glyburide and quinine

glyburide has been researched along with quinine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19904 (11.11)18.7374
1990's8 (22.22)18.2507
2000's13 (36.11)29.6817
2010's11 (30.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Abe, T; Itoh, T; Kato, Y; Kusuhara, H; Meier, PJ; Shitara, Y; Sugiyama, D; Sugiyama, Y1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN1
Bedoya, M; Decher, N; González, W; Kiper, AK; Ramírez, D; Rinné, S1
Rahav, G; Shalev, O; Tsur, A1
Baeyens, JM; Barrios, M; Del Pozo, E; Ocaña, M; Robles, LI1
Rosario, LM1
Castle, NA; Haylett, DG1
Herchuelz, A; Lebrun, P; Malaisse, WJ1
Atwater, I; Rojas, E; Rosario, LM1
Devor, DC; Frizzell, RA1
Atwater, I; Carroll, PB; Moura, AS; Rojas, E1
Belyaeva, EA; Wojtczak, L1
Borowitz, JL; Isom, GE; Kanthasamy, A; Latha, MV; Yim, GK1
Boutellier, S; Lutz, TA; Rossi, R; Scharrer, E; Seebacher, MC; Sutter, DA1
Rao, VS; Santos, FA1
Huang, DY; Osswald, H; Vallon, V1
Furuichi, K; Inamura, K; Kitada, C; Matsushime, H; Miyake, A; Mochizuki, S; Nozawa, K; Okada, H; Sano, Y; Yokoi, H1
Anapolski, M; Barfield, JP; Cooper, TG; Yeung, CH1
Faggio, C; Trischitta, F1
Espinosa-Garcia, MT; Flores-Herrera, O; Martinez, F; Milan, R; Olvera-Sanchez, S1
Nishimura-Danjobara, Y; Oyama, K; Oyama, Y; Yokoigawa, K1

Reviews

3 review(s) available for glyburide and quinine

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
TASK Channels Pharmacology: New Challenges in Drug Design.
    Journal of medicinal chemistry, 2019, 11-27, Volume: 62, Issue:22

    Topics: Animals; Drug Design; Drug Discovery; Humans; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Tandem Pore Domain

2019

Other Studies

33 other study(ies) available for glyburide and quinine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Comparative inhibitory effects of different compounds on rat oatpl (slc21a1)- and Oatp2 (Slc21a5)-mediated transport.
    Pharmaceutical research, 2002, Volume: 19, Issue:2

    Topics: Algorithms; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antibiotics, Antitubercular; Antimalarials; Biological Transport, Active; Digoxin; Enzyme Inhibitors; Estradiol; Ibuprofen; LLC-PK1 Cells; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Organic Cation Transport Proteins; Quinidine; Quinine; Rats; Rifampin; Swine

2002
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
    Chemical biology & drug design, 2016, Volume: 88, Issue:6

    Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain

2016
Falciparum malaria-induced hypoglycaemia in a diabetic patient.
    Postgraduate medical journal, 1992, Volume: 68, Issue:798

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Glucose Solution, Hypertonic; Glyburide; Humans; Hypoglycemia; Malaria, Falciparum; Male; Middle Aged; Quinine

1992
An ATP-dependent potassium channel blocker antagonizes morphine analgesia.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: Adenosine Triphosphate; Analgesia; Animals; Female; Glyburide; Injections, Intraventricular; Mice; Morphine; Pain Measurement; Potassium Channels; Quinine; Tetraethylammonium; Tetraethylammonium Compounds

1990
Electrophysiological measurements show marked differences in the properties of the pancreatic beta-cell K-channels from albino mice and a strain of ob/ob (obese) mice.
    Advances in experimental medicine and biology, 1986, Volume: 211

    Topics: Animals; Glucose; Glyburide; In Vitro Techniques; Ion Channels; Islets of Langerhans; Membrane Potentials; Mice; Mice, Obese; Potassium; Quinine; Species Specificity; Tolbutamide

1986
Effect of channel blockers on potassium efflux from metabolically exhausted frog skeletal muscle.
    The Journal of physiology, 1987, Volume: 383

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Apamin; Barium; Cell Membrane Permeability; Decamethonium Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Glyburide; In Vitro Techniques; Ion Channels; Muscles; Potassium; Quinine; Rana temporaria; Rubidium; Scorpion Venoms; Tetraethylammonium Compounds; Tolbutamide

1987
Do hypoglycemic sulfonylureas inhibit Na+,K+-ATPase activity in pancreatic islets?
    The American journal of physiology, 1985, Volume: 248, Issue:5 Pt 1

    Topics: Animals; Calcimycin; Calcium; Cell Membrane Permeability; Drug Synergism; Glucose; Glyburide; Insulin; Ion Channels; Islets of Langerhans; Ouabain; Potassium; Quinine; Rats; Rubidium; Sodium-Potassium-Exchanging ATPase; Tolbutamide

1985
Membrane potential measurements in islets of Langerhans from ob/ob obese mice suggest an alteration in [Ca2+]i-activated K+ permeability.
    Quarterly journal of experimental physiology (Cambridge, England), 1985, Volume: 70, Issue:1

    Topics: Animals; Calcium; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cell Membrane Permeability; Glucose; Glyburide; Intracellular Membranes; Islets of Langerhans; Membrane Potentials; Mice; Mice, Obese; Potassium; Quinine; Reference Values

1985
Calcium-mediated agonists activate an inwardly rectified K+ channel in colonic secretory cells.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 1

    Topics: 4-Aminopyridine; Animals; Apamin; Barium; Calcium; Cell Line; Charybdotoxin; Colon; Cytosol; Glyburide; Hydrogen-Ion Concentration; Kinetics; Membrane Potentials; Potassium Channels; Quinine; Scorpion Venoms; Sodium; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors

1993
The diabetogenic agent alloxan increases K+ permeability by a mechanism involving activation of ATP-sensitive K(+)-channels in mouse pancreatic beta-cells.
    Molecular and cellular biochemistry, 1994, Nov-23, Volume: 140, Issue:2

    Topics: Alloxan; Animals; Electric Conductivity; Electrophysiology; Evoked Potentials; Female; Glucose; Glyburide; In Vitro Techniques; Islets of Langerhans; Kinetics; Membrane Potentials; Mice; Potassium Channel Blockers; Potassium Channels; Quinine; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors

1994
An attempt to quantify K+ fluxes in rat liver mitochondria.
    Biochemistry and molecular biology international, 1994, Volume: 33, Issue:1

    Topics: Animals; Calcimycin; Glyburide; In Vitro Techniques; Kinetics; Magnesium; Male; Membrane Potentials; Mitochondria, Liver; Potassium; Potassium Channels; Quinine; Rats; Rats, Wistar

1994
Plasma membrane hyperpolarization by cyanide in chromaffin cells: role of potassium channels.
    Archives of toxicology, 1994, Volume: 68, Issue:6

    Topics: Animals; Calcium; Chromaffin System; Glyburide; Membrane Potentials; Neurons; PC12 Cells; Potassium Channels; Potassium Chloride; Quinine; Rats; Sodium Cyanide

1994
Hyperpolarization of hepatocytes by 2,5-AM: implications for hepatic control of food intake.
    The American journal of physiology, 1997, Volume: 272, Issue:3 Pt 2

    Topics: Amiloride; Animals; Apamin; Appetite; Azepines; Barium; Bicarbonates; Chlorides; Female; Flufenamic Acid; Glyburide; Homeostasis; In Vitro Techniques; Liver; Male; Mannitol; Membrane Potentials; Mice; Mice, Inbred ICR; Ouabain; Potassium Channel Blockers; Potassium Channels; Quinine; Rats; Rats, Sprague-Dawley; Sodium

1997
Quinine-induced inhibition of gastrointestinal transit in mice: possible involvement of endogenous opioids.
    European journal of pharmacology, 1999, Jan-08, Volume: 364, Issue:2-3

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Gastrointestinal Transit; Glyburide; Male; Mice; Minoxidil; Morphine; Naloxone; Narcotic Antagonists; Opioid Peptides; Potassium Channels; Quinine; Yohimbine

1999
Sodium reabsorption in thick ascending limb of Henle's loop: effect of potassium channel blockade in vivo.
    British journal of pharmacology, 2000, Volume: 130, Issue:6

    Topics: Adamantane; Animals; Barium; Cesium; Charybdotoxin; Dose-Response Relationship, Drug; Glyburide; Loop of Henle; Male; Models, Biological; Morpholines; Potassium; Potassium Channel Blockers; Potassium Channels; Quinine; Rats; Rats, Wistar; Sodium; Verapamil

2000
A novel two-pore domain K+ channel, TRESK, is localized in the spinal cord.
    The Journal of biological chemistry, 2003, Jul-25, Volume: 278, Issue:30

    Topics: Amino Acid Sequence; Analgesics, Non-Narcotic; Animals; Anti-Arrhythmia Agents; Arachidonic Acid; Barium; Cell Line; Cloning, Molecular; Docosahexaenoic Acids; Electrophysiology; Ethanolamines; Fatty Acids; Fatty Acids, Nonesterified; Glyburide; Humans; Hydrogen-Ion Concentration; Lidocaine; Mice; Models, Biological; Molecular Sequence Data; Patch-Clamp Techniques; Phylogeny; Potassium Channels; Propafenone; Protein Structure, Tertiary; Quinidine; Quinine; Reverse Transcriptase Polymerase Chain Reaction; Spinal Cord; Tissue Distribution; Transfection

2003
Volume regulation of mature and immature spermatozoa in a primate model, and possible ion channels involved.
    Human reproduction (Oxford, England), 2004, Volume: 19, Issue:11

    Topics: 4-Aminopyridine; Animals; Apamin; Cell Size; Cells, Cultured; Charybdotoxin; Ejaculation; Epididymis; Glyburide; Ion Channels; Macaca fascicularis; Male; Neurotoxins; Nitrobenzoates; Potassium Channel Blockers; Quaternary Ammonium Compounds; Quinine; Scorpion Venoms; Spermatozoa; Tetraethylammonium

2004
Gossypol affects ion transport in the isolated intestine of the seawater adapted eel, Anguilla anguilla.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2008, Volume: 151, Issue:1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Adaptation, Physiological; Anguilla; Animals; Buffers; Calcium; Electric Conductivity; Epithelial Cells; Glyburide; Gossypol; In Vitro Techniques; Intestines; Ion Channel Gating; Ion Transport; Mucous Membrane; Nitrobenzoates; Perfusion; Quinine; Seawater; Serous Membrane

2008
Contribution of potassium in human placental steroidogenesis.
    Placenta, 2010, Volume: 31, Issue:10

    Topics: Blotting, Western; Cholesterol; Female; Glyburide; Humans; Ionophores; KATP Channels; Membrane Potential, Mitochondrial; Mitochondria; Placenta; Potassium; Pregnancy; Progesterone; Quinine; Valinomycin

2010
Hyperpolarization by N-(3-oxododecanoyl)-l-homoserine-lactone, a quorum sensing molecule, in rat thymic lymphocytes.
    Chemico-biological interactions, 2018, Mar-01, Volume: 283

    Topics: 4-Butyrolactone; Animals; Calcium; Cell Polarity; Charybdotoxin; Flow Cytometry; Glyburide; Homoserine; KATP Channels; Lymphocytes; Permeability; Potassium; Potassium Channels, Voltage-Gated; Quinine; Quorum Sensing; Rats; Rats, Wistar; Thymocytes

2018