glyburide has been researched along with nifedipine in 87 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (1.15) | 18.7374 |
1990's | 39 (44.83) | 18.2507 |
2000's | 19 (21.84) | 29.6817 |
2010's | 23 (26.44) | 24.3611 |
2020's | 5 (5.75) | 2.80 |
Authors | Studies |
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Topliss, JG; Yoshida, F | 1 |
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Andricopulo, AD; Moda, TL; Montanari, CA | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M | 1 |
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
Sen, S; Sinha, N | 1 |
Barber, J; Dawson, S; Kenna, JG; Paul, N; Stahl, S | 1 |
Caradonna, NP; Hallifax, D; Houston, JB; Turlizzi, E; Zanelli, U | 1 |
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Aleo, MD; Bonin, PD; Luo, Y; Potter, DM; Swiss, R; Will, Y | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF | 1 |
Chang, G; Mathialagan, S; Ryu, S; Varma, MVS; Woody, N | 1 |
Fukata, Y; Fukushima, H; Jinno, Y; Kaneta, S; Nishikori, K; Ogawa, N | 1 |
Karim, OM; Mostwin, JL; Seki, N | 1 |
Aiyar, N; Gleason, MM; Griffin, EC; Nambi, P | 1 |
Brown, TJ; Raeburn, D | 1 |
Asano, M; Masuzawa, K; Matsuda, T | 1 |
McHarg, AD; Southerton, JS; Weston, AH | 1 |
Abu-Jayyab, AR; al-Bekairi, AM; el-Denshary, ES; el-Sawaf, HA | 1 |
Satoh, E; Taira, N; Yanagisawa, T | 1 |
Wilson, C | 1 |
Mizusawa, H; Omote, M | 2 |
Hiramatsu, T; Kotlikoff, MI; Kume, H; Takagi, K | 1 |
Maggi, CA; Meini, S; Santicioli, P | 1 |
Fukushima, H; Jinno, Y; Kaneta, S; Miwa, A; Ogawa, N | 1 |
Boev, KK; Duridanova, DB; Gagov, HS | 1 |
Ginkawa, M; Kontani, H; Sakai, T | 1 |
Kam, KL; Pfaffendorf, M; van Zwieten, PA | 2 |
Gonzalez de la Fuente, P; Marthan, R; Savineau, JP | 1 |
Kojima, I; Miyazaki, J; Mogami, H; Nobusawa, R; Ohnota, H; Satou, F; Shibata, H | 1 |
Izawa, T; Jinno, Y; Miwa, A; Ogawa, N; Yokoyama, T | 1 |
Cahill, AL; Perlman, RL | 1 |
Aizawa, T; Hashizume, K; Ishihara, F; Komatsu, M; Nishii, N; Sato, Y; Suzuki, N; Yamada, T | 1 |
Jinkawa, M; Kontani, H; Sakai, T | 1 |
McMurtry, IF; Morris, KG; Oka, M | 1 |
Freed, AN; Lindeman, KS | 1 |
Ko, FN; Lin, CH; Lu, ST; Teng, CM; Wu, YC | 1 |
Arvola, P; Kähönen, M; Mäkynen, H; Pörsti, I; Wu, X | 1 |
Angus, JA; Fujiwara, T | 1 |
Kume, H; Mikawa, K; Takagi, K | 1 |
Fukunari, A; Kawahara, K; Miyai, H; Nakajima, T; Shinagawa, K | 1 |
Buus, C; Mulvany, MJ; Nilsson, H; Prieto, D | 1 |
Högemann, A; Jonkman, JH; Lins, R; Sennewald, R; van Heiningen, PN; van Lier, JJ | 1 |
Houchi, H; Nakaya, Y; Oka, M; Shono, M | 1 |
Bouskela, E; Conde, CM; Cyrino, FZ; Garcia, AA | 1 |
Brading, AF; Teramoto, N | 1 |
Benes, C; Creuzet, C; Fagard, R; Miyazaki, J; Roisin, MP; Van Tan, H | 1 |
Brennecke, SP; Coleman, HA; Davies, NK; Parkington, HC; Tonta, MA | 1 |
Araki, E; Kaneko, K; Kishikawa, H; Motoshima, H; Motoyoshi, S; Sakai, K; Shichiri, M; Shirakami, A; Shirotani, T; Yoshizato, K | 1 |
Kang, SY; Kim, MJ; Kim, ND; Park, JH; Schini-Kerth, VB | 1 |
Inoue, Y; Kondo, A; Li, JW; Miyazaki, M; Namba, M; Pu, H | 1 |
Golledge, J; Gosling, M; Powell, JT; Standfield, NJ; Turner, RJ | 1 |
Miller, DV; Paterson, WG; Zhang, Y | 1 |
Ikawa, S; Ito, Y; Naito, S; Seki, N; Takano, N; Tanaka, K; Teramoto, N; Yunoki, T | 1 |
Chang, IY; Choi, S; Jun, JY; Kim, KW; Kim, MJ; Kim, MY; Kong, ID; Lee, KP; Park, CK; So, I; Yeum, CH; You, HJ | 1 |
Kito, Y; Sanders, KM; Ward, SM | 1 |
Kwon, G; Liu, H; Marshall, CA; McDaniel, ML; Pappan, KL; Remedi, MS | 1 |
Mishra, SK; Prakash, VR; Ross, GR; Sathishkumar, K | 1 |
Dkhar, SA; Krishna, PR; Ramaswamy, S; Sandhiya, S | 1 |
Basak, F; Cehreli, SB; Cehreli, ZC; Guven, G; Kaya, E; Seyrek, M; Ulku, C; Vural, IM; Yildiz, O | 1 |
Fan, CL; Huang, Y; Lau, CW; Li, Y; Lin, SM; Wang, J; Ye, WC; Yiu, A; Zhang, DM | 1 |
Chuan, P; Lluch, S; Mauricio, MD; Medina, P; Segarra, G; Vila, JM | 1 |
Cehreli, ZC; Guven, G; Seyrek, M; Vural, IM; Yildiz, O | 1 |
Matsumoto, A; Miki, T; Nakaya, H; Nishida, A; Seino, S; Takizawa, T | 1 |
Buttigieg, J; Livermore, S; Nurse, CA; Piskuric, NA; Zhang, M | 1 |
Khaertdinov, NN; Sitdikova, GF; Zefirov, AL | 1 |
Choi, DS; Chokshi, H; Hu, Q; Sandhu, H; Shah, N | 1 |
Holstein-Rathlou, NH; Jensen, LJ; Ngo, AT; Riemann, M; Torp-Pedersen, C | 1 |
Ghasemi, A; Godini, A; Zahediasl, S | 1 |
Hoshmandi, E; Karbalaei, N; Noorafshan, A | 1 |
Jiang, Y; Peng, C; Tao, X; Wang, LP; Xie, HH; Yang, H; Zhang, C | 1 |
Carbonell-Barrachina, ÁA; Gur, S; Kaya-Sezginer, E; Onder, A; Oztekin, CV; Yilmaz-Oral, D; Zor, M | 1 |
Ajebli, M; Amssayef, A; Eddouks, M | 1 |
Berezina, TP; Evlakhov, VI; Poyasov, IZ | 1 |
2 review(s) available for glyburide and nifedipine
Article | Year |
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DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells | 2022 |
1 trial(s) available for glyburide and nifedipine
Article | Year |
---|---|
Pharmacokinetic drug interaction studies with candesartan cilexetil.
Topics: Adolescent; Adult; Angiotensin Receptor Antagonists; Antihypertensive Agents; Benzimidazoles; Biphenyl Compounds; Digoxin; Drug Interactions; Female; Glyburide; Humans; Hydrochlorothiazide; Male; Middle Aged; Nifedipine; Tetrazoles; Warfarin | 1997 |
84 other study(ies) available for glyburide and nifedipine
Article | Year |
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QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration | 2004 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Hologram QSAR model for the prediction of human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2007 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship | 2008 |
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship | 2011 |
In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Cholestasis; Drug-Related Side Effects and Adverse Reactions; Humans; Insecta; Rats; Risk Factors | 2012 |
Comparison of cryopreserved HepaRG cells with cryopreserved human hepatocytes for prediction of clearance for 26 drugs.
Topics: Cell Line, Tumor; Cryopreservation; Female; Hepatocytes; Humans; Male; Metabolic Clearance Rate; Pharmaceutical Preparations; Predictive Value of Tests | 2012 |
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection | 2012 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Human drug-induced liver injury severity is highly associated with dual inhibition of liver mitochondrial function and bile salt export pump.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Chemical and Drug Induced Liver Injury; Humans; Male; Mitochondria, Liver; Rats; Rats, Sprague-Dawley; Severity of Illness Index | 2014 |
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain | 2016 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
Identification of Organic Anion Transporter 2 Inhibitors: Screening, Structure-Based Analysis, and Clinical Drug Interaction Risk Assessment.
Topics: Drug Interactions; HEK293 Cells; Humans; Liver; Organic Anion Transporters, Sodium-Independent; Risk Assessment | 2022 |
Comparison of KRN2391 with nicorandil and nifedipine on canine coronary blood flow: antagonism by glibenclamide.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Female; Glyburide; Heart Rate; Male; Niacinamide; Nicorandil; Nifedipine; Potassium Channels; Pyridines; Vascular Resistance | 1992 |
Effect of pinacidil on the membrane electrical activity of guinea pig detrusor muscle.
Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Glyburide; Guanidines; Guinea Pigs; Membrane Potentials; Muscle, Smooth; Nifedipine; Pinacidil; Urinary Bladder; Vasodilator Agents | 1992 |
Endothelin stimulates 86Rb efflux in rat glioma C6-Bu-1 cells.
Topics: Alkaloids; Analysis of Variance; Animals; Calcium; Diltiazem; Endothelins; Glioma; Glyburide; Nifedipine; Pertussis Toxin; Potassium; Potassium Channels; Protein Kinase C; Rats; Rubidium; Staurosporine; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1991 |
RP 49356 and cromakalim relax airway smooth muscle in vitro by opening a sulphonylurea-sensitive K+ channel: a comparison with nifedipine.
Topics: Animals; Benzopyrans; Calcium; Cromakalim; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Picolines; Potassium Channels; Pyrans; Pyrroles; Trachea | 1991 |
Evidence that pinacidil may promote the opening of ATP-sensitive K+ channels yet inhibit the opening of Ca2(+)-activated K+ channels in K(+)-contracted canine mesenteric artery.
Topics: Adenosine Triphosphate; Animals; Benzopyrans; Calcium; Cromakalim; Dogs; Female; Glyburide; Guanidines; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Pinacidil; Potassium; Potassium Channels; Pyrroles; Rubidium Radioisotopes | 1990 |
A comparison of the actions of cromakalim and nifedipine on rabbit isolated mesenteric artery.
Topics: Animals; Benzopyrans; Blood Pressure; Cell Membrane; Cromakalim; Electric Stimulation; Glyburide; Humans; In Vitro Techniques; Infant, Newborn; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Perfusion; Potassium Channels; Pyrroles; Rabbits | 1990 |
Counteraction of nifedipine-induced hyperglycaemia by metformin.
Topics: Animals; Glyburide; Hyperglycemia; Male; Metformin; Nifedipine; Rats | 1990 |
Specific antagonism by glibenclamide of negative inotropic effects of potassium channel openers in canine atrial muscle.
Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dogs; Female; Glyburide; Guanidines; Heart Atria; Male; Myocardial Contraction; Niacinamide; Nicorandil; Nifedipine; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents | 1990 |
Inhibition by sulphonylureas of vasorelaxation induced by K+ channel activators in vitro.
Topics: Animals; Antihypertensive Agents; Benzopyrans; Cromakalim; Drug Interactions; Glipizide; Glyburide; Guanidines; In Vitro Techniques; Male; Nifedipine; Norepinephrine; Pinacidil; Potassium Channels; Potassium Chloride; Pyrroles; Rabbits; Sulfonylurea Compounds; Tolbutamide; Vasodilator Agents | 1989 |
Phenylephrine-induced rhythmic activity in the rabbit ear artery.
Topics: Animals; Arginine; Arteries; Charybdotoxin; Ear, External; Endothelium, Vascular; Glyburide; In Vitro Techniques; Indomethacin; Male; Nifedipine; Nitric Oxide; Nitroarginine; omega-N-Methylarginine; Periodicity; Phenylephrine; Potassium Channel Blockers; Prostaglandin Antagonists; Rabbits; Scorpion Venoms; Vasoconstriction | 1993 |
Role of calcium-activated potassium channels in the relaxation of tracheal smooth muscles by forskolin.
Topics: Animals; Apamin; Calcium; Carbachol; Charybdotoxin; Colforsin; Cyclic AMP; Drug Interactions; Electrophysiology; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Trachea | 1994 |
Propagation of impulses in the guinea-pig ureter and its blockade by calcitonin gene-related peptide (CGRP).
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Cromakalim; Electric Stimulation; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyrroles; Tetrodotoxin; Ureter | 1995 |
Effect of KRN2391 on venous return: comparison with other vasodilators.
Topics: Animals; Benzopyrans; Cromakalim; Dogs; Female; Glyburide; Hemodynamics; Male; Niacinamide; Nicorandil; Nifedipine; Nitroglycerin; Potassium Channels; Pyridines; Pyrroles; Vasodilator Agents; Veins | 1993 |
Participation of calcium, released from the IP3-sensitive Ca-store in activation of Ca-dependent potassium conductance of ileal smooth muscle cells.
Topics: Animals; Apamin; Calcium; Charybdotoxin; Egtazic Acid; Glyburide; Guinea Pigs; Heparin; Ileum; In Vitro Techniques; Indoles; Inositol 1,4,5-Trisphosphate; Membrane Potentials; Muscle, Smooth; Nifedipine; Potassium Channels; Ruthenium Red; Scorpion Venoms | 1993 |
A simple method for measurement of ureteric peristaltic function in vivo and the effects of drugs acting on ion channels applied from the ureter lumen in anesthetized rats.
Topics: 4-Aminopyridine; Anesthesia; Animals; Benzopyrans; Cromakalim; Glyburide; Ion Channels; Lidocaine; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyrroles; Rats; Rats, Sprague-Dawley; Ureter; Vasodilator Agents | 1993 |
Drug-induced endothelium-dependent and -independent relaxations in isolated resistance vessels taken from simultaneously hypertensive and streptozotocin-diabetic rats.
Topics: Animals; Benzopyrans; Bradykinin; Calcium; Cromakalim; Diabetes Mellitus, Experimental; Endothelium, Vascular; Glyburide; Histamine; Hypertension; Male; Mesenteric Arteries; Methacholine Chloride; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Nitroprusside; Potassium Channels; Potassium Chloride; Pyrroles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Streptozocin; Vascular Resistance; Vasodilation; Vasodilator Agents | 1994 |
Cellular mechanisms of hypoxia-induced contraction in human and rat pulmonary arteries.
Topics: Aged; Animals; Benzopyrans; Calcium; Calcium Channels; Cromakalim; Glyburide; Humans; Hypoxia; In Vitro Techniques; Iodoacetates; Iodoacetic Acid; Male; Middle Aged; Muscle, Smooth, Vascular; Nifedipine; Potassium Channels; Pulmonary Artery; Pyrroles; Rats; Rats, Wistar; Vasoconstriction; Verapamil | 1995 |
Inhibition of ATP-sensitive K+ channel by a non-sulfonylurea compound KAD-1229 in a pancreatic beta-cell line, MIN 6 cell.
Topics: Action Potentials; Adenosine Triphosphate; Binding, Competitive; Calcium; Cell Membrane; Cobalt; Dose-Response Relationship, Drug; Drug Synergism; Fura-2; Glucose; Glyburide; Humans; Hypoglycemic Agents; Indoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Isoindoles; Membrane Potentials; Nifedipine; Pancreatic Neoplasms; Patch-Clamp Techniques; Potassium Channel Blockers; Tumor Cells, Cultured | 1994 |
Pharmacological analysis of the effect of KRN2391 on coronary vasculature in perfused rat heart.
Topics: Animals; Benzopyrans; Coronary Circulation; Cromakalim; Dose-Response Relationship, Drug; Glyburide; In Vitro Techniques; Male; Nifedipine; Perfusion; Potassium Channels; Pyridines; Pyrroles; Rats; Rats, Wistar; Vasodilator Agents | 1994 |
Tetraethylammonium selectively stimulates secretion from noradrenergic bovine chromaffin cells.
Topics: 4-Aminopyridine; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; Drug Interactions; Drug Synergism; Epinephrine; Glyburide; Nifedipine; Norepinephrine; Ouabain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tolbutamide | 1994 |
Insulin secretion by the pancreatic beta cell of aged rats.
Topics: Aging; Animals; Colforsin; Dose-Response Relationship, Drug; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Potassium; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1994 |
Effects of levcromakalim on ureteral peristaltic function and cystometrogram in rats.
Topics: Administration, Topical; Animals; Benzopyrans; Cromakalim; Glyburide; Injections, Intraperitoneal; Injections, Intravenous; Male; Nifedipine; Parasympatholytics; Pyrroles; Rats; Rats, Sprague-Dawley; Ureter; Urinary Bladder | 1993 |
NIP-121 is more effective than nifedipine in acutely reversing chronic pulmonary hypertension.
Topics: Altitude; Animals; Chronic Disease; Glyburide; Hemodynamics; Hypertension, Pulmonary; Hypoxia; Male; Nifedipine; Oxadiazoles; Piperidines; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasodilation | 1993 |
Lemakalim attenuates hypocapnia- and dry air-induced bronchoconstriction in canine peripheral airways.
Topics: Acetylcholine; Adenosine Triphosphate; Aerosols; Airway Resistance; Albuterol; Animals; Benzopyrans; Blood Pressure; Bronchoconstriction; Bronchodilator Agents; Cromakalim; Dogs; Glyburide; Heart Rate; Humidity; Hypocapnia; Injections, Intravenous; Lung; Male; Nifedipine; Potassium Channels; Pyrroles | 1993 |
The relaxant actions on guinea-pig trachealis of atherosperminine isolated from Fissistigma glaucescens.
Topics: Alkaloids; Animals; Benzopyrans; Calcium; Calmodulin; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Egtazic Acid; Epithelium; Female; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Nitroprusside; Phenanthrenes; Plants, Medicinal; Propranolol; Pyrroles; Theophylline; Trachea; Vasodilator Agents | 1993 |
Endothelial function in deoxycorticosterone-NaCl hypertension: effect of calcium supplementation.
Topics: Acetylcholine; Adenosine Diphosphate; Animals; Apamin; Arginine; Blood Pressure; Calcium, Dietary; Desoxycorticosterone; Endothelium, Vascular; Glyburide; Hypertension; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nifedipine; Nitroprusside; Norepinephrine; Potassium Channels; Rats; Rats, Inbred WKY; Serotonin; Sodium Chloride; Vasodilation | 1996 |
Pharmacodynamic behaviour of isolated resistance vessels obtained from hypertensive-diabetic rats.
Topics: Animals; Benzopyrans; Blood Glucose; Calcium Channels; Calcium Chloride; Cromakalim; Glyburide; Hypertension; In Vitro Techniques; Male; Mesenteric Arteries; Methacholine Chloride; Methoxamine; Muscle Contraction; Muscle, Smooth; Nifedipine; Nitroprusside; Norepinephrine; Obesity; Potassium Channels; Potassium Chloride; Pyrroles; Rats; Rats, Zucker; Serotonin; Tunica Media; Vascular Resistance; Vasoconstrictor Agents; Vasodilator Agents | 1996 |
Analysis of relaxation and repolarization mechanisms of nicorandil in rat mesenteric artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Benzopyrans; Calcium Channel Blockers; Cromakalim; Electrophysiology; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Nifedipine; Potassium Channels; Prostaglandin Endoperoxides, Synthetic; Pyrroles; Rats; Rats, Sprague-Dawley; Thromboxane A2; Vasoconstrictor Agents; Vasodilator Agents | 1996 |
Interaction between the L-type Ca2+ channel and the Ca(2+)-activated K+ channel in the fluctuating myogenic contraction in the rabbit basilar artery.
Topics: Animals; Basilar Artery; Calcium; Calcium Channel Blockers; Calcium Channels; Charybdotoxin; Glyburide; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Nifedipine; Potassium Channel Blockers; Potassium Channels; Rabbits; Vasoconstriction | 1996 |
Effects of BKCa channels on the reduction of cytosolic Ca2+ in cGMP-induced relaxation of guinea-pig trachea.
Topics: Animals; Apamin; Atrial Natriuretic Factor; Calcium; Cyclic GMP; Cytosol; Extracellular Space; Glyburide; Guinea Pigs; Intracellular Fluid; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nifedipine; Peptides; Potassium; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Trachea | 1997 |
Y-26763 protects the canine heart from a stunning injury through opening of the KATP channels.
Topics: Adenosine Triphosphate; Animals; Antihypertensive Agents; Benzopyrans; Calcium Channel Blockers; Dogs; Female; Glyburide; Hemodynamics; Male; Myocardial Stunning; Nifedipine; Potassium Channels | 1997 |
Interactions between neuropeptide Y and the adenylate cyclase pathway in rat mesenteric small arteries: role of membrane potential.
Topics: 4-Aminopyridine; Acetylcholine; Adenylyl Cyclases; Animals; Charybdotoxin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dichlororibofuranosylbenzimidazole; Gadolinium; Glyburide; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Nifedipine; Potassium Channels; Rats; Rats, Wistar; Thionucleotides | 1997 |
Effects of nitroprusside and nicorandil on catecholamine secretion and calcium mobilization in cultured bovine adrenal chromaffin cells.
Topics: Adrenal Medulla; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin Cells; Glyburide; Niacinamide; Nicorandil; Nifedipine; Nitroprusside; Vasodilator Agents | 1997 |
Microvascular permeability with sulfonylureas in normal and diabetic hamsters.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Capillary Permeability; Cricetinae; Dextrans; Diabetes Mellitus, Experimental; Diazoxide; Disease Models, Animal; Dose-Response Relationship, Drug; Fluorescein-5-isothiocyanate; Gliclazide; Glyburide; Histamine; Hypoglycemic Agents; Insulin; Macromolecular Substances; Male; Mesocricetus; Nifedipine; Potassium Channels; Reperfusion Injury; Streptozocin; Sulfonylurea Compounds | 1997 |
The effects of nifedipine and other calcium antagonists on the glibenclamide-sensitive K+ currents in smooth muscle cells from pig urethra.
Topics: Animals; Barium; Calcium Channel Blockers; Cromakalim; Female; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Muscle, Smooth; Nifedipine; Patch-Clamp Techniques; Potassium Channels; Swine; Urethra | 1998 |
Rapid activation and nuclear translocation of mitogen-activated protein kinases in response to physiological concentration of glucose in the MIN6 pancreatic beta cell line.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Nucleus; Colforsin; Egtazic Acid; Enzyme Activation; Glucose; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Kainic Acid; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nifedipine; Potassium; Receptors, Glutamate | 1998 |
Hyperpolarization and slowing of the rate of contraction in human uterus in pregnancy by prostaglandins E2 and f2alpha: involvement of the Na+ pump.
Topics: Albuterol; Calcium; Calcium Channel Blockers; Charybdotoxin; Cyclic AMP; Dinoprost; Dinoprostone; Enzyme Inhibitors; Female; Glyburide; Humans; Hypoglycemic Agents; Iloprost; Membrane Potentials; Myometrium; Nifedipine; Ouabain; Potassium; Potassium Channel Blockers; Potassium Channels; Pregnancy; Sodium-Potassium-Exchanging ATPase; Sympathomimetics; Tetraethylammonium; Uterine Contraction; Vasodilator Agents | 1999 |
Cellular characterization of pituitary adenoma cell line (AtT20 cell) transfected with insulin, glucose transporter type 2 (GLUT2) and glucokinase genes: insulin secretion in response to physiological concentrations of glucose.
Topics: Adenoma; Calcium Channel Blockers; Corticotropin-Releasing Hormone; Diazoxide; Gene Expression; Glucokinase; Glucose; Glucose Transporter Type 2; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Monosaccharide Transport Proteins; Nifedipine; Pituitary Neoplasms; Potassium Chloride; Transfection; Tumor Cells, Cultured | 1998 |
The ginsenoside Rg3 evokes endothelium-independent relaxation in rat aortic rings: role of K+ channels.
Topics: Animals; Antineoplastic Agents, Phytogenic; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Cromakalim; Dose-Response Relationship, Drug; Endothelium, Vascular; Ginsenosides; Glyburide; In Vitro Techniques; Male; Muscle Relaxation; Nifedipine; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Rats; Rats, Sprague-Dawley; Rubidium Radioisotopes; Saponins; Tetraethylammonium; Vasodilator Agents | 1999 |
Growth inhibitory effects of ATP and its derivatives on human fibroblasts immortalized with 60Co-gamma rays.
Topics: Adenosine Triphosphate; Cell Division; Cell Line; DNA Fragmentation; Gamma Rays; Glyburide; Humans; Nifedipine; Receptors, Purinergic P2 | 2000 |
Arterial flow induces changes in saphenous vein endothelium proteins transduced by cation channels.
Topics: Arteries; Biomarkers; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Endothelium, Vascular; Glyburide; Humans; In Vitro Techniques; Intercellular Adhesion Molecule-1; Nifedipine; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Perfusion; Potassium Channel Blockers; Potassium Channels; Proteins; Regional Blood Flow; Saphenous Vein; Tetraethylammonium; Thromboplastin; Vascular Cell Adhesion Molecule-1 | 2000 |
Opposing roles of K(+) and Cl(-) channels in maintenance of opossum lower esophageal sphincter tone.
Topics: 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Action Potentials; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Chloride Channels; Esophagogastric Junction; Glyburide; Isometric Contraction; Microelectrodes; Muscle, Smooth; Nifedipine; Niflumic Acid; Opossums; Potassium Channels | 2000 |
The involvement of L-type Ca(2+) channels in the relaxant effects of the ATP-sensitive K(+) channel opener ZD6169 on pig urethral smooth muscle.
Topics: Adenosine Triphosphate; Amides; Animals; Barium; Benzophenones; Calcium Channel Blockers; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gene Expression; Glyburide; In Vitro Techniques; Membrane Potentials; Muscle Relaxation; Muscle, Smooth; Nifedipine; Potassium Channels; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Swine; Urethra | 2001 |
Substance P induces inward current and regulates pacemaker currents through tachykinin NK1 receptor in cultured interstitial cells of Cajal of murine small intestine.
Topics: 4-Aminopyridine; Action Potentials; Alkaloids; Animals; Benzophenanthridines; Calcium; Cations, Divalent; Cells, Cultured; Electrophysiology; Enteric Nervous System; Female; Glyburide; Intestine, Small; Ion Channels; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nifedipine; Phenanthridines; Receptors, Neurokinin-1; Sinoatrial Node; Sodium; Substance P; Tachykinins; Tetraethylammonium; Tetrodotoxin | 2004 |
Pacemaker potentials generated by interstitial cells of Cajal in the murine intestine.
Topics: Animals; Anti-Arrhythmia Agents; Biological Clocks; Caffeine; Calcium Channel Blockers; Central Nervous System Stimulants; Electrophysiology; Glyburide; In Vitro Techniques; Intestine, Small; Membrane Potentials; Mibefradil; Mice; Mice, Inbred BALB C; Myocytes, Smooth Muscle; Nifedipine; Pinacidil; Vasodilator Agents | 2005 |
Glucose-stimulated DNA synthesis through mammalian target of rapamycin (mTOR) is regulated by KATP channels: effects on cell cycle progression in rodent islets.
Topics: Animals; Blotting, Western; Calcium; Cell Cycle; Cell Division; Cell Proliferation; Cells, Cultured; Cytosol; Diazoxide; Dose-Response Relationship, Drug; Flow Cytometry; G2 Phase; Glucose; Glyburide; Islets of Langerhans; Male; Nifedipine; Potassium; Potassium Channels; Protein Kinases; Rats; Rats, Sprague-Dawley; S Phase; Sirolimus; Thymidine; TOR Serine-Threonine Kinases | 2006 |
Relative contribution of intracellular and extracellular Ca2+ to alpha2-adrenoceptor-mediated contractions of ovine pulmonary artery.
Topics: Adrenergic alpha-Agonists; Animals; Calcium; Calcium Channel Blockers; Cyclic AMP; Cyclic GMP; Glyburide; Guanfacine; Indoles; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nucleotides, Cyclic; Pulmonary Artery; Receptors, Adrenergic, alpha-2; Sheep; Vasoconstriction; Vasodilator Agents | 2006 |
Role of ion channel modifiers in reversal of morphine-induced gastrointestinal inertia by prokinetic agents in mice.
Topics: Analgesics, Opioid; Animals; Benzamides; Calcium Channels; Domperidone; Gastrointestinal Tract; Glyburide; Intestine, Small; Ion Channels; Kinetics; Mice; Minoxidil; Morphine; Morpholines; Nifedipine; Time Factors | 2008 |
Vasorelaxant effect of a self-etch adhesive system through calcium antagonistic action.
Topics: 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Dentin-Bonding Agents; Endothelium, Vascular; Enzyme Inhibitors; Epoprostenol; Glyburide; Indomethacin; Male; Materials Testing; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Potassium Channels, Voltage-Gated; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Time Factors; Vasoconstrictor Agents; Vasodilator Agents | 2008 |
Anemoside A3-induced relaxation in rat renal arteries: role of endothelium and Ca2+ channel inhibition.
Topics: Animals; Apamin; Arteries; Biological Factors; Calcium; Calcium Channel Blockers; Capsaicin; Charybdotoxin; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Glyburide; Kidney; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myography; Nifedipine; Plant Extracts; Plant Roots; Potassium Channels; Potassium Chloride; Pulsatilla; Rats; Rats, Sprague-Dawley; Saponins; Tetraethylammonium; Triterpenes; Vasodilator Agents | 2010 |
Modulation of adrenergic responses of human vas deferens by K+ channel inhibitors.
Topics: Adult; Apamin; Calcium; Calcium Channels, L-Type; Charybdotoxin; Electric Stimulation; Glyburide; Humans; Ion Transport; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Peptides; Potassium; Potassium Channel Blockers; Potassium Channels; Receptors, Adrenergic, alpha-1; Tetraethylammonium; Vas Deferens | 2010 |
Vasodilatory effect of hydroxyethyl methacrylate and triethylene glycol dimethacrylate in rat aorta through calcium antagonistic action.
Topics: 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Calcium Chloride; Composite Resins; Cyclooxygenase Inhibitors; Dental Materials; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Indomethacin; Male; Methacrylates; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide Synthase; Polyethylene Glycols; Polymethacrylic Acids; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Transducers; Vasoconstrictor Agents; Vasodilator Agents | 2011 |
Inhibition of ATP-sensitive K+ channels and L-type Ca2+ channels by amiodarone elicits contradictory effect on insulin secretion in MIN6 cells.
Topics: Amiodarone; Animals; Anti-Arrhythmia Agents; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; KATP Channels; Membrane Potentials; Mice; Nifedipine; Osmolar Concentration; Patch-Clamp Techniques; Potassium Channel Blockers; Quinidine | 2011 |
Low glucose sensitivity and polymodal chemosensing in neonatal rat adrenomedullary chromaffin cells.
Topics: Animals; Animals, Newborn; Calcium; Calcium Channel Blockers; Catecholamines; Cell Hypoxia; Cells, Cultured; Chromaffin Cells; Glucose; Glyburide; Hypercapnia; Membrane Potentials; Nickel; Nifedipine; Potassium Channels; Rats; Rats, Wistar | 2011 |
Role of calcium and potassium channels in effects of hydrogen sulfide on frog myocardial contractility.
Topics: 4-Aminopyridine; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Electric Stimulation; Glyburide; Heart; Hydrogen Sulfide; In Vitro Techniques; KATP Channels; Minoxidil; Myocardial Contraction; Myocardium; Nifedipine; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Rana ridibunda; Tetraethylammonium | 2011 |
Highly efficient miniaturized coprecipitation screening (MiCoS) for amorphous solid dispersion formulation development.
Topics: Acrylic Resins; Chemical Precipitation; Chemistry, Pharmaceutical; Felodipine; Glyburide; Methylcellulose; Miniaturization; Nifedipine; Polymethacrylic Acids; Powders; Solubility | 2013 |
Significance of K(ATP) channels, L-type Ca²⁺ channels and CYP450-4A enzymes in oxygen sensing in mouse cremaster muscle arterioles in vivo.
Topics: Animals; Arterioles; Calcium Channels, L-Type; Cromakalim; Cytochrome P-450 Enzyme System; Glyburide; Hydroxyeicosatetraenoic Acids; KATP Channels; Male; Mice; Mice, Inbred C57BL; Muscle, Skeletal; Muscle, Smooth, Vascular; Nifedipine; Nitric Oxide Synthase; Oxygen; Retinoic Acid 4-Hydroxylase; Vasoconstriction; Vasodilation | 2013 |
The Possible Mechanisms of the Impaired Insulin Secretion in Hypothyroid Rats.
Topics: Acetylcholine; Animals; Blood Glucose; Glucokinase; Glyburide; Hexokinase; Hypoglycemic Agents; Hypothyroidism; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Rats; Rats, Wistar; Thyroxine; Triiodothyronine | 2015 |
Impaired glucose-stimulated insulin secretion and reduced β-cell mass in pancreatic islets of hyperthyroid rats.
Topics: Animals; Calcium Channels, L-Type; Diazoxide; Glucose; Glucose Tolerance Test; Glyburide; Hyperthyroidism; Hypoglycemic Agents; Insulin; Insulin-Secreting Cells; KATP Channels; Male; Nifedipine; Rats; Rats, Sprague-Dawley; Thyroid Hormones; Thyroxine | 2016 |
Combination Therapy of Nifedipine and Sulphonylureas Exhibits a Mutual Antagonistic Effect on the Endothelial Cell Dysfunction Induced by Hyperglycemia Linked to Vascular Disease.
Topics: Antihypertensive Agents; Biphenyl Compounds; Cell Movement; Diabetic Angiopathies; Drug Synergism; Endothelial Cells; Glucose; Glyburide; Human Umbilical Vein Endothelial Cells; Humans; Hyperglycemia; Hypoglycemic Agents; Irbesartan; Metformin; Nifedipine; Oxygen; Sulfonylurea Compounds; Tetrazoles | 2016 |
The beneficial effect of clove essential oil and its major component, eugenol, on erectile function in diabetic rats.
Topics: Animals; Clove Oil; Diabetes Mellitus, Experimental; Erectile Dysfunction; Eugenol; Glyburide; In Vitro Techniques; Injections; Male; Nifedipine; Nitric Oxide Synthase; Oils, Volatile; Penile Erection; Penis; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Soluble Guanylyl Cyclase; Tetraethylammonium | 2020 |
Aqueous extract of oakmoss produces antihypertensive activity in L-NAME-induced hypertensive rats through sGC-cGMP pathway.
Topics: Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Aorta, Thoracic; Arterial Pressure; Blood Pressure; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Glyburide; Hypertension; KATP Channels; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide Synthase; Parmeliaceae; Plant Extracts; Propranolol; Rats; Rats, Wistar; Resins, Plant; Terpenes; Vasodilator Agents | 2021 |
Pulmonary Microcirculation in Experimental Model of Pulmonary Thromboembolism after Pretreatment with Chloroquine.
Topics: Adenosine Triphosphate; Animals; Chloroquine; Glyburide; Lung; Microcirculation; Models, Theoretical; Nifedipine; Pulmonary Embolism; Rabbits; Vascular Resistance | 2023 |