glyburide and nifedipine

glyburide has been researched along with nifedipine in 87 studies

Research

Studies (87)

TimeframeStudies, this research(%)All Research%
pre-19901 (1.15)18.7374
1990's39 (44.83)18.2507
2000's19 (21.84)29.6817
2010's23 (26.44)24.3611
2020's5 (5.75)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Sen, S; Sinha, N1
Barber, J; Dawson, S; Kenna, JG; Paul, N; Stahl, S1
Caradonna, NP; Hallifax, D; Houston, JB; Turlizzi, E; Zanelli, U1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Aleo, MD; Bonin, PD; Luo, Y; Potter, DM; Swiss, R; Will, Y1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF1
Chang, G; Mathialagan, S; Ryu, S; Varma, MVS; Woody, N1
Fukata, Y; Fukushima, H; Jinno, Y; Kaneta, S; Nishikori, K; Ogawa, N1
Karim, OM; Mostwin, JL; Seki, N1
Aiyar, N; Gleason, MM; Griffin, EC; Nambi, P1
Brown, TJ; Raeburn, D1
Asano, M; Masuzawa, K; Matsuda, T1
McHarg, AD; Southerton, JS; Weston, AH1
Abu-Jayyab, AR; al-Bekairi, AM; el-Denshary, ES; el-Sawaf, HA1
Satoh, E; Taira, N; Yanagisawa, T1
Wilson, C1
Mizusawa, H; Omote, M2
Hiramatsu, T; Kotlikoff, MI; Kume, H; Takagi, K1
Maggi, CA; Meini, S; Santicioli, P1
Fukushima, H; Jinno, Y; Kaneta, S; Miwa, A; Ogawa, N1
Boev, KK; Duridanova, DB; Gagov, HS1
Ginkawa, M; Kontani, H; Sakai, T1
Kam, KL; Pfaffendorf, M; van Zwieten, PA2
Gonzalez de la Fuente, P; Marthan, R; Savineau, JP1
Kojima, I; Miyazaki, J; Mogami, H; Nobusawa, R; Ohnota, H; Satou, F; Shibata, H1
Izawa, T; Jinno, Y; Miwa, A; Ogawa, N; Yokoyama, T1
Cahill, AL; Perlman, RL1
Aizawa, T; Hashizume, K; Ishihara, F; Komatsu, M; Nishii, N; Sato, Y; Suzuki, N; Yamada, T1
Jinkawa, M; Kontani, H; Sakai, T1
McMurtry, IF; Morris, KG; Oka, M1
Freed, AN; Lindeman, KS1
Ko, FN; Lin, CH; Lu, ST; Teng, CM; Wu, YC1
Arvola, P; Kähönen, M; Mäkynen, H; Pörsti, I; Wu, X1
Angus, JA; Fujiwara, T1
Kume, H; Mikawa, K; Takagi, K1
Fukunari, A; Kawahara, K; Miyai, H; Nakajima, T; Shinagawa, K1
Buus, C; Mulvany, MJ; Nilsson, H; Prieto, D1
Högemann, A; Jonkman, JH; Lins, R; Sennewald, R; van Heiningen, PN; van Lier, JJ1
Houchi, H; Nakaya, Y; Oka, M; Shono, M1
Bouskela, E; Conde, CM; Cyrino, FZ; Garcia, AA1
Brading, AF; Teramoto, N1
Benes, C; Creuzet, C; Fagard, R; Miyazaki, J; Roisin, MP; Van Tan, H1
Brennecke, SP; Coleman, HA; Davies, NK; Parkington, HC; Tonta, MA1
Araki, E; Kaneko, K; Kishikawa, H; Motoshima, H; Motoyoshi, S; Sakai, K; Shichiri, M; Shirakami, A; Shirotani, T; Yoshizato, K1
Kang, SY; Kim, MJ; Kim, ND; Park, JH; Schini-Kerth, VB1
Inoue, Y; Kondo, A; Li, JW; Miyazaki, M; Namba, M; Pu, H1
Golledge, J; Gosling, M; Powell, JT; Standfield, NJ; Turner, RJ1
Miller, DV; Paterson, WG; Zhang, Y1
Ikawa, S; Ito, Y; Naito, S; Seki, N; Takano, N; Tanaka, K; Teramoto, N; Yunoki, T1
Chang, IY; Choi, S; Jun, JY; Kim, KW; Kim, MJ; Kim, MY; Kong, ID; Lee, KP; Park, CK; So, I; Yeum, CH; You, HJ1
Kito, Y; Sanders, KM; Ward, SM1
Kwon, G; Liu, H; Marshall, CA; McDaniel, ML; Pappan, KL; Remedi, MS1
Mishra, SK; Prakash, VR; Ross, GR; Sathishkumar, K1
Dkhar, SA; Krishna, PR; Ramaswamy, S; Sandhiya, S1
Basak, F; Cehreli, SB; Cehreli, ZC; Guven, G; Kaya, E; Seyrek, M; Ulku, C; Vural, IM; Yildiz, O1
Fan, CL; Huang, Y; Lau, CW; Li, Y; Lin, SM; Wang, J; Ye, WC; Yiu, A; Zhang, DM1
Chuan, P; Lluch, S; Mauricio, MD; Medina, P; Segarra, G; Vila, JM1
Cehreli, ZC; Guven, G; Seyrek, M; Vural, IM; Yildiz, O1
Matsumoto, A; Miki, T; Nakaya, H; Nishida, A; Seino, S; Takizawa, T1
Buttigieg, J; Livermore, S; Nurse, CA; Piskuric, NA; Zhang, M1
Khaertdinov, NN; Sitdikova, GF; Zefirov, AL1
Choi, DS; Chokshi, H; Hu, Q; Sandhu, H; Shah, N1
Holstein-Rathlou, NH; Jensen, LJ; Ngo, AT; Riemann, M; Torp-Pedersen, C1
Ghasemi, A; Godini, A; Zahediasl, S1
Hoshmandi, E; Karbalaei, N; Noorafshan, A1
Jiang, Y; Peng, C; Tao, X; Wang, LP; Xie, HH; Yang, H; Zhang, C1
Carbonell-Barrachina, ÁA; Gur, S; Kaya-Sezginer, E; Onder, A; Oztekin, CV; Yilmaz-Oral, D; Zor, M1
Ajebli, M; Amssayef, A; Eddouks, M1
Berezina, TP; Evlakhov, VI; Poyasov, IZ1

Reviews

2 review(s) available for glyburide and nifedipine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells

2022

Trials

1 trial(s) available for glyburide and nifedipine

ArticleYear
Pharmacokinetic drug interaction studies with candesartan cilexetil.
    Journal of human hypertension, 1997, Volume: 11 Suppl 2

    Topics: Adolescent; Adult; Angiotensin Receptor Antagonists; Antihypertensive Agents; Benzimidazoles; Biphenyl Compounds; Digoxin; Drug Interactions; Female; Glyburide; Humans; Hydrochlorothiazide; Male; Middle Aged; Nifedipine; Tetrazoles; Warfarin

1997

Other Studies

84 other study(ies) available for glyburide and nifedipine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Cholestasis; Drug-Related Side Effects and Adverse Reactions; Humans; Insecta; Rats; Risk Factors

2012
Comparison of cryopreserved HepaRG cells with cryopreserved human hepatocytes for prediction of clearance for 26 drugs.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:1

    Topics: Cell Line, Tumor; Cryopreservation; Female; Hepatocytes; Humans; Male; Metabolic Clearance Rate; Pharmaceutical Preparations; Predictive Value of Tests

2012
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Human drug-induced liver injury severity is highly associated with dual inhibition of liver mitochondrial function and bile salt export pump.
    Hepatology (Baltimore, Md.), 2014, Volume: 60, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Chemical and Drug Induced Liver Injury; Humans; Male; Mitochondria, Liver; Rats; Rats, Sprague-Dawley; Severity of Illness Index

2014
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
    Chemical biology & drug design, 2016, Volume: 88, Issue:6

    Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain

2016
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Identification of Organic Anion Transporter 2 Inhibitors: Screening, Structure-Based Analysis, and Clinical Drug Interaction Risk Assessment.
    Journal of medicinal chemistry, 2022, 11-10, Volume: 65, Issue:21

    Topics: Drug Interactions; HEK293 Cells; Humans; Liver; Organic Anion Transporters, Sodium-Independent; Risk Assessment

2022
Comparison of KRN2391 with nicorandil and nifedipine on canine coronary blood flow: antagonism by glibenclamide.
    Journal of cardiovascular pharmacology, 1992, Volume: 20, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Female; Glyburide; Heart Rate; Male; Niacinamide; Nicorandil; Nifedipine; Potassium Channels; Pyridines; Vascular Resistance

1992
Effect of pinacidil on the membrane electrical activity of guinea pig detrusor muscle.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Glyburide; Guanidines; Guinea Pigs; Membrane Potentials; Muscle, Smooth; Nifedipine; Pinacidil; Urinary Bladder; Vasodilator Agents

1992
Endothelin stimulates 86Rb efflux in rat glioma C6-Bu-1 cells.
    Neuropeptides, 1991, Volume: 20, Issue:1

    Topics: Alkaloids; Analysis of Variance; Animals; Calcium; Diltiazem; Endothelins; Glioma; Glyburide; Nifedipine; Pertussis Toxin; Potassium; Potassium Channels; Protein Kinase C; Rats; Rubidium; Staurosporine; Tumor Cells, Cultured; Virulence Factors, Bordetella

1991
RP 49356 and cromakalim relax airway smooth muscle in vitro by opening a sulphonylurea-sensitive K+ channel: a comparison with nifedipine.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Animals; Benzopyrans; Calcium; Cromakalim; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Picolines; Potassium Channels; Pyrans; Pyrroles; Trachea

1991
Evidence that pinacidil may promote the opening of ATP-sensitive K+ channels yet inhibit the opening of Ca2(+)-activated K+ channels in K(+)-contracted canine mesenteric artery.
    British journal of pharmacology, 1990, Volume: 100, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Calcium; Cromakalim; Dogs; Female; Glyburide; Guanidines; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Pinacidil; Potassium; Potassium Channels; Pyrroles; Rubidium Radioisotopes

1990
A comparison of the actions of cromakalim and nifedipine on rabbit isolated mesenteric artery.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: Animals; Benzopyrans; Blood Pressure; Cell Membrane; Cromakalim; Electric Stimulation; Glyburide; Humans; In Vitro Techniques; Infant, Newborn; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Perfusion; Potassium Channels; Pyrroles; Rabbits

1990
Counteraction of nifedipine-induced hyperglycaemia by metformin.
    Diabete & metabolisme, 1990, Volume: 16, Issue:6

    Topics: Animals; Glyburide; Hyperglycemia; Male; Metformin; Nifedipine; Rats

1990
Specific antagonism by glibenclamide of negative inotropic effects of potassium channel openers in canine atrial muscle.
    Japanese journal of pharmacology, 1990, Volume: 54, Issue:2

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dogs; Female; Glyburide; Guanidines; Heart Atria; Male; Myocardial Contraction; Niacinamide; Nicorandil; Nifedipine; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents

1990
Inhibition by sulphonylureas of vasorelaxation induced by K+ channel activators in vitro.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: Animals; Antihypertensive Agents; Benzopyrans; Cromakalim; Drug Interactions; Glipizide; Glyburide; Guanidines; In Vitro Techniques; Male; Nifedipine; Norepinephrine; Pinacidil; Potassium Channels; Potassium Chloride; Pyrroles; Rabbits; Sulfonylurea Compounds; Tolbutamide; Vasodilator Agents

1989
Phenylephrine-induced rhythmic activity in the rabbit ear artery.
    The Japanese journal of physiology, 1993, Volume: 43, Issue:4

    Topics: Animals; Arginine; Arteries; Charybdotoxin; Ear, External; Endothelium, Vascular; Glyburide; In Vitro Techniques; Indomethacin; Male; Nifedipine; Nitric Oxide; Nitroarginine; omega-N-Methylarginine; Periodicity; Phenylephrine; Potassium Channel Blockers; Prostaglandin Antagonists; Rabbits; Scorpion Venoms; Vasoconstriction

1993
Role of calcium-activated potassium channels in the relaxation of tracheal smooth muscles by forskolin.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:5

    Topics: Animals; Apamin; Calcium; Carbachol; Charybdotoxin; Colforsin; Cyclic AMP; Drug Interactions; Electrophysiology; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Trachea

1994
Propagation of impulses in the guinea-pig ureter and its blockade by calcitonin gene-related peptide (CGRP).
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 351, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Cromakalim; Electric Stimulation; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyrroles; Tetrodotoxin; Ureter

1995
Effect of KRN2391 on venous return: comparison with other vasodilators.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:1

    Topics: Animals; Benzopyrans; Cromakalim; Dogs; Female; Glyburide; Hemodynamics; Male; Niacinamide; Nicorandil; Nifedipine; Nitroglycerin; Potassium Channels; Pyridines; Pyrroles; Vasodilator Agents; Veins

1993
Participation of calcium, released from the IP3-sensitive Ca-store in activation of Ca-dependent potassium conductance of ileal smooth muscle cells.
    General physiology and biophysics, 1993, Volume: 12, Issue:3

    Topics: Animals; Apamin; Calcium; Charybdotoxin; Egtazic Acid; Glyburide; Guinea Pigs; Heparin; Ileum; In Vitro Techniques; Indoles; Inositol 1,4,5-Trisphosphate; Membrane Potentials; Muscle, Smooth; Nifedipine; Potassium Channels; Ruthenium Red; Scorpion Venoms

1993
A simple method for measurement of ureteric peristaltic function in vivo and the effects of drugs acting on ion channels applied from the ureter lumen in anesthetized rats.
    Japanese journal of pharmacology, 1993, Volume: 62, Issue:4

    Topics: 4-Aminopyridine; Anesthesia; Animals; Benzopyrans; Cromakalim; Glyburide; Ion Channels; Lidocaine; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyrroles; Rats; Rats, Sprague-Dawley; Ureter; Vasodilator Agents

1993
Drug-induced endothelium-dependent and -independent relaxations in isolated resistance vessels taken from simultaneously hypertensive and streptozotocin-diabetic rats.
    Blood pressure, 1994, Volume: 3, Issue:6

    Topics: Animals; Benzopyrans; Bradykinin; Calcium; Cromakalim; Diabetes Mellitus, Experimental; Endothelium, Vascular; Glyburide; Histamine; Hypertension; Male; Mesenteric Arteries; Methacholine Chloride; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Nitroprusside; Potassium Channels; Potassium Chloride; Pyrroles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Streptozocin; Vascular Resistance; Vasodilation; Vasodilator Agents

1994
Cellular mechanisms of hypoxia-induced contraction in human and rat pulmonary arteries.
    Respiration physiology, 1995, Volume: 99, Issue:2

    Topics: Aged; Animals; Benzopyrans; Calcium; Calcium Channels; Cromakalim; Glyburide; Humans; Hypoxia; In Vitro Techniques; Iodoacetates; Iodoacetic Acid; Male; Middle Aged; Muscle, Smooth, Vascular; Nifedipine; Potassium Channels; Pulmonary Artery; Pyrroles; Rats; Rats, Wistar; Vasoconstriction; Verapamil

1995
Inhibition of ATP-sensitive K+ channel by a non-sulfonylurea compound KAD-1229 in a pancreatic beta-cell line, MIN 6 cell.
    European journal of pharmacology, 1994, Nov-15, Volume: 269, Issue:3

    Topics: Action Potentials; Adenosine Triphosphate; Binding, Competitive; Calcium; Cell Membrane; Cobalt; Dose-Response Relationship, Drug; Drug Synergism; Fura-2; Glucose; Glyburide; Humans; Hypoglycemic Agents; Indoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Isoindoles; Membrane Potentials; Nifedipine; Pancreatic Neoplasms; Patch-Clamp Techniques; Potassium Channel Blockers; Tumor Cells, Cultured

1994
Pharmacological analysis of the effect of KRN2391 on coronary vasculature in perfused rat heart.
    General pharmacology, 1994, Volume: 25, Issue:3

    Topics: Animals; Benzopyrans; Coronary Circulation; Cromakalim; Dose-Response Relationship, Drug; Glyburide; In Vitro Techniques; Male; Nifedipine; Perfusion; Potassium Channels; Pyridines; Pyrroles; Rats; Rats, Wistar; Vasodilator Agents

1994
Tetraethylammonium selectively stimulates secretion from noradrenergic bovine chromaffin cells.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:3

    Topics: 4-Aminopyridine; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; Drug Interactions; Drug Synergism; Epinephrine; Glyburide; Nifedipine; Norepinephrine; Ouabain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tolbutamide

1994
Insulin secretion by the pancreatic beta cell of aged rats.
    Pancreas, 1994, Volume: 9, Issue:4

    Topics: Aging; Animals; Colforsin; Dose-Response Relationship, Drug; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Potassium; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate

1994
Effects of levcromakalim on ureteral peristaltic function and cystometrogram in rats.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:4

    Topics: Administration, Topical; Animals; Benzopyrans; Cromakalim; Glyburide; Injections, Intraperitoneal; Injections, Intravenous; Male; Nifedipine; Parasympatholytics; Pyrroles; Rats; Rats, Sprague-Dawley; Ureter; Urinary Bladder

1993
NIP-121 is more effective than nifedipine in acutely reversing chronic pulmonary hypertension.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 75, Issue:3

    Topics: Altitude; Animals; Chronic Disease; Glyburide; Hemodynamics; Hypertension, Pulmonary; Hypoxia; Male; Nifedipine; Oxadiazoles; Piperidines; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasodilation

1993
Lemakalim attenuates hypocapnia- and dry air-induced bronchoconstriction in canine peripheral airways.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 75, Issue:1

    Topics: Acetylcholine; Adenosine Triphosphate; Aerosols; Airway Resistance; Albuterol; Animals; Benzopyrans; Blood Pressure; Bronchoconstriction; Bronchodilator Agents; Cromakalim; Dogs; Glyburide; Heart Rate; Humidity; Hypocapnia; Injections, Intravenous; Lung; Male; Nifedipine; Potassium Channels; Pyrroles

1993
The relaxant actions on guinea-pig trachealis of atherosperminine isolated from Fissistigma glaucescens.
    European journal of pharmacology, 1993, Jun-11, Volume: 237, Issue:1

    Topics: Alkaloids; Animals; Benzopyrans; Calcium; Calmodulin; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Egtazic Acid; Epithelium; Female; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Nitroprusside; Phenanthrenes; Plants, Medicinal; Propranolol; Pyrroles; Theophylline; Trachea; Vasodilator Agents

1993
Endothelial function in deoxycorticosterone-NaCl hypertension: effect of calcium supplementation.
    Circulation, 1996, Mar-01, Volume: 93, Issue:5

    Topics: Acetylcholine; Adenosine Diphosphate; Animals; Apamin; Arginine; Blood Pressure; Calcium, Dietary; Desoxycorticosterone; Endothelium, Vascular; Glyburide; Hypertension; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nifedipine; Nitroprusside; Norepinephrine; Potassium Channels; Rats; Rats, Inbred WKY; Serotonin; Sodium Chloride; Vasodilation

1996
Pharmacodynamic behaviour of isolated resistance vessels obtained from hypertensive-diabetic rats.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Animals; Benzopyrans; Blood Glucose; Calcium Channels; Calcium Chloride; Cromakalim; Glyburide; Hypertension; In Vitro Techniques; Male; Mesenteric Arteries; Methacholine Chloride; Methoxamine; Muscle Contraction; Muscle, Smooth; Nifedipine; Nitroprusside; Norepinephrine; Obesity; Potassium Channels; Potassium Chloride; Pyrroles; Rats; Rats, Zucker; Serotonin; Tunica Media; Vascular Resistance; Vasoconstrictor Agents; Vasodilator Agents

1996
Analysis of relaxation and repolarization mechanisms of nicorandil in rat mesenteric artery.
    British journal of pharmacology, 1996, Volume: 119, Issue:8

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Benzopyrans; Calcium Channel Blockers; Cromakalim; Electrophysiology; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Nifedipine; Potassium Channels; Prostaglandin Endoperoxides, Synthetic; Pyrroles; Rats; Rats, Sprague-Dawley; Thromboxane A2; Vasoconstrictor Agents; Vasodilator Agents

1996
Interaction between the L-type Ca2+ channel and the Ca(2+)-activated K+ channel in the fluctuating myogenic contraction in the rabbit basilar artery.
    The Japanese journal of physiology, 1996, Volume: 46, Issue:4

    Topics: Animals; Basilar Artery; Calcium; Calcium Channel Blockers; Calcium Channels; Charybdotoxin; Glyburide; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Nifedipine; Potassium Channel Blockers; Potassium Channels; Rabbits; Vasoconstriction

1996
Effects of BKCa channels on the reduction of cytosolic Ca2+ in cGMP-induced relaxation of guinea-pig trachea.
    Clinical and experimental pharmacology & physiology, 1997, Volume: 24, Issue:2

    Topics: Animals; Apamin; Atrial Natriuretic Factor; Calcium; Cyclic GMP; Cytosol; Extracellular Space; Glyburide; Guinea Pigs; Intracellular Fluid; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nifedipine; Peptides; Potassium; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Trachea

1997
Y-26763 protects the canine heart from a stunning injury through opening of the KATP channels.
    European journal of pharmacology, 1997, Apr-04, Volume: 323, Issue:2-3

    Topics: Adenosine Triphosphate; Animals; Antihypertensive Agents; Benzopyrans; Calcium Channel Blockers; Dogs; Female; Glyburide; Hemodynamics; Male; Myocardial Stunning; Nifedipine; Potassium Channels

1997
Interactions between neuropeptide Y and the adenylate cyclase pathway in rat mesenteric small arteries: role of membrane potential.
    The Journal of physiology, 1997, Jul-15, Volume: 502 ( Pt 2)

    Topics: 4-Aminopyridine; Acetylcholine; Adenylyl Cyclases; Animals; Charybdotoxin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dichlororibofuranosylbenzimidazole; Gadolinium; Glyburide; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Nifedipine; Potassium Channels; Rats; Rats, Wistar; Thionucleotides

1997
Effects of nitroprusside and nicorandil on catecholamine secretion and calcium mobilization in cultured bovine adrenal chromaffin cells.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:4

    Topics: Adrenal Medulla; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin Cells; Glyburide; Niacinamide; Nicorandil; Nifedipine; Nitroprusside; Vasodilator Agents

1997
Microvascular permeability with sulfonylureas in normal and diabetic hamsters.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:12 Suppl 1

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Capillary Permeability; Cricetinae; Dextrans; Diabetes Mellitus, Experimental; Diazoxide; Disease Models, Animal; Dose-Response Relationship, Drug; Fluorescein-5-isothiocyanate; Gliclazide; Glyburide; Histamine; Hypoglycemic Agents; Insulin; Macromolecular Substances; Male; Mesocricetus; Nifedipine; Potassium Channels; Reperfusion Injury; Streptozocin; Sulfonylurea Compounds

1997
The effects of nifedipine and other calcium antagonists on the glibenclamide-sensitive K+ currents in smooth muscle cells from pig urethra.
    British journal of pharmacology, 1998, Volume: 123, Issue:8

    Topics: Animals; Barium; Calcium Channel Blockers; Cromakalim; Female; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Muscle, Smooth; Nifedipine; Patch-Clamp Techniques; Potassium Channels; Swine; Urethra

1998
Rapid activation and nuclear translocation of mitogen-activated protein kinases in response to physiological concentration of glucose in the MIN6 pancreatic beta cell line.
    The Journal of biological chemistry, 1998, Jun-19, Volume: 273, Issue:25

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Nucleus; Colforsin; Egtazic Acid; Enzyme Activation; Glucose; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Kainic Acid; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nifedipine; Potassium; Receptors, Glutamate

1998
Hyperpolarization and slowing of the rate of contraction in human uterus in pregnancy by prostaglandins E2 and f2alpha: involvement of the Na+ pump.
    The Journal of physiology, 1999, Jan-01, Volume: 514 ( Pt 1)

    Topics: Albuterol; Calcium; Calcium Channel Blockers; Charybdotoxin; Cyclic AMP; Dinoprost; Dinoprostone; Enzyme Inhibitors; Female; Glyburide; Humans; Hypoglycemic Agents; Iloprost; Membrane Potentials; Myometrium; Nifedipine; Ouabain; Potassium; Potassium Channel Blockers; Potassium Channels; Pregnancy; Sodium-Potassium-Exchanging ATPase; Sympathomimetics; Tetraethylammonium; Uterine Contraction; Vasodilator Agents

1999
Cellular characterization of pituitary adenoma cell line (AtT20 cell) transfected with insulin, glucose transporter type 2 (GLUT2) and glucokinase genes: insulin secretion in response to physiological concentrations of glucose.
    Diabetologia, 1998, Volume: 41, Issue:12

    Topics: Adenoma; Calcium Channel Blockers; Corticotropin-Releasing Hormone; Diazoxide; Gene Expression; Glucokinase; Glucose; Glucose Transporter Type 2; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Monosaccharide Transport Proteins; Nifedipine; Pituitary Neoplasms; Potassium Chloride; Transfection; Tumor Cells, Cultured

1998
The ginsenoside Rg3 evokes endothelium-independent relaxation in rat aortic rings: role of K+ channels.
    European journal of pharmacology, 1999, Feb-12, Volume: 367, Issue:1

    Topics: Animals; Antineoplastic Agents, Phytogenic; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Cromakalim; Dose-Response Relationship, Drug; Endothelium, Vascular; Ginsenosides; Glyburide; In Vitro Techniques; Male; Muscle Relaxation; Nifedipine; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Rats; Rats, Sprague-Dawley; Rubidium Radioisotopes; Saponins; Tetraethylammonium; Vasodilator Agents

1999
Growth inhibitory effects of ATP and its derivatives on human fibroblasts immortalized with 60Co-gamma rays.
    International journal of molecular medicine, 2000, Volume: 5, Issue:1

    Topics: Adenosine Triphosphate; Cell Division; Cell Line; DNA Fragmentation; Gamma Rays; Glyburide; Humans; Nifedipine; Receptors, Purinergic P2

2000
Arterial flow induces changes in saphenous vein endothelium proteins transduced by cation channels.
    European journal of vascular and endovascular surgery : the official journal of the European Society for Vascular Surgery, 2000, Volume: 19, Issue:5

    Topics: Arteries; Biomarkers; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Endothelium, Vascular; Glyburide; Humans; In Vitro Techniques; Intercellular Adhesion Molecule-1; Nifedipine; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Perfusion; Potassium Channel Blockers; Potassium Channels; Proteins; Regional Blood Flow; Saphenous Vein; Tetraethylammonium; Thromboplastin; Vascular Cell Adhesion Molecule-1

2000
Opposing roles of K(+) and Cl(-) channels in maintenance of opossum lower esophageal sphincter tone.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 279, Issue:6

    Topics: 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Action Potentials; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Chloride Channels; Esophagogastric Junction; Glyburide; Isometric Contraction; Microelectrodes; Muscle, Smooth; Nifedipine; Niflumic Acid; Opossums; Potassium Channels

2000
The involvement of L-type Ca(2+) channels in the relaxant effects of the ATP-sensitive K(+) channel opener ZD6169 on pig urethral smooth muscle.
    British journal of pharmacology, 2001, Volume: 134, Issue:7

    Topics: Adenosine Triphosphate; Amides; Animals; Barium; Benzophenones; Calcium Channel Blockers; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gene Expression; Glyburide; In Vitro Techniques; Membrane Potentials; Muscle Relaxation; Muscle, Smooth; Nifedipine; Potassium Channels; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Swine; Urethra

2001
Substance P induces inward current and regulates pacemaker currents through tachykinin NK1 receptor in cultured interstitial cells of Cajal of murine small intestine.
    European journal of pharmacology, 2004, Jul-08, Volume: 495, Issue:1

    Topics: 4-Aminopyridine; Action Potentials; Alkaloids; Animals; Benzophenanthridines; Calcium; Cations, Divalent; Cells, Cultured; Electrophysiology; Enteric Nervous System; Female; Glyburide; Intestine, Small; Ion Channels; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nifedipine; Phenanthridines; Receptors, Neurokinin-1; Sinoatrial Node; Sodium; Substance P; Tachykinins; Tetraethylammonium; Tetrodotoxin

2004
Pacemaker potentials generated by interstitial cells of Cajal in the murine intestine.
    American journal of physiology. Cell physiology, 2005, Volume: 288, Issue:3

    Topics: Animals; Anti-Arrhythmia Agents; Biological Clocks; Caffeine; Calcium Channel Blockers; Central Nervous System Stimulants; Electrophysiology; Glyburide; In Vitro Techniques; Intestine, Small; Membrane Potentials; Mibefradil; Mice; Mice, Inbred BALB C; Myocytes, Smooth Muscle; Nifedipine; Pinacidil; Vasodilator Agents

2005
Glucose-stimulated DNA synthesis through mammalian target of rapamycin (mTOR) is regulated by KATP channels: effects on cell cycle progression in rodent islets.
    The Journal of biological chemistry, 2006, Feb-10, Volume: 281, Issue:6

    Topics: Animals; Blotting, Western; Calcium; Cell Cycle; Cell Division; Cell Proliferation; Cells, Cultured; Cytosol; Diazoxide; Dose-Response Relationship, Drug; Flow Cytometry; G2 Phase; Glucose; Glyburide; Islets of Langerhans; Male; Nifedipine; Potassium; Potassium Channels; Protein Kinases; Rats; Rats, Sprague-Dawley; S Phase; Sirolimus; Thymidine; TOR Serine-Threonine Kinases

2006
Relative contribution of intracellular and extracellular Ca2+ to alpha2-adrenoceptor-mediated contractions of ovine pulmonary artery.
    Pharmacological research, 2006, Volume: 54, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Calcium; Calcium Channel Blockers; Cyclic AMP; Cyclic GMP; Glyburide; Guanfacine; Indoles; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nucleotides, Cyclic; Pulmonary Artery; Receptors, Adrenergic, alpha-2; Sheep; Vasoconstriction; Vasodilator Agents

2006
Role of ion channel modifiers in reversal of morphine-induced gastrointestinal inertia by prokinetic agents in mice.
    Indian journal of experimental biology, 2008, Volume: 46, Issue:1

    Topics: Analgesics, Opioid; Animals; Benzamides; Calcium Channels; Domperidone; Gastrointestinal Tract; Glyburide; Intestine, Small; Ion Channels; Kinetics; Mice; Minoxidil; Morphine; Morpholines; Nifedipine; Time Factors

2008
Vasorelaxant effect of a self-etch adhesive system through calcium antagonistic action.
    Journal of endodontics, 2008, Volume: 34, Issue:10

    Topics: 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Dentin-Bonding Agents; Endothelium, Vascular; Enzyme Inhibitors; Epoprostenol; Glyburide; Indomethacin; Male; Materials Testing; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Potassium Channels, Voltage-Gated; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Time Factors; Vasoconstrictor Agents; Vasodilator Agents

2008
Anemoside A3-induced relaxation in rat renal arteries: role of endothelium and Ca2+ channel inhibition.
    Planta medica, 2010, Volume: 76, Issue:16

    Topics: Animals; Apamin; Arteries; Biological Factors; Calcium; Calcium Channel Blockers; Capsaicin; Charybdotoxin; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Glyburide; Kidney; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myography; Nifedipine; Plant Extracts; Plant Roots; Potassium Channels; Potassium Chloride; Pulsatilla; Rats; Rats, Sprague-Dawley; Saponins; Tetraethylammonium; Triterpenes; Vasodilator Agents

2010
Modulation of adrenergic responses of human vas deferens by K+ channel inhibitors.
    Urology, 2010, Volume: 76, Issue:6

    Topics: Adult; Apamin; Calcium; Calcium Channels, L-Type; Charybdotoxin; Electric Stimulation; Glyburide; Humans; Ion Transport; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Peptides; Potassium; Potassium Channel Blockers; Potassium Channels; Receptors, Adrenergic, alpha-1; Tetraethylammonium; Vas Deferens

2010
Vasodilatory effect of hydroxyethyl methacrylate and triethylene glycol dimethacrylate in rat aorta through calcium antagonistic action.
    Journal of endodontics, 2011, Volume: 37, Issue:3

    Topics: 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Calcium Chloride; Composite Resins; Cyclooxygenase Inhibitors; Dental Materials; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Indomethacin; Male; Methacrylates; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide Synthase; Polyethylene Glycols; Polymethacrylic Acids; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Transducers; Vasoconstrictor Agents; Vasodilator Agents

2011
Inhibition of ATP-sensitive K+ channels and L-type Ca2+ channels by amiodarone elicits contradictory effect on insulin secretion in MIN6 cells.
    Journal of pharmacological sciences, 2011, Volume: 116, Issue:1

    Topics: Amiodarone; Animals; Anti-Arrhythmia Agents; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; KATP Channels; Membrane Potentials; Mice; Nifedipine; Osmolar Concentration; Patch-Clamp Techniques; Potassium Channel Blockers; Quinidine

2011
Low glucose sensitivity and polymodal chemosensing in neonatal rat adrenomedullary chromaffin cells.
    American journal of physiology. Cell physiology, 2011, Volume: 301, Issue:5

    Topics: Animals; Animals, Newborn; Calcium; Calcium Channel Blockers; Catecholamines; Cell Hypoxia; Cells, Cultured; Chromaffin Cells; Glucose; Glyburide; Hypercapnia; Membrane Potentials; Nickel; Nifedipine; Potassium Channels; Rats; Rats, Wistar

2011
Role of calcium and potassium channels in effects of hydrogen sulfide on frog myocardial contractility.
    Bulletin of experimental biology and medicine, 2011, Volume: 151, Issue:2

    Topics: 4-Aminopyridine; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Electric Stimulation; Glyburide; Heart; Hydrogen Sulfide; In Vitro Techniques; KATP Channels; Minoxidil; Myocardial Contraction; Myocardium; Nifedipine; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Rana ridibunda; Tetraethylammonium

2011
Highly efficient miniaturized coprecipitation screening (MiCoS) for amorphous solid dispersion formulation development.
    International journal of pharmaceutics, 2013, Jun-25, Volume: 450, Issue:1-2

    Topics: Acrylic Resins; Chemical Precipitation; Chemistry, Pharmaceutical; Felodipine; Glyburide; Methylcellulose; Miniaturization; Nifedipine; Polymethacrylic Acids; Powders; Solubility

2013
Significance of K(ATP) channels, L-type Ca²⁺ channels and CYP450-4A enzymes in oxygen sensing in mouse cremaster muscle arterioles in vivo.
    BMC physiology, 2013, May-12, Volume: 13

    Topics: Animals; Arterioles; Calcium Channels, L-Type; Cromakalim; Cytochrome P-450 Enzyme System; Glyburide; Hydroxyeicosatetraenoic Acids; KATP Channels; Male; Mice; Mice, Inbred C57BL; Muscle, Skeletal; Muscle, Smooth, Vascular; Nifedipine; Nitric Oxide Synthase; Oxygen; Retinoic Acid 4-Hydroxylase; Vasoconstriction; Vasodilation

2013
The Possible Mechanisms of the Impaired Insulin Secretion in Hypothyroid Rats.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: Acetylcholine; Animals; Blood Glucose; Glucokinase; Glyburide; Hexokinase; Hypoglycemic Agents; Hypothyroidism; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Rats; Rats, Wistar; Thyroxine; Triiodothyronine

2015
Impaired glucose-stimulated insulin secretion and reduced β-cell mass in pancreatic islets of hyperthyroid rats.
    Experimental physiology, 2016, 08-01, Volume: 101, Issue:8

    Topics: Animals; Calcium Channels, L-Type; Diazoxide; Glucose; Glucose Tolerance Test; Glyburide; Hyperthyroidism; Hypoglycemic Agents; Insulin; Insulin-Secreting Cells; KATP Channels; Male; Nifedipine; Rats; Rats, Sprague-Dawley; Thyroid Hormones; Thyroxine

2016
Combination Therapy of Nifedipine and Sulphonylureas Exhibits a Mutual Antagonistic Effect on the Endothelial Cell Dysfunction Induced by Hyperglycemia Linked to Vascular Disease.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2016, Volume: 38, Issue:6

    Topics: Antihypertensive Agents; Biphenyl Compounds; Cell Movement; Diabetic Angiopathies; Drug Synergism; Endothelial Cells; Glucose; Glyburide; Human Umbilical Vein Endothelial Cells; Humans; Hyperglycemia; Hypoglycemic Agents; Irbesartan; Metformin; Nifedipine; Oxygen; Sulfonylurea Compounds; Tetrazoles

2016
The beneficial effect of clove essential oil and its major component, eugenol, on erectile function in diabetic rats.
    Andrologia, 2020, Volume: 52, Issue:6

    Topics: Animals; Clove Oil; Diabetes Mellitus, Experimental; Erectile Dysfunction; Eugenol; Glyburide; In Vitro Techniques; Injections; Male; Nifedipine; Nitric Oxide Synthase; Oils, Volatile; Penile Erection; Penis; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Soluble Guanylyl Cyclase; Tetraethylammonium

2020
Aqueous extract of oakmoss produces antihypertensive activity in L-NAME-induced hypertensive rats through sGC-cGMP pathway.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2021, Jan-02, Volume: 43, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Aorta, Thoracic; Arterial Pressure; Blood Pressure; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Glyburide; Hypertension; KATP Channels; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide Synthase; Parmeliaceae; Plant Extracts; Propranolol; Rats; Rats, Wistar; Resins, Plant; Terpenes; Vasodilator Agents

2021
Pulmonary Microcirculation in Experimental Model of Pulmonary Thromboembolism after Pretreatment with Chloroquine.
    Bulletin of experimental biology and medicine, 2023, Volume: 175, Issue:3

    Topics: Adenosine Triphosphate; Animals; Chloroquine; Glyburide; Lung; Microcirculation; Models, Theoretical; Nifedipine; Pulmonary Embolism; Rabbits; Vascular Resistance

2023