardiology, 1995, Jul-13, Volume: 76, Issue:2

    Topics: Administration, Oral; Anticholesteremic Agents; Blood Glucose; C-Peptide; Diabetes Mellitus, Type 2; Diclofenac; Drug Interactions; Fatty Acids, Monounsaturated; Fluvastatin; Glyburide; Humans; Hydroxymethylglutaryl CoA Reductases; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Indoles; Insulin; Lovastatin; Placebos; Simvastatin; Tolbutamide

1995
Effects of a new oral hypoglycaemic agent, repaglinide, on metabolic control in sulphonylurea-treated patients with NIDDM.
    European journal of clinical pharmacology, 1993, Volume: 45, Issue:2

    Topics: Aged; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Female; Fructosamine; Gliclazide; Glyburide; Glycated Hemoglobin; Hexosamines; Humans; Hypoglycemic Agents; Lipids; Male; Middle Aged; Piperidines; Tolbutamide

1993
An importance of carbohydrate ingestion for the expression of the effect of alpha-glucosidase inhibitor in NIDDM.
    Diabetes care, 1996, Volume: 19, Issue:6

    Topics: Biomarkers; Blood Glucose; C-Peptide; Circadian Rhythm; Diabetes Mellitus, Type 2; Dietary Carbohydrates; Energy Intake; Enzyme Inhibitors; Follow-Up Studies; Glyburide; Glycated Hemoglobin; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Inpatients; Insulin; Middle Aged; Regression Analysis; Retrospective Studies; Sulfonylurea Compounds; Tolbutamide

1996

Other Studies

379 other study(ies) available for glyburide and tolbutamide

ArticleYear
Sulfonyliminoimidazolidines. A new class of oral hypoglycemic agents. 1. 1-[[p-[2-(acylamino)ethyl]phenyl]sulfonyl]-2-iminoimidazolidines.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:7

    Topics: Animals; Biological Assay; Blood Glucose; Diabetes Mellitus, Experimental; Hypoglycemic Agents; Imidazoles; Indicators and Reagents; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Sulfones

1983
Reconstitution of IKATP: an inward rectifier subunit plus the sulfonylurea receptor.
    Science (New York, N.Y.), 1995, Nov-17, Volume: 270, Issue:5239

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; ATP-Binding Cassette Transporters; Base Sequence; Cell Line; Chromosome Mapping; Chromosomes, Human, Pair 11; Cloning, Molecular; Cricetinae; Diazoxide; Humans; Islets of Langerhans; KATP Channels; Mice; Molecular Sequence Data; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Rubidium; Sulfonylurea Compounds; Sulfonylurea Receptors

1995
A novel sulfonylurea receptor forms with BIR (Kir6.2) a smooth muscle type ATP-sensitive K+ channel.
    The Journal of biological chemistry, 1996, Oct-04, Volume: 271, Issue:40

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; ATP-Binding Cassette Transporters; Base Sequence; Cell Line; Cloning, Molecular; DNA, Complementary; Humans; Mice; Molecular Sequence Data; Muscle, Smooth; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sulfonylurea Receptors

1996
Inhibitory effect of anti-diabetic agents on rat organic anion transporter rOAT1.
    European journal of pharmacology, 2000, Jun-16, Volume: 398, Issue:2

    Topics: Animals; Anion Transport Proteins; Binding, Competitive; Carbon Radioisotopes; Carrier Proteins; Chlorpropamide; Cyclohexanes; Dose-Response Relationship, Drug; Female; Glyburide; Hypoglycemic Agents; Kinetics; Nateglinide; Oocytes; p-Aminohippuric Acid; Phenylalanine; Rats; RNA, Complementary; Sulfonylurea Compounds; Tolbutamide; Xenopus

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Comparative inhibitory effects of different compounds on rat oatpl (slc21a1)- and Oatp2 (Slc21a5)-mediated transport.
    Pharmaceutical research, 2002, Volume: 19, Issue:2

    Topics: Algorithms; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antibiotics, Antitubercular; Antimalarials; Biological Transport, Active; Digoxin; Enzyme Inhibitors; Estradiol; Ibuprofen; LLC-PK1 Cells; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Organic Cation Transport Proteins; Quinidine; Quinine; Rats; Rifampin; Swine

2002
Citrus juices inhibit the function of human organic anion-transporting polypeptide OATP-B.
    Drug metabolism and disposition: the biological fate of chemicals, 2005, Volume: 33, Issue:4

    Topics: Beverages; Cell Line; Citrus paradisi; Citrus sinensis; Estrone; Glyburide; Humans; Organic Anion Transporters; Transfection

2005
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions.
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Binding Sites; Crystallography, X-Ray; Drug Interactions; Humans; Pharmaceutical Preparations; Protein Binding; Protein Structure, Tertiary; Serum Albumin; Spectrometry, Fluorescence

2010
In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Cholestasis; Drug-Related Side Effects and Adverse Reactions; Humans; Insecta; Rats; Risk Factors

2012
Comparison of cryopreserved HepaRG cells with cryopreserved human hepatocytes for prediction of clearance for 26 drugs.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:1

    Topics: Cell Line, Tumor; Cryopreservation; Female; Hepatocytes; Humans; Male; Metabolic Clearance Rate; Pharmaceutical Preparations; Predictive Value of Tests

2012
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
    Chemical biology & drug design, 2016, Volume: 88, Issue:6

    Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain

2016
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
High-performance liquid chromatographic determination of glipizide and some other sulfonylurea drugs in serum.
    Journal of chromatography, 1979, Dec-01, Volume: 164, Issue:4

    Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Glipizide; Glyburide; Humans; Hydrogen-Ion Concentration; Sulfonylurea Compounds; Tolbutamide

1979
Effects of chronic and acute treatment with sulfonylureas on plasma insulin and glucose levels in the rat.
    Diabete & metabolisme, 1978, Volume: 4, Issue:1

    Topics: Acetoacetates; Animals; Blood Glucose; Fasting; Female; Glyburide; Hydroxybutyrates; Insulin; Kinetics; Rats; Sulfonylurea Compounds; Tolbutamide

1978
Glycogen phosphorylase activities in sulfonylureas treated rats.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1978, Volume: 10, Issue:4

    Topics: Animals; Female; Glyburide; Liver; Muscles; Phosphorylases; Rats; Sulfonylurea Compounds; Tolbutamide

1978
Studies on the effect of tolbutamide, glibenclamide, HB 699, and glucose on serum insulin and blood glucose in gastro-enterectomized dogs.
    Archives internationales de pharmacodynamie et de therapie, 1978, Volume: 234, Issue:1

    Topics: Animals; Blood Glucose; Digestive System Physiological Phenomena; Dogs; Female; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Male; Pancreas; Regional Blood Flow; Sulfonylurea Compounds; Time Factors; Tolbutamide; Vagotomy

1978
Changes in plasma amino acids levels and "in vivo" gluconeogenesis from alanine in rats chronically treated with sulfonylureas.
    Diabete & metabolisme, 1978, Volume: 4, Issue:3

    Topics: Alanine; Amino Acids; Animals; Blood Glucose; Female; Gluconeogenesis; Glyburide; Glycerides; Glycerol; Hypoglycemic Agents; Liver; Liver Glycogen; Rats; Sulfonylurea Compounds; Tolbutamide

1978
Effect of sulfonylurea treatment and fasting on the levels of plasma amino acids in the rat.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1978, Volume: 10, Issue:6

    Topics: Amino Acids; Animals; Fasting; Female; Glyburide; Hydroxyproline; Proline; Rats; Sulfonylurea Compounds; Tolbutamide

1978
Gas chromatographic determination of glibenclamide in plasma.
    Clinica chimica acta; international journal of clinical chemistry, 1979, Apr-16, Volume: 93, Issue:2

    Topics: Administration, Oral; Chromatography, Gas; Glyburide; Humans; Microchemistry; Tolbutamide

1979
Insulin release by tolbutamide and glibenclamide. A comparative study on the perfused rat pancreas.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 306, Issue:3

    Topics: Animals; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Pancreas; Rats; Time Factors; Tolbutamide

1979
Release of gastrin from the skeletal muscles and from the antral mucosa in cats induced by sulfonuric drugs.
    Acta physiologica Scandinavica, 1979, Volume: 106, Issue:3

    Topics: Animals; Cats; Gastric Mucosa; Gastrins; Glyburide; Hindlimb; Muscles; Perfusion; Pyloric Antrum; Secretory Rate; Tolbutamide

1979
[Comparative use of gliquidone and tolbutamide administered intravenously].
    MMW, Munchener medizinische Wochenschrift, 1975, Sep-05, Volume: 117, Issue:36

    Topics: Basal Metabolism; Blood Glucose; Fasting; Fatty Acids, Nonesterified; Glyburide; Humans; Injections, Intravenous; Insulin; Insulin Secretion; Sulfonylurea Compounds; Time Factors; Tolbutamide

1975
Dynamics of sulfonylurea-induced insulin release from the isolated perfused rat pancreas.
    Diabetologia, 1976, Volume: 12, Issue:4

    Topics: Animals; Glipizide; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Perfusion; Rats; Sulfonylurea Compounds; Tolbutamide

1976
Hyaluronidase-induced inhibition of the insulinotropic action of sulfonylureas, leucine, and glucagon in rodent isolated pancreatic islets.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1976, Volume: 8, Issue:2

    Topics: Animals; Chlorpropamide; Cricetinae; Female; Glucagon; Glucose; Glyburide; Hyaluronoglucosaminidase; Insulin; Islets of Langerhans; Leucine; Mice; Microbial Collagenase; Rats; Species Specificity; Sulfonylurea Compounds; Tolbutamide

1976
[The role of cyclic AMP in the control of insulin secretion (author's transl)].
    MMW, Munchener medizinische Wochenschrift, 1977, Sep-23, Volume: 119, Issue:38

    Topics: Animals; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mannose; Phosphodiesterase Inhibitors; Rats; Receptors, Drug; Time Factors; Tolbutamide; Xanthines

1977
Inhibition of vasopressin-stimulated prostaglandin E biosynthesis by chlorpropamide in the toad urinary bladder. Mechanism of enhancement of vasopressin-stimulated water flow.
    The Journal of clinical investigation, 1977, Volume: 60, Issue:6

    Topics: Animals; Anura; Arginine Vasopressin; Chlorpropamide; Chromatography, Thin Layer; Cyclic AMP; Glyburide; Lipid Metabolism; Permeability; Prostaglandins E; Stimulation, Chemical; Structure-Activity Relationship; Theophylline; Tolbutamide; Urinary Bladder; Vasopressins; Water

1977
The positive inotropic action of sulfonylureas. A mechanism independent of cyclic adenosine 3',5'-monophosphate.
    Diabetes, 1978, Volume: 27, Issue:6

    Topics: Adenylyl Cyclases; Animals; Atrial Function; Cyclic AMP; Dose-Response Relationship, Drug; Glyburide; Guinea Pigs; Heart; Isoproterenol; Male; Myocardial Contraction; Myocardium; Rabbits; Rats; Species Specificity; Tolbutamide; Ventricular Function

1978
Cyclic AMP and insulin release.
    Acta paediatrica Scandinavica. Supplement, 1977, Issue:270

    Topics: Animals; Cricetinae; Cyclic AMP; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Tolbutamide

1977
Modification of diuresis in the rat by chlorpropamide, glibenclamide and tolbutamide.
    Experientia, 1975, May-15, Volume: 31, Issue:5

    Topics: Administration, Oral; Animals; Body Water; Chlorpropamide; Diabetes Mellitus; Diuresis; Glyburide; Hydrogen-Ion Concentration; Male; Potassium; Rats; Sodium; Streptozocin; Time Factors; Tolbutamide

1975
Side effects of therapy in diabetes evaluated by a self-administered questionnaire.
    Journal of chronic diseases, 1977, Volume: 30, Issue:1

    Topics: Chlorpropamide; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Patient Acceptance of Health Care; Phenformin; Surveys and Questionnaires; Tolbutamide

1977
The pharmacology of a new hypoglycaemic agent N-[4-(2-(2,3-dihydrobenzo(b)furan-m-carboxamido)-ethyl)-benzenesulphonyl]-N'-cyclohexylurea (NOVO CS 476). I. Pharmacological studies on the hypoglycaemic effect.
    Acta pharmacologica et toxicologica, 1977, Volume: 40, Issue:2

    Topics: Administration, Oral; Animals; Blood Glucose; Dogs; Drug Evaluation, Preclinical; Glucose Tolerance Test; Glyburide; Hypoglycemic Agents; Injections, Intravenous; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred Strains; Rabbits; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide

1977
The pharmacology of a new hypoglycaemic agent N-[4-(2-(2,3-dihydrobenzo(b)furan-7-carboxamid o)-ethyl)-benzenesulphonyl]-N'-cyclohexlurea (NOVO CS 476). III. General pharmacological studies.
    Acta pharmacologica et toxicologica, 1977, Volume: 40, Issue:2

    Topics: Animals; Blood Pressure; Cats; Chlorpropamide; Diuresis; Dogs; Female; Glyburide; Guinea Pigs; Heart; Hypoglycemic Agents; Male; Muscle Contraction; Muscle, Smooth; Papillary Muscles; Rats; Sulfonylurea Compounds; Tolbutamide

1977
[Clinico-statistical studies of the use of oral hypoglycemic agents in the therapy of diabetes: critical evaluation of their effectiveness and tolerance].
    La Clinica terapeutica, 1977, Jul-15, Volume: 82, Issue:1

    Topics: Adult; Aged; Chlorpropamide; Diabetes Mellitus; Drug Evaluation; Drug Therapy, Combination; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Phenformin; Tolbutamide

1977
[Hypoglycemic sulfonylurea metabolites: clinical interest. Experiences with glibenclamide in the rat].
    Schweizerische medizinische Wochenschrift, 1977, Sep-17, Volume: 107, Issue:37

    Topics: Animals; Biotransformation; Blood Glucose; Chlorpropamide; Glyburide; Injections, Intraperitoneal; Rats; Tolbutamide

1977
Long-term actions of sulfonylureas on (pro-) insulin biosynthesis and secretion: I. Lack of evidence for a compensatory increase in (pro-) insulin biosynthesis after exposure of isolated pancreatic rat islets to tolbutamide and glibenclamide in vitro.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1977, Volume: 9, Issue:6

    Topics: Animals; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Proinsulin; Rats; Time Factors; Tolbutamide

1977
[Insulin and pro-insulin secretion following intravenous administration of tolbutamide, glisoxepide and glibenclamide].
    Arzneimittel-Forschung, 1978, Volume: 28, Issue:1

    Topics: Blood Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Proinsulin; Sulfonylurea Compounds; Time Factors; Tolbutamide

1978
Long-term actions of sulfonylureas on (pro-)insulin biosynthesis and secretion. II. Studies after administration of tolbutamide and glibenclamide to rats in vivo.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1978, Volume: 10, Issue:1

    Topics: Animals; Body Weight; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Male; Proinsulin; Rats; Time Factors; Tolbutamide

1978
Sulfonylurea-induced factitious hypoglycemia in a nondiabetic nurse.
    Canadian Medical Association journal, 1975, Jan-11, Volume: 112, Issue:1

    Topics: Adult; Blood Glucose; Female; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemia; Insulin; Munchausen Syndrome; Sulfonylurea Compounds; Tolbutamide

1975
[Experimental studies on the mechanism of thrombocyte aggregation inhibition caused by sulfonylurea compounds. 2. Modification of blood sugar and thrombocyte aggregation by oral antidiabetics].
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:2

    Topics: Adenosine Monophosphate; Administration, Oral; Animals; Biguanides; Blood Glucose; Carbutamide; Depression, Chemical; Dose-Response Relationship, Drug; Glyburide; Hypoglycemic Agents; Injections, Intravenous; Platelet Adhesiveness; Platelet Aggregation; Pyrimidines; Rats; Semicarbazides; Sulfonylurea Compounds; Tolazamide; Tolbutamide

1975
[Effect of methylpyrazole-carboxylic acid on carbohydrate and lipid metabolisms in patients with diabetes mellitus].
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:1

    Topics: Aged; Blood Glucose; Carbutamide; Cholesterol; Diabetes Mellitus; Drug Evaluation; Fatty Acids, Nonesterified; Female; Glyburide; Glycosuria; Humans; Hypoglycemic Agents; Male; Middle Aged; Pyrazoles; Stimulation, Chemical; Tolbutamide; Triglycerides

1975
Myocardial infarction in diabetics.
    The Quarterly journal of medicine, 1975, Volume: 44, Issue:173

    Topics: Administration, Oral; Adult; Aged; Chlorpropamide; Coronary Care Units; Diabetes Complications; Diabetes Mellitus; Diabetic Retinopathy; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Myocardial Infarction; Phenformin; Sex Factors; Sulfonylurea Compounds; Tolbutamide

1975
Gliflumide, a new oral antidiabetic of high potency and efficacy.
    International journal of clinical pharmacology and biopharmacy, 1975, Volume: 12, Issue:1-2

    Topics: Administration, Oral; Animals; Blood Glucose; Cricetinae; Dogs; Fatty Acids, Nonesterified; Glucose; Glyburide; Humans; Hypoglycemic Agents; Injections, Intravenous; Insulin; Insulin Secretion; Kinetics; Pyrimidines; Rats; Stereoisomerism; Sulfonamides; Theophylline; Tolbutamide

1975
[Studies on new sulfonylurea derivatives and their metabolites in isolated Langerhans's islets of the rat pancreas (author's transl].
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:8

    Topics: Animals; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Stimulation, Chemical; Sulfonylurea Compounds; Time Factors; Tolbutamide

1975
[The importance of serum insulin determination in the diagnosis and treatment of diabetes mellitus (author's transl)].
    MMW, Munchener medizinische Wochenschrift, 1975, Oct-10, Volume: 117, Issue:41

    Topics: Blood Glucose; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diet Therapy; Dose-Response Relationship, Drug; Glucose Tolerance Test; Glyburide; Humans; Insulin; Obesity; Prediabetic State; Prognosis; Radioimmunoassay; Sulfonylurea Compounds; Tolbutamide

1975
(Pro-) insulin biosynthesis and release of newly synthesized (pro-) insulin from isolated islets of rat pancreas in the presence of amino acids and sulphonylureas.
    European journal of clinical investigation, 1975, Nov-21, Volume: 5, Issue:6

    Topics: Amino Acids; Animals; Arginine; Glyburide; In Vitro Techniques; Insulin; Islets of Langerhans; Lysine; Male; Proinsulin; Rats; Sulfonylurea Compounds; Tolbutamide

1975
[Relation of uric acid and arteriosclerosis on an experimental model of chickens fed with eggs. Influence of insulin and oral antidiabetics (glibenclamide and tolbutamide)].
    Revista clinica espanola, 1975, Nov-15, Volume: 139, Issue:3

    Topics: Animals; Arteriosclerosis; Chickens; Cholesterol, Dietary; Disease Models, Animal; Eggs; Glyburide; Insulin; Sex Factors; Tolbutamide; Uric Acid

1975
[Effect of tolbutamide and glibenclamide on glucagon secretion in subjects with normal metabolism and in diabetics].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1975, Volume: 81

    Topics: Adult; Diabetes Mellitus; Glucagon; Glyburide; Humans; Male; Tolbutamide

1975
Circular dichroism studies on the interaction of sulfonylureas with bovine and human serum albumin.
    Research communications in chemical pathology and pharmacology, 1976, Volume: 13, Issue:3

    Topics: Binding Sites; Binding, Competitive; Carbutamide; Chlorpropamide; Circular Dichroism; Glipizide; Glyburide; Humans; In Vitro Techniques; Optical Rotatory Dispersion; Protein Binding; Serum Albumin; Serum Albumin, Bovine; Sulfonylurea Compounds; Tolbutamide

1976
Displacement of tolbutamide, glibencalmide and chlorpropamide from serum albumin by anionic drugs.
    Biochemical pharmacology, 1976, May-15, Volume: 25, Issue:10

    Topics: Acetaminophen; Animals; Cattle; Chlorpropamide; Dialysis; Glyburide; Humans; Phenylbutazone; Protein Binding; Salicylates; Serum Albumin; Serum Albumin, Bovine; Sulfaphenazole; Tolbutamide; Warfarin

1976
[Experimental study of glipizide. A comparison with other hypoglycemic sulfonamides (author's transl)].
    Diabete & metabolisme, 1975, Volume: 1

    Topics: Administration, Oral; Ammonia; Animals; Dogs; Dose-Response Relationship, Drug; Female; Glipizide; Glyburide; Injections, Intravenous; Insulin; Islets of Langerhans; Mice; Purine-Pyrimidine Metabolism, Inborn Errors; Rats; Seizures; Sulfonylurea Compounds; Time Factors; Tolbutamide

1975
[Non-saturable cooperative binding of tolbutamide to rat endocrine pancreas. Criteria of specificity].
    Comptes rendus hebdomadaires des seances de l'Academie des sciences. Serie D: Sciences naturelles, 1976, Jul-19, Volume: 283, Issue:3

    Topics: Animals; Diazoxide; Drug Interactions; Glipizide; Glucose; Glyburide; Islets of Langerhans; Kinetics; Rats; Tolbutamide

1976
[The insulin-secreting and proliferative activity of established islet cells in the presence of sulfonylurea].
    Biulleten' eksperimental'noi biologii i meditsiny, 1992, Volume: 114, Issue:10

    Topics: Animals; Cell Division; Cell Line; Cell Line, Transformed; Cells, Cultured; Cricetinae; Gliclazide; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Rats; Sulfonylurea Compounds; Time Factors; Tolbutamide

1992
Therapeutical concentrations of tolbutamide, glibenclamide, gliclazide and gliquidone at different glucose levels: in vitro effects on pancreatic A- and B-cell function.
    Diabetes research and clinical practice, 1992, Volume: 18, Issue:3

    Topics: Animals; Blood Glucose; Dose-Response Relationship, Drug; Gliclazide; Glucagon; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Perfusion; Rats; Rats, Sprague-Dawley; Sulfonylurea Compounds; Time Factors; Tolbutamide

1992
Influence of KATP channel modulation on net potassium efflux from ischaemic mammalian cardiac tissue.
    Cardiovascular research, 1992, Volume: 26, Issue:11

    Topics: Action Potentials; Animals; Barium; Benzopyrans; Cromakalim; Glyburide; Guinea Pigs; Hydrogen-Ion Concentration; Muscles; Myocardial Ischemia; Oxygen; Papillary Muscles; Potassium; Potassium Channels; Pyrroles; Tolbutamide; Vasodilator Agents

1992
Pharmacological evidence for a role of ATP-dependent potassium channels in myocardial stunning.
    Circulation, 1992, Volume: 86, Issue:1

    Topics: Adenosine Triphosphate; Animals; Blood Glucose; Dogs; Female; Glyburide; Hemodynamics; Male; Myocardial Contraction; Myocardial Reperfusion Injury; Myocardium; Picolines; Potassium Channels; Pyrans; Risk Factors; Tolbutamide

1992
Effect of tolbutamide and glyburide on pyruvate kinase flux in isolated rat hepatocytes.
    Life sciences, 1992, Volume: 50, Issue:23

    Topics: Animals; Bicarbonates; Carbon Radioisotopes; Glucose; Glyburide; Lactates; Liver; Male; Pyruvate Kinase; Rats; Rats, Inbred Strains; Sensitivity and Specificity; Sodium; Sodium Bicarbonate; Sulfonylurea Compounds; Time Factors; Tolbutamide

1992
Opposing actions of tolbutamide and glibenclamide on hypoxic pulmonary vasoconstriction.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 102, Issue:3

    Topics: Animals; Benzopyrans; Cromakalim; Diazoxide; Glyburide; Hypoxia; In Vitro Techniques; Lung; Male; Potassium Channels; Pyrroles; Rats; Tolbutamide; Vasoconstriction

1992
Glyburide and tolbutamide induce desensitization of insulin release in rat pancreatic islets by different mechanisms.
    Endocrinology, 1992, Volume: 131, Issue:4

    Topics: Animals; Calcium; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Wistar; Rubidium; Tolbutamide

1992
Lack of evidence for coupling of the dopamine D2 receptor to an adenosine triphosphate-sensitive potassium (ATP-K+) channel in dopaminergic neurones of the rat substantia nigra.
    Neuroscience letters, 1992, Jul-20, Volume: 141, Issue:2

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Dopamine; Electrophysiology; Glyburide; Male; Neurons; Potassium Channels; Pyrroles; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Dopamine D2; Substantia Nigra; Tolbutamide

1992
High external Ca2+ levels trigger membrane potential oscillations in mouse pancreatic beta-cells during blockade of K(ATP) channels.
    Biochemical and biophysical research communications, 1992, Sep-16, Volume: 187, Issue:2

    Topics: Adenosine Triphosphate; Animals; Calcium; Cell Membrane; Drug Synergism; Fluorescent Dyes; Fura-2; Glyburide; Ionomycin; Islets of Langerhans; Membrane Potentials; Mice; Potassium Channels; Tolbutamide

1992
Inhibition of ATP-sensitive K+ channels in cardiac muscle by the sulphonylurea drug glibenclamide.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:2

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Dihydropyridines; Glyburide; Guinea Pigs; Heart Ventricles; Muscle, Smooth, Vascular; Potassium Channels; Tolbutamide; Vasodilator Agents

1992
Role of ATP-sensitive K+ channels during anoxia: major differences between rat (newborn and adult) and turtle neurons.
    The Journal of physiology, 1992, Volume: 448

    Topics: Animals; Brain Stem; Dose-Response Relationship, Drug; Glyburide; Homeostasis; Membrane Potentials; Oxygen; Potassium; Potassium Channels; Rats; Tolbutamide; Turtles

1992
Effects of pH upon the inhibition by sulphonylurea drugs of ATP-sensitive K+ channels in cardiac muscle.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Dihydropyridines; Drug Interactions; Glyburide; Guinea Pigs; Hydrogen-Ion Concentration; Kinetics; Membrane Potentials; Muscle, Smooth, Vascular; Potassium Channels; Tolbutamide; Vasodilator Agents

1992
ATP/ADP binding sites are present in the sulfonylurea binding protein associated with brain ATP-sensitive K+ channels.
    Biochemistry, 1992, Jul-14, Volume: 31, Issue:27

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Binding Sites; Binding, Competitive; Brain; Glyburide; Kinetics; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors; Swine; Tolbutamide

1992
Specificity of photolabeling of beta-cell membrane proteins with an 125I-labeled glyburide analog.
    The Journal of biological chemistry, 1992, Jul-25, Volume: 267, Issue:21

    Topics: Animals; Binding Sites; Cell Membrane; Chromatography, Gel; Cricetinae; Electrophoresis, Polyacrylamide Gel; Glipizide; Glyburide; Iodine Radioisotopes; Islets of Langerhans; Membrane Proteins; Photochemistry; Substrate Specificity; Tolbutamide; Tumor Cells, Cultured

1992
Adverse effect on diabetes control of concomitant glibenclamide and tolbutamide.
    Lancet (London, England), 1991, Mar-09, Volume: 337, Issue:8741

    Topics: Diabetes Mellitus, Type 2; Drug Interactions; Drug Therapy, Combination; Glyburide; Humans; Male; Middle Aged; Patient Acceptance of Health Care; Tolbutamide

1991
Sulfonylurea enhances insulin-induced acetyl coenzyme A carboxylase activity in rat adipocytes.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1991, Volume: 23, Issue:5

    Topics: Acetyl-CoA Carboxylase; Adipose Tissue; Animals; Enzyme Induction; Epinephrine; Glucagon; Glyburide; In Vitro Techniques; Insulin; Male; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide

1991
Co-secretion of amylin and insulin from cultured islet beta-cells: modulation by nutrient secretagogues, islet hormones and hypoglycemic agents.
    Biochemical and biophysical research communications, 1991, Aug-30, Volume: 179, Issue:1

    Topics: Amyloid; Animals; Arginine; Cell Line; Cricetinae; Glucagon; Glucose; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islet Amyloid Polypeptide; Islets of Langerhans; Kinetics; Metformin; Somatostatin; Tolbutamide

1991
Ion channels of glucose-responsive and -unresponsive beta-cells.
    Diabetes, 1991, Volume: 40, Issue:8

    Topics: Animals; Cobalt; Electrophysiology; Glucose; Glyburide; Hemolytic Plaque Technique; In Vitro Techniques; Ion Channels; Islets of Langerhans; Male; Membrane Potentials; Potassium Channels; Potassium Chloride; Rats; Rats, Inbred Strains; Sodium Channels; Tolbutamide

1991
Effects of glibenclamide and tolbutamide on ischemia- and ouabain-induced arrhythmias and membrane potentials of ventricular myocardium from rat and guinea pig.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1991, Volume: 12, Issue:5

    Topics: Animals; Arrhythmias, Cardiac; Dose-Response Relationship, Drug; Female; Glyburide; Guinea Pigs; Hypoxia; Ischemia; Male; Membrane Potentials; Ouabain; Rats; Species Specificity; Tolbutamide; Ventricular Fibrillation

1991
Activation by adrenaline of a low-conductance G protein-dependent K+ channel in mouse pancreatic B cells.
    Nature, 1991, Jan-03, Volume: 349, Issue:6304

    Topics: Animals; Clonidine; Epinephrine; Glucose; Glyburide; Islets of Langerhans; Membrane Potentials; Mice; Potassium Channels; Tolbutamide; Yohimbine

1991
Sulfonylureas activate glucose transport and protein kinase C in rat adipocytes.
    Metabolism: clinical and experimental, 1991, Volume: 40, Issue:2

    Topics: Adipose Tissue; Animals; Biological Transport; Deoxyglucose; Glucose; Glyburide; Insulin; Male; Protein Kinase C; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tetradecanoylphorbol Acetate; Time Factors; Tolbutamide

1991
Inhibitory effect of cyclosporine A on the activity of oral hypoglycemic agents in rats.
    The Journal of pharmacology and experimental therapeutics, 1991, Jul-01, Volume: 258, Issue:1

    Topics: Administration, Oral; Animals; Blood Glucose; Cyclosporins; Dose-Response Relationship, Drug; Drug Interactions; Glyburide; Insulin; Male; Rats; Tissue Distribution; Tolbutamide

1991
Possibility of ideal blood glucose control by a new oral hypoglycemic agent, N-[(trans-4-isopropylcyclohexyl)-carbonyl]-D-phenylalanine (A-4166), and its stimulatory effect on insulin secretion in animals.
    Diabetes research and clinical practice, 1991, Volume: 12, Issue:1

    Topics: Animals; Blood Glucose; Cyclohexanes; Diabetes Mellitus, Experimental; Dogs; Glucose Tolerance Test; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Male; Mice; Mice, Mutant Strains; Nateglinide; Phenylalanine; Rats; Rats, Inbred Strains; Tolbutamide

1991
Chronic exposure to glibenclamide impairs insulin secretion in isolated rat pancreatic islets.
    Journal of endocrinological investigation, 1991, Volume: 14, Issue:4

    Topics: Animals; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Time Factors; Tolbutamide

1991
Characterization of the solubilized glibenclamide receptor in a hamster pancreatic beta-cell line, HIT T15.
    The Biochemical journal, 1991, Aug-01, Volume: 277 ( Pt 3)

    Topics: Affinity Labels; Animals; Benzamides; Cell Line; Cricetinae; Glyburide; Islets of Langerhans; Photochemistry; Potassium Channels; Protein Binding; Receptors, Drug; Solubility; Tolbutamide

1991
Sulfonylureas, ATP-sensitive K+ channels, and cellular K+ loss during hypoxia, ischemia, and metabolic inhibition in mammalian ventricle.
    Circulation research, 1991, Volume: 69, Issue:3

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Binding Sites; Coronary Disease; Female; Glyburide; Guinea Pigs; Heart; In Vitro Techniques; Male; Myocardium; Oxygen Consumption; Potassium; Potassium Channels; Rabbits; Sulfonylurea Compounds; Tolbutamide

1991
Effects of ATP-sensitive K+ channel blockers on the action potential shortening in hypoxic and ischaemic myocardium.
    British journal of pharmacology, 1991, Volume: 103, Issue:1

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Coronary Circulation; Coronary Disease; Dogs; Female; Glyburide; Guanidines; Guinea Pigs; Hypoxia; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Perfusion; Pinacidil; Potassium Channels; Sulfonylurea Compounds; Tolbutamide

1991
Hyperpolarization of denervated skeletal muscle by lemakalim and its antagonism by glybenclamide and tolbutamide.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: Animals; Benzopyrans; Calcium Channel Blockers; Cesium; Cromakalim; Female; Glyburide; Male; Membrane Potentials; Mice; Muscle Denervation; Muscles; Pyrroles; Tolbutamide

1991
B cell adrenoceptors and sulphonylurea-induced insulin release in mouse islets.
    Diabetologia, 1990, Volume: 33, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Female; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Metoprolol; Mice; Mice, Inbred Strains; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tolbutamide

1990
Divergent cardiac effects of the first and second generation hypoglycemic sulfonylurea compounds.
    Diabetes research and clinical practice, 1990, Volume: 8, Issue:2

    Topics: Animals; Arrhythmias, Cardiac; Blood Glucose; Carbutamide; Dose-Response Relationship, Drug; Electrocardiography; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Male; Myocardial Infarction; Potassium; Rats; Rats, Inbred Strains; Reference Values; Structure-Activity Relationship; Tolbutamide

1990
The potentiating effect of the simultaneous administration of tolbutamide, glibenclamide, and gliclazide on the development of alloxan-induced diabetes in rats.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1990, Volume: 22, Issue:1

    Topics: Animals; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Drug Synergism; Gliclazide; Glucose Tolerance Test; Glyburide; Insulin; Male; Pancreas; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide

1990
Action of cromakalim on potassium membrane conductance in isolated heart myocytes of frog.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Adenosine Triphosphate; Animals; Barium; Benzopyrans; Cesium; Cromakalim; Glyburide; In Vitro Techniques; Membranes; Myocardium; Potassium Channels; Pyrroles; Rana esculenta; Sulfonylurea Compounds; Tolbutamide

1990
A screening test for detecting sulfonylureas in plasma.
    Therapeutic drug monitoring, 1990, Volume: 12, Issue:4

    Topics: Aged; Aged, 80 and over; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1990
Sulfonylurea-stimulated glucose transport association with diacylglycerollike activation of protein kinase C in BC3H1 myocytes.
    Diabetes, 1990, Volume: 39, Issue:11

    Topics: Alkaloids; Animals; Biological Transport; Cell Line; Cells, Cultured; Deoxyglucose; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Glucose; Glyburide; Insulin; Muscles; Protein Kinase C; Staurosporine; Sulfonylurea Compounds; Tetradecanoylphorbol Acetate; Tolbutamide

1990
Hypoglycemic sulfonylureas antagonize the effects of cromakalim and pinacidil on 86Rb fluxes and contractile activity in the rat aorta.
    Pharmacology, 1990, Volume: 41, Issue:1

    Topics: Animals; Aorta, Thoracic; Benzopyrans; Cromakalim; Glyburide; Guanidines; Hypoglycemic Agents; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Parasympatholytics; Pinacidil; Potassium Channels; Pyrroles; Rats; Rats, Inbred Strains; Rubidium Radioisotopes; Sulfonylurea Compounds; Tetraethylammonium Compounds; Tolbutamide; Vasodilator Agents

1990
Adenosine triphosphate-sensitive potassium channels in anoxia.
    Stroke, 1990, Volume: 21, Issue:11 Suppl

    Topics: Adenosine Triphosphate; Animals; Diazoxide; Electrophysiology; Glyburide; Hippocampus; Hypoxia; Neurons; Potassium Channels; Tolbutamide

1990
Effect of sulphonylurea therapy on insulin sensitivity in non insulin dependent diabetics.
    The Journal of the Association of Physicians of India, 1990, Volume: 38, Issue:7

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Insulin Resistance; Middle Aged; Sulfonylurea Compounds; Time Factors; Tolbutamide

1990
Tolbutamide excites rat glucoreceptive ventromedial hypothalamic neurones by indirect inhibition of ATP-K+ channels.
    British journal of pharmacology, 1990, Volume: 101, Issue:3

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Binding Sites; Cerebral Cortex; Glyburide; In Vitro Techniques; Male; Potassium Channels; Rats; Rats, Inbred Strains; Tolbutamide; Ventromedial Hypothalamic Nucleus

1990
Mechanism of potassium efflux and action potential shortening during ischaemia in isolated mammalian cardiac muscle.
    The Journal of physiology, 1990, Volume: 431

    Topics: Action Potentials; Animals; Bumetanide; Chlorides; Coronary Disease; Coumaric Acids; Deoxyglucose; Female; Glyburide; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Membrane Potentials; Myocardial Contraction; Papillary Muscles; Potassium; Purkinje Fibers; Sheep; Time Factors; Tolbutamide

1990
Glibenclamide is a competitive antagonist of the thromboxane A2 receptor in dog coronary artery in vitro.
    British journal of pharmacology, 1990, Volume: 100, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Coronary Vessels; Dogs; Endothelins; Endothelium, Vascular; Female; Glyburide; In Vitro Techniques; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Peptides; Potassium Chloride; Prostaglandin Endoperoxides, Synthetic; Receptors, Prostaglandin; Receptors, Thromboxane; Thromboxane A2; Tolbutamide

1990
The sulphonylurea receptor may be an ATP-sensitive potassium channel.
    Lancet (London, England), 1985, Aug-31, Volume: 2, Issue:8453

    Topics: Adenosine Triphosphate; Animals; Cell Line; Cell Membrane; Glyburide; Insulin; Ion Channels; Islets of Langerhans; Rats; Sulfonylurea Compounds; Tolbutamide

1985
Direct measurements of increased free cytoplasmic Ca2+ in mouse pancreatic beta-cells following stimulation by hypoglycemic sulfonylureas.
    FEBS letters, 1985, Oct-07, Volume: 190, Issue:1

    Topics: Aminoquinolines; Animals; Calcium; Cytoplasm; Female; Fluorescent Dyes; Glyburide; Hypoglycemic Agents; Ion Channels; Islets of Langerhans; Male; Mice; Mice, Obese; Potassium; Sulfonylurea Compounds; Tolbutamide

1985
Opposite effects of tolbutamide and diazoxide on the ATP-dependent K+ channel in mouse pancreatic beta-cells.
    Pflugers Archiv : European journal of physiology, 1986, Volume: 407, Issue:5

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Cells, Cultured; Diazoxide; Glucose; Glyburide; Ion Channels; Islets of Langerhans; Mice; Potassium; Tolbutamide

1986
Electrophysiological measurements show marked differences in the properties of the pancreatic beta-cell K-channels from albino mice and a strain of ob/ob (obese) mice.
    Advances in experimental medicine and biology, 1986, Volume: 211

    Topics: Animals; Glucose; Glyburide; In Vitro Techniques; Ion Channels; Islets of Langerhans; Membrane Potentials; Mice; Mice, Obese; Potassium; Quinine; Species Specificity; Tolbutamide

1986
Effect of channel blockers on potassium efflux from metabolically exhausted frog skeletal muscle.
    The Journal of physiology, 1987, Volume: 383

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Apamin; Barium; Cell Membrane Permeability; Decamethonium Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Glyburide; In Vitro Techniques; Ion Channels; Muscles; Potassium; Quinine; Rana temporaria; Rubidium; Scorpion Venoms; Tetraethylammonium Compounds; Tolbutamide

1987
Concentration-dependent effects of tolbutamide, meglitinide, glipizide, glibenclamide and diazoxide on ATP-regulated K+ currents in pancreatic B-cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:2

    Topics: Adenosine Triphosphate; Animals; Benzamides; Diazoxide; Glipizide; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Ion Channels; Islets of Langerhans; Mice; Mice, Inbred Strains; Potassium; Sulfonylurea Compounds; Tolbutamide

1988
Inhibition by sulphonylureas of vasorelaxation induced by K+ channel activators in vitro.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: Animals; Antihypertensive Agents; Benzopyrans; Cromakalim; Drug Interactions; Glipizide; Glyburide; Guanidines; In Vitro Techniques; Male; Nifedipine; Norepinephrine; Pinacidil; Potassium Channels; Potassium Chloride; Pyrroles; Rabbits; Sulfonylurea Compounds; Tolbutamide; Vasodilator Agents

1989
The inotropic action of tolbutamide and glyburide.
    Clinical pharmacology and therapeutics, 1989, Volume: 45, Issue:6

    Topics: Administration, Oral; Adult; Blood Glucose; Blood Pressure; Dobutamine; Epinephrine; Glyburide; Humans; Male; Myocardial Contraction; Norepinephrine; Propranolol; Stroke Volume; Tolbutamide

1989
Glucose and sulfonylureas modify different phases of the membrane potential change during hypoxia in rat hippocampal slices.
    Brain research, 1989, Jun-12, Volume: 489, Issue:2

    Topics: Action Potentials; Animals; Cell Survival; Glucose; Glyburide; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide

1989
Hyperpolarizing vasodilators activate ATP-sensitive K+ channels in arterial smooth muscle.
    Science (New York, N.Y.), 1989, Jul-14, Volume: 245, Issue:4914

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Benzopyrans; Cerebral Arteries; Cromakalim; Diazoxide; Glyburide; Guanidines; Mesenteric Arteries; Muscle, Smooth, Vascular; Pinacidil; Potassium Channels; Pyrroles; Rabbits; Rats; Tolbutamide; Vasoactive Intestinal Peptide; Vasodilator Agents

1989
Effects of tolbutamide, glibenclamide and diazoxide upon action potentials recorded from rat ventricular muscle.
    Biochimica et biophysica acta, 1989, Aug-21, Volume: 984, Issue:1

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Diazoxide; Glyburide; Heart; In Vitro Techniques; Male; Potassium Channels; Rats; Rats, Inbred Strains; Tolbutamide

1989
Influence of ATP-sensitive potassium channel modulators on ischemia-induced fibrillation in isolated rat hearts.
    Journal of molecular and cellular cardiology, 1989, Volume: 21, Issue:8

    Topics: Adenosine Triphosphate; Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Benzopyrans; Coronary Circulation; Coronary Disease; Cromakalim; Glyburide; Guanidines; Heart; Heart Rate; In Vitro Techniques; Male; Perfusion; Pinacidil; Potassium Channels; Pyrroles; Rats; Rats, Inbred Strains; Tolbutamide; Vascular Resistance

1989
Effects of sulfonamides on a metabolite-regulated ATPi-sensitive K+ channel in rat pancreatic B-cells.
    The American journal of physiology, 1989, Volume: 257, Issue:6 Pt 1

    Topics: Adenosine Triphosphate; Animals; Cells, Cultured; Diazoxide; Electric Conductivity; Glucose; Glyburide; Islets of Langerhans; Kinetics; Mathematics; Membrane Potentials; Models, Biological; Potassium Channels; Rats; Tolbutamide

1989
ATP-sensitive K-channels in HIT T15 beta-cells studied by patch-clamp methods, 86Rb efflux and glibenclamide binding.
    Pflugers Archiv : European journal of physiology, 1989, Volume: 415, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Binding Sites; Cell Line, Transformed; Cell Membrane Permeability; Cricetinae; Electric Conductivity; Glyburide; Islets of Langerhans; Potassium Channels; Rubidium Radioisotopes; Tolbutamide

1989
[Effect of antidiabetics on post-exercise alaninemia in patients with non-insulin-dependent diabetes mellitus (type 2)].
    Polskie Archiwum Medycyny Wewnetrznej, 1989, Volume: 81, Issue:4

    Topics: Adult; Alanine; Diabetes Mellitus, Type 2; Drug Interactions; Drug Therapy, Combination; Exercise; Exercise Test; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Phenformin; Tolbutamide

1989
Do hypoglycemic sulfonylureas inhibit Na+,K+-ATPase activity in pancreatic islets?
    The American journal of physiology, 1985, Volume: 248, Issue:5 Pt 1

    Topics: Animals; Calcimycin; Calcium; Cell Membrane Permeability; Drug Synergism; Glucose; Glyburide; Insulin; Ion Channels; Islets of Langerhans; Ouabain; Potassium; Quinine; Rats; Rubidium; Sodium-Potassium-Exchanging ATPase; Tolbutamide

1985
Effect of tolbutamide and glyburide on cAMP-dependent protein kinase activity in rat liver cytosol.
    Diabetes, 1988, Volume: 37, Issue:7

    Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Cyclic AMP; Cytosol; Dose-Response Relationship, Drug; Glyburide; Histones; Kinetics; Liver; Male; Protein Kinases; Rats; Rats, Inbred Strains; Tolbutamide

1988
Interaction of sulfonylureas with pancreatic beta-cells. A study with glyburide.
    Diabetes, 1988, Volume: 37, Issue:8

    Topics: Animals; Cyclic AMP; Glucagon; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Male; Oxidation-Reduction; Rats; Rats, Inbred Strains; Tolbutamide

1988
Effects of sulphonylureas on spontaneous motility and induced contractions in rat isolated uterus.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:10

    Topics: Animals; Calcium; Female; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide; Uterine Contraction; Vanadates; Vanadium

1986
Differential activities of tolbutamide, tolazamide, and glyburide in vitro on rabbit myocardial membrane Ca2+-transporting ATPase activity.
    Diabetes, 1986, Volume: 35, Issue:9

    Topics: Animals; Calcium; Calcium-Transporting ATPases; Calmodulin; Cell Membrane; Female; Glyburide; Heart; In Vitro Techniques; Male; Milrinone; Myocardium; Pyridones; Rabbits; Thyroxine; Tolazamide; Tolbutamide

1986
Increased cytosolic calcium. A signal for sulfonylurea-stimulated insulin release from beta cells.
    The Journal of biological chemistry, 1987, Feb-25, Volume: 262, Issue:6

    Topics: Animals; Calcium; Cells, Cultured; Colforsin; Cricetinae; Cyclic AMP; Glyburide; Insulin; Islets of Langerhans; Tolbutamide; Verapamil

1987
Relaxant effects of sulfonylureas on induced contractions of rat uterine smooth muscle: role of intracellular calcium.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 279, Issue:2

    Topics: Acetylcholine; Animals; Calcium; Female; Glyburide; In Vitro Techniques; Muscle, Smooth; Oxytocin; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide; Uterine Contraction

1986
Potentiating effect of glibenclamide on the occurrence of alloxan diabetes in rats.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1986, Volume: 18, Issue:4

    Topics: Alloxan; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Drug Synergism; Glyburide; Male; Rats; Rats, Inbred Strains; Tolbutamide

1986
Effect of sulfonylureas on hepatic fatty acid oxidation.
    The American journal of physiology, 1986, Volume: 251, Issue:2 Pt 1

    Topics: Animals; Carnitine O-Palmitoyltransferase; Fatty Acids; Glyburide; Ketone Bodies; Liver; Male; Mitochondria, Liver; Oleic Acid; Oleic Acids; Oxidation-Reduction; Perfusion; Rats; Rats, Inbred Strains; Tolbutamide

1986
[Importance of calcium in the interaction between prostaglandins E and sulfonylureas in utero].
    Archivos de farmacologia y toxicologia, 1986, Volume: 12, Issue:1

    Topics: Animals; Calcium; Dose-Response Relationship, Drug; Drug Interactions; Female; Glyburide; Muscle Relaxation; Oxytocin; Potassium Chloride; Pregnancy; Prostaglandins E; Rats; Rats, Inbred Strains; Tolbutamide; Uterine Contraction

1986
Evidence for direct effect of tolbutamide on hepatic glycogenolysis induced by Ca2+-dependent hormones.
    Biochemical pharmacology, 1986, Sep-15, Volume: 35, Issue:18

    Topics: Angiotensin II; Animals; Calcium; Gluconeogenesis; Glyburide; Hormones; Liver Glycogen; Male; Phenylephrine; Rats; Rats, Inbred Strains; Tolbutamide; Trifluoperazine; Vasopressins

1986
Mutagenic evaluation of tolbutamide and glybenclamide on the bone marrow cells of mice.
    Toxicology letters, 1986, Volume: 34, Issue:2-3

    Topics: Animals; Bone Marrow; Dose-Response Relationship, Drug; Erythrocytes; Female; Glyburide; Male; Mice; Mutagenicity Tests; Mutagens; Tolbutamide

1986
The hypoglycemic sulfonylureas glyburide and tolbutamide inhibit fatty acid oxidation by inhibiting carnitine palmitoyltransferase.
    The Journal of biological chemistry, 1987, Apr-15, Volume: 262, Issue:11

    Topics: Acyltransferases; Animals; Carnitine O-Palmitoyltransferase; Diabetes Mellitus, Experimental; Fatty Acids; Glyburide; Male; Malonyl Coenzyme A; Mitochondria, Liver; Muscles; Myocardium; Rats; Rats, Inbred Strains; Tolbutamide

1987
Regulation of muscle fructose 2, 6-bisphosphate levels by sulfonylureas.
    Endocrinologia japonica, 1986, Volume: 33, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Fructosediphosphates; Glyburide; Hexosediphosphates; Mice; Muscles; Perfusion; Sulfonylurea Compounds; Tolbutamide

1986
Stimulation of biliary glutathione secretion by sulfonylureas.
    Molecular pharmacology, 1987, Volume: 31, Issue:6

    Topics: Animals; Bile; Biotransformation; Gallbladder; Glutathione; Glutathione Disulfide; Glyburide; Kinetics; Male; Perfusion; Rats; Rats, Inbred Strains; Tolbutamide

1987
Direct effects of sulfonylurea agents on glucose transport in the BC3H-1 myocyte.
    Diabetes, 1987, Volume: 36, Issue:11

    Topics: Animals; Cell Line; Deoxy Sugars; Deoxyglucose; Glipizide; Glyburide; Hypoglycemic Agents; Insulin; Kinetics; Mice; Muscles; Tolbutamide

1987
Effect of PGE2 on sulfonylurea induced insulin release.
    Journal de physiologie, 1987, Volume: 82, Issue:1

    Topics: Animals; Blood Glucose; Dinoprostone; Female; Glyburide; Insulin; Insulin Secretion; Kinetics; Prostaglandins E; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide

1987
Characterization of the sulfonylurea receptor on beta cell membranes.
    The Journal of biological chemistry, 1988, Feb-25, Volume: 263, Issue:6

    Topics: Animals; ATP-Binding Cassette Transporters; Cell Line; Cell Membrane; Cricetinae; Glipizide; Glyburide; Insulin; Islets of Langerhans; Kinetics; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Temperature; Tolazamide; Tolbutamide

1988
Effects of hypoglycemic sulfonylureas on catecholamine secretion and calcium uptake in cultured bovine adrenal chromaffin cells.
    Biochemical pharmacology, 1988, Mar-01, Volume: 37, Issue:5

    Topics: Adrenal Medulla; Animals; Calcimycin; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Glyburide; Hypoglycemic Agents; Sulfonylurea Compounds; Tolbutamide

1988
Sulfonylureas inhibit metabolic flux through rat liver pyruvate carboxylase reaction.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: Acetyl Coenzyme A; Adenine Nucleotides; Animals; Coenzyme A; Glyburide; Kinetics; Male; Mitochondria, Liver; Oxygen Consumption; Pyruvate Carboxylase; Rats; Rats, Inbred Strains; Tolbutamide

1988
Effects of sulphonylureas and diazoxide on insulin secretion and nucleotide-sensitive channels in an insulin-secreting cell line.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Adenosine Triphosphate; Animals; Cell Line; Diazoxide; Electrophysiology; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Leucine; Nucleotides; Potassium Channels; Rats; Sulfonylurea Compounds; Tolbutamide

1988
[Correlation between the levels of CA19-9 and fasting plasma glucose in a case of diabetes mellitus].
    Nihon Naika Gakkai zasshi. The Journal of the Japanese Society of Internal Medicine, 1988, Volume: 77, Issue:9

    Topics: Aged; Antigens, Tumor-Associated, Carbohydrate; Blood Glucose; Diabetes Mellitus; Female; Glyburide; Humans; Tolbutamide

1988
Suppression by 2-ketoisocaproate of the insulinotropic action of hypoglycemic sulfonylureas.
    Research communications in chemical pathology and pharmacology, 1985, Volume: 47, Issue:2

    Topics: Animals; Calcium; Gliclazide; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Insulin Secretion; Ionophores; Keto Acids; Oxidation-Reduction; Rats; Sulfonylurea Compounds; Tolbutamide

1985
Stimulation of insulin secretion from isolated rat islets by SaRI 59-801.
    Diabetes, 1985, Volume: 34, Issue:6

    Topics: Administration, Oral; Animals; Dose-Response Relationship, Drug; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Isoxazoles; Male; Mannoheptulose; Oxazoles; Proinsulin; Rats; Rats, Inbred Strains; Tolbutamide

1985
Determination of glibenclamide, chlorpropamide and tolbutamide in plasma by high-performance liquid chromatography with ultraviolet detection.
    Journal of chromatography, 1985, Apr-12, Volume: 339, Issue:1

    Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Diabetes Mellitus; Dinitrofluorobenzene; Gas Chromatography-Mass Spectrometry; Glyburide; Humans; Spectrophotometry, Ultraviolet; Tolbutamide

1985
Effects of various hypoglycaemic sulphonylureas on the cardiotoxicity of glycosides.
    European journal of clinical pharmacology, 1985, Volume: 28, Issue:4

    Topics: Aged; Animals; Carbutamide; Cardiac Glycosides; Dose-Response Relationship, Drug; Female; Glyburide; Heart; Humans; Hypoglycemic Agents; Male; Middle Aged; Rabbits; Tolbutamide

1985
Sulfonylurea stimulates liver fructose-2,6-bisphosphate formation in proportion to its hypoglycemic action.
    Diabetes research and clinical practice, 1985, Volume: 1, Issue:1

    Topics: Acetohexamide; Animals; Buformin; Chlorpropamide; Fructosediphosphates; Gliclazide; Gluconeogenesis; Glyburide; Glycolysis; Hexosediphosphates; In Vitro Techniques; Liver; Male; Rats; Rats, Inbred Strains; Stimulation, Chemical; Sulfamethoxazole; Sulfonylurea Compounds; Tolbutamide

1985
Antidiuretic action of chlorpropamide.
    Lancet (London, England), 1973, Volume: 2, Issue:7822

    Topics: Chlorpropamide; Diuresis; Female; Glyburide; Humans; Male; Tolbutamide

1973
[Thyroid gland function of patients with diabetes in long-term use of glibornuride].
    Arzneimittel-Forschung, 1972, Volume: 22

    Topics: Camphanes; Carbutamide; Diabetes Mellitus; Female; Glyburide; Goiter; Humans; Hypoglycemic Agents; Male; Middle Aged; Sulfonylurea Compounds; Thyroid Function Tests; Thyroid Gland; Tolbutamide

1972
The binding of sulphonylureas to serum albumin.
    The Journal of pharmacy and pharmacology, 1974, Volume: 26, Issue:5

    Topics: Animals; Carbon Radioisotopes; Cattle; Chlorpropamide; Glyburide; Humans; Hydrogen-Ion Concentration; Protein Binding; Serum Albumin; Serum Albumin, Bovine; Sulfonylurea Compounds; Tolazamide; Tolbutamide

1974
Different amounts of insulin secretion following an equal total decrease of blood glucose as an indication of possible extrapancreatic activities of different sulfonylurea drugs.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1973, Volume: 5, Issue:1

    Topics: Animals; Antigens; Autoanalysis; Blood Glucose; Camphanes; Computers; Diabetes Mellitus; Dogs; Fasting; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Pancreas; Sulfonylurea Compounds; Time Factors; Tolbutamide

1973
The pancreatic -cell recognition of insulin secretagogues. IV. Islet uptake of sulfonylureas.
    Diabetologia, 1973, Volume: 9, Issue:3

    Topics: Animals; Antimycin A; Carbon Isotopes; Chlorpromazine; Diazoxide; Glucose; Glyburide; In Vitro Techniques; Islets of Langerhans; Leucine; Male; Mice; Serum Albumin; Sulfur Isotopes; Tolbutamide

1973
[Insulin secretion after oral and intravenous administration of various 1st and 2d generation sulfonylurea derivatives in equipotential dosage].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1972, Volume: 78

    Topics: Administration, Oral; Glyburide; Humans; Injections, Intravenous; Insulin; Insulin Secretion; Sulfonylurea Compounds; Tolbutamide

1972
[Betacytotropic and antilipolytic effect of critical doses of tolbutamide and glibenclamide].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1972, Volume: 78

    Topics: Blood Glucose; Fatty Acids, Nonesterified; Glyburide; Humans; Insulin; Tolbutamide

1972
[Glibornuride, a new high-effective antidiabetic agent. Pharmacological and biochemical comparative studies in various animal species and animal experimental models].
    Arzneimittel-Forschung, 1972, Volume: 22

    Topics: Administration, Oral; Animals; Blood Glucose; Camphanes; Chemical Phenomena; Chemistry; Cholesterol; Disease Models, Animal; Dogs; Dose-Response Relationship, Drug; Female; Glyburide; Hyperglycemia; Hypoglycemia; Hypoglycemic Agents; Injections, Intravenous; Liver Glycogen; Mice; Microsomes, Liver; Oxidoreductases; Phospholipids; Rabbits; Rats; Sulfonylurea Compounds; Tolbutamide; Triglycerides

1972
[Extrapancreatic effects of sulfonylurea compounds. 3. Studies on the additional blood sugar decreasing and antilipolytic effect of tolbutamide, glibornuride, and glibenclamide on completely pancreatectomized dogs, chronically treated with insulin during
    Arzneimittel-Forschung, 1972, Volume: 22

    Topics: Animals; Blood Glucose; Camphanes; Dogs; Fatty Acids, Nonesterified; Glyburide; Glycerol; Hyperglycemia; Hypoglycemic Agents; Infusions, Parenteral; Insulin; Lipid Metabolism; Pancreatectomy; Sulfonylurea Compounds; Time Factors; Tolbutamide

1972
[Extrapancreatic effects of sulfonylurea compounds. IV. Increase of the effect of insulin due to tolbutamide, glibornuride, and glibenclamide in vitro].
    Arzneimittel-Forschung, 1972, Volume: 22

    Topics: Animals; Camphanes; Diaphragm; Dose-Response Relationship, Drug; Drug Interactions; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Mice; Sulfonylurea Compounds; Tolbutamide

1972
[Insulin liberation by blood sugar decreasing sulfonamides and by glucose in adult diabetic patients].
    Arzneimittel-Forschung, 1972, Volume: 22

    Topics: Adult; Azepines; Blood Glucose; Diabetes Mellitus; Drug Interactions; Fatty Acids, Nonesterified; Glucose; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Oxazoles; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide

1972
[Studies on dose-response relationship of various sulfonylurea derivatives of the old and the new generation with further hints to extrapancreatic mechanisms of decreasing blood sugar].
    Arzneimittel-Forschung, 1972, Volume: 22

    Topics: Administration, Oral; Azepines; Blood Glucose; Dose-Response Relationship, Drug; Glyburide; Humans; Hypoglycemic Agents; Injections, Intravenous; Insulin; Insulin Secretion; Oxazoles; Sulfonylurea Compounds; Tolbutamide

1972
Interrelationship of islet metabolism, adenosine triphosphate content and insulin release.
    The Biochemical journal, 1973, Volume: 132, Issue:2

    Topics: Adenosine Triphosphate; Animals; Carbon Isotopes; Glucose; Glyburide; Glyceraldehyde; Heptoses; Hexoses; Insulin; Insulin Secretion; Islets of Langerhans; Leucine; Male; Mice; Models, Biological; Nitriles; Oxidative Phosphorylation; Phenylhydrazines; Time Factors; Tolbutamide; Uncoupling Agents

1973
Observations of the mechanism of action of the sulfonylureas under clinical conditions.
    Metabolism: clinical and experimental, 1973, Volume: 22, Issue:9

    Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Fasting; Female; Glyburide; Humans; Hypoglycemia; Insulin; Male; Middle Aged; Time Factors; Tolbutamide

1973
The effect of glibenclamide on non-esterified fatty acid levels in the plasma of the severely alloxan diabetic rat.
    Experientia, 1973, Aug-15, Volume: 29, Issue:8

    Topics: Animals; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Experimental; Fatty Acids, Nonesterified; Glyburide; Insulin; Male; Rats; Tolbutamide

1973
[Secretion of insulin under the influence of sulfonylurea derivates (SH)].
    Wiener Zeitschrift fur innere Medizin und ihre Grenzgebiete, 1973, Volume: 54, Issue:2

    Topics: Animals; Blood Glucose; Diabetes Mellitus; Glucose Tolerance Test; Glyburide; Humans; Insulin; Insulin Secretion; Pancreas; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide

1973
Effects of feeding and fasting on the insulin secretory response to glucose and sulfonylureas in intact rats and isolated perfused rat pancreas.
    Diabetologia, 1973, Volume: 9, Issue:4

    Topics: Animal Nutritional Physiological Phenomena; Animals; Fasting; Glucose; Glucose Tolerance Test; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Male; Pancreas; Perfusion; Rats; Rats, Inbred Strains; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide

1973
[A comparison of intravenous tolbutamide and insulin administration during and after operation in patients with maturity-onset diabetes (author's transl)].
    Deutsche medizinische Wochenschrift (1946), 1974, Jan-25, Volume: 99, Issue:4

    Topics: Administration, Oral; Age Factors; Aged; Anesthesia, General; Blood Glucose; Carbohydrates; Carbutamide; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Diet Therapy; Fructose; Glyburide; Glycosuria; Humans; Injections, Intravenous; Insulin; Ketone Bodies; Plasma Substitutes; Postoperative Care; Preoperative Care; Surgical Procedures, Operative; Tolbutamide

1974
Insulinotrophic drugs. Effect on intestinal abosorption of sugar.
    Diabetes, 1974, Volume: 23, Issue:2

    Topics: Animals; Azepines; Biological Transport; Ethers; Galactose; Glyburide; Hypoglycemic Agents; Ileum; Intestinal Absorption; Intestine, Small; Oxazoles; Perfusion; Pyrimidines; Rats; Sulfonamides; Sulfonylurea Compounds; Tolbutamide

1974
Effect of sulfonylureas on the secretion of pancreatic immunoreactive glucagon and enteric glucagon-like immunoreactivity.
    Canadian journal of physiology and pharmacology, 1973, Volume: 51, Issue:12

    Topics: Animals; Antibody Formation; Antigens; Arginine; Glucagon; Glucose; Glyburide; In Vitro Techniques; Insulin Antibodies; Pancreas; Radioimmunoassay; Rats; Sulfonylurea Compounds; Theophylline; Tolbutamide

1973
[Pharmacological aspects of comparative studies on different blood sugar-lowering sulfonylureas].
    Arzneimittel-Forschung, 1973, Volume: 23, Issue:11

    Topics: Administration, Oral; Animals; Autoanalysis; Biopharmaceutics; Blood Glucose; Dogs; Dose-Response Relationship, Drug; Glyburide; Humans; Hypoglycemic Agents; Injections, Intravenous; Insulin; Sulfonylurea Compounds; Time Factors; Tolbutamide

1973
[Hypoglycemia caused by oral antidiabetic agents].
    Nederlands tijdschrift voor geneeskunde, 1973, Jul-07, Volume: 117, Issue:27

    Topics: Adult; Aged; Chlorpropamide; Delayed-Action Preparations; Diet; Female; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Kidney Diseases; Liver Diseases; Male; Middle Aged; Phenformin; Tolazamide; Tolbutamide

1973
Interactions of sulfonylureas with plasma proteins.
    Journal of pharmaceutical sciences, 1974, Volume: 63, Issue:4

    Topics: Acetohexamide; Acridines; Aniline Compounds; Animals; Binding Sites; Blood Proteins; Cattle; Chlorpropamide; Cyclohexanes; Glyburide; Humans; Hypoglycemic Agents; Naphthalenesulfonates; Protein Binding; Pyrazines; Serum Albumin; Serum Albumin, Bovine; Spectrometry, Fluorescence; Sulfonylurea Compounds; Tolbutamide; Warfarin

1974
[Insulin secretion following combined administration of glucose and different sulfonylurea compounds in equipotential doses in metabolically healthy persons].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1973, Volume: 79

    Topics: Camphanes; Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Sulfonylurea Compounds; Tolbutamide

1973
Effects of hypoglycemic sulfonamides on glucagon and insulin secretion in ducks and dogs.
    Diabetes, 1974, Volume: 23, Issue:5

    Topics: Animals; Antigens; Arteries; Blood Glucose; Carboxylic Acids; Dogs; Ducks; Ethers; Femoral Artery; Glucagon; Glyburide; Hypoglycemic Agents; Injections, Intravenous; Insulin; Insulin Secretion; Pancreas; Pyrimidines; Species Specificity; Sulfonamides; Tolbutamide; Veins

1974
An inhibitory effect of tolbutamide and glibenclamide (glyburide) on the pancreatic islets of normal animals.
    Diabetologia, 1974, Volume: 10, Issue:1

    Topics: Animals; Blood Glucose; Carbon Radioisotopes; Female; Glucose; Glyburide; Insulin; Islets of Langerhans; Leucine; Tolbutamide

1974
In vitro secretion of insulin after glucose, sulphonylureas, adrenergic and cholinergic substances studied by isolated perfused rat pancreas.
    Endocrinologia experimentalis, 1974, Volume: 8, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Diazoxide; Epinephrine; Glucagon; Glucose; Glyburide; Heptoses; In Vitro Techniques; Insulin; Insulin Secretion; Isoproterenol; Ketoses; Norepinephrine; Pancreas; Parasympathomimetics; Perfusion; Phenoxybenzamine; Practolol; Propranolol; Sulfonylurea Compounds; Theophylline; Tolbutamide

1974
[Insulin secretion after administration of sulfonylurea in normal and diabetic subjects].
    Nihon Naibunpi Gakkai zasshi, 1974, Jan-20, Volume: 50, Issue:1

    Topics: Diabetes Mellitus; Fatty Acids, Nonesterified; Female; Glucose Tolerance Test; Glyburide; Growth Hormone; Humans; Insulin; Insulin Secretion; Male; Radioimmunoassay; Tolbutamide

1974
Clinical assessment of glybenclamide (daonil) in diabetes mellitus.
    The Journal of the Association of Physicians of India, 1973, Volume: 21, Issue:3

    Topics: Chlorpropamide; Diabetes Mellitus; Female; Glyburide; Humans; Male; Tolbutamide

1973
Uptake of glibornuride by microdissected pancreatic islets.
    Hormone research, 1974, Volume: 5, Issue:4

    Topics: Animals; Biological Transport; Camphanes; Carbon Radioisotopes; Female; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Obesity; Pancreas; Sucrose; Sulfonylurea Compounds; Time Factors; Tolbutamide; Tritium

1974
[Single intravenous glibenclamide-glucose loading as a prediction test (author's transl)].
    Deutsche medizinische Wochenschrift (1946), 1974, Jun-14, Volume: 99, Issue:24

    Topics: Adult; Age Factors; Aged; Diabetes Mellitus; Female; Glucose Tolerance Test; Glyburide; Humans; Insulin; Insulin Antibodies; Insulin Secretion; Long-Term Care; Male; Middle Aged; Tolbutamide

1974
[Pharmacologic study with glisoxepide and other blood sugar reducing sulfonamide derivatives in metabolically healthy subjects and diabetics].
    Arzneimittel-Forschung, 1974, Volume: 24, Issue:0

    Topics: Administration, Oral; Autoanalysis; Azepines; Blood Glucose; Depression, Chemical; Diabetes Mellitus; Dose-Response Relationship, Drug; Drug Evaluation; Glyburide; Humans; Hypoglycemic Agents; Injections, Intravenous; Insulin; Oxazoles; Sulfonamides; Sulfonylurea Compounds; Time Factors; Tolbutamide

1974
Potentiating effects of drugs on the binding of glibenclamide to pancreatic beta cells.
    Metabolism: clinical and experimental, 1974, Volume: 23, Issue:9

    Topics: Animals; Binding Sites; Drug Synergism; Female; Glyburide; Hyperglycemia; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Phenylbutazone; Serum Albumin; Sucrose; Sulfaphenazole; Sulfisomidine; Sulfisoxazole; Sulfonamides; Tolbutamide

1974
Effect of hypoglycemic sulfonylureas on hepatic fructose metabolism in the rat.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1974, Volume: 6, Issue:4

    Topics: Acetoacetates; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Chlorpropamide; Fasting; Flavoproteins; Fructose; Gluconeogenesis; Glyburide; Hydrogen-Ion Concentration; Hydroxybutyrates; Hypoglycemia; Ketone Bodies; Liver; Male; Mitochondria, Liver; Oxidation-Reduction; Perfusion; Rats; Spectrometry, Fluorescence; Sulfonylurea Compounds; Time Factors; Tolbutamide

1974
[The glibenclamide-phenformin combination in the therapy of diabetes mellitus].
    Minerva medica, 1974, Aug-29, Volume: 65, Issue:59

    Topics: Adult; Aged; Biguanides; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Drug Combinations; Drug Evaluation; Drug Synergism; Female; Glyburide; Humans; Insulin; Male; Middle Aged; Phenformin; Tolbutamide

1974
[Oral antidiabetic therapy with delayed-action glibenclamide and phenformin in fixed combination].
    Minerva medica, 1974, Sep-01, Volume: 65, Issue:60

    Topics: Adult; Aged; Blood Glucose; Carbutamide; Cholesterol; Delayed-Action Preparations; Diabetes Mellitus; Drug Combinations; Evaluation Studies as Topic; Fatty Acids, Nonesterified; Female; Glyburide; Glycosuria; Humans; Lipids; Male; Metformin; Middle Aged; Phenformin; Tolbutamide; Triglycerides

1974
Zinc and insulin content in pancreatic islets of rats after administration of hypoglycemic sulfonamides.
    Bulletin of experimental biology and medicine, 1974, Volume: 77, Issue:6

    Topics: Animals; Blood Glucose; Chlorpropamide; Glyburide; Histocytochemistry; Hypoglycemic Agents; Insulin; Islets of Langerhans; Male; Rats; Tolbutamide; Zinc

1974
Investigations on the antilipolytic activity of sulfonylureas in man with indications on limit dosages concerning their insulin-secreting properties.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1974, Volume: 6, Issue:6

    Topics: Blood Glucose; Body Weight; Dose-Response Relationship, Drug; Fatty Acids, Nonesterified; Glyburide; Humans; Insulin; Lipid Mobilization; Male; Time Factors; Tolbutamide

1974
Oral management of uncomplicated maturity onset diabetes.
    The Journal of the Egyptian Medical Association, 1974, Volume: 57, Issue:7-8

    Topics: Adult; Aged; Biguanides; Chlorpropamide; Diabetes Mellitus; Diet; Drug Combinations; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemic Agents; Insulin; Middle Aged; Obesity; Sulfonylurea Compounds; Tolbutamide

1974
[Studies on the course of mass screening in discovered diabetic patients].
    Zeitschrift fur die gesamte innere Medizin und ihre Grenzgebiete, 1974, Jul-01, Volume: 29, Issue:13

    Topics: Adolescent; Adult; Aged; Biguanides; Child; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Humans; Insulin; Male; Mass Screening; Middle Aged; Obesity; Tolbutamide

1974
[Recent pharmacologic aspects of sulfamides modifying insulin secretion (hypoglycemic and hyperglycemic sulfamides)].
    Actualites de physiologie pathologique, 1973, Volume: 4

    Topics: Animals; Catecholamines; Diazoxide; Dogs; Dose-Response Relationship, Drug; Drug Antagonism; Drug Synergism; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Isoproterenol; Pancreas; Pancreatectomy; Phenoxybenzamine; Propranolol; Rats; Tolbutamide

1973
[Propranolol and hypoglycemic sulfonamides. Study on insulin secretion and blood sugar].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1971, Volume: 165, Issue:6

    Topics: Animals; Blood Glucose; Dogs; Drug Antagonism; Drug Synergism; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Perfusion; Propranolol; Radioimmunoassay; Rats; Tolbutamide

1971
Proceedings: Half-life of phenprocoumarol (Marcumar R) during treatment with insulin and sulfonylureas in diabetics.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:Suppl

    Topics: Benzyl Compounds; Blood Glucose; Coumarins; Diabetes Mellitus; Glyburide; Half-Life; Humans; Insulin; Prothrombin Time; Sulfonylurea Compounds; Tolbutamide

1974
Biochemical and morphological events associated with the development of fetal rat pancreas "in vivo" and "in vitro": effect of glucagon and of other agents.
    Acta isotopica, 1970, Volume: 10, Issue:3

    Topics: Animals; Caffeine; Cell Differentiation; Culture Techniques; Cyclic AMP; Glucagon; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Pancreas; Pyruvates; Rats; Sulfonylurea Compounds; Tolbutamide

1970
The mode of action of adenosine 3':5'-cyclic monophosphate in mammalian islets of Langerhans. Effects of insulin secretagogues on islet-cell protein kinase activity.
    The Biochemical journal, 1973, Volume: 134, Issue:1

    Topics: Animals; Arginine; Caffeine; Cyclic AMP; Diazoxide; Epinephrine; Glucagon; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Leucine; Male; Phosphorus Isotopes; Phosphotransferases; Protein Kinases; Rats; Theophylline; Time Factors; Tolbutamide; Xanthines; Xylitol

1973
Inhibition of glucose-induced insulin secretion in trypsin-treated islets of Langerhans.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1973, Volume: 5, Issue:5

    Topics: Animals; Calcium; Cells, Cultured; Cellulose; Electrophoresis; Glucose; Glyburide; Humans; In Vitro Techniques; Insulin; Insulin Antibodies; Insulin Secretion; Islets of Langerhans; Magnesium; Male; Methods; Microbial Collagenase; Radioimmunoassay; Rats; Time Factors; Tolbutamide; Trypsin

1973
Significance of acid amyloglucosidase in sulphonylurea-induced insulin release.
    Diabetologia, 1974, Volume: 10, Issue:6

    Topics: Adenylyl Cyclases; Albumins; Amylases; Animals; Blood Glucose; Carbutamide; Cyclic AMP; Dose-Response Relationship, Drug; Fasting; Female; Glucuronidase; Glyburide; Glycoside Hydrolases; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred Strains; Norepinephrine; Phosphoric Diester Hydrolases; Rats; Secretin; Sulfonylurea Compounds; Tolbutamide; Xanthines

1974
Role of calcium and cyclic adenosine 3',5'-monophosphate in the antilipolytic effect of tolbutamide and glibenclamide.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 286, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adipose Tissue; Adrenocorticotropic Hormone; Animals; Bucladesine; Calcium; Carboxylic Acids; Cyclic AMP; Epinephrine; Glucagon; Glyburide; Isoproterenol; Lipid Metabolism; Male; Norepinephrine; Rats; Theophylline; Tolbutamide

1974
[Influence of an alpha- and beta-receptor blockade on the dynamics of insulin secretion in dogs following increased dosage of various sulfonylureas].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1971, Volume: 77

    Topics: 1-Propanol; Adrenergic beta-Antagonists; Amino Alcohols; Animals; Blood Glucose; Cresols; Dogs; Glyburide; Insulin; Insulin Secretion; Phentolamine; Propylamines; Sulfonylurea Compounds; Tolbutamide

1971
Haemolytic anaemia associated with antibodies to tolbutamide and phenacetin.
    British medical journal, 1972, Mar-18, Volume: 1, Issue:5802

    Topics: Anemia, Hemolytic; Antibodies; Chlorpropamide; Coombs Test; Cross Reactions; Female; Glyburide; Humans; Middle Aged; Phenacetin; Tolbutamide

1972
[Advantages and hazards of oral antidiabetics].
    Deutsches medizinisches Journal, 1972, Feb-10, Volume: 23, Issue:2

    Topics: Administration, Oral; Diabetes Mellitus; Diet Therapy; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Tolbutamide

1972
[Role of glibenclamide in the therapy of diabetes].
    Minerva medica, 1972, Apr-14, Volume: 63, Issue:28

    Topics: Adult; Chlorpropamide; Diabetes Mellitus; Evaluation Studies as Topic; Glyburide; Glycosuria; Humans; Insulin; Insulin Secretion; Sulfonylurea Compounds; Tolbutamide

1972
A dose equivalence study of glybenclamide (daonil)--a new hypoglycaemic agent.
    The Journal of the Association of Physicians of India, 1972, Volume: 20, Issue:3

    Topics: Adult; Chlorpropamide; Diabetes Mellitus; Female; Glyburide; Humans; Male; Sulfonylurea Compounds; Therapeutic Equivalency; Tolbutamide

1972
[Infantile diabetes and treatment with oral hypoglycemizing agents (function tests of the endocrine pancreatic before and after one year of therapy)].
    Minerva pediatrica, 1972, Jun-02, Volume: 24, Issue:20

    Topics: Child; Child, Preschool; Diabetes Mellitus, Type 1; Female; Glucose Tolerance Test; Glyburide; Humans; Insulin; Male; Pancreas; Phenformin; Sulfonylurea Compounds; Tolbutamide

1972
Oral therapy in diabetes.
    Journal of the Royal College of Physicians of London, 1972, Volume: 7, Issue:1

    Topics: Acetohexamide; Administration, Oral; Animals; Chlorpropamide; Diabetes Mellitus; Diet Therapy; Evaluation Studies as Topic; Glyburide; Humans; Hypoglycemic Agents; Insulin; Metformin; Obesity; Phenformin; Pyrimidines; Sulfonamides; Time Factors; Tolbutamide

1972
The effect of tolbutamide and glibenclamide on the incorporation of ( 3 H)leucine and on the conversion of proinsulin to insulin in isolated pancreatic islets.
    FEBS letters, 1972, Oct-01, Volume: 26, Issue:1

    Topics: Animals; Chromatography, Gel; Depression, Chemical; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Isotope Labeling; Leucine; Male; Mice; Proinsulin; Rats; Time Factors; Tolbutamide; Tritium

1972
The effects of tolbutamide and glibenclamide on intestinal glucose absorption.
    Biochemical pharmacology, 1972, Jul-01, Volume: 21, Issue:13

    Topics: Aerobiosis; Anaerobiosis; Animals; Blood Glucose; Body Weight; Glucose; Glyburide; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Jejunum; Male; Rats; Sulfonylurea Compounds; Time Factors; Tolbutamide

1972
Diabetes mellitus: the thin maturity-onset diabetic.
    British medical journal, 1972, Sep-16, Volume: 3, Issue:5828

    Topics: Acetohexamide; Body Weight; Chlorpropamide; Diabetes Mellitus; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Middle Aged; Tolazamide; Tolbutamide

1972
[Recent findings in the use of 1st and 2nd generation hypoglycemic sulfonamides].
    Klinische Wochenschrift, 1973, Jan-15, Volume: 51, Issue:2

    Topics: Adult; Azepines; Blood Glucose; Dose-Response Relationship, Drug; Glucose; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemic Agents; Insulin; Oxazoles; Pancreas; Sulfonylurea Compounds; Tolbutamide

1973
[The effect of oral antidiabetics on the biosynthesis of proinsulin in the rat].
    Arzneimittel-Forschung, 1972, Volume: 22, Issue:11

    Topics: Animals; Chromatography, Gel; Electrophoresis, Disc; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Islets of Langerhans; Leucine; Male; Proinsulin; Pyrimidines; Rats; Sulfonic Acids; Sulfonylurea Compounds; Tolbutamide; Tritium

1972
[Incidence and severity of treatment-induced hypoglycemias in diabetics].
    Deutsche medizinische Wochenschrift (1946), 1971, Nov-12, Volume: 96, Issue:46

    Topics: Aged; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Hemiplegia; Humans; Hypoglycemia; Insulin; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1971
[ADH-like mechanism of action of chlorpropamide in diabetes insipidus (a comparison with the antidiuretic effect of other blood glucose decreasing sulfonamides and hydrochlorothiazide)].
    Klinische Wochenschrift, 1970, Jul-15, Volume: 48, Issue:14

    Topics: Aged; Blood Glucose; Body Weight; Chlorpropamide; Depression, Chemical; Diabetes Insipidus; Diuresis; Female; Glyburide; Humans; Hydrochlorothiazide; Hypoglycemic Agents; Male; Middle Aged; Natriuresis; Osmolar Concentration; Potassium; Sulfonylurea Compounds; Tolbutamide; Vasopressins

1970
In vitro effect of various hypoglycemic agents on the hepatic and pancreatic protein synthesis in the rat.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1971, Volume: 3, Issue:5

    Topics: Animals; Cell-Free System; Depression, Chemical; Ethers; Female; Glyburide; Hypoglycemic Agents; Leucine; Liver; Male; Metabolism; Pancreas; Protein Biosynthesis; Pyrimidines; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Terpenes; Tolbutamide; Tritium

1971
Treatment with glibenclamide in maturity-onset diabetes mellitus.
    Geriatrics, 1971, Volume: 26, Issue:5

    Topics: Age Factors; Aged; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1971
Immunohistological demonstration of insulin in islets of langerhans after stimulation of insulin secretion by glucose, sulphonylureas and insulin antibodies.
    Diabetologia, 1971, Volume: 7, Issue:6

    Topics: Animals; Fluorescent Antibody Technique; Formaldehyde; Freeze Drying; Glucose; Glyburide; Histological Techniques; Insulin; Insulin Antibodies; Insulin Secretion; Islets of Langerhans; Male; Methods; Pancreas; Rats; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide

1971
Pharmacodynamic aspects of tolbutamide, glibenclamide, glibornuride and glisoxepide. I. Dose response relations and repeated administration in diabetic subjects.
    Diabetologia, 1971, Volume: 7, Issue:6

    Topics: Adult; Blood Glucose; Diabetes Mellitus; Glyburide; Humans; Injections, Intravenous; Insulin; Insulin Secretion; Sulfonylurea Compounds; Tolbutamide

1971
Pharmacodynamic aspects of tolbutamide, glibenclamide, glibornuride, and glisoxepide. II. Repeated administration in combination with glucose.
    Diabetologia, 1971, Volume: 7, Issue:6

    Topics: Adult; Blood Glucose; Glucose; Glyburide; Humans; Injections, Intravenous; Insulin; Insulin Secretion; Sulfonylurea Compounds; Tolbutamide

1971
[Synergism between oral diabetics and insulin].
    Bollettino della Societa italiana di biologia sperimentale, 1971, Nov-30, Volume: 47, Issue:22

    Topics: Animals; Biguanides; Blood Glucose; Chlorpropamide; Columbidae; Drug Synergism; Glyburide; Hypoglycemia; Hypoglycemic Agents; Insulin; Tolbutamide

1971
Clinical experiences in oral antidiabetic therapy with sulphonylureas and biguanides.
    Australian and New Zealand journal of medicine, 1971, Volume: 1

    Topics: Aged; Biguanides; Blood Glucose; Diabetes Mellitus; Glyburide; Humans; Insulin; Middle Aged; Phenformin; Sulfonylurea Compounds; Tolbutamide

1971
[Studies on the effect of various sulfonylureas during adrenergic blockade of the insulin secretion in man].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1971, Volume: 77

    Topics: Blood Glucose; Catecholamines; Drug Antagonism; Epinephrine; Fatty Acids, Nonesterified; Glyburide; Glycerol; Humans; Insulin; Insulin Secretion; Norepinephrine; Sulfonylurea Compounds; Tolbutamide

1971
[Changes of blood sugar, serum insulin and free fatty acids following tolbutamide and glibenclamide in subjects of normal metabolism, pretreated with alpha and beta receptor blockaders].
    Verhandlungen der Deutschen Gesellschaft fur Innere Medizin, 1971, Volume: 77

    Topics: Blood Glucose; Fatty Acids, Nonesterified; Glyburide; Humans; Insulin; Phentolamine; Propranolol; Tolbutamide

1971
Suppressive effect of long term sulfonylurea treatment on A, B, and D cells of normal rat pancreas.
    Endocrinology, 1983, Volume: 113, Issue:6

    Topics: Animals; Arginine; Glucagon; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Somatostatin; Time Factors; Tolbutamide

1983
Glibenclamide is exceptional among hypoglycaemic sulphonylureas in accumulating progressively in beta-cell-rich pancreatic islets.
    Acta endocrinologica, 1984, Volume: 105, Issue:3

    Topics: Animals; Carbutamide; Chlorpropamide; Glipizide; Glyburide; Islets of Langerhans; Mice; Mice, Obese; Sulfonylurea Compounds; Tolbutamide

1984
Effects of sulfonylureas on membrane-bound low Km cyclic AMP phosphodiesterase in rat fat cells.
    Biochimica et biophysica acta, 1982, Nov-17, Volume: 721, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Acetohexamide; Adipose Tissue; Animals; Buformin; Glyburide; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide

1982
Thiol-dependent and non-thiol-dependent stimulations of insulin release.
    Diabetes, 1984, Volume: 33, Issue:3

    Topics: Animals; Bucladesine; Calcimycin; Calcium; Diamide; Dose-Response Relationship, Drug; Female; Glucose; Glutathione; Glyburide; Glyceraldehyde; Insulin; Insulin Secretion; Islets of Langerhans; Isoproterenol; Leucine; Male; Rats; Rats, Inbred Strains; Sulfhydryl Compounds; Tolbutamide

1984
Tolbutamide and glyburide differ in effectiveness to displace alpha- and beta-adrenergic radioligands in pancreatic islet cells and membranes.
    Diabetes, 1984, Volume: 33, Issue:5

    Topics: Alprenolol; Animals; Cell Membrane; Clonidine; Dihydroalprenolol; Epinephrine; Glyburide; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tolbutamide

1984
Clinical pharmacology of glipizide.
    The American journal of medicine, 1983, Nov-30, Volume: 75, Issue:5B

    Topics: Biological Availability; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Half-Life; Humans; Kinetics; Structure-Activity Relationship; Sulfonylurea Compounds; Tolbutamide

1983
[Hypoglycemic effects of the blended Chinese traditional medicines in genetically and chemically diabetic mice].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1984, Volume: 83, Issue:1

    Topics: Alloxan; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Glyburide; Hypoglycemic Agents; Male; Medicine, Chinese Traditional; Medicine, East Asian Traditional; Metformin; Mice; Tolbutamide

1984
Effects of cations, ionophores and hypoglycemic sulfonylureas on the fluorescence of fluorescein-labelled pancreatic islets.
    Research communications in chemical pathology and pharmacology, 1984, Volume: 44, Issue:1

    Topics: Animals; Calcimycin; Calcium; Fluoresceins; Fluorescence; Glyburide; Hydrogen-Ion Concentration; Hypoglycemic Agents; Islets of Langerhans; Lasalocid; Potassium; Rats; Tolbutamide

1984
Effect of glibenclamide on the osmotic resistance of pancreatic beta-cells.
    Acta physiologica Scandinavica, 1984, Volume: 120, Issue:3

    Topics: Animals; Cell Membrane; Culture Media; Glyburide; Imipramine; Islets of Langerhans; Mice; Mice, Obese; Osmolar Concentration; Tetracaine; Tolbutamide

1984
The control of 86Rb efflux from rat isolated pancreatic islets by the sulphonylureas tolbutamide and glibenclamide.
    British journal of pharmacology, 1984, Volume: 82, Issue:3

    Topics: Animals; Biological Transport; Calcium; Cell Membrane; Cell Membrane Permeability; Cobalt; Glyburide; In Vitro Techniques; Islets of Langerhans; Male; Potassium; Radioisotopes; Rats; Rats, Inbred Strains; Rubidium; Tolbutamide

1984
Effects of tolbutamide and glyburide on glucose and acetate incorporation into aortic lipids of the dog.
    Blood vessels, 1980, Volume: 17, Issue:4

    Topics: Acetates; Animals; Aorta; Dogs; Glucose; Glyburide; Lipid Metabolism; Tolbutamide

1980
Glipizide: experimental study and comparison with other sulfonylureas.
    Acta endocrinologica. Supplementum, 1980, Volume: 239

    Topics: Animals; Blood Glucose; Dogs; Dose-Response Relationship, Drug; Glipizide; Glyburide; Hypoglycemia; Insulin; Islets of Langerhans; Mice; Rats; Sulfonylurea Compounds; Tolbutamide

1980
Kinetics-effect relations of glipizide and other sulfonylureas.
    Acta endocrinologica. Supplementum, 1980, Volume: 239

    Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus; Dose-Response Relationship, Drug; Fasting; Feeding Behavior; Glipizide; Glyburide; Humans; Kidney; Sulfonylurea Compounds; Tolbutamide

1980
Comparative single-dose kinetics and effects of four sulfonylureas in healthy volunteers.
    Acta medica Scandinavica, 1980, Volume: 208, Issue:4

    Topics: Adult; Blood Glucose; Chlorpropamide; Fasting; Glipizide; Glyburide; Humans; Insulin; Kinetics; Male; Sulfonylurea Compounds; Time Factors; Tolbutamide

1980
The pharmacology of sulfonylureas.
    The American journal of medicine, 1981, Volume: 70, Issue:2

    Topics: Acetohexamide; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Glyburide; Humans; Insulin; Sulfonylurea Compounds; Tolazamide; Tolbutamide

1981
Lipoprotein patterns in diet, sulphonylurea, and insulin treated diabetics.
    Diabetologia, 1981, Volume: 20, Issue:2

    Topics: Adult; Aged; Blood Glucose; Body Weight; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Humans; Insulin; Lipoproteins; Male; Middle Aged; Tolbutamide

1981
IRI-secretion in MOD with and without SU (5 year control).
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1980, Volume: 12, Issue:12

    Topics: Blood Glucose; Diabetes Mellitus; Glucagon; Glyburide; Humans; Insulin; Middle Aged; Tolbutamide

1980
Long-term actions of sulfonylureas on (Pro-) insulin biosynthesis and secretion. III. Functional state of isolated pancreatic rat islets after culture in the presence of tolbutamide and glibenclamide.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1981, Volume: 13, Issue:7

    Topics: Animals; Cells, Cultured; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Proinsulin; Rats; Tolbutamide

1981
Serum glycohydrolases in compensated & decompensated alloxan diabetic rabbits.
    Indian journal of experimental biology, 1981, Volume: 19, Issue:8

    Topics: Animals; Diabetes Mellitus, Experimental; Glyburide; Glycoside Hydrolases; Insulin; Kinetics; Male; Rabbits; Tolbutamide

1981
[The effect of tolbutamide and glibenclamide on HDL-cholesterol levels].
    Orvosi hetilap, 1982, Dec-26, Volume: 123, Issue:52

    Topics: Glyburide; Humans; Lipoproteins, HDL; Tolbutamide

1982
Reconstitution of a KATP channel from basolateral membranes of Necturus enterocytes.
    The American journal of physiology, 1995, Volume: 269, Issue:2 Pt 1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Diazoxide; Glyburide; Intestine, Small; Membranes; Necturus; Potassium Channels; Tolbutamide

1995
Inhibition of liver microsomal carnitine acyltransferases by sulphonylurea drugs.
    FEBS letters, 1995, Sep-04, Volume: 371, Issue:2

    Topics: Animals; Carnitine Acyltransferases; Glyburide; Lipoproteins, VLDL; Liposomes; Male; Malonyl Coenzyme A; Microsomes, Liver; Rats; Rats, Sprague-Dawley; Tolbutamide; Triglycerides

1995
Dissociation of KATP channel and sulphonylurea receptor in the rat clonal insulin-secreting cell line, CRI-D11.
    Proceedings. Biological sciences, 1993, Sep-22, Volume: 253, Issue:1338

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Cell Membrane; Clone Cells; Glyburide; Insulin; Insulin Secretion; Insulinoma; Membrane Potentials; Pancreatic Neoplasms; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sulfonylurea Receptors; Tetradecanoylphorbol Acetate; Tolbutamide; Tumor Cells, Cultured

1993
Regulation of a potassium conductance in rat midbrain dopamine neurons by intracellular adenosine triphosphate (ATP) and the sulfonylureas tolbutamide and glibenclamide.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:6

    Topics: Adenosine Triphosphate; Animals; Dopamine; Electric Conductivity; Glyburide; Homeostasis; In Vitro Techniques; Male; Membrane Potentials; Mesencephalon; Neurons; Patch-Clamp Techniques; Potassium; Potassium Channels; Rats; Rats, Wistar; Tolbutamide

1995
Characterization of ATP-sensitive potassium channel-blocking activity of ZENECA ZM181,037, a eukalemic diuretic.
    Pharmacology, 1994, Volume: 49, Issue:4

    Topics: Acetamides; Adenosine Triphosphate; Administration, Oral; Animals; Benzopyrans; Blood Glucose; Blood Pressure; Cromakalim; Diuretics; Dogs; Dose-Response Relationship, Drug; Electrophysiology; Glyburide; Guinea Pigs; Hypertension; In Vitro Techniques; Injections, Intravenous; Male; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Potassium Channel Blockers; Pyrroles; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Stereoisomerism; Tolbutamide

1994
Location of the sulphonylurea receptor at the cytoplasmic face of the beta-cell membrane.
    British journal of pharmacology, 1994, Volume: 113, Issue:3

    Topics: Animals; ATP-Binding Cassette Transporters; Cells, Cultured; Cytoplasm; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Solubility; Sulfonylurea Receptors; Tolbutamide

1994
Tolbutamide suppresses slow and medium afterhyperpolarization in hippocampal slices.
    Neuroreport, 1994, Oct-27, Volume: 5, Issue:16

    Topics: Animals; Electric Stimulation; Evoked Potentials; Glyburide; Hippocampus; In Vitro Techniques; Neurons; Rats; Rats, Sprague-Dawley; Tolbutamide

1994
Influence of ranitidine on the hypoglycaemic activity of glibenclamide and tolbutamide in rabbits.
    Indian journal of physiology and pharmacology, 1994, Volume: 38, Issue:4

    Topics: Animals; Drug Interactions; Glyburide; Hypoglycemia; Rabbits; Ranitidine; Tolbutamide

1994
Spontaneous activation of KATP current in rat dorsal vagal neurones.
    Neuroreport, 1994, Jun-02, Volume: 5, Issue:10

    Topics: Adenosine Triphosphate; Animals; Diazoxide; Diffusion; Female; Glyburide; Male; Membrane Potentials; Neurons; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium Compounds; Tolbutamide; Vagus Nerve

1994
Tetraethylammonium selectively stimulates secretion from noradrenergic bovine chromaffin cells.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:3

    Topics: 4-Aminopyridine; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; Drug Interactions; Drug Synergism; Epinephrine; Glyburide; Nifedipine; Norepinephrine; Ouabain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tolbutamide

1994
Mg(2+)-dependent inhibition of KATP by sulphonylureas in CRI-G1 insulin-secreting cells.
    British journal of pharmacology, 1994, Volume: 111, Issue:2

    Topics: Adenosine Triphosphate; Animals; Benzamides; Cell Line; Cell Membrane; Electrophysiology; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Ligands; Magnesium; Potassium Channels; Rats; Sulfonylurea Compounds; Thiopental; Tolbutamide

1994
The ATP-regulated potassium channel in ischemia-reperfusion injury.
    Annals of the New York Academy of Sciences, 1994, Jun-17, Volume: 723

    Topics: Adenosine Triphosphate; Animals; Dogs; Glyburide; Ion Channel Gating; Myocardial Contraction; Myocardial Infarction; Myocardial Reperfusion Injury; Niacinamide; Nicorandil; Picolines; Potassium Channels; Pyrans; Tolbutamide

1994
Photoaffinity labeling of the cerebral sulfonylurea receptor using a novel radioiodinated azidoglibenclamide analogue.
    Journal of neurochemistry, 1994, Volume: 63, Issue:2

    Topics: Affinity Labels; Animals; ATP-Binding Cassette Transporters; Binding, Competitive; Cell Fractionation; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Glipizide; Glyburide; Iodine Radioisotopes; Kinetics; Microsomes; Molecular Weight; Photolysis; Potassium Channels; Potassium Channels, Inwardly Rectifying; Radioligand Assay; Receptors, Drug; Sulfonylurea Receptors; Swine; Tolbutamide; Tritium

1994
The effects of trypsin on ATP-sensitive potassium channel properties and sulfonylurea receptors in the CRI-G1 insulin-secreting cell line.
    Molecular pharmacology, 1994, Volume: 46, Issue:1

    Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Cell Line; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sulfonylurea Receptors; Tolbutamide; Trypsin

1994
Comparative placental transport of oral hypoglycemic agents in humans: a model of human placental drug transfer.
    American journal of obstetrics and gynecology, 1994, Volume: 171, Issue:3

    Topics: Administration, Oral; Analysis of Variance; Antipyrine; Biological Transport; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Maternal-Fetal Exchange; Models, Biological; Molecular Weight; Placenta; Pregnancy; Regression Analysis; Tolbutamide

1994
Tolbutamide suppresses anoxic outward current of hippocampal neurons.
    Neuroscience letters, 1993, Nov-12, Volume: 162, Issue:1-2

    Topics: Adenosine Triphosphate; Animals; Glyburide; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Kynurenic Acid; Neurons; Potassium Channels; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Tolbutamide

1993
Effects of sulphonylureas on cAMP-stimulated Cl- transport via the cystic fibrosis gene product in human epithelial cells.
    Pflugers Archiv : European journal of physiology, 1994, Volume: 426, Issue:3-4

    Topics: Adenosine Triphosphate; Blood Proteins; Cell Line; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Diazoxide; Electrophysiology; Glyburide; Humans; Sulfonylurea Compounds; Tolbutamide

1994
Tolbutamide, but not glyburide, affects the excitability and contractility of unfatigued frog sartorius muscle.
    European journal of pharmacology, 1993, Sep-21, Volume: 242, Issue:1

    Topics: Action Potentials; Animals; Electric Stimulation; Glyburide; Hydrogen-Ion Concentration; Muscle Contraction; Muscle, Smooth; Potassium Channels; Rana pipiens; Tolbutamide

1993
Sulfonylurea-binding sites and ATP-sensitive K+ channels in alpha-TC glucagonoma and beta-TC insulinoma cells.
    Diabetes, 1993, Volume: 42, Issue:12

    Topics: Adenosine Triphosphate; Animals; Binding Sites; Binding, Competitive; Diazoxide; Glucagon; Glucagonoma; Glyburide; Insulinoma; Kinetics; Membrane Potentials; Mice; Pancreatic Neoplasms; Potassium Channels; Tolbutamide; Tritium; Tumor Cells, Cultured

1993
Multiple sulfonylurea-sensitive potassium channels: a novel subtype modulated by dopamine.
    Molecular pharmacology, 1993, Volume: 44, Issue:5

    Topics: Animals; Dopamine; Glyburide; In Vitro Techniques; Male; Membrane Potentials; Neostriatum; Neurons; Potassium Channels; Rats; Rats, Sprague-Dawley; Tolbutamide

1993
Whole-cell recordings of inwardly rectifying K+ currents activated by 5-HT1A receptors on dorsal raphe neurones of the adult rat.
    The Journal of physiology, 1993, Volume: 469

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Barium; Cyclic AMP; Electrophysiology; Glyburide; In Vitro Techniques; Ion Channel Gating; Masoprocol; Membrane Potentials; Neurons; Pertussis Toxin; Potassium; Potassium Channels; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Tolbutamide; Virulence Factors, Bordetella

1993
Characterization and solubilization of the sulphonylurea receptor in rat brain.
    Neuropharmacology, 1993, Volume: 32, Issue:10

    Topics: Adenine Nucleotides; Adenosine Triphosphatases; Animals; ATP-Binding Cassette Transporters; Benzamides; Binding, Competitive; Brain Chemistry; Ca(2+) Mg(2+)-ATPase; Diazoxide; Glyburide; Guanine Nucleotides; Hypoglycemic Agents; In Vitro Techniques; Membranes; Microsomes; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sulfonylurea Receptors; Tolbutamide

1993
Sulphonylurea drugs no longer inhibit ATP-sensitive K+ channels during metabolic stress in cardiac muscle.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Cells, Cultured; Dihydropyridines; Dinitrophenols; Glyburide; Heart; Membrane Potentials; Myocardial Contraction; Myocardium; Potassium Channels; Rats; Sensitivity and Specificity; Stress, Physiological; Sulfonylurea Compounds; Tolbutamide

1993
Effects of potassium channel openers and their antagonists on rat locus coeruleus neurones.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Barium; Benzopyrans; Cromakalim; Electrophysiology; Glyburide; In Vitro Techniques; Kynurenic Acid; Locus Coeruleus; Male; Membrane Potentials; Neurons; Parasympatholytics; Potassium Channels; Pyridines; Pyrroles; Rats; Rats, Wistar; Substantia Nigra; Tetrodotoxin; Tolbutamide

1993
Potassium channel-mediated relaxation to acetylcholine in rabbit arteries.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Acetylcholine; Animals; Aorta, Abdominal; Aorta, Thoracic; Arginine; Cyclic GMP; Endothelium, Vascular; Glyburide; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Potassium; Potassium Channels; Rabbits; Stimulation, Chemical; Tetraethylammonium; Tetraethylammonium Compounds; Tolbutamide

1993
Adenosine release is a major cause of failure of synaptic transmission during hypoglycaemia in rat hippocampal slices.
    Neuroscience letters, 1993, Jun-11, Volume: 155, Issue:2

    Topics: Action Potentials; Adenosine; Animals; Caffeine; Cell Hypoxia; Energy Metabolism; Evoked Potentials; Glucose; Glyburide; Hippocampus; Hypoglycemia; Neural Inhibition; Potassium; Potassium Channels; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Theophylline; Tolbutamide

1993
Enhanced stimulus-secretion coupling in polyamine-depleted rat insulinoma cells. An effect involving increased cytoplasmic Ca2+, inositol phosphate generation, and phorbol ester sensitivity.
    The Journal of clinical investigation, 1993, Volume: 92, Issue:4

    Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Channels; Carbachol; Cytoplasm; Diazoxide; DNA, Neoplasm; Eflornithine; Glucose; Glyburide; Inositol Phosphates; Insulin; Insulin Secretion; Insulinoma; Kinetics; Pancreatic Neoplasms; Polyamines; Potassium; Putrescine; Rats; RNA, Messenger; Spermidine; Spermine; Tetradecanoylphorbol Acetate; Theophylline; Tolbutamide; Tumor Cells, Cultured

1993
Sulphonylureas reduce the slowly inactivating D-type outward current in rat hippocampal neurons.
    The Journal of physiology, 1993, Volume: 466

    Topics: Adenosine Triphosphate; Animals; Electric Conductivity; Glyburide; Hippocampus; Hypoglycemic Agents; In Vitro Techniques; Male; Membrane Potentials; Neurons; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Sulfonylurea Compounds; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tolbutamide

1993
ATP-inhibited and Ca(2+)-dependent K+ channels in the soma membrane of cultured leech Retzius neurons.
    The Journal of membrane biology, 1993, Volume: 134, Issue:2

    Topics: Adenosine Triphosphate; Animals; Barium; Calcium; Cells, Cultured; Cesium; Electric Stimulation; Glyburide; Hydrogen-Ion Concentration; Leeches; Membrane Potentials; Neurons; Potassium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Tolbutamide

1993
Tolbutamide-sensitive potassium conductance in the basolateral membrane of A6 cells.
    The Journal of membrane biology, 1993, Volume: 134, Issue:3

    Topics: Adenosine Triphosphate; Amphibians; Animals; Cell Line; Cell Membrane; Epithelium; Glucose; Glyburide; Insulin; Kidney; Membrane Potentials; Potassium Channels; Sulfonylurea Compounds; Tolbutamide

1993
Potentiating effects of combined usage of three sulfonylurea drugs on the occurrence of alloxan diabetes in rats.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1993, Volume: 25, Issue:2

    Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Drug Combinations; Drug Synergism; Gliclazide; Glyburide; Hypoglycemic Agents; Rats; Rats, Wistar; Sulfonylurea Compounds; Tolbutamide

1993
Mechanosensitive gating of atrial ATP-sensitive potassium channels.
    Circulation research, 1993, Volume: 72, Issue:5

    Topics: Adenosine Triphosphate; Animals; Electrophysiology; Glyburide; Guanidines; Heart Atria; Ion Channel Gating; Myocardium; Pinacidil; Potassium Channels; Pressure; Rats; Rats, Wistar; Tolbutamide

1993
Glibenclamide and meglitinide block the transport of low molecular weight solutes into malaria-infected erythrocytes.
    FEBS letters, 1993, May-24, Volume: 323, Issue:1-2

    Topics: Animals; Benzamides; Biological Transport; Cells, Cultured; Chlorides; Choline; Erythrocytes; Glyburide; Humans; Kinetics; Molecular Weight; Plasmodium falciparum; Sorbitol; Threonine; Tolbutamide

1993
PKC-dependent stimulation of exocytosis by sulfonylureas in pancreatic beta cells.
    Science (New York, N.Y.), 1996, Feb-09, Volume: 271, Issue:5250

    Topics: Animals; Calcium; Cells, Cultured; Cytoplasmic Granules; Electric Conductivity; Exocytosis; Glipizide; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Protein Kinase C; Sulfonylurea Compounds; Tolbutamide

1996
Gliclazide hydroxylation by rat liver microsomes.
    Xenobiotica; the fate of foreign compounds in biological systems, 1995, Volume: 25, Issue:12

    Topics: Animals; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2D6; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Enzyme Inhibitors; Gliclazide; Glipizide; Glyburide; Hydroxylation; Hypoglycemic Agents; Kinetics; Male; Microsomes, Liver; Mixed Function Oxygenases; Rats; Rats, Sprague-Dawley; Tolbutamide

1995
Tolbutamide blocks Ca(2+)- and voltage-dependent K+ currents of hippocampal Ca1 neurons.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Animals; Calcium Channels; Depression, Chemical; Dose-Response Relationship, Drug; Evoked Potentials; Glyburide; Hippocampus; In Vitro Techniques; Membrane Potentials; Patch-Clamp Techniques; Potassium Channels; Rats; Rats, Sprague-Dawley; Tolbutamide

1996
ATP-sensitive K+ channels are functional in expiratory neurones of normoxic cats.
    The Journal of physiology, 1996, Jul-15, Volume: 494 ( Pt 2)

    Topics: Adenosine Triphosphate; Animals; Bicuculline; Blood-Brain Barrier; Brain Stem; Cats; Female; Glyburide; Hypoxia; Male; Membrane Potentials; Neurons; Phrenic Nerve; Potassium Channels; Reference Values; Respiration; Tolbutamide

1996
Sulphonylureas do not increase insulin secretion by a mechanism other than a rise in cytoplasmic Ca2+ in pancreatic B-cells.
    European journal of pharmacology, 1996, Mar-18, Volume: 298, Issue:3

    Topics: Adenosine Triphosphate; Animals; Calcium; Cytoplasm; Cytosol; Female; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Potassium; Sulfonylurea Compounds; Tolbutamide; Type C Phospholipases

1996
Membrane potentials and microenvironment of rat dorsal vagal cells in vitro during energy depletion.
    The Journal of physiology, 1996, Sep-15, Volume: 495 ( Pt 3)

    Topics: Animals; Brain Stem; Cell Hypoxia; Diazoxide; Electric Stimulation; Glucose; Glyburide; Hydrogen-Ion Concentration; In Vitro Techniques; Membrane Potentials; Neuroglia; Neurons; Oxygen Consumption; Potassium; Rats; Synaptic Transmission; Tolbutamide; Vagus Nerve

1996
Photohemolytic potency of oral antidiabetic drugs in vitro: effects of antioxidants and a nitrogen atmosphere.
    Photodermatology, photoimmunology & photomedicine, 1996, Volume: 12, Issue:4

    Topics: Antioxidants; Ascorbic Acid; Carbutamide; Chlorpropamide; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glyburide; Hemolysis; Humans; Hypoglycemic Agents; Nitrogen; Radiation-Sensitizing Agents; Reactive Oxygen Species; Sulfonamides; Sulfonylurea Compounds; Superoxide Dismutase; Tolazamide; Tolbutamide; Ultraviolet Rays; Vitamin E

1996
Inhibitory effect of sulfonylureas on protein phosphatase activity in rat pancreatic islets.
    Acta diabetologica, 1997, Volume: 34, Issue:1

    Topics: Animals; Cytosol; Gliclazide; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Kinetics; Male; Okadaic Acid; Phosphoprotein Phosphatases; Rats; Rats, Wistar; Sulfonylurea Compounds; Tolbutamide

1997
Rates of hypoglycemia in users of sulfonylureas.
    Journal of clinical epidemiology, 1997, Volume: 50, Issue:6

    Topics: Adult; Aged; Chlorpropamide; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Incidence; Male; Middle Aged; Poisson Distribution; Risk; Risk Factors; Sulfonylurea Compounds; Surveys and Questionnaires; Time Factors; Tolbutamide

1997
Antidiabetic sulphonylureas stimulate acetylcholine release from striatal cholinergic interneurones through inhibition of K(ATP) channel activity.
    Journal of neurochemistry, 1997, Volume: 69, Issue:4

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Corpus Striatum; Glyburide; Hypoglycemic Agents; Interneurons; Male; Parasympathetic Nervous System; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Tolbutamide

1997
Ca2+-activated K+ currents in rat locus coeruleus neurons induced by experimental ischemia, anoxia, and hypoglycemia.
    Journal of neurophysiology, 1997, Volume: 78, Issue:5

    Topics: Animals; Brain Ischemia; Calcium; Calcium Channels; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Charybdotoxin; Glucose; Glyburide; Hypoglycemia; Hypoxia, Brain; In Vitro Techniques; Locus Coeruleus; Membrane Potentials; N-Methylaspartate; Neurons; Oxygen; Partial Pressure; Rats; Rats, Wistar; Ryanodine; Sodium Cyanide; Thapsigargin; Tolbutamide

1997
KATP channels contribute to beta- and adenosine receptor-mediated pulmonary vasorelaxation.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Acetylcholine; Adenosine; Adenylyl Cyclases; Animals; ATP-Binding Cassette Transporters; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Glyburide; In Vitro Techniques; Isoproterenol; KATP Channels; Kinetics; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Tolbutamide; Vasodilation

1997
Effects of glycosylation of hypoglycaemic drug binding to serum albumin.
    Biopharmaceutics & drug disposition, 1997, Volume: 18, Issue:9

    Topics: Acetohexamide; Binding Sites; Binding, Competitive; Gliclazide; Glyburide; Glycated Serum Albumin; Glycation End Products, Advanced; Glycosylation; Humans; Hypoglycemic Agents; Metformin; Serum Albumin; Spectrometry, Fluorescence; Structure-Activity Relationship; Tolbutamide

1997
The effects of gliclazide and other sulfonylureas on low-density lipoprotein oxidation in vitro.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:12 Suppl 1

    Topics: Administration, Oral; Adult; Antioxidants; Ascorbic Acid; Coronary Artery Disease; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Lipoproteins, LDL; Male; Middle Aged; Oxidation-Reduction; Sulfonylurea Compounds; Tolbutamide

1997
Treatment of NIDDM in youth.
    Clinical pediatrics, 1998, Volume: 37, Issue:2

    Topics: Adolescent; Child; Diabetes Mellitus, Type 2; Female; Glyburide; Humans; Hypoglycemic Agents; Japan; Male; School Health Services; Tolbutamide

1998
Whole cell patch-clamp recordings of rat midbrain dopaminergic neurons isolate a sulphonylurea- and ATP-sensitive component of potassium currents activated by hypoxia.
    Journal of neurophysiology, 1998, Volume: 79, Issue:3

    Topics: Adenosine Triphosphate; Animals; Barium Compounds; Cell Hypoxia; Charybdotoxin; Chlorides; Dopamine; Glipizide; Glyburide; In Vitro Techniques; Membrane Potentials; Mesencephalon; Microelectrodes; Neurons; Patch-Clamp Techniques; Potassium Channels; Rats; Rats, Wistar; Reaction Time; Sulfonylurea Compounds; Tolbutamide

1998
Insulin secretion from isolated rat islets induced by the novel hypoglycemic agent A-4166, a derivative of D-phenylalanine.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1998, Volume: 30, Issue:1

    Topics: Animals; ATP-Binding Cassette Transporters; Biological Availability; Calcium; Cell Line; Cyclohexanes; Diazoxide; Epinephrine; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nateglinide; Phenylalanine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rubidium; Somatostatin; Stereoisomerism; Sulfonylurea Receptors; Tolbutamide

1998
Hypoxia activates ATP-dependent potassium channels in inspiratory neurones of neonatal mice.
    The Journal of physiology, 1998, Jun-15, Volume: 509 ( Pt 3)

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Calcium; Diazoxide; Electric Stimulation; Glyburide; Hypoglycemic Agents; Hypoxia; Hypoxia, Brain; Ion Channel Gating; Medulla Oblongata; Membrane Potentials; Mice; Neurons; Patch-Clamp Techniques; Potassium Channels; Respiration; Tolbutamide; Vasodilator Agents

1998
Identification of an ATP-sensitive potassium channel current in rat striatal cholinergic interneurones.
    The Journal of physiology, 1998, Jul-15, Volume: 510 ( Pt 2)

    Topics: Adenosine Triphosphate; Animals; Diazoxide; Diuretics; Electric Stimulation; Electrophysiology; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Interneurons; Male; Membrane Potentials; Neostriatum; Parasympathetic Nervous System; Patch-Clamp Techniques; Potassium Channels; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Sodium Chloride Symporter Inhibitors; Tolbutamide

1998
Tissue specificity of sulfonylureas: studies on cloned cardiac and beta-cell K(ATP) channels.
    Diabetes, 1998, Volume: 47, Issue:9

    Topics: Animals; ATP-Binding Cassette Transporters; Benzamides; Cloning, Molecular; Female; Glyburide; Heart; Hypoglycemic Agents; Islets of Langerhans; Membrane Potentials; Mice; Myocardium; Oocytes; Organ Specificity; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Recombinant Proteins; Sulfonylurea Receptors; Tolbutamide; Xenopus laevis

1998
Sulfonylureas enhance exocytosis from pancreatic beta-cells by a mechanism that does not involve direct activation of protein kinase C.
    Diabetes, 1998, Volume: 47, Issue:11

    Topics: Animals; Calcium; Enzyme Activation; Exocytosis; Glyburide; Guanosine 5'-O-(3-Thiotriphosphate); Hypoglycemic Agents; Insulinoma; Islets of Langerhans; Isoenzymes; Mice; Pancreatic Neoplasms; Phosphatidylserines; Potassium Channels; Protein Kinase C; Sulfonylurea Compounds; Tetradecanoylphorbol Acetate; Tolbutamide; Tumor Cells, Cultured

1998
Reconstituted human cardiac KATP channels: functional identity with the native channels from the sarcolemma of human ventricular cells.
    Circulation research, 1998, Nov-30, Volume: 83, Issue:11

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adolescent; Adult; Animals; ATP-Binding Cassette Transporters; Child; CHO Cells; Cloning, Molecular; COS Cells; Cricetinae; Cromakalim; Diazoxide; DNA, Complementary; Gene Library; Glyburide; Heart Ventricles; Humans; Magnesium; Middle Aged; Myocardium; Patch-Clamp Techniques; Pinacidil; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sarcolemma; Sulfonylurea Receptors; Tolbutamide; Transfection

1998
Effects of sulphonylureas on the volume-sensitive anion channel in rat pancreatic beta-cells.
    British journal of pharmacology, 1998, Volume: 125, Issue:4

    Topics: Animals; Anions; Benzamides; Cells, Cultured; Dose-Response Relationship, Drug; Evoked Potentials; Glyburide; Hypoglycemic Agents; Ion Channels; Ion Transport; Islets of Langerhans; Rats; Sulfonylurea Compounds; Taurine; Tolbutamide

1998
Sodium influx plays a major role in the membrane depolarization induced by oxygen and glucose deprivation in rat striatal spiny neurons.
    Stroke, 1999, Volume: 30, Issue:1

    Topics: Adenosine Triphosphate; Animals; Brain Ischemia; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Chelating Agents; Corpus Striatum; Egtazic Acid; Glucose; Glyburide; Hypoglycemic Agents; Magnesium; Membrane Potentials; Neurons; Organ Culture Techniques; Oxygen; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Receptors, Glutamate; Sodium; Sodium Channel Blockers; Sodium Channels; Tetrodotoxin; Tolbutamide

1999
Sulfonylureas stimulate renin secretion from the perfused kidney of the rat.
    Nephron, 1999, Volume: 81, Issue:1

    Topics: Animals; Blood Pressure; Chlorpropamide; Cyclic AMP; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Kidney; Male; Perfusion; Rats; Rats, Wistar; Renin; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide

1999
Endothelium-dependent blunted membrane potential responses to ATP-sensitive K+ channel modulators in aortae from rats with cirrhosis.
    Journal of hepatology, 1999, Volume: 30, Issue:1

    Topics: Adenosine Triphosphate; Animals; Aorta; Bosentan; Cromakalim; Diazoxide; Endothelin-1; Endothelium, Vascular; Glyburide; Liver Cirrhosis, Experimental; Male; Membrane Potentials; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Sulfonamides; Tolbutamide

1999
JTT-608 controls blood glucose by enhancement of glucose-stimulated insulin secretion in normal and diabetes mellitus rats.
    European journal of pharmacology, 1999, Feb-12, Volume: 367, Issue:1

    Topics: Administration, Oral; Animals; Animals, Newborn; Blood Glucose; Butyrates; Cyclohexanes; Diabetes Mellitus, Experimental; Fasting; Glucose; Glucose Tolerance Test; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Male; Rats; Rats, Sprague-Dawley; Rats, Wistar; Tolbutamide

1999
Characterization of low-affinity binding sites for glibenclamide on the Kir6.2 subunit of the beta-cell KATP channel.
    Biochemical and biophysical research communications, 1999, Apr-21, Volume: 257, Issue:3

    Topics: Animals; ATP-Binding Cassette Transporters; Binding Sites; Blotting, Northern; Cell Line; Cell Membrane; COS Cells; Gliclazide; Glipizide; Glyburide; Islets of Langerhans; Kinetics; Organelles; Phentolamine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Recombinant Fusion Proteins; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide; Transfection

1999
Glucose regulation of insulin secretion independent of the opening or closure of adenosine triphosphate-sensitive K+ channels in beta cells.
    Endocrinology, 1999, Volume: 140, Issue:5

    Topics: Adenosine Triphosphate; Animals; Calcium; Diazoxide; Exocytosis; Female; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Ion Channel Gating; Islets of Langerhans; Mice; Potassium Channels; Sulfonylurea Compounds; Tolbutamide

1999
The stimulatory action of tolbutamide on Ca2+-dependent exocytosis in pancreatic beta cells is mediated by a 65-kDa mdr-like P-glycoprotein.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, May-11, Volume: 96, Issue:10

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Antibodies, Monoclonal; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Calcium; Cells, Cultured; Cytoplasmic Granules; Diabetes Mellitus, Type 2; Drug Resistance, Multiple; Exocytosis; Glyburide; Islets of Langerhans; Mice; Mice, Inbred Strains; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors; Tolbutamide

1999
A role for KATP+-channels in mediating the elevations of cerebral blood flow and arterial pressure by hypoxic stimulation of oxygen-sensitive neurons of rostral ventrolateral medulla.
    Brain research, 1999, May-08, Volume: 827, Issue:1-2

    Topics: Adenosine Triphosphate; Animals; Blood Pressure; Brain Chemistry; Cerebrovascular Circulation; Glyburide; Hypoglycemic Agents; Hypoxia; Hypoxia, Brain; Male; Medulla Oblongata; Neurons; Oxygen; Potassium Channels; Rats; Rats, Sprague-Dawley; Respiratory Center; Tolbutamide

1999
The effect of an insulin releasing agent, BTS 67582, on advanced glycation end product formation in vitro.
    Life sciences, 1999, Volume: 64, Issue:16

    Topics: Ferrous Compounds; Glucose; Glucose-6-Phosphate; Glyburide; Glycation End Products, Advanced; Guanidines; Lysine; Serum Albumin, Bovine; Tolbutamide

1999
Identification of the high-affinity tolbutamide site on the SUR1 subunit of the K(ATP) channel.
    Diabetes, 1999, Volume: 48, Issue:6

    Topics: Adenosine Diphosphate; Amino Acid Substitution; Animals; ATP-Binding Cassette Transporters; Binding Sites; COS Cells; Glyburide; Hypoglycemic Agents; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide; Transfection; Xenopus

1999
Effect of hypoxia on membrane potential and resting conductance in rat hippocampal neurons.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: Adenosine Triphosphate; Animals; Cell Hypoxia; Dantrolene; Dizocilpine Maleate; Electric Conductivity; Glyburide; Hippocampus; Hypoglycemia; In Vitro Techniques; Membrane Potentials; Potassium Chloride; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Time Factors; Tolbutamide

1999
Potentiation of quantal catecholamine secretion by glibenclamide: evidence for a novel role of sulphonylurea receptors in regulating the Ca(2+) sensitivity of exocytosis.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-15, Volume: 19, Issue:14

    Topics: Animals; ATP-Binding Cassette Transporters; Caffeine; Calcium; Catecholamines; Cromakalim; Egtazic Acid; Electrochemistry; Exocytosis; Glyburide; Kinetics; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pinacidil; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quantum Theory; Rats; Receptors, Drug; Sulfonylurea Receptors; Tolbutamide

1999
Alterations of insulin secretion from mouse islets treated with sulphonylureas: perturbations of Ca2+ regulation prevail over changes in insulin content.
    British journal of pharmacology, 1999, Volume: 127, Issue:8

    Topics: Adenosine Triphosphate; Animals; Calcium; Cells, Cultured; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Potassium Channels; Tolbutamide

1999
Different effects of tolbutamide and diazoxide in alpha, beta-, and delta-cells within intact islets of Langerhans.
    Diabetes, 1999, Volume: 48, Issue:12

    Topics: Animals; Boron Compounds; Calcium; Diazoxide; Fluorescent Dyes; Glucose; Glyburide; In Vitro Techniques; Islets of Langerhans; Kinetics; Mice; Mice, Inbred Strains; Potassium Channels; Receptors, Drug; Signal Transduction; Tolbutamide

1999
Involvement of adenosine triphosphate-sensitive K+ channels in glucose-sensing in the rat solitary tract nucleus.
    Neuroscience letters, 2000, Jan-07, Volume: 278, Issue:1-2

    Topics: Adenosine Triphosphate; Animals; Blood Glucose; Diazoxide; Glyburide; Homeostasis; Hypoglycemia; Hypoglycemic Agents; Male; Nerve Tissue Proteins; Neurons; Pinacidil; Potassium Channels; Rats; Rats, Wistar; Solitary Nucleus; Tolbutamide

2000
Pharmacological identification of the K(+) currents mediating the hypoglycemic hyperpolarization of rat midbrain dopaminergic neurones.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: Animals; Barium; Charybdotoxin; Dopamine; Extracellular Space; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Mesencephalon; Neurons; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Strophanthidin; Tolbutamide

2000
Pharmacology of human sulphonylurea receptor SUR1 and inward rectifier K(+) channel Kir6.2 combination expressed in HEK-293 cells.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: ATP-Binding Cassette Transporters; Binding, Competitive; Cations; Cell Line; Deoxyglucose; Diazoxide; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Fluorescence; Gene Expression; Glipizide; Glyburide; Humans; Membrane Potentials; Oligomycins; Potassium Channels; Potassium Channels, Inwardly Rectifying; Radioligand Assay; Receptors, Drug; Recombinant Fusion Proteins; RNA, Messenger; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolazamide; Tolbutamide; Tritium

2000
Inhibitory effects of glibenclamide on the contraction of human arterial conduits used in coronary artery bypass surgery.
    The Journal of pharmacy and pharmacology, 2000, Volume: 52, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Calcium; Coronary Artery Bypass; Dose-Response Relationship, Drug; Glyburide; Humans; In Vitro Techniques; Indomethacin; Mammary Arteries; Phenylephrine; Potassium; Radial Artery; Tolbutamide; Vasoconstriction; Vasoconstrictor Agents

2000
Glibenclamide but not other sulphonylureas stimulates release of neuropeptide Y from perifused rat islets and hamster insulinoma cells.
    The Journal of endocrinology, 2000, Volume: 165, Issue:2

    Topics: Animals; Blotting, Northern; Cricetinae; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Neuropeptide Y; Pancreatic Neoplasms; Perfusion; Radioimmunoassay; Rats; Stimulation, Chemical; Tolbutamide; Tumor Cells, Cultured

2000
Identification of sulfonylureas in serum by electrospray mass spectrometry.
    Analytical biochemistry, 2000, Jun-15, Volume: 282, Issue:1

    Topics: Calibration; Chlorpropamide; Chromatography, Liquid; Glipizide; Glyburide; Humans; Mass Spectrometry; Models, Chemical; Sulfonylurea Compounds; Tolbutamide; Ultraviolet Rays

2000
Sensitivity of Kir6.2-SUR1 currents, in the absence and presence of sodium azide, to the K(ATP) channel inhibitors, ciclazindol and englitazone.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Benzopyrans; Cell Line; Dose-Response Relationship, Drug; Female; Glyburide; Humans; Indoles; Membrane Potentials; Mice; Microinjections; Oocytes; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; RNA, Complementary; Sodium Azide; Sulfonylurea Receptors; Thiazoles; Thiazolidinediones; Tolbutamide; Xenopus laevis

2000
Activation of sulphonylurea-sensitive channels and the NO-cGMP pathway decreases the heart rate response to sympathetic nerve stimulation.
    Cardiovascular research, 2000, Volume: 47, Issue:1

    Topics: Analysis of Variance; Animals; Cyclic GMP; Diazoxide; Electric Stimulation; Enzyme Inhibitors; Glyburide; Guinea Pigs; Heart Atria; Heart Rate; Hypoxia; In Vitro Techniques; Male; Nitric Oxide; Norepinephrine; Potassium Channel Blockers; Potassium Channels; Stellate Ganglion; Sympathetic Nervous System; Tolbutamide

2000
Sulphonylurea drugs reduce hypoxic damage in the isolated perfused rat kidney.
    British journal of pharmacology, 2000, Volume: 130, Issue:7

    Topics: Analysis of Variance; Animals; ATP-Binding Cassette Transporters; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Ischemia; KATP Channels; Kidney; Male; Perfusion; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protective Agents; Rats; Rats, Wistar; Tolbutamide

2000
Sulphonylurea-sensitive channels and NO-cGMP pathway modulate the heart rate response to vagal nerve stimulation in vitro.
    Journal of molecular and cellular cardiology, 2000, Volume: 32, Issue:11

    Topics: Acetylcholine; Animals; Cyclic GMP; Diazoxide; Electric Stimulation; Glyburide; Guinea Pigs; Heart Conduction System; Heart Rate; Ion Transport; Male; Muscle Proteins; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Potassium; Potassium Channels; Signal Transduction; Sulfonylurea Compounds; Tolbutamide; Vagus Nerve

2000
Analysis of single K(ATP) channels in mammalian dentate gyrus granule cells.
    Journal of neurophysiology, 2000, Volume: 84, Issue:5

    Topics: Animals; Antihypertensive Agents; Dentate Gyrus; Diazoxide; Glyburide; Hypoglycemia; Hypoglycemic Agents; Hypoxia; Ion Channel Gating; Kinetics; Male; Mammals; Membrane Potentials; Neurons; Organ Culture Techniques; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tolbutamide

2000
Desensitization of sulphonylurea- and nutrient-induced insulin secretion following prolonged treatment with glibenclamide.
    European journal of pharmacology, 2000, Nov-24, Volume: 408, Issue:3

    Topics: Adenosine Triphosphate; Alanine; Animals; Arginine; Cell Line; Culture Media; Dose-Response Relationship, Drug; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Keto Acids; Potassium Channels; Potassium Chloride; Sulfonylurea Compounds; Tolbutamide

2000
Activation of Na(+), K(+), Cl(-)-cotransport mediates intracellular Ca(2+) increase and apoptosis induced by Pinacidil in HepG2 human hepatoblastoma cells.
    Biochemical and biophysical research communications, 2001, Feb-23, Volume: 281, Issue:2

    Topics: Adenosine Triphosphate; Amiloride; Apoptosis; Bepridil; Bumetanide; Calcium; Carrier Proteins; DNA Fragmentation; Dose-Response Relationship, Drug; Furosemide; Glyburide; Hepatoblastoma; Humans; Pinacidil; Potassium; Potassium Channel Blockers; Potassium Channels; Sodium; Sodium-Calcium Exchanger; Sodium-Potassium-Chloride Symporters; Time Factors; Tolbutamide; Tumor Cells, Cultured

2001
Interaction of sulfonylurea-conjugated polymer with insulinoma cell line of MIN6 and its effect on insulin secretion.
    Journal of biomedical materials research, 2001, Volume: 55, Issue:1

    Topics: Acrylic Resins; Animals; Biocompatible Materials; Culture Media, Conditioned; Diazoxide; Glucose; Glyburide; Insulin; Insulin Secretion; Insulinoma; Kinetics; Magnetic Resonance Spectroscopy; Materials Testing; Molecular Structure; Pancreatic Neoplasms; Povidone; Sulfonylurea Compounds; Tolbutamide; Tumor Cells, Cultured

2001
Sulfonylurea receptors inhibit the epithelial sodium channel (ENaC) by reducing surface expression.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 442, Issue:5

    Topics: Animals; ATP-Binding Cassette Transporters; Cystic Fibrosis Transmembrane Conductance Regulator; Diazoxide; Diuretics; Epithelial Sodium Channels; Glyburide; Hypoglycemic Agents; Oocytes; Patch-Clamp Techniques; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sodium Channel Blockers; Sodium Channels; Sodium Chloride Symporter Inhibitors; Sulfonylurea Receptors; Time Factors; Tolbutamide; Vasodilator Agents; Xenopus laevis

2001
Dibutyryl-cyclic GMP induces peripheral antinociception via activation of ATP-sensitive K(+) channels in the rat PGE2-induced hyperalgesic paw.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: 4-Aminopyridine; Adenosine Triphosphate; Analgesics; Animals; Apamin; Cesium; Charybdotoxin; Dibutyryl Cyclic GMP; Dinoprostone; Dose-Response Relationship, Drug; Glyburide; Hindlimb; Hyperalgesia; Male; Pain; Pain Measurement; Pain Threshold; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide

2001
The effects of mitiglinide (KAD-1229), a new anti-diabetic drug, on ATP-sensitive K+ channels and insulin secretion: comparison with the sulfonylureas and nateglinide.
    European journal of pharmacology, 2001, Nov-09, Volume: 431, Issue:1

    Topics: Animals; ATP-Binding Cassette Transporters; Cell Line; COS Cells; Cyclohexanes; Glyburide; Hypoglycemic Agents; Indoles; Insulin; Isoindoles; Nateglinide; Patch-Clamp Techniques; Phenylalanine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide; Transfection

2001
Novel properties of peptides derived from the sequence coded by exon 26A of human elastin.
    The international journal of biochemistry & cell biology, 2002, Volume: 34, Issue:2

    Topics: 4-Aminopyridine; Animals; Aorta; Dose-Response Relationship, Drug; Elastin; Enzyme Inhibitors; Exons; Glyburide; Humans; Hypoglycemic Agents; In Vitro Techniques; Lactose; Male; Models, Biological; Muscle, Smooth, Vascular; Nitroarginine; Peptides; Phenylephrine; Potassium Channel Blockers; Rats; Rats, Wistar; Tolbutamide; Vasoconstrictor Agents; Virulence Factors, Bordetella

2002
Pharmacological evidence for the activation of K(+) channels by diclofenac.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: 4-Aminopyridine; Analgesics; Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Behavior, Animal; Charybdotoxin; Diclofenac; Dose-Response Relationship, Drug; Female; Formaldehyde; Glyburide; Hindlimb; Morphine; Pain; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide

2002
Involvement of ATP-sensitive K(+) channels in the peripheral antinociceptive effect induced by dipyrone.
    European journal of pharmacology, 2002, May-24, Volume: 444, Issue:1-2

    Topics: Adenosine Triphosphate; Analgesia; Animals; Anti-Inflammatory Agents, Non-Steroidal; Dipyrone; Drug Interactions; Glyburide; Male; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tolbutamide

2002
A novel simple method for the investigation of drug binding to the K(ATP) channel sulfonylurea receptor.
    Analytical biochemistry, 2002, Aug-15, Volume: 307, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Gliclazide; Glyburide; Hypoglycemic Agents; Kinetics; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Rats; Receptors, Drug; Spodoptera; Sulfonylurea Receptors; Tolbutamide

2002
The molecular site of action of K(ATP) channel inhibitors determines their ability to inhibit iNOS-mediated relaxation in rat aorta.
    Cardiovascular research, 2002, Volume: 56, Issue:1

    Topics: 4-Aminopyridine; Adenosine Triphosphate; Aminopyridines; Analysis of Variance; Animals; Aorta; Arginine; Barium; Endothelium, Vascular; Glyburide; Guanidines; Lipopolysaccharides; Male; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitrites; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Tolbutamide; Vasodilator Agents

2002
The peripheral antinociceptive effect of resveratrol is associated with activation of potassium channels.
    Neuropharmacology, 2002, Volume: 43, Issue:5

    Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; ATP-Binding Cassette Transporters; Charybdotoxin; Female; Glipizide; Glyburide; KATP Channels; Morphine; Narcotics; Peripheral Nervous System; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Resveratrol; Stilbenes; Tetraethylammonium; Tolbutamide

2002
The cytoplasmic C-terminus of the sulfonylurea receptor is important for KATP channel function but is not key for complex assembly or trafficking.
    European journal of biochemistry, 2002, Volume: 269, Issue:21

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Biotinylation; Cell Line; Cell Membrane; Cricetinae; Diazoxide; Fluorescent Antibody Technique; Glyburide; Humans; Kidney; Macromolecular Substances; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Protein Structure, Tertiary; Protein Transport; Receptors, Drug; Sequence Deletion; Structure-Activity Relationship; Sulfonylurea Receptors; Tolbutamide

2002
Role of the nitric oxide-cyclic GMP-K+ channel pathway in the antinociception induced by atrial natriuretic peptide (ANP) and diclofenac.
    Proceedings of the Western Pharmacology Society, 2002, Volume: 45

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Atrial Natriuretic Factor; Charybdotoxin; Cyclic GMP; Diclofenac; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Formaldehyde; Glyburide; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Pain Measurement; Potassium Channels; Quinoxalines; Rats; Rats, Wistar; Tolbutamide

2002
Possible involvement of potassium channels in peripheral antinociception induced by metamizol: lack of participation of ATP-sensitive K+ channels.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 74, Issue:2

    Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Area Under Curve; ATP-Binding Cassette Transporters; Charybdotoxin; Dipyrone; Drug Interactions; Female; Formaldehyde; Glyburide; KATP Channels; Pain Measurement; Peripheral Nerves; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide

2003
Dimethyl disulfide exerts insecticidal neurotoxicity through mitochondrial dysfunction and activation of insect K(ATP) channels.
    Journal of neurophysiology, 2003, Volume: 90, Issue:1

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Axons; Coleoptera; Disulfides; Electron Transport Complex IV; Electrophysiology; Fumigation; Glyburide; Insecticides; Male; Mice; Mitochondria; Neurons; Neurotoxins; Patch-Clamp Techniques; Periplaneta; Potassium Channel Blockers; Potassium Channels; Synaptic Transmission; Tolbutamide

2003
Functional coupling between sulfonylurea receptor type 1 and a nonselective cation channel in reactive astrocytes from adult rat brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Sep-17, Volume: 23, Issue:24

    Topics: Adenosine Triphosphate; Animals; Antibodies; Astrocytes; ATP-Binding Cassette Transporters; Binding, Competitive; Brain; Brain Injuries; Cell Size; Cells, Cultured; Diazoxide; Gliosis; Glyburide; Ion Channels; Membrane Potentials; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; Sodium Azide; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide; Trypsin

2003
Sulfonylureas rapidly cross phospholipid bilayer membranes by a free-diffusion mechanism.
    Diabetes, 2003, Volume: 52, Issue:10

    Topics: Albumins; Diffusion; Fluoresceins; Fluorescence; Fluorescent Dyes; Fluorometry; Glyburide; Hydrogen-Ion Concentration; Lipid Bilayers; Magnetic Resonance Spectroscopy; Phospholipids; Sulfonylurea Compounds; Time Factors; Titrimetry; Tolbutamide

2003
Diclofenac-induced peripheral antinociception is associated with ATP-sensitive K+ channels activation.
    Life sciences, 2004, Apr-02, Volume: 74, Issue:20

    Topics: Analgesia; Animals; Anti-Inflammatory Agents, Non-Steroidal; Diclofenac; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Hyperalgesia; Indomethacin; Male; Naloxone; Narcotic Antagonists; Pain Measurement; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tolbutamide

2004
Chronic exposure to tolbutamide and glibenclamide impairs insulin secretion but not transcription of K(ATP) channel components.
    Pharmacological research, 2004, Volume: 50, Issue:1

    Topics: Animals; ATP-Binding Cassette Transporters; Cells, Cultured; Clone Cells; Gene Expression Regulation; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Multidrug Resistance-Associated Proteins; Pancreas; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2004
Study of the involvement of K+ channels in the peripheral antinociception of the kappa-opioid receptor agonist bremazocine.
    European journal of pharmacology, 2004, Jun-28, Volume: 494, Issue:2-3

    Topics: 4-Aminopyridine; Analgesics; Animals; ATP-Binding Cassette Transporters; Benzomorphans; Charybdotoxin; Cyclic GMP; Dequalinium; Glyburide; Hyperalgesia; KATP Channels; Male; Naltrexone; Nitric Oxide; Peripheral Nervous System; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Opioid, kappa; Signal Transduction; Tetraethylammonium; Tolbutamide

2004
Taurine block of cloned ATP-sensitive K+ channels with different sulfonylurea receptor subunits expressed in Xenopus laevis oocytes.
    Biochemical pharmacology, 2004, Sep-01, Volume: 68, Issue:5

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Drug Interactions; Female; Gene Expression; Gliclazide; Glyburide; Hypoglycemic Agents; Membrane Proteins; Mice; Oocytes; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Subunits; Rats; Receptors, Drug; Sulfonylurea Receptors; Taurine; Tolbutamide; Xenopus laevis

2004
Testosterone modulates K(+)ATP channels in Sertoli cell membrane via the PLC-PIP2 pathway.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2004, Volume: 36, Issue:8

    Topics: Adenosine Triphosphate; Androgens; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Electric Impedance; Glyburide; Male; Membrane Potentials; Membrane Proteins; Pertussis Toxin; Phosphatidylinositol 4,5-Diphosphate; Potassium Channels; Rats; Rats, Wistar; Sertoli Cells; Static Electricity; Testosterone; Tolbutamide; Type C Phospholipases

2004
Pharmacological evidence for the activation of Ca2+-activated K+ channels by meloxicam in the formalin test.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:4

    Topics: 4-Aminopyridine; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Apamin; Behavior, Animal; Charybdotoxin; Dose-Response Relationship, Drug; Female; Formaldehyde; Glyburide; Meloxicam; Pain; Pain Measurement; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tetraethylammonium; Thiazines; Thiazoles; Tolbutamide

2005
ATP and sulfonylurea sensitivity of mutant ATP-sensitive K+ channels in neonatal diabetes: implications for pharmacogenomic therapy.
    Diabetes, 2005, Volume: 54, Issue:9

    Topics: Adenosine Triphosphate; Animals; Cell Line; Diabetes Mellitus, Type 1; Glyburide; Humans; Hypoglycemic Agents; Mutation; Pharmacogenetics; Potassium Channels, Inwardly Rectifying; Tolbutamide

2005
Partial mitochondrial inhibition causes striatal dopamine release suppression and medium spiny neuron depolarization via H2O2 elevation, not ATP depletion.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Oct-26, Volume: 25, Issue:43

    Topics: Adenosine Triphosphate; Analysis of Variance; Animals; Catalase; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Fluoresceins; Glyburide; Guinea Pigs; Hydrogen Peroxide; Hypoglycemic Agents; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Rotenone; Sodium Channel Blockers; Tetrodotoxin; Time Factors; Tolbutamide; Uncoupling Agents

2005
Inhibition of 1-methyl-4-phenylpyridinium-induced mitochondrial dysfunction and cell death in PC12 cells by sulfonylurea glibenclamide.
    European journal of pharmacology, 2005, Dec-19, Volume: 527, Issue:1-3

    Topics: 1-Methyl-4-phenylpyridinium; Acetylcysteine; Animals; Apoptosis; Benzoates; Caspase 3; Caspases; Catalase; Cell Nucleus; Cell Survival; Cytochromes c; DNA Fragmentation; Dose-Response Relationship, Drug; Enzyme Activation; Glutathione; Glyburide; Imidazoles; Mitochondrial Membranes; PC12 Cells; Permeability; Porphyrins; Rats; Reactive Oxygen Species; Tolbutamide

2005
KATP channels in mouse spermatogenic cells and sperm, and their role in capacitation.
    Developmental biology, 2006, Jan-15, Volume: 289, Issue:2

    Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Barium; Diazoxide; Dose-Response Relationship, Drug; Glyburide; KATP Channels; Male; Membrane Potentials; Mice; Microscopy, Confocal; Multidrug Resistance-Associated Proteins; Pinacidil; Potassium Channels, Inwardly Rectifying; Receptors, Drug; RNA, Messenger; Sperm Capacitation; Spermatogenesis; Spermatozoa; Sulfonylurea Receptors; Time Factors; Tolbutamide

2006
Probable activation of the opioid receptor-nitric oxide-cyclic GMP-K+ channels pathway by codeine.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 82, Issue:4

    Topics: 4-Aminopyridine; Analgesics, Opioid; Animals; Codeine; Cyclic GMP; Female; Glyburide; Methylene Blue; Naloxone; NG-Nitroarginine Methyl Ester; Nitric Oxide; Potassium Channels; Rats; Rats, Wistar; Receptors, Opioid; Tetraethylammonium; Tolbutamide

2005
Hybrid assemblies of ATP-sensitive K+ channels determine their muscle-type-dependent biophysical and pharmacological properties.
    Proceedings of the National Academy of Sciences of the United States of America, 2006, Jan-24, Volume: 103, Issue:4

    Topics: Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; ATP-Binding Cassette Transporters; Biophysics; Cromakalim; Diazoxide; DNA Primers; Dose-Response Relationship, Drug; Gene Expression Regulation; Glyburide; Hypoglycemic Agents; KATP Channels; Kinetics; Male; Models, Statistical; Muscle Fibers, Skeletal; Muscle, Skeletal; Muscles; Patch-Clamp Techniques; Phenotype; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Drug; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; Sulfonylurea Receptors; Tolbutamide

2006
Possible activation of the NO-cyclic GMP-protein kinase G-K+ channels pathway by gabapentin on the formalin test.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 83, Issue:3

    Topics: 4-Aminopyridine; Amines; Analgesics; Animals; Apamin; Carbazoles; Charybdotoxin; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Cyclohexanecarboxylic Acids; Female; Gabapentin; gamma-Aminobutyric Acid; Glyburide; Indoles; Naloxone; NG-Nitroarginine Methyl Ester; Nitric Oxide; Pain Measurement; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tolbutamide

2006
Switching from insulin to oral sulfonylureas in patients with diabetes due to Kir6.2 mutations.
    The New England journal of medicine, 2006, Aug-03, Volume: 355, Issue:5

    Topics: ATP-Binding Cassette Transporters; Cohort Studies; Diabetes Mellitus; Female; Glyburide; Glycated Hemoglobin; Heterozygote; Humans; Hypoglycemic Agents; Infant; Infant, Newborn; Insulin; Insulin-Secreting Cells; Male; Mutation; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2006
First phase of glucose-stimulated insulin secretion from MIN 6 cells does not always require extracellular calcium influx.
    Journal of pharmacological sciences, 2006, Volume: 101, Issue:4

    Topics: Animals; Calcium; Calcium Isotopes; Cell Line, Tumor; Cell Survival; Dantrolene; Diazoxide; Dose-Response Relationship, Drug; Extracellular Fluid; Glucose; Glyburide; Insulin; Insulin Antagonists; Insulin Secretion; Insulin-Secreting Cells; L-Lactate Dehydrogenase; Male; Mice; Potassium Channels; Sodium Channels; Tetrodotoxin; Tolbutamide; Verapamil

2006
Peripheral antinociceptive effect of pertussis toxin: activation of the arginine/NO/cGMP/PKG/ ATP-sensitive K channel pathway.
    The European journal of neuroscience, 2006, Volume: 24, Issue:4

    Topics: Adenosine Triphosphate; Analgesia; Analgesics; Animals; Arginine; Bucladesine; Carbazoles; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dinoprostone; Enzyme Inhibitors; Ganglia, Spinal; Glyburide; Indoles; KATP Channels; Male; Neurons; Nitric Oxide; omega-N-Methylarginine; Oxadiazoles; Pain; Pain Measurement; Pertussis Toxin; Potassium Channels, Inwardly Rectifying; Quinoxalines; Rats; Rats, Wistar; Signal Transduction; Tolbutamide

2006
Baclofen, an agonist at peripheral GABAB receptors, induces antinociception via activation of TEA-sensitive potassium channels.
    British journal of pharmacology, 2006, Volume: 149, Issue:6

    Topics: Analgesics; Animals; Baclofen; Bicuculline; Cesium; Charybdotoxin; Dequalinium; GABA Agonists; GABA-B Receptor Agonists; Glyburide; Male; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide

2006
Investigation of the effects of sulfonylurea exposure on pancreatic beta cell metabolism.
    The FEBS journal, 2006, Volume: 273, Issue:22

    Topics: Animals; Carbon Radioisotopes; Cells, Cultured; Glucose; Glyburide; Hypoglycemic Agents; Insulin-Secreting Cells; Magnetic Resonance Spectroscopy; Models, Biological; Rats; Sulfonylurea Compounds; Tolbutamide

2006
Transgenic expression of a dominant negative K(ATP) channel subunit in the mouse endothelium: effects on coronary flow and endothelin-1 secretion.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2007, Volume: 21, Issue:9

    Topics: Adenosine Triphosphate; Animals; Bradykinin; Coronary Circulation; Diazoxide; Electrocardiography; Endothelin-1; Endothelium, Vascular; Ergonovine; Exocytosis; Gene Expression Regulation; Genes, Synthetic; Glyburide; KATP Channels; Mice; Mice, Transgenic; Point Mutation; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Pressure; Rats; Rats, Sprague-Dawley; Tolbutamide; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2007
Regulation by glucose of oscillatory electrical activity and 5-HT/insulin release from single mouse pancreatic islets in absence of functional K(ATP) channels.
    Endocrine journal, 2008, Volume: 55, Issue:4

    Topics: Adenosine Triphosphate; Animals; Calcium; Cells, Cultured; Glucose; Glyburide; Insulin; Insulin Secretion; Insulin-Secreting Cells; Keto Acids; Membrane Potentials; Mice; Patch-Clamp Techniques; Potassium Channels; Serotonin; Tolbutamide

2008
The cAMP sensor Epac2 is a direct target of antidiabetic sulfonylurea drugs.
    Science (New York, N.Y.), 2009, Jul-31, Volume: 325, Issue:5940

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Blood Glucose; Carrier Proteins; Cell Line; Chlorocebus aethiops; COS Cells; Cyclic AMP; Fluorescence Resonance Energy Transfer; Glucose; Glyburide; Guanine Nucleotide Exchange Factors; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred C57BL; rap1 GTP-Binding Proteins; Sulfonylurea Compounds; Tolbutamide

2009
Adenosine inhibits paraventricular pre-sympathetic neurons through ATP-dependent potassium channels.
    Journal of neurochemistry, 2010, Volume: 113, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adenosine; Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glyburide; Guanosine Diphosphate; In Vitro Techniques; KATP Channels; Male; Membrane Potentials; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Sodium Channel Blockers; Tetrodotoxin; Thionucleotides; Tolbutamide; Triazines; Triazoles; Xanthines

2010
Effects of K openers on the QT prolongation induced by HERG-blocking drugs in guinea-pigs.
    The Journal of pharmacy and pharmacology, 2010, Volume: 62, Issue:7

    Topics: Animals; Benzothiadiazines; Cromakalim; Decanoic Acids; Ether-A-Go-Go Potassium Channels; Glyburide; Guinea Pigs; Heart; Humans; Hydroxy Acids; Intracellular Membranes; KATP Channels; Long QT Syndrome; Male; Membrane Transport Modulators; Mitochondrial Membranes; Picolines; Pinacidil; Potassium Channel Blockers; Pyrans; Sarcolemma; Tolbutamide

2010
Effects of metformin on BRIN-BD11 beta-cell insulin secretory desensitization induced by prolonged exposure to sulphonylureas.
    Diabetes, obesity & metabolism, 2010, Volume: 12, Issue:12

    Topics: Cell Line; Culture Media; Glyburide; Humans; Insulin-Secreting Cells; Metformin; Sulfonylurea Compounds; Tolbutamide

2010
Exchange protein directly activated by cyclic AMP isoform 2 is not a direct target of sulfonylurea drugs.
    Assay and drug development technologies, 2011, Volume: 9, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Blood Glucose; Carrier Proteins; Cell Line; Chlorocebus aethiops; COS Cells; Cyclic AMP; Fluorescence Resonance Energy Transfer; Glucose; Glyburide; Guanine Nucleotide Exchange Factors; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred C57BL; rap1 GTP-Binding Proteins; Sulfonylurea Compounds; Tolbutamide

2011
Comparable long-term mortality risk associated with individual sulfonylureas in diabetes patients with heart failure.
    Diabetes research and clinical practice, 2011, Volume: 94, Issue:1

    Topics: Aged; Aged, 80 and over; Diabetes Mellitus; Female; Glipizide; Glyburide; Heart Failure; Humans; Hypoglycemic Agents; Male; Sulfonylurea Compounds; Tolbutamide

2011
Expression and functional properties of TRPM2 channels in dopaminergic neurons of the substantia nigra of the rat.
    Journal of neurophysiology, 2011, Volume: 106, Issue:6

    Topics: Adenosine Diphosphate Ribose; Adenosine Triphosphate; Animals; Biophysics; Calcium; Clusterin; Dopaminergic Neurons; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Glyburide; Hydrogen Peroxide; In Vitro Techniques; Isoquinolines; Membrane Potentials; Oxidants; Patch-Clamp Techniques; Piperidines; Potassium Channel Blockers; Rats; Reactive Oxygen Species; RNA, Messenger; Substantia Nigra; Tetraethylammonium; Tolbutamide; Tyrosine 3-Monooxygenase

2011
Structural nucleotide analogs are potent activators/inhibitors of pancreatic β cell KATP channels: an emerging mechanism supporting their use as antidiabetic drugs.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:2

    Topics: Animals; Area Under Curve; Benzoxazines; Blood Glucose; Dose-Response Relationship, Drug; Electrophysiological Phenomena; Fasting; Glucose; Glucose Tolerance Test; Glyburide; HEK293 Cells; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; KATP Channels; Membrane Potentials; Mice; Mice, Inbred Strains; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Sodium Azide; Tolbutamide

2012
Protein phosphorylation involved in the gene expression of the hydrogen sulphide producing enzyme cystathionine γ-lyase in the pancreatic β-cell.
    Molecular and cellular endocrinology, 2012, Mar-05, Volume: 350, Issue:1

    Topics: Animals; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Cells, Cultured; Cystathionine beta-Synthase; Cystathionine gamma-Lyase; ets-Domain Protein Elk-1; Gene Expression; Gene Expression Regulation; Glucose; Glyburide; Hydrogen Sulfide; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; Male; Mice; Mice, Inbred ICR; Mitogen-Activated Protein Kinases; Phosphorylation; Promoter Regions, Genetic; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Sp1 Transcription Factor; Thapsigargin; Tolbutamide

2012
Differential contribution of TM6 and TM12 to the pore of CFTR identified by three sulfonylurea-based blockers.
    Pflugers Archiv : European journal of physiology, 2012, Volume: 463, Issue:3

    Topics: Alanine; Amino Acid Sequence; Animals; Benzamides; Cystic Fibrosis Transmembrane Conductance Regulator; Glipizide; Glyburide; Ion Channel Gating; Kinetics; Mutagenesis; Oocytes; Patch-Clamp Techniques; Sulfonylurea Compounds; Tolbutamide; Xenopus

2012
Pharmacogenomic analysis of ATP-sensitive potassium channels coexpressing the common type 2 diabetes risk variants E23K and S1369A.
    Pharmacogenetics and genomics, 2012, Volume: 22, Issue:3

    Topics: ATP-Binding Cassette Transporters; Chlorpropamide; Cyclohexanes; Diabetes Mellitus, Type 2; Gene Expression Regulation; Gliclazide; Glyburide; Haplotypes; Homozygote; Humans; Isoindoles; Nateglinide; Patch-Clamp Techniques; Phenylalanine; Polymorphism, Single Nucleotide; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Structure-Activity Relationship; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2012
Synthesis, antidiabetic and hypolipidemic activities of new diethylamine and triethoxysilyl derivatives of tolbutamide on rats.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2012, Volume: 8, Issue:5

    Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Diethylamines; Glyburide; Hypoglycemic Agents; Lipoproteins, VLDL; Male; Rats; Rats, Wistar; Silanes; Streptozocin; Tolbutamide; Triglycerides

2012
Activation of glibenclamide-sensitive ATP-sensitive K+ channels during β-adrenergically induced metabolic stress produces a substrate for atrial tachyarrhythmia.
    Circulation. Arrhythmia and electrophysiology, 2012, Volume: 5, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Disease Models, Animal; Electrophysiologic Techniques, Cardiac; Glyburide; Heart Atria; Heart Conduction System; Isoproterenol; KATP Channels; Male; Potassium Channel Blockers; Rats; Stress, Physiological; Tachycardia; Time Factors; Tolbutamide

2012
Mortality outcomes of different sulphonylurea drugs: the results of a 14-year cohort study of type 2 diabetic patients.
    European journal of endocrinology, 2013, Volume: 169, Issue:1

    Topics: Adult; Aged; Cardiovascular Diseases; Cause of Death; Cohort Studies; Confounding Factors, Epidemiologic; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Kaplan-Meier Estimate; Male; Metformin; Middle Aged; Neoplasms; Odds Ratio; Proportional Hazards Models; Research Design; Retrospective Studies; Risk Assessment; Risk Factors; Sulfonylurea Compounds; Tolbutamide

2013
Mechanosynthesis of pharmaceutically relevant sulfonyl-(thio)ureas.
    Chemical communications (Cambridge, England), 2014, May-25, Volume: 50, Issue:40

    Topics: Catalysis; Chlorpropamide; Copper; Glyburide; Hypoglycemic Agents; Isothiocyanates; Molecular Structure; Sulfonamides; Tolbutamide

2014
Effect of tolbutamide, glyburide and glipizide administered supraspinally on CA3 hippocampal neuronal cell death and hyperglycemia induced by kainic acid in mice.
    Brain research, 2014, May-20, Volume: 1564

    Topics: Animals; Blood Glucose; CA3 Region, Hippocampal; Cell Death; Glipizide; Glyburide; Hyperglycemia; Hypoglycemic Agents; Infusions, Intraventricular; Kainic Acid; Male; Mice; Mice, Inbred ICR; Neurons; Sulfonylurea Compounds; Tolbutamide

2014
Metformin in combination with various insulin secretagogues in type 2 diabetes and associated risk of cardiovascular morbidity and mortality--a retrospective nationwide study.
    Diabetes research and clinical practice, 2015, Volume: 107, Issue:1

    Topics: Aged; Carbamates; Cardiovascular Diseases; Denmark; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Morbidity; Myocardial Infarction; Piperidines; Registries; Retrospective Studies; Risk Factors; Stroke; Sulfonylurea Compounds; Tolbutamide

2015
Evidence for a KATP Channel in Rough Endoplasmic Reticulum (rerKATP Channel) of Rat Hepatocytes.
    PloS one, 2015, Volume: 10, Issue:5

    Topics: Adenosine Triphosphate; Animals; Calcium; Cells, Cultured; Charybdotoxin; Endoplasmic Reticulum, Rough; Glyburide; Hepatocytes; KATP Channels; Male; Membrane Potentials; Peptides; Rats; Tolbutamide

2015
Sulphonylurea receptor-1, sulphonylureas and amplification of insulin secretion by Epac activation in β cells.
    Diabetes, obesity & metabolism, 2016, Volume: 18, Issue:7

    Topics: Acetylcysteine; Animals; Bucladesine; Cyclic AMP-Dependent Protein Kinases; Erythromycin; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mice, Inbred C57BL; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2016
On-Line two dimensional liquid chromatography based on skeleton type molecularly imprinted column for selective determination of sulfonylurea additive in Chinese patent medicines or functional foods.
    Journal of pharmaceutical and biomedical analysis, 2017, Nov-30, Volume: 146

    Topics: Chromatography, Liquid; Counterfeit Drugs; Dietary Supplements; Drugs, Chinese Herbal; Functional Food; Glyburide; Hypoglycemic Agents; Medicine, Chinese Traditional; Nonprescription Drugs; Online Systems; Sulfonylurea Compounds; Tolbutamide

2017
β-Cell-intrinsic β-arrestin 1 signaling enhances sulfonylurea-induced insulin secretion.
    The Journal of clinical investigation, 2019, 06-11, Volume: 129, Issue:9

    Topics: Animals; beta-Arrestin 1; beta-Arrestin 2; Genotype; Glyburide; Guanine Nucleotide Exchange Factors; Hypoglycemic Agents; Insulin Secretion; Insulin-Secreting Cells; Male; Mice; Mice, Knockout; Mice, Transgenic; Phenotype; Signal Transduction; Sulfonylurea Compounds; Tolbutamide

2019
Analysis of Hypoglycemic Drugs by Liquid Chromatography-Tandem Mass Spectrometry.
    Methods in molecular biology (Clifton, N.J.), 2024, Volume: 2737

    Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Chromatography, Liquid; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Nateglinide; Pioglitazone; Rosiglitazone; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Tolazamide; Tolbutamide

2024