glyburide and glipizide

glyburide has been researched along with glipizide in 185 studies

Research

Studies (185)

TimeframeStudies, this research(%)All Research%
pre-199042 (22.70)18.7374
1990's59 (31.89)18.2507
2000's37 (20.00)29.6817
2010's39 (21.08)24.3611
2020's8 (4.32)2.80

Authors

AuthorsStudies
Gehlert, DR; Krushinski, JH; Mais, DE; Robertson, DW; Schober, DA; Thompson, DC1
Topliss, JG; Yoshida, F1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Barton, P; Luker, T; Wenlock, MC1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Melander, A; Wåhlin-Boll, E2
Balant, L1
Blohmé, G; Waldenström, J1
Abdel-Hay, MM; Ghanem, MH; Guirgis, FK1
Gotfredsen, CF1
Codaccioni, JL; Fontaine, G1
Ceretti, AP; Emanueli, A; Losi, S; Orsini, G1
Müller, WE; Wollert, U1
Brunová, E1
Balant, L; Fabre, J; Zahnd, GR1
Alric, R; Loubatières, AL; Loubatieres-Mariani, MM; Ribes, G; Sorial, G; Tarasco, A1
Alric, R; Lignon, F; Loubatières, A; Manteghetti, M; Puech, R1
Madhavan, R; Sankaran, JR; Seshasaianam, C; Seshiah, V; Shanker, R; Sundaram, A; Venkataraman, S1
Carter, BL; Helling, DK; McCormick, WC; Noyes, MA; Ramirez, R1
Gwilt, M; Henderson, CG; Orme, J; Rourke, JD2
Bird, DM; Cameron, DP; Ma, A; McIntyre, HD; Patterson, CA1
Aguilar-Bryan, L; Bryan, J; Nelson, DA1
Lazdunski, M; Schaeffer, P1
Brodows, RG1
Harrower, AD2
Bemis, KG; Ertel, PJ; Robertson, DW; Steinberg, MI; Wiest, SA; Zimmerman, KM1
Brown, TJ; Raeburn, D1
Gackenheimer, SL; Gehlert, DR; Mais, DE; Robertson, DW1
Kidd, GS; McDermott, MT; Simcic, KJ; White, JC1
Feng, JG; Shi, MZ; Zheng, JJ1
Aranyi, Z; Ballagi-Pordány, G; Koltai, MZ; Köszeghy, A; Pogátsa, G1
Antal, EJ; Jaber, LA; Komanicky, P; Wenzloff, NJ1
Huupponen, R; Karvonen, I; Rytömaa, K; Sotaniemi, EA; Vierimaa, E; Vuoti, MJ1
Boutagy, JS; Shenfield, GM; Webb, C1
Dash, RJ; Khandekar, S; Sethi, BK1
Harrower, AD; Wong, C1
Reckless, JP; Simpson, HC; Stirling, CA; Sturley, R1
Lenzen, S; Männer, K; Panten, U; Trube, G; Zünkler, BJ1
Schmitt, JK1
Wilson, C1
Morrison, AD; Shank, WA1
Kure, J1
Pollet, RJ; Rogers, BJ; Standaert, ML1
DeFronzo, RA; Groop, L; Groop, PH; Luzi, L; Melander, A; Ratheiser, K; Simonson, DC1
Boyd, AE; Gaines, KL; Hamilton, S1
Adamson, U; Lins, PE; Lundblad, S; Persson-Trotzig, E1
Borisova, AM; Georgieva, R; Koev, D; Taneva, T1
Kuhn, T1
Groop, L; Salo, S1
Lenzen, S; Panten, U; Schwanstecher, M; Wallasch, A1
Kilo, C1
Arner, P; Bolinder, J; Ostman, J1
Gerich, JE1
Pearson, JG1
Fyhrqvist, F; Groop, L; Groop, PH; Melander, A; Tolppanen, EM; Tötterman, KJ; Wåhlin-Boll, E1
Baker, DE; Campbell, RK1
Hellman, B; Sehlin, J; Täljedal, IB1
Ahrén, B; Scherstén, B1
Delawter, DE; Moss, JM1
Chadwick, T; Harkness, J; Hartog, M; Paisey, RB1
Loubatieres-Mariani, MM1
Melander, A; Sartor, G; Scherstén, B; Wåhlin-Boll, E2
Groop, L; Harno, K1
Chow, CC; Cockram, CS; Sorensen, JP; Tsang, LW1
Akkan, AG; Malaisse, WJ; Sener, A1
Balabolkin, MI; Maksumova, MA; Orekhov, AN; Slavina, ES; Sobenin, IA1
Bachmann, C; Chudziak, F; Löser, S; Panten, U; Schwanstecher, M1
Elliott, BD; Johnson, R; Langer, O; Prihoda, T; Schenker, S1
Birkeland, KI; Furuseth, K; Melander, A; Mowinckel, P; Vaaler, S1
Nielsen-Kudsk, JE; Thirstrup, S1
Amoroso, S; Bernardi, H; De Weille, JR; Epelbaum, J; Fosset, M; Lazdunski, M; Mourre, C; Slama, A1
Chen, H; Duckworth, WC; Hamel, FG; Siford, G1
Miller, JL; Rose, LI; Salman, K; Shulman, LH1
Jaber, LA; Lewis, NJ; Neale, AV; Slaughter, RL1
Hong, KW; Kwon, YJ; Lee, WS; Rhim, BY; Yu, SS1
Ammälä, C; Berggren, PO; Bertorello, AM; Bokvist, K; Chibalin, A; Deeney, JT; Eliasson, L; Flatt, PR; Gäbel, J; Gromada, J; Larsson, O; Lindström, P; Renström, E; Rhodes, CJ; Rorsman, P1
Ferguson, JE; Jacob, G; Landers, JP; Lawson, GM; Machacek, D; Núñez, M; Oda, RP1
Gross, AS; Rieutord, A; Shenfield, GM; Stupans, I1
Grenhoff, J; Johnson, SW1
Selvaag, E; Thune, P1
Kivistö, KT; Laine, K; Lehto, P; Neuvonen, PJ1
Selvaag, E1
Banerjee, A; Cain, BS; Cleveland, JC; Harken, AH; Meldrum, DR1
Abenhaim, L; Monette, J; van Staa, T1
Anderson, BD; Anderson, DL; Fenn, J; Gorman, SE; Krenzelok, EP; Muir, SJ; Rodgers, GC; Rose, SR; Spiller, HA; Villalobos, D1
Landers, JP; Lawson, GM; Oda, RP; Roche, ME1
Anderson, D; Briscoe, TA; Cooper, GS; Usifo, OS1
Aubin, R; Lajeunesse, D; Lapointe, JY; Moreau, R1
Luo, M; O'Brien, RC1
Burge, MR; Fischette, C; Qualls, CR; Schade, DS; Schmitz-Fiorentino, K1
Bernardi, G; Federici, M; Guatteo, E; Knöpfel, T; Mercuri, NB; Siniscalchi, A1
Shorr, RI1
Bernabei, R; Carbonin, P; Gambassi, G1
Nadel, HL1
Bataille, D; Blache, P; Gros, L; Salazar, G; Virsolvy, A1
André, P1
Brioni, JD; Gopalakrishnan, M; Miller, TR; Molinari, EJ; Monteggia, LM; Scott, VE; Sullivan, JP; Taber, RD; Whiteaker, KL1
Ersöz, B; Girgin, FK; Menteş, G; Sözmen, EY; Tüzün, S1
Courtois, P; Herbaut, C; Malaisse, WJ; Sener, A; Turc, A1
Chugh, SN; Kakkar, R; Kharb, S; Sharma, A; Singh, GP1
Gomis, R; Jones, NP; Patwardhan, RN; Squatrito, S; Wolffenbuttel, BH1
Brioni, JD; Gopalakrishnan, M; Molinari, EJ; Monteggia, LM; Roch, JM; Scott, VE; Shieh, CC; Sullivan, JP; Whiteaker, KL1
Bryer-Ash, M; Bush, A; Fisher, JN; Kaminska, E; Kitabchi, AE; Pitts, K; Sherman, A1
Galli Kienle, M; Magni, F; Marazzini, L; Monti, L; Pereira, S1
Eisenhofer, G; Harvey-White, J; He, LP; Hrycyna, C; Kopin, IJ; Lamensdorf, I; Nechushtan, A; Rojas, E; Tjurmina, O1
de Smet, PA; Fischer, HR1
Chan, JC; Cockram, CS; Critchley, JA; Hallengren, B; Jönsson, A; Melander, A; Rydberg, T; Vaaler, S1
Backman, JT; Kivistö, KT; Neuvonen, M; Neuvonen, PJ; Niemi, M1
Gottsäter, M; Lindberg, G; Lindwall, K; Melander, A; Olsson, J; Tisell, A1
Cozma, LS; Dunseath, GJ; Langendorg, KW; Luzio, SD; Owens, DR; Pieber, T1
Bussing, R; Gende, A1
Argüelles, CF; Granados-Soto, V; Ortiz, MI1
Mutalik, S; Udupa, N2
Aronson, D; Burger, AJ; Mittleman, MA1
Rochester, CD; Samuel, J1
Bell, CF; Botteman, MF; Braunstein, SN; Devine, ST; Ramsdell, JW; Stephens, JM1
Aburuz, S; McElnay, J; Millership, J1
Debska, G; Kunz, WS; Skalska, J; Szewczyk, A1
Ambrose, PJ; Briggs, GG; Donat, DJ; Feig, DS; Klein, J; Koren, G; Kraemer, JM; Moskovitz, DN; Nageotte, M; Padilla, G; Wan, S1
Boettner, WA; Flynn, DM; Gernhardt, SS; Knight, DR; Levy, CB; Plowchalk, DR; Smith, AH; Soeller, WC; Tracey, WR; Treadway, JL; Wisniecki, P1
Choudhury, H; Harisudhan, T; Mullangi, R; Srinivas, NR; Venkatesh, P1
Jin, SH; Li, ZR; Shi, YQ; Yao, J1
Krishnarajah, G; Lyu, R; Mavros, P; Vexiau, P; Yin, D1
Mogensen, CE; Sadikot, SM1
Djokanovic, N; Finkelstein, Y; Garcia-Bournissen, F; Glatstein, MM; Koren, G1
Ee, JW; Kwon, SW; Lee, J; Lee, WJ; Park, JH; Shaodong, J1
Arrigain, S; Atreja, A; Jain, A; Kattan, MW; Pantalone, KM; Wells, BJ; Yu, C; Zimmerman, RS2
Bartley, EP; Hurren, KM; O'Neill, JL; Ronis, DL1
Bilker, WB; Brensinger, CM; Hennessy, S; Schelleman, H; Wan, F1
Heikkilä, P; Huupponen, R; Laine, K; Tirkkonen, T1
Aguilera, E; Fasano, CJ; Heard, K; O'Malley, GF; Rowden, AK1
Chan, JC; Chow, CC; Ko, GT; Kong, AP; Luk, AO; Ma, RC; Ng, VW; Ozaki, R; So, WY; Tong, PC; Yang, X; Yu, LW1
Andersson, C; Gislason, GH; Hansen, PR; Jørgensen, CH; Køber, L; Mérie, C; Norgaard, ML; Olesen, JB; Schmiegelow, M; Sørensen, R; Torp-Pedersen, C; Vaag, A; Weeke, P1
Burns, BD; Levine, M; Lovecchio, F; Pizon, AF; Riley, BD; Ruha, AM; Thomas, SH1
Abdelmoneim, AS; Brocks, DR; Hasenbank, SE; Light, PE; Seubert, JM; Simpson, SH1
Cantrell, M; Egge, JA; Shaw, RF; Skoff, RA; Waterbury, NV1
Cui, G; McCarty, NA; Song, B; Turki, HW1
Arrigain, S; Atreja, A; Jain, A; Kattan, MW; Nutter, B; Pantalone, KM; Wells, BJ; Yu, C; Zimmerman, RS1
Coley, KC; Deusenberry, CM; Donihi, AC; Korytkowski, MT1
Binz, TM; Neels, H; Schneider, S; Villani, N1
AbuKhader, MM; Alqtaishat, S; Khanfar, MA; Taha, MO1
Boyko, EJ; Floyd, JS; Forsberg, CW; Moore, K; Riley, K; Smith, NL; Wheeler, S1
Bilker, WB; Brensinger, CM; Flockhart, DA; Han, X; Hennessy, S; Li, L; Quinney, SK; Schelleman, H1
Jung, JS; Kim, CH; Kim, SJ; Kim, SS; Lim, SM; Park, SH; Sim, YB; Suh, HW1
Goodwin, JS; Holmes, HM; Kuo, YF; Raji, MA; Tan, A1
Goodwin, JS; Kuo, YF; Lin, YL; Parekh, TM; Raji, M; Tan, A1
Andersson, C; Fosbøl, EL; Gislason, G; Køber, L; Mogensen, UM; Scheller, NM; Schramm, TK; Torp-Pedersen, C; Vaag, A1
Bilker, WB; Brensinger, CM; Cardillo, S; Flockhart, DA; Flory, JH; Gagne, JJ; Han, X; Hennessy, S; Leonard, CE1
Bilker, WB; Brensinger, CM; Chiang, C; Han, X; Hennessy, S; Leonard, CE; Li, L1
Bergström, CAS; Edueng, K; Larsson, P; Mahlin, D1
Archdeacon, P; Axtman, S; Carnahan, RM; Cavagnaro, E; Chrischilles, EA; Fuller, C; Gagne, JJ; Hampp, C; Hennessy, S; Iyer, A; Leonard, CE; Panozzo, CA; Toh, S; Wang, SV; Woodworth, TS; Zhou, M1
Abdel-Kader, K; Greevy, RA; Griffin, MR; Horner, J; Hung, AM; Ikizler, TA; Matheny, ME; Parr, SK; Perkins, AM; Roumie, CL; Siew, ED; Speroff, T; Wilson, OD1
Ahmed, T; Punde, R; Sahu, R; Sangana, R; Subudhi, BB1
Aquilante, CL; Bilker, WB; Boudreau, DM; Brensinger, CM; Deo, R; Flory, JH; Gagne, JJ; Hennessy, S; Leonard, CE; Mangaali, MJ1
Cordiner, RLM; Pearson, ER1
Huang, HK; Yeh, JI1
Campillo, NE; García-Pérez, CA; Haupt, VJ; Herrera-Mayorga, V; Juárez-Saldivar, A; Reyes-Espinosa, F; Rivera, G; Saavedra, E; Salentin, S; Schroeder, M; Vázquez, C; Villalobos-Rocha, JC1
Bilker, WB; Brensinger, CM; Dawwas, GK; Dhopeshwarkar, N; Flory, JH; Gagne, JJ; Hennessy, S; Leonard, CE; Soprano, SE1
Chiriac, FL; Iancu, VI; Radu, GL; Scutariu, RE1
Bilker, WB; Brensinger, CM; Flory, JH; Hee Nam, Y; Hennessy, S; Leonard, CE1
Khasipo, AZ; Sagandira, CR; Watts, P1
Berry, SD; Hayes, KN; Munshi, MN; Riester, MR; Zullo, AR1
Gayakvad, B; Kothari, C; Patel, C; Patel, R; Solanki, R; Wadhwana, P1
Jannetto, PJ; Langman, LJ1

Reviews

12 review(s) available for glyburide and glipizide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
["First" and "second" generation sulfonylureas: distinction or difference? (author's transl)].
    Diabete & metabolisme, 1978, Volume: 4, Issue:2

    Topics: Animals; Chlorpropamide; Dose-Response Relationship, Drug; Glipizide; Glyburide; Half-Life; Humans; Hypoglycemic Agents; Kinetics; Structure-Activity Relationship; Sulfonylurea Compounds; Tolbutamide

1978
[Glipizide a new oral antidiabetic agent (comprehensive review)].
    Vnitrni lekarstvi, 1976, Volume: 22, Issue:6

    Topics: Animals; Blood Glucose; Chemical Phenomena; Chemistry; Diabetes Mellitus; Dogs; Drug Evaluation; Glipizide; Glyburide; Humans; Insulin; Insulin Secretion; Sulfonylurea Compounds

1976
Oral sulfonylureas for the treatment of type II diabetes: an update.
    Southern medical journal, 1986, Volume: 79, Issue:3

    Topics: Administration, Oral; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Hypersensitivity; Glipizide; Glyburide; Humans; Insulin Resistance; Kinetics; Liver; Nausea; Patient Education as Topic; Sulfonylurea Compounds

1986
The second generation oral sulfonylureas: glyburide and glipizide.
    American pharmacy, 1988, Volume: NS28, Issue:10

    Topics: Administration, Oral; Drug Interactions; Glipizide; Glyburide; Humans; Sulfonylurea Compounds

1988
Sulfonylureas in the treatment of diabetes mellitus--1985.
    Mayo Clinic proceedings, 1985, Volume: 60, Issue:7

    Topics: Blood Glucose; Body Weight; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Glipizide; Glyburide; Humans; Hypoglycemia; Insulin; Pancreas; Sulfonylurea Compounds

1985
Pharmacological and molecular characterization of ATP-sensitive K+ channels in the TE671 human medulloblastoma cell line.
    European journal of pharmacology, 1999, Apr-09, Volume: 370, Issue:2

    Topics: Adenosine Triphosphate; Animals; Barbiturates; Cells, Cultured; Cromakalim; Fluorescent Dyes; Fluorometry; Glipizide; Glyburide; Humans; Insulinoma; Isoxazoles; Medulloblastoma; Membrane Potentials; Muscle, Smooth; Parasympatholytics; Potassium Channels; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured

1999
[Timing of administration of sulfonyl urea derivatives].
    Nederlands tijdschrift voor geneeskunde, 2000, Jun-17, Volume: 144, Issue:25

    Topics: Biological Availability; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Drug Administration Schedule; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Tolbutamide

2000
Combination agents for diabetes.
    Advance for nurse practitioners, 2003, Volume: 11, Issue:6

    Topics: Adult; Diabetes Mellitus, Type 2; Drug Combinations; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Metformin; Rosiglitazone; Thiazoles; Thiazolidinediones

2003
Use of hypoglycemic drugs during lactation.
    Canadian family physician Medecin de famille canadien, 2009, Volume: 55, Issue:4

    Topics: Administration, Oral; Breast Feeding; Diabetes Mellitus, Type 2; Drug-Related Side Effects and Adverse Reactions; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Infant, Newborn; Lactation; Maternal Welfare; Milk, Human; Pregnancy; Pregnancy in Diabetics; Risk Assessment; Sulfonylurea Compounds

2009
Variations in tissue selectivity amongst insulin secretagogues: a systematic review.
    Diabetes, obesity & metabolism, 2012, Volume: 14, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Cardiovascular Diseases; Cricetinae; Cyclohexanes; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Ischemic Preconditioning, Myocardial; Isoindoles; Mice; Muscle, Smooth, Vascular; Myocytes, Cardiac; Nateglinide; Phenylalanine; Piperidines; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Risk Factors; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2012
Reflections on the sulphonylurea story: A drug class at risk of extinction or a drug class worth reviving?
    Diabetes, obesity & metabolism, 2019, Volume: 21, Issue:4

    Topics: Diabetes Mellitus; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glucagon-Like Peptide-1 Receptor; Glyburide; History, 20th Century; History, 21st Century; Humans; Hypoglycemic Agents; Insulin Secretion; Insulin-Secreting Cells; Metformin; Sodium-Glucose Transporter 2 Inhibitors; Sulfonylurea Compounds; Treatment Failure

2019

Trials

28 trial(s) available for glyburide and glipizide

ArticleYear
Glibenclamide and glipizide in maturity onset diabetes. A double-blind cross-over study.
    Acta medica Scandinavica, 1979, Volume: 206, Issue:4

    Topics: Aged; Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus; Double-Blind Method; Female; Glipizide; Glyburide; Humans; Insulin; Lipids; Male; Middle Aged; Placebos; Random Allocation; Sulfonylurea Compounds

1979
A controlled study of the hypoglycemic and insulinopoietic effect of glipizide and glibenclamide in non-diabetic human subjects.
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:4

    Topics: Adult; Blood Glucose; Clinical Trials as Topic; Female; Glipizide; Glyburide; Humans; Insulin; Middle Aged; Sulfonylurea Compounds; Time Factors

1975
Evaluation of glipizide and glyburide in a health maintenance organization.
    The Annals of pharmacotherapy, 1992, Volume: 26, Issue:10

    Topics: Adult; Aged; Blood Glucose; Diabetes Mellitus, Type 2; Drug Costs; Evaluation Studies as Topic; Female; Glipizide; Glyburide; Health Maintenance Organizations; Humans; Male; Middle Aged; Retrospective Studies; Texas

1992
Chronic sulfonylurea therapy augments basal and meal-stimulated insulin secretion while attenuating insulin responses to sulfonylurea per se.
    Diabetes care, 1992, Volume: 15, Issue:11

    Topics: Adult; Aged; Analysis of Variance; Blood Glucose; Body Mass Index; C-Peptide; Diabetes Mellitus, Type 2; Eating; Fasting; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Insulin; Insulin Secretion; Kinetics; Middle Aged; Time Factors

1992
Benefits and risks with glyburide and glipizide in elderly NIDDM patients.
    Diabetes care, 1992, Volume: 15, Issue:1

    Topics: Aged; Blood Glucose; C-Peptide; Diabetes Mellitus, Type 2; Eating; Fasting; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Male

1992
Efficacy of gliclazide in comparison with other sulphonylureas in the treatment of NIDDM.
    Diabetes research and clinical practice, 1991, Volume: 14 Suppl 2

    Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Diet, Diabetic; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Tolbutamide

1991
An evaluation of the therapeutic effects and dosage equivalence of glyburide and glipizide.
    Journal of clinical pharmacology, 1990, Volume: 30, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Blood Glucose; Diabetes Mellitus, Type 2; Double-Blind Method; Female; Glipizide; Glyburide; Humans; Male; Middle Aged; Random Allocation; Sulfonylurea Compounds; Therapeutic Equivalency

1990
Insulin and sulphonylurea in the therapy of type 2 diabetes.
    Diabetes research and clinical practice, 1990, Volume: 8, Issue:3

    Topics: Aged; Blood Glucose; C-Peptide; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Double-Blind Method; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Insulin; Lipids; Male; Metformin; Middle Aged; Placebos; Random Allocation; Sulfonylurea Compounds

1990
Comparison of secondary failure rate between three second generation sulphonylureas.
    Diabetes research (Edinburgh, Scotland), 1990, Volume: 13, Issue:1

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Diet, Diabetic; Follow-Up Studies; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Random Allocation

1990
Combination of insulin with glipizide increases peripheral glucose disposal in secondary failure type 2 diabetic patients.
    Diabetic medicine : a journal of the British Diabetic Association, 1990, Volume: 7, Issue:2

    Topics: Aged; Blood Glucose; C-Peptide; Cholesterol; Cholesterol Esters; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glipizide; Glucagon; Glucose Clamp Technique; Glyburide; Glycated Hemoglobin; Humans; Insulin; Lipoproteins; Male; Middle Aged; Sulfonylurea Compounds

1990
Clinical comparison of glipizide and glyburide.
    Diabetes care, 1989, Volume: 12, Issue:1

    Topics: Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Fasting; Glipizide; Glyburide; Humans; Middle Aged; Random Allocation; Sulfonylurea Compounds

1989
Glibenclamide improves the response to insulin treatment in non-insulin-dependent diabetics with second failure to sulfonylurea therapy.
    Acta medica Scandinavica, 1988, Volume: 223, Issue:2

    Topics: Adult; Aged; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Double-Blind Method; Drug Therapy, Combination; Female; Glipizide; Glyburide; Humans; Insulin; Male; Middle Aged; Sulfonylurea Compounds

1988
Combination of two sulfonylureas. Does it make sense.
    Diabetes care, 1988, Volume: 11, Issue:9

    Topics: Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glipizide; Glyburide; Glycated Hemoglobin; Glycosuria; Humans; Male; Middle Aged; Obesity; Sulfonylurea Compounds

1988
Multicenter comparison of glyburide and glipizide in the treatment of non-insulin-dependent diabetes mellitus.
    Clinical therapeutics, 1988, Volume: 10, Issue:3

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Glycated Hemoglobin; Hepatitis B Surface Antigens; Humans; Male; Middle Aged; Multicenter Studies as Topic; Randomized Controlled Trials as Topic; Sulfonylurea Compounds

1988
Pharmacokinetics and metabolic effects of glibenclamide and glipizide in type 2 diabetics.
    European journal of clinical pharmacology, 1985, Volume: 28, Issue:6

    Topics: Aged; Blood Glucose; Body Weight; C-Peptide; Diabetes Mellitus, Type 2; Double-Blind Method; Erythrocytes; Female; Gastric Inhibitory Polypeptide; Glipizide; Glucagon; Glyburide; Glycosuria; Humans; Insulin; Insulin Resistance; Kinetics; Male; Middle Aged; Random Allocation; Sulfonylurea Compounds

1985
Comparison of diabetic control in type 2 (non-insulin dependent) diabetic patients treated with different sulphonylureas.
    Current medical research and opinion, 1985, Volume: 9, Issue:10

    Topics: Aged; Chlorpropamide; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Middle Aged; Random Allocation; Sulfonylurea Compounds

1985
Comparison of insulin with or without continuation of oral hypoglycemic agents in the treatment of secondary failure in NIDDM patients.
    Diabetes care, 1995, Volume: 18, Issue:3

    Topics: Analysis of Variance; Biomarkers; Blood Glucose; Body Mass Index; C-Peptide; Cholesterol; Cholesterol, HDL; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Fructosamine; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Hexosamines; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Treatment Failure; Triglycerides

1995
Long-term randomized placebo-controlled double-blind therapeutic comparison of glipizide and glyburide. Glycemic control and insulin secretion during 15 months.
    Diabetes care, 1994, Volume: 17, Issue:1

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Double-Blind Method; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Insulin; Insulin Secretion; Male; Middle Aged; Time Factors

1994
The effect of stress on glycemic control in patients with type II diabetes during glyburide and glipizide therapy.
    Journal of clinical pharmacology, 1993, Volume: 33, Issue:3

    Topics: Adult; Aged; Aged, 80 and over; Blood Glucose; Diabetes Mellitus, Type 2; Double-Blind Method; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hyperglycemia; Male; Middle Aged; Stress, Physiological; Stress, Psychological; Surveys and Questionnaires

1993
A prospective trial of risk factors for sulfonylurea-induced hypoglycemia in type 2 diabetes mellitus.
    JAMA, 1998, Jan-14, Volume: 279, Issue:2

    Topics: Age Factors; Aged; Analysis of Variance; Blood Chemical Analysis; Blood Glucose; Diabetes Mellitus, Type 2; Double-Blind Method; Epinephrine; Fasting; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Peptides; Prospective Studies; Risk Factors

1998
Intensive blood-glucose control with sulphonylureas or insulin compared with conventional treatment and risk of complications in patients with type 2 diabetes (UKPDS 33). UK Prospective Diabetes Study (UKPDS) Group.
    Lancet (London, England), 1998, Sep-12, Volume: 352, Issue:9131

    Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Prospective Studies; Risk Factors; Sulfonylurea Compounds

1998
Evaluation of oxidative stress before and after control of glycemia and after vitamin E supplementation in diabetic patients.
    Metabolism: clinical and experimental, 2000, Volume: 49, Issue:2

    Topics: Adult; Blood Glucose; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Female; Glipizide; Glutathione; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Oxidative Stress; Thiobarbituric Acid Reactive Substances; Vitamin E

2000
Addition of low-dose rosiglitazone to sulphonylurea therapy improves glycaemic control in Type 2 diabetic patients.
    Diabetic medicine : a journal of the British Diabetic Association, 2000, Volume: 17, Issue:1

    Topics: Adult; Aged; Blood Glucose; C-Peptide; Cholesterol; Cholesterol, HDL; Cholesterol, LDL; Diabetes Mellitus, Type 2; Double-Blind Method; Drug Therapy, Combination; Europe; Female; Fructosamine; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Rosiglitazone; Safety; Thiazoles; Thiazolidinediones; Triglycerides

2000
Comparative efficacy and potency of long-term therapy with glipizide or glyburide in patients with type 2 diabetes mellitus.
    The American journal of the medical sciences, 2000, Volume: 319, Issue:3

    Topics: Adult; Aged; Blood Glucose; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Postprandial Period; Prospective Studies; Therapeutic Equivalency; Time Factors; Treatment Outcome

2000
Effects and pharmacokinetics of oral glibenclamide and glipizide in Caucasian and Chinese patients with type-2 diabetes.
    European journal of clinical pharmacology, 2000, Volume: 56, Issue:9-10

    Topics: Adult; Aged; Asian People; Blood Glucose; Diabetes Mellitus, Type 2; Female; Glipizide; Glucose Tolerance Test; Glyburide; Glycated Hemoglobin; Half-Life; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Proinsulin; White People

2000
Effects of rifampin on the pharmacokinetics and pharmacodynamics of glyburide and glipizide.
    Clinical pharmacology and therapeutics, 2001, Volume: 69, Issue:6

    Topics: Adult; Antibiotics, Antitubercular; Area Under Curve; Blood Glucose; Female; Glipizide; Glyburide; Half-Life; Humans; Hypoglycemic Agents; Male; Rifampin

2001
Comparison of the effects of three insulinotropic drugs on plasma insulin levels after a standard meal.
    Diabetes care, 2002, Volume: 25, Issue:8

    Topics: Aged; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Double-Blind Method; Eating; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Middle Aged; Piperidines

2002
Effects of sulfonylurea hypoglycemic agents and adenosine triphosphate dependent potassium channel antagonists on ventricular arrhythmias in patients with decompensated heart failure.
    Pacing and clinical electrophysiology : PACE, 2003, Volume: 26, Issue:5

    Topics: Aged; Analysis of Variance; Anti-Arrhythmia Agents; Chi-Square Distribution; Diabetes Complications; Diabetes Mellitus; Electrocardiography, Ambulatory; Female; Glipizide; Glyburide; Heart Failure; Humans; Hypoglycemic Agents; Male; Middle Aged; Potassium Channels; Regression Analysis; Sulfonylurea Compounds; Vasodilator Agents; Ventricular Fibrillation

2003

Other Studies

145 other study(ies) available for glyburide and glipizide

ArticleYear
Expedient synthesis and biochemical properties of an [125I]-labeled analogue of glyburide, a radioligand for ATP-inhibited potassium channels.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Adenosine Triphosphate; Animals; Brain; Cell Membrane; Glyburide; Iodine Radioisotopes; Male; Molecular Structure; Potassium Channels; Rats; Rats, Inbred Strains

1990
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Lipophilicity of acidic compounds: impact of ion pair partitioning on drug design.
    Bioorganic & medicinal chemistry letters, 2011, Jun-15, Volume: 21, Issue:12

    Topics: Acids; Albumins; Drug Design; Humans; Hydrogen-Ion Concentration; Lipids; Molecular Structure; Pharmaceutical Preparations; Protein Binding

2011
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
High-performance liquid chromatographic determination of glipizide and some other sulfonylurea drugs in serum.
    Journal of chromatography, 1979, Dec-01, Volume: 164, Issue:4

    Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Glipizide; Glyburide; Humans; Hydrogen-Ion Concentration; Sulfonylurea Compounds; Tolbutamide

1979
Comparative study of the hypoglycaemic and antilipolytic effects of four antidiabetic agents administered i.v.
    Arzneimittel-Forschung, 1976, Volume: 26, Issue:3

    Topics: Adult; Blood Glucose; Diabetes Mellitus; Fatty Acids, Nonesterified; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Injections, Intravenous; Male; Middle Aged; Sulfonamides; Thiadiazoles

1976
Dynamics of sulfonylurea-induced insulin release from the isolated perfused rat pancreas.
    Diabetologia, 1976, Volume: 12, Issue:4

    Topics: Animals; Glipizide; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Perfusion; Rats; Sulfonylurea Compounds; Tolbutamide

1976
[Diabetes: new drugs?].
    La semaine des hopitaux : organe fonde par l'Association d'enseignement medical des hopitaux de Paris, 1976, May-23, Volume: 52, Issue:20

    Topics: Biguanides; Diabetes Mellitus; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Sulfonylurea Compounds

1976
Circular dichroism studies on the interaction of sulfonylureas with bovine and human serum albumin.
    Research communications in chemical pathology and pharmacology, 1976, Volume: 13, Issue:3

    Topics: Binding Sites; Binding, Competitive; Carbutamide; Chlorpropamide; Circular Dichroism; Glipizide; Glyburide; Humans; In Vitro Techniques; Optical Rotatory Dispersion; Protein Binding; Serum Albumin; Serum Albumin, Bovine; Sulfonylurea Compounds; Tolbutamide

1976
Comparison of the pharmacokinetics of glipizide and glibenclamide in man.
    European journal of clinical pharmacology, 1975, Volume: 8, Issue:1

    Topics: Administration, Oral; Adult; Blood Glucose; Female; Glipizide; Glyburide; Half-Life; Humans; Injections, Intravenous; Insulin; Intestinal Absorption; Kinetics; Male; Sulfonylurea Compounds; Tablets

1975
[Experimental study of glipizide. A comparison with other hypoglycemic sulfonamides (author's transl)].
    Diabete & metabolisme, 1975, Volume: 1

    Topics: Administration, Oral; Ammonia; Animals; Dogs; Dose-Response Relationship, Drug; Female; Glipizide; Glyburide; Injections, Intravenous; Insulin; Islets of Langerhans; Mice; Purine-Pyrimidine Metabolism, Inborn Errors; Rats; Seizures; Sulfonylurea Compounds; Time Factors; Tolbutamide

1975
[Non-saturable cooperative binding of tolbutamide to rat endocrine pancreas. Criteria of specificity].
    Comptes rendus hebdomadaires des seances de l'Academie des sciences. Serie D: Sciences naturelles, 1976, Jul-19, Volume: 283, Issue:3

    Topics: Animals; Diazoxide; Drug Interactions; Glipizide; Glucose; Glyburide; Islets of Langerhans; Kinetics; Rats; Tolbutamide

1976
Effect of bed time intermediate acting insulin in NIDDM subjects refractory to a combination of sulphonylureas and biguanides.
    The Journal of the Association of Physicians of India, 1992, Volume: 40, Issue:10

    Topics: Biguanides; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Combinations; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Injections, Subcutaneous; Insulin, Long-Acting; Lipids; Male; Metformin; Middle Aged; Phenformin; Sulfonylurea Compounds; Time Factors

1992
Effects of drugs on ventricular fibrillation and ischaemic K+ loss in a model of ischaemia in perfused guinea-pig hearts in vitro.
    European journal of pharmacology, 1992, Sep-22, Volume: 220, Issue:2-3

    Topics: 4-Aminopyridine; Animals; Anti-Arrhythmia Agents; Benzothiazoles; Calcium Channel Blockers; Disease Models, Animal; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Myocardial Ischemia; Piperidines; Potassium; Potassium Channels; Pyrazines; Pyridines; Sympatholytics; Thiazoles; Ventricular Fibrillation

1992
Specificity of photolabeling of beta-cell membrane proteins with an 125I-labeled glyburide analog.
    The Journal of biological chemistry, 1992, Jul-25, Volume: 267, Issue:21

    Topics: Animals; Binding Sites; Cell Membrane; Chromatography, Gel; Cricetinae; Electrophoresis, Polyacrylamide Gel; Glipizide; Glyburide; Iodine Radioisotopes; Islets of Langerhans; Membrane Proteins; Photochemistry; Substrate Specificity; Tolbutamide; Tumor Cells, Cultured

1992
K+ efflux pathways and neurotransmitter release associated to hippocampal ischemia: effects of glucose and of K+ channel blockers.
    Brain research, 1991, Jan-18, Volume: 539, Issue:1

    Topics: 4-Aminopyridine; Animals; Apamin; Aspartic Acid; Barium; Barium Compounds; Brain Ischemia; Calcium Chloride; Charybdotoxin; Chlorides; Elapid Venoms; gamma-Aminobutyric Acid; Glipizide; Glucose; Glyburide; Hippocampus; In Vitro Techniques; Kinetics; Potassium; Potassium Channels; Rats; Rats, Inbred Strains; Rubidium; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds

1991
Chiral recognition of pinacidil and its 3-pyridyl isomer by canine cardiac and smooth muscle: antagonism by sulfonylureas.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Adenosine Triphosphate; Animals; Dogs; Dose-Response Relationship, Drug; Female; Glipizide; Glyburide; Guanidines; Heart; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Pinacidil; Potassium Channels; Purkinje Fibers; Rubidium Radioisotopes; Stereoisomerism; Sulfonylurea Compounds; Vasodilator Agents

1991
RP 49356 and cromakalim relax airway smooth muscle in vitro by opening a sulphonylurea-sensitive K+ channel: a comparison with nifedipine.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Animals; Benzopyrans; Calcium; Cromakalim; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Picolines; Potassium Channels; Pyrans; Pyrroles; Trachea

1991
Quantitative autoradiography of the binding sites for [125I] iodoglyburide, a novel high-affinity ligand for ATP-sensitive potassium channels in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:2

    Topics: Affinity Labels; Animals; Autoradiography; Binding Sites; Brain; Glipizide; Glyburide; Guanidines; Iodine Radioisotopes; Male; Pinacidil; Potassium Channels; Rats; Rats, Inbred Strains; Vasodilator Agents

1991
Crossover comparison of maximum dose glyburide and glipizide.
    Southern medical journal, 1991, Volume: 84, Issue:6

    Topics: Blood Glucose; Cholesterol; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Female; Glipizide; Glyburide; Humans; Lipoproteins; Male; Middle Aged; Triglycerides

1991
[A comparison between glibenclamide and glipizide in the treatment of type II diabetes].
    Zhonghua nei ke za zhi, 1991, Volume: 30, Issue:2

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Male; Middle Aged; Platelet Adhesiveness; Platelet Aggregation

1991
Divergent cardiac effects of the first and second generation hypoglycemic sulfonylurea compounds.
    Diabetes research and clinical practice, 1990, Volume: 8, Issue:2

    Topics: Animals; Arrhythmias, Cardiac; Blood Glucose; Carbutamide; Dose-Response Relationship, Drug; Electrocardiography; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Male; Myocardial Infarction; Potassium; Rats; Rats, Inbred Strains; Reference Values; Structure-Activity Relationship; Tolbutamide

1990
A screening test for detecting sulfonylureas in plasma.
    Therapeutic drug monitoring, 1990, Volume: 12, Issue:4

    Topics: Aged; Aged, 80 and over; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide

1990
Effect of sulphonylurea therapy on insulin sensitivity in non insulin dependent diabetics.
    The Journal of the Association of Physicians of India, 1990, Volume: 38, Issue:7

    Topics: Blood Glucose; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Insulin Resistance; Middle Aged; Sulfonylurea Compounds; Time Factors; Tolbutamide

1990
Concentration-dependent effects of tolbutamide, meglitinide, glipizide, glibenclamide and diazoxide on ATP-regulated K+ currents in pancreatic B-cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:2

    Topics: Adenosine Triphosphate; Animals; Benzamides; Diazoxide; Glipizide; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Ion Channels; Islets of Langerhans; Mice; Mice, Inbred Strains; Potassium; Sulfonylurea Compounds; Tolbutamide

1988
Inhibition by sulphonylureas of vasorelaxation induced by K+ channel activators in vitro.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: Animals; Antihypertensive Agents; Benzopyrans; Cromakalim; Drug Interactions; Glipizide; Glyburide; Guanidines; In Vitro Techniques; Male; Nifedipine; Norepinephrine; Pinacidil; Potassium Channels; Potassium Chloride; Pyrroles; Rabbits; Sulfonylurea Compounds; Tolbutamide; Vasodilator Agents

1989
Glipizide and glyburide.
    North Carolina medical journal, 1986, Volume: 47, Issue:3

    Topics: Diabetes Mellitus, Type 2; Drug Interactions; Glipizide; Glyburide; Humans; Kinetics; Sulfonylurea Compounds

1986
Direct effects of sulfonylurea agents on glucose transport in the BC3H-1 myocyte.
    Diabetes, 1987, Volume: 36, Issue:11

    Topics: Animals; Cell Line; Deoxy Sugars; Deoxyglucose; Glipizide; Glyburide; Hypoglycemic Agents; Insulin; Kinetics; Mice; Muscles; Tolbutamide

1987
Different effects of glyburide and glipizide on insulin secretion and hepatic glucose production in normal and NIDDM subjects.
    Diabetes, 1987, Volume: 36, Issue:11

    Topics: Adult; Aged; Blood Glucose; C-Peptide; Diabetes Mellitus, Type 2; Gastric Inhibitory Polypeptide; Glipizide; Glucagon; Glucose; Glyburide; Humans; Hyperglycemia; Insulin; Insulin Secretion; Kinetics; Liver; Sulfonylurea Compounds

1987
Characterization of the sulfonylurea receptor on beta cell membranes.
    The Journal of biological chemistry, 1988, Feb-25, Volume: 263, Issue:6

    Topics: Animals; ATP-Binding Cassette Transporters; Cell Line; Cell Membrane; Cricetinae; Glipizide; Glyburide; Insulin; Islets of Langerhans; Kinetics; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Temperature; Tolazamide; Tolbutamide

1988
[Clinical efficacy of a Minidiab preparation (glipizide) in an acute experiment].
    Vutreshni bolesti, 1988, Volume: 27, Issue:2

    Topics: Adult; Aged; Blood Glucose; Diabetes Mellitus, Type 2; Drug Evaluation; Female; Glipizide; Glyburide; Humans; Insulin Antibodies; Male; Middle Aged; Sulfonylurea Compounds; Time Factors

1988
Glucose both inhibits and stimulates insulin secretion from isolated pancreatic islets exposed to maximally effective concentrations of sulfonylureas.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:4

    Topics: Animals; Cell Membrane; Glipizide; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Iodine Radioisotopes; Islets of Langerhans; Keto Acids; Male; Mice; Sulfonylurea Compounds

1988
Reversal of insulin resistance in adipose tissue of non-insulin-dependent diabetics by treatment with diet and sulphonylurea.
    Acta endocrinologica, 1985, Volume: 108, Issue:1

    Topics: Adipose Tissue; Diabetes Mellitus, Type 2; Female; Glipizide; Glucose; Glyburide; Humans; Insulin; Insulin Resistance; Male; Middle Aged; Oxidation-Reduction; Receptor, Insulin; Sulfonylurea Compounds

1985
Pharmacokinetics of glyburide.
    The American journal of medicine, 1985, Sep-20, Volume: 79, Issue:3B

    Topics: Acute Kidney Injury; Blood Glucose; Dose-Response Relationship, Drug; Fasting; Glipizide; Glyburide; Humans; Kidney; Kinetics; Liver

1985
The second generation sulfonylureas: glipizide and glyburide.
    The Diabetes educator, 1985,Fall, Volume: 11, Issue:3

    Topics: Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Insulin; Sulfonylurea Compounds

1985
Glibenclamide is exceptional among hypoglycaemic sulphonylureas in accumulating progressively in beta-cell-rich pancreatic islets.
    Acta endocrinologica, 1984, Volume: 105, Issue:3

    Topics: Animals; Carbutamide; Chlorpropamide; Glipizide; Glyburide; Islets of Langerhans; Mice; Mice, Obese; Sulfonylurea Compounds; Tolbutamide

1984
Clinical pharmacology of glipizide.
    The American journal of medicine, 1983, Nov-30, Volume: 75, Issue:5B

    Topics: Biological Availability; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Half-Life; Humans; Kinetics; Structure-Activity Relationship; Sulfonylurea Compounds; Tolbutamide

1983
Effect of sulfonylurea on glucose, insulin and C-peptide responses to a meal stimulus in a patient with type 2 diabetes and liver disease.
    Acta medica Scandinavica, 1984, Volume: 215, Issue:5

    Topics: Aged; Blood Glucose; C-Peptide; Diabetes Mellitus, Type 2; Fasting; Female; Food; Glipizide; Glyburide; Humans; Insulin; Liver Diseases; Liver Neoplasms; Sulfonylurea Compounds

1984
Glyburide and glipizide.
    The Medical letter on drugs and therapeutics, 1984, Aug-31, Volume: 26, Issue:669

    Topics: Diabetes Mellitus; Glipizide; Glyburide; Humans; Sulfonylurea Compounds

1984
The new oral antidiabetic drugs.
    American family physician, 1984, Volume: 30, Issue:5

    Topics: Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Sulfonylurea Compounds

1984
The effect of improvement in diabetic control on plasma and whole blood viscosity.
    Diabetologia, 1980, Volume: 19, Issue:4

    Topics: Adolescent; Adult; Blood; Blood Glucose; Diabetes Mellitus; Female; Glipizide; Glyburide; Hemoglobin A; Humans; Insulin; Male; Middle Aged; Plasma; Viscosity

1980
Glipizide: experimental study and comparison with other sulfonylureas.
    Acta endocrinologica. Supplementum, 1980, Volume: 239

    Topics: Animals; Blood Glucose; Dogs; Dose-Response Relationship, Drug; Glipizide; Glyburide; Hypoglycemia; Insulin; Islets of Langerhans; Mice; Rats; Sulfonylurea Compounds; Tolbutamide

1980
Kinetics-effect relations of glipizide and other sulfonylureas.
    Acta endocrinologica. Supplementum, 1980, Volume: 239

    Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus; Dose-Response Relationship, Drug; Fasting; Feeding Behavior; Glipizide; Glyburide; Humans; Kidney; Sulfonylurea Compounds; Tolbutamide

1980
Diurnal pattern of plasma insulin and blood glucose during glibenclamide and glipizide therapy in elderly diabetics.
    Acta endocrinologica. Supplementum, 1980, Volume: 239

    Topics: Aged; Blood Glucose; Circadian Rhythm; Diabetes Mellitus; Female; Glipizide; Glyburide; Humans; Insulin; Male; Middle Aged; Sulfonylurea Compounds

1980
Comparative single-dose kinetics and effects of four sulfonylureas in healthy volunteers.
    Acta medica Scandinavica, 1980, Volume: 208, Issue:4

    Topics: Adult; Blood Glucose; Chlorpropamide; Fasting; Glipizide; Glyburide; Humans; Insulin; Kinetics; Male; Sulfonylurea Compounds; Time Factors; Tolbutamide

1980
Standardized procedure for the assay and identification of hypoglycemic sulfonylureas in human plasma.
    Acta diabetologica, 1995, Volume: 32, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diabetes Mellitus, Type 2; Drug Monitoring; Forensic Medicine; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Reproducibility of Results; Sensitivity and Specificity; Sulfonylurea Compounds

1995
Sulfonylureas induce cholesterol accumulation in cultured human intimal cells and macrophages.
    Atherosclerosis, 1994, Volume: 105, Issue:2

    Topics: Adult; Animals; Cells, Cultured; Cholesterol; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glyburide; Humans; Macrophages, Peritoneal; Male; Mice; Mice, Inbred BALB C; Middle Aged; Muscle, Smooth, Vascular; Sulfonylurea Compounds; Tunica Intima

1994
Photoaffinity labeling of the cerebral sulfonylurea receptor using a novel radioiodinated azidoglibenclamide analogue.
    Journal of neurochemistry, 1994, Volume: 63, Issue:2

    Topics: Affinity Labels; Animals; ATP-Binding Cassette Transporters; Binding, Competitive; Cell Fractionation; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Glipizide; Glyburide; Iodine Radioisotopes; Kinetics; Microsomes; Molecular Weight; Photolysis; Potassium Channels; Potassium Channels, Inwardly Rectifying; Radioligand Assay; Receptors, Drug; Sulfonylurea Receptors; Swine; Tolbutamide; Tritium

1994
Comparative placental transport of oral hypoglycemic agents in humans: a model of human placental drug transfer.
    American journal of obstetrics and gynecology, 1994, Volume: 171, Issue:3

    Topics: Administration, Oral; Analysis of Variance; Antipyrine; Biological Transport; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Maternal-Fetal Exchange; Models, Biological; Molecular Weight; Placenta; Pregnancy; Regression Analysis; Tolbutamide

1994
K(+)-channel blockers and coronary vasoconstriction in guinea-pig perfused hearts in-vitro.
    The Journal of pharmacy and pharmacology, 1993, Volume: 45, Issue:7

    Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Coronary Vessels; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Perfusion; Phentolamine; Potassium Channels; Pyrazines; Pyridines; Vasoconstriction

1993
Effects of antidiabetic sulphonylureas, cromakalim and their interaction in guinea-pig isolated tracheal smooth muscle.
    Pulmonary pharmacology, 1993, Volume: 6, Issue:3

    Topics: Animals; Benzopyrans; Cromakalim; Drug Interactions; Glipizide; Glyburide; Guinea Pigs; Hypoglycemic Agents; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Pyrroles; Sulfonylurea Compounds; Trachea

1993
ATP-modulated K+ channels sensitive to antidiabetic sulfonylureas are present in adenohypophysis and are involved in growth hormone release.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Feb-15, Volume: 90, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Affinity Labels; Animals; Calcium; Cells, Cultured; Diazoxide; Female; Glipizide; Glyburide; Growth Hormone; Hypoglycemic Agents; Kinetics; Membrane Potentials; Oligomycins; Pituitary Gland, Anterior; Potassium Channels; Rats; Receptors, Drug; Sulfonylurea Compounds

1993
Alteration of rat hepatic insulin metabolism by glyburide and glipizide.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:3

    Topics: Animals; Glipizide; Glyburide; In Vitro Techniques; Insulin; Liver; Male; Perfusion; Rats; Rats, Sprague-Dawley

1993
Bedtime insulin added to daytime sulfonylureas improves glycemic control in uncontrolled type II diabetes.
    Clinical pharmacology and therapeutics, 1993, Volume: 53, Issue:3

    Topics: Adult; Aged; Diabetes Mellitus; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Glipizide; Glyburide; Humans; Insulin, Isophane; Middle Aged; Obesity; Prospective Studies; Time Factors

1993
Disturbances in autoregulatory responses of rat pial arteries by sulfonylureas.
    Life sciences, 1993, Volume: 52, Issue:19

    Topics: Animals; Arterioles; Blood Pressure; Cerebral Arteries; Glipizide; Glyburide; Pia Mater; Rats; Rats, Sprague-Dawley; Vasodilation

1993
PKC-dependent stimulation of exocytosis by sulfonylureas in pancreatic beta cells.
    Science (New York, N.Y.), 1996, Feb-09, Volume: 271, Issue:5250

    Topics: Animals; Calcium; Cells, Cultured; Cytoplasmic Granules; Electric Conductivity; Exocytosis; Glipizide; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Protein Kinase C; Sulfonylurea Compounds; Tolbutamide

1996
Detection of hypoglycemic drugs in human urine using micellar electrokinetic chromatography.
    Analytical chemistry, 1995, Oct-15, Volume: 67, Issue:20

    Topics: Chromatography, High Pressure Liquid; Electrophoresis, Capillary; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Micelles; Reproducibility of Results; Sulfonylurea Compounds

1995
Gliclazide hydroxylation by rat liver microsomes.
    Xenobiotica; the fate of foreign compounds in biological systems, 1995, Volume: 25, Issue:12

    Topics: Animals; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2D6; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Enzyme Inhibitors; Gliclazide; Glipizide; Glyburide; Hydroxylation; Hypoglycemic Agents; Kinetics; Male; Microsomes, Liver; Mixed Function Oxygenases; Rats; Rats, Sprague-Dawley; Tolbutamide

1995
Sulfonylureas enhance GABAA synaptic potentials in rat midbrain dopamine neurones.
    Acta physiologica Scandinavica, 1996, Volume: 156, Issue:2

    Topics: Animals; Dopamine; Electric Stimulation; Glipizide; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Male; Membrane Potentials; Mesencephalon; Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfonylurea Compounds; Synapses

1996
Photodegradation products of sulphonamide-derived oral antidiabetics and diuretics are not phototoxic in vitro.
    Photodermatology, photoimmunology & photomedicine, 1996, Volume: 12, Issue:2

    Topics: Bendroflumethiazide; Dermatitis, Phototoxic; Diuretics; Furosemide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Photochemistry; Photosensitizing Agents; Sulfonamides; Tumor Cells, Cultured

1996
The effect of pH on the in-vitro dissolution of three second-generation sulphonylurea preparations: mechanism of antacid-sulphonylurea interaction.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:9

    Topics: Antacids; Glipizide; Glyburide; Hydrogen-Ion Concentration; Hypoglycemic Agents; Solubility; Tablets

1996
Photohemolytic potency of oral antidiabetic drugs in vitro: effects of antioxidants and a nitrogen atmosphere.
    Photodermatology, photoimmunology & photomedicine, 1996, Volume: 12, Issue:4

    Topics: Antioxidants; Ascorbic Acid; Carbutamide; Chlorpropamide; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glyburide; Hemolysis; Humans; Hypoglycemic Agents; Nitrogen; Radiation-Sensitizing Agents; Reactive Oxygen Species; Sulfonamides; Sulfonylurea Compounds; Superoxide Dismutase; Tolazamide; Tolbutamide; Ultraviolet Rays; Vitamin E

1996
Oral sulfonylurea hypoglycemic agents prevent ischemic preconditioning in human myocardium. Two paradoxes revisited.
    Circulation, 1997, Jul-01, Volume: 96, Issue:1

    Topics: Administration, Oral; Aged; Diabetes Mellitus; Female; Glipizide; Glyburide; Heart Atria; Humans; Hypoglycemic Agents; In Vitro Techniques; Ischemic Preconditioning, Myocardial; Male; Middle Aged; Myocardial Contraction; Potassium Channels; Sulfonylurea Compounds

1997
Rates of hypoglycemia in users of sulfonylureas.
    Journal of clinical epidemiology, 1997, Volume: 50, Issue:6

    Topics: Adult; Aged; Chlorpropamide; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Incidence; Male; Middle Aged; Poisson Distribution; Risk; Risk Factors; Sulfonylurea Compounds; Surveys and Questionnaires; Time Factors; Tolbutamide

1997
Prospective multicenter study of sulfonylurea ingestion in children.
    The Journal of pediatrics, 1997, Volume: 131, Issue:1 Pt 1

    Topics: Accidents; Administration, Oral; Blood Glucose; Body Weight; Child; Child, Preschool; Confidence Intervals; Dose-Response Relationship, Drug; Drug Monitoring; Female; Forecasting; Gastrointestinal Agents; Glipizide; Glucagon; Glucose; Glyburide; Hospitalization; Humans; Hypoglycemia; Hypoglycemic Agents; Infant; Infusions, Intravenous; Male; Patient Admission; Poison Control Centers; Prospective Studies; Risk Factors; Sensitivity and Specificity; Sulfonylurea Compounds; Time Factors; Treatment Outcome

1997
Capillary electrophoretic detection of metabolites in the urine of patients receiving hypoglycemic drug therapy.
    Electrophoresis, 1997, Volume: 18, Issue:10

    Topics: Electrophoresis, Capillary; Glipizide; Glyburide; Humans; Hypoglycemia; Sulfonylurea Compounds

1997
A retrospective analysis of the efficacy and safety of metformin in the African-American patient.
    Journal of the National Medical Association, 1997, Volume: 89, Issue:11

    Topics: Adult; Aged; Aged, 80 and over; Black People; Body Weight; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Insulin, Isophane; Male; Metformin; Middle Aged; Prognosis; Retrospective Studies

1997
Pharmacological and biochemical evidence for the regulation of osteocalcin secretion by potassium channels in human osteoblast-like MG-63 cells.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 1997, Volume: 12, Issue:12

    Topics: Adenosine Triphosphate; Antihypertensive Agents; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Diazoxide; Dose-Response Relationship, Drug; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Osteoblasts; Osteocalcin; Osteosarcoma; Potassium Channels; Tumor Cells, Cultured

1997
The effects of gliclazide and other sulfonylureas on low-density lipoprotein oxidation in vitro.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:12 Suppl 1

    Topics: Administration, Oral; Adult; Antioxidants; Ascorbic Acid; Coronary Artery Disease; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Lipoproteins, LDL; Male; Middle Aged; Oxidation-Reduction; Sulfonylurea Compounds; Tolbutamide

1997
Whole cell patch-clamp recordings of rat midbrain dopaminergic neurons isolate a sulphonylurea- and ATP-sensitive component of potassium currents activated by hypoxia.
    Journal of neurophysiology, 1998, Volume: 79, Issue:3

    Topics: Adenosine Triphosphate; Animals; Barium Compounds; Cell Hypoxia; Charybdotoxin; Chlorides; Dopamine; Glipizide; Glyburide; In Vitro Techniques; Membrane Potentials; Mesencephalon; Microelectrodes; Neurons; Patch-Clamp Techniques; Potassium Channels; Rats; Rats, Wistar; Reaction Time; Sulfonylurea Compounds; Tolbutamide

1998
Hypoglycemia from glipizide and glyburide.
    JAMA, 1998, May-13, Volume: 279, Issue:18

    Topics: Glipizide; Glyburide; Humans; Hypoglycemia; Risk

1998
Hypoglycemia from glipizide and glyburide.
    JAMA, 1998, May-13, Volume: 279, Issue:18

    Topics: Aged; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Hypoglycemia; Risk

1998
Formulary conversion from glipizide to glyburide: a cost-minimization analysis.
    Hospital pharmacy, 1995, Volume: 30, Issue:6

    Topics: Aged; Cost Savings; Drug Costs; Formularies, Hospital as Topic; Glipizide; Glyburide; Hospitals, Municipal; Humans; Hypoglycemic Agents; New York City; Pharmacy Service, Hospital

1995
Characterization of low-affinity binding sites for glibenclamide on the Kir6.2 subunit of the beta-cell KATP channel.
    Biochemical and biophysical research communications, 1999, Apr-21, Volume: 257, Issue:3

    Topics: Animals; ATP-Binding Cassette Transporters; Binding Sites; Blotting, Northern; Cell Line; Cell Membrane; COS Cells; Gliclazide; Glipizide; Glyburide; Islets of Langerhans; Kinetics; Organelles; Phentolamine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Recombinant Fusion Proteins; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide; Transfection

1999
[Impact of intensive blood glucose control with hypoglycemic sulfamides, metformin or insulin on complications of non-insulin dependent diabetes].
    Revue d'epidemiologie et de sante publique, 1999, Volume: 47, Issue:1

    Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Metformin; Multicenter Studies as Topic; Randomized Controlled Trials as Topic; Risk Factors

1999
Antioxidant status in experimental type 2 diabetes mellitus: effects of glibenclamide and glipizide on various rat tissues.
    Experimental and toxicologic pathology : official journal of the Gesellschaft fur Toxikologische Pathologie, 1999, Volume: 51, Issue:4-5

    Topics: Animals; Antioxidants; Brain; Catalase; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Hypoglycemic Agents; Kidney; Liver; Lung; Male; Malondialdehyde; Myocardium; Rats

1999
Pharmacokinetics of gliquidone, glibenclamide, gliclazide and glipizide in middle-aged and aged subjects.
    Research communications in molecular pathology and pharmacology, 1999, Volume: 103, Issue:2

    Topics: Aged; Female; Gliclazide; Glipizide; Glyburide; Half-Life; Humans; Hypoglycemic Agents; Male; Middle Aged; Sulfonylurea Compounds

1999
Pharmacology of human sulphonylurea receptor SUR1 and inward rectifier K(+) channel Kir6.2 combination expressed in HEK-293 cells.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: ATP-Binding Cassette Transporters; Binding, Competitive; Cations; Cell Line; Deoxyglucose; Diazoxide; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Fluorescence; Gene Expression; Glipizide; Glyburide; Humans; Membrane Potentials; Oligomycins; Potassium Channels; Potassium Channels, Inwardly Rectifying; Radioligand Assay; Receptors, Drug; Recombinant Fusion Proteins; RNA, Messenger; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolazamide; Tolbutamide; Tritium

2000
Identification of sulfonylureas in serum by electrospray mass spectrometry.
    Analytical biochemistry, 2000, Jun-15, Volume: 282, Issue:1

    Topics: Calibration; Chlorpropamide; Chromatography, Liquid; Glipizide; Glyburide; Humans; Mass Spectrometry; Models, Chemical; Sulfonylurea Compounds; Tolbutamide; Ultraviolet Rays

2000
Acidic dopamine metabolites are actively extruded from PC12 cells by a novel sulfonylurea-sensitive transporter.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 361, Issue:6

    Topics: 3,4-Dihydroxyphenylacetic Acid; 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport, Active; Dopamine; Glipizide; Glyburide; Homovanillic Acid; Male; Mice; Microdialysis; Multidrug Resistance-Associated Proteins; PC12 Cells; Potassium Channels; Potassium Channels, Inwardly Rectifying; Probenecid; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rhodamines; RNA, Messenger; Sulfonylurea Receptors; Transfection

2000
Differences in pharmacotherapy and in glucose control of type 2 diabetes patients in two neighbouring towns: a longitudinal population-based study.
    Diabetes, obesity & metabolism, 2001, Volume: 3, Issue:4

    Topics: Aged; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Longitudinal Studies; Male; Retrospective Studies; Sweden; Time Factors; Urban Population

2001
Severe hypoglycemia from clarithromycin-sulfonylurea drug interaction.
    Diabetes care, 2002, Volume: 25, Issue:9

    Topics: Aged; Aged, 80 and over; Anti-Bacterial Agents; Clarithromycin; Drug Interactions; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male

2002
The peripheral antinociceptive effect of resveratrol is associated with activation of potassium channels.
    Neuropharmacology, 2002, Volume: 43, Issue:5

    Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; ATP-Binding Cassette Transporters; Charybdotoxin; Female; Glipizide; Glyburide; KATP Channels; Morphine; Narcotics; Peripheral Nervous System; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Resveratrol; Stilbenes; Tetraethylammonium; Tolbutamide

2002
Transdermal delivery of glibenclamide and glipizide: in vitro permeation studies through mouse skin.
    Die Pharmazie, 2002, Volume: 57, Issue:12

    Topics: Administration, Cutaneous; Animals; Chemical Phenomena; Chemistry, Physical; Glipizide; Glyburide; Hypoglycemic Agents; Mice; Skin Absorption; Solubility

2002
Economic model of first-line drug strategies to achieve recommended glycaemic control in newly diagnosed type 2 diabetes mellitus.
    PharmacoEconomics, 2003, Volume: 21, Issue:11

    Topics: Carbamates; Cohort Studies; Decision Trees; Diabetes Mellitus, Type 2; Direct Service Costs; Drug Costs; Drug Therapy, Combination; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Managed Care Programs; Markov Chains; Metformin; Models, Economic; Piperidines; Rosiglitazone; Thiazoles; Thiazolidinediones; United States

2003
Effect of some penetration enhancers on the permeation of glibenclamide and glipizide through mouse skin.
    Die Pharmazie, 2003, Volume: 58, Issue:12

    Topics: Animals; Ethanol; Excipients; Glipizide; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Mice; Skin Absorption; Solubility; Solvents

2003
The development and validation of liquid chromatography method for the simultaneous determination of metformin and glipizide, gliclazide, glibenclamide or glimperide in plasma.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2005, Mar-25, Volume: 817, Issue:2

    Topics: Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Metformin; Reference Standards; Sensitivity and Specificity

2005
Antidiabetic sulphonylureas activate mitochondrial permeability transition in rat skeletal muscle.
    British journal of pharmacology, 2005, Volume: 145, Issue:6

    Topics: Animals; Calcium; Cyclosporine; Glipizide; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Membrane Potentials; Mitochondria, Muscle; Mitochondrial Swelling; Muscle, Skeletal; Oxygen; Permeability; Rats; Sulfonylurea Compounds

2005
Transfer of glyburide and glipizide into breast milk.
    Diabetes care, 2005, Volume: 28, Issue:8

    Topics: Adult; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Infant; Infant Food; Milk, Human

2005
The sulfonylurea glipizide does not inhibit ischemic preconditioning in anesthetized rabbits.
    Cardiovascular drugs and therapy, 2005, Volume: 19, Issue:5

    Topics: Animals; Glipizide; Glyburide; Heart; Hypnotics and Sedatives; Hypoglycemic Agents; Insulin; Insulin-Secreting Cells; Ischemic Preconditioning, Myocardial; Ketamine; Male; Models, Animal; Myocardial Infarction; Rabbits; Xylazine

2005
Simultaneous estimation of six anti-diabetic drugs--glibenclamide, gliclazide, glipizide, pioglitazone, repaglinide and rosiglitazone: development of a novel HPLC method for use in the analysis of pharmaceutical formulations and its application to human p
    Biomedical chromatography : BMC, 2006, Volume: 20, Issue:10

    Topics: Carbamates; Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Molecular Structure; Pioglitazone; Piperidines; Reproducibility of Results; Rosiglitazone; Thiazolidinediones

2006
Development of a RP-HPLC method for screening potentially counterfeit anti-diabetic drugs.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2007, Jun-15, Volume: 853, Issue:1-2

    Topics: Carbamates; Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Molecular Structure; Piperidines; Reproducibility of Results; Sulfonylurea Compounds

2007
Sitagliptin: new drug. Type 2 diabetes: limited efficacy, too many unknown risks.
    Prescrire international, 2008, Volume: 17, Issue:93

    Topics: Clinical Trials as Topic; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Drug Therapy, Combination; Europe; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Metformin; Pyrazines; Triazoles

2008
Hypoglycaemia in patients with type 2 diabetes treated with a combination of metformin and sulphonylurea therapy in France.
    Diabetes, obesity & metabolism, 2008, Volume: 10 Suppl 1

    Topics: Cross-Sectional Studies; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; France; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Metformin; Middle Aged; Quality of Life; Stress, Psychological; Sulfonylurea Compounds

2008
Risk of coronary artery disease associated with initial sulphonylurea treatment of patients with type 2 diabetes: a matched case-control study.
    Diabetes research and clinical practice, 2008, Volume: 82, Issue:3

    Topics: Adult; Case-Control Studies; Coronary Artery Disease; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Metformin; Middle Aged; Risk; Sulfonylurea Compounds

2008
Comparison of ultraviolet detection, evaporative light scattering detection and charged aerosol detection methods for liquid-chromatographic determination of anti-diabetic drugs.
    Journal of pharmaceutical and biomedical analysis, 2010, Mar-11, Volume: 51, Issue:4

    Topics: Aerosols; Chromatography, High Pressure Liquid; Chromatography, Reverse-Phase; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Light; Reproducibility of Results; Scattering, Radiation; Spectrophotometry, Ultraviolet; Sulfonylurea Compounds

2010
The risk of overall mortality in patients with type 2 diabetes receiving glipizide, glyburide, or glimepiride monotherapy: a retrospective analysis.
    Diabetes care, 2010, Volume: 33, Issue:6

    Topics: Aged; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Multivariate Analysis; Retrospective Studies; Sulfonylurea Compounds

2010
Effect of sulfonylurea dose escalation on hemoglobin A1c in Veterans Affairs patients with type 2 diabetes.
    Acta diabetologica, 2013, Volume: 50, Issue:2

    Topics: Aged; Creatinine; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Male; Middle Aged; Retrospective Studies; United States; United States Department of Veterans Affairs; Veterans

2013
Anti-infectives and the risk of severe hypoglycemia in users of glipizide or glyburide.
    Clinical pharmacology and therapeutics, 2010, Volume: 88, Issue:2

    Topics: Adolescent; Adult; Aged; Anti-Infective Agents; Antifungal Agents; Aryl Hydrocarbon Hydroxylases; Blood Glucose; Case-Control Studies; Cross-Over Studies; Cytochrome P-450 CYP2C9; Drug Interactions; Enzyme Inhibitors; Ethnicity; Female; Fluconazole; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Middle Aged; Risk; Trimethoprim, Sulfamethoxazole Drug Combination; Young Adult

2010
Potential CYP2C9-mediated drug-drug interactions in hospitalized type 2 diabetes mellitus patients treated with the sulphonylureas glibenclamide, glimepiride or glipizide.
    Journal of internal medicine, 2010, Volume: 268, Issue:4

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Aryl Hydrocarbon Hydroxylases; Cytochrome P-450 CYP2C9; Diabetes Mellitus, Type 2; Drug Interactions; Female; Glipizide; Glyburide; Hospitalization; Humans; Hypoglycemic Agents; Male; Middle Aged; Sulfonylurea Compounds; Young Adult

2010
Quantitative insulin and C-peptide levels among ED patients with sulfonylurea-induced hypoglycemia-a prospective case series.
    The American journal of emergency medicine, 2010, Volume: 28, Issue:8

    Topics: Aged; Aged, 80 and over; C-Peptide; Cross-Sectional Studies; Drug Overdose; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Middle Aged; Prospective Studies; Sulfonylurea Compounds

2010
Use of sulphonylurea and cancer in type 2 diabetes-The Hong Kong Diabetes Registry.
    Diabetes research and clinical practice, 2010, Volume: 90, Issue:3

    Topics: Aged; Asian People; Cohort Studies; Diabetes Mellitus, Type 2; Female; Gliclazide; Glipizide; Glyburide; Hong Kong; Humans; Male; Middle Aged; Neoplasms; Proportional Hazards Models; Prospective Studies; Registries; Risk Factors; Sulfonylurea Compounds

2010
Comparable long-term mortality risk associated with individual sulfonylureas in diabetes patients with heart failure.
    Diabetes research and clinical practice, 2011, Volume: 94, Issue:1

    Topics: Aged; Aged, 80 and over; Diabetes Mellitus; Female; Glipizide; Glyburide; Heart Failure; Humans; Hypoglycemic Agents; Male; Sulfonylurea Compounds; Tolbutamide

2011
Hypoglycemia after accidental pediatric sulfonylurea ingestions.
    Pediatric emergency care, 2011, Volume: 27, Issue:9

    Topics: Accidents, Home; Arizona; Blood Glucose; Child, Preschool; Emergency Service, Hospital; Glipizide; Glucose; Glyburide; Hospitals, Pediatric; Hospitals, Teaching; Hospitals, Urban; Humans; Hypoglycemia; Hypoglycemic Agents; Incidence; Infant; Poisoning; Retrospective Studies; Sulfonylurea Compounds; Time Factors

2011
Glycemic control and hypoglycemia in Veterans Health Administration patients converted from glyburide to glipizide.
    Journal of managed care pharmacy : JMCP, 2011, Volume: 17, Issue:9

    Topics: Aged; Blood Glucose; Creatinine; Diabetes Mellitus; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Middle Aged; Renal Insufficiency; Retrospective Studies; United States; United States Department of Veterans Affairs

2011
Differential contribution of TM6 and TM12 to the pore of CFTR identified by three sulfonylurea-based blockers.
    Pflugers Archiv : European journal of physiology, 2012, Volume: 463, Issue:3

    Topics: Alanine; Amino Acid Sequence; Animals; Benzamides; Cystic Fibrosis Transmembrane Conductance Regulator; Glipizide; Glyburide; Ion Channel Gating; Kinetics; Mutagenesis; Oocytes; Patch-Clamp Techniques; Sulfonylurea Compounds; Tolbutamide; Xenopus

2012
The risk of overall mortality in patients with Type 2 diabetes receiving different combinations of sulfonylureas and metformin: a retrospective analysis.
    Diabetic medicine : a journal of the British Diabetic Association, 2012, Volume: 29, Issue:8

    Topics: Aged; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Retrospective Studies; Risk Factors; Sulfonylurea Compounds

2012
Increase in overall mortality risk in patients with type 2 diabetes receiving glipizide, glyburide or glimepiride monotherapy versus metformin: a retrospective analysis.
    Diabetes, obesity & metabolism, 2012, Volume: 14, Issue:9

    Topics: Adult; Aged; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Kaplan-Meier Estimate; Male; Metformin; Middle Aged; Propensity Score; Retrospective Studies; Sulfonylurea Compounds; Young Adult

2012
Hypoglycemia in hospitalized patients treated with sulfonylureas.
    Pharmacotherapy, 2012, Volume: 32, Issue:7

    Topics: Academic Medical Centers; Age Factors; Aged; Blood Glucose; Case-Control Studies; Drug Therapy, Combination; Female; Glipizide; Glomerular Filtration Rate; Glyburide; Hospitalization; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Middle Aged; Multivariate Analysis; Regression Analysis; Retrospective Studies; Risk Factors; Sulfonylurea Compounds

2012
Rapid extraction, identification and quantification of oral hypoglycaemic drugs in serum and hair using LC-MS/MS.
    Forensic science international, 2012, Nov-30, Volume: 223, Issue:1-3

    Topics: Acetonitriles; Chromatography, Liquid; Female; Forensic Toxicology; Gliclazide; Glipizide; Glyburide; Hair; Humans; Hypoglycemic Agents; Limit of Detection; Male; Mass Spectrometry; Metformin; Methanol; Middle Aged; Molecular Structure; Solvents; Sulfonylurea Compounds

2012
Pharmacophore modeling, homology modeling, and in silico screening reveal mammalian target of rapamycin inhibitory activities for sotalol, glyburide, metipranolol, sulfamethizole, glipizide, and pioglitazone.
    Journal of molecular graphics & modelling, 2013, Volume: 42

    Topics: Adrenergic beta-Antagonists; Amino Acid Sequence; Anti-Infective Agents; Catalytic Domain; Crystallography, X-Ray; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Metipranolol; Models, Molecular; Molecular Docking Simulation; Phosphatidylinositol 3-Kinases; Pioglitazone; Quantitative Structure-Activity Relationship; ROC Curve; Sequence Alignment; Sotalol; Sulfamethizole; Thiazolidinediones; TOR Serine-Threonine Kinases

2013
Mortality among veterans with type 2 diabetes initiating metformin, sulfonylurea or rosiglitazone monotherapy.
    Diabetologia, 2013, Volume: 56, Issue:9

    Topics: Diabetes Mellitus, Type 2; Female; Follow-Up Studies; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Proportional Hazards Models; Retrospective Studies; Risk Factors; Rosiglitazone; Sulfonylurea Compounds; Thiazolidinediones; Time Factors; United States; Veterans

2013
Pharmacoepidemiologic and in vitro evaluation of potential drug-drug interactions of sulfonylureas with fibrates and statins.
    British journal of clinical pharmacology, 2014, Volume: 78, Issue:3

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Area Under Curve; Case-Control Studies; Cytochrome P-450 Enzyme Inhibitors; Drug Interactions; Female; Fibric Acids; Glipizide; Glyburide; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypoglycemia; Hypoglycemic Agents; Male; Middle Aged; Pharmacoepidemiology; Sulfonylurea Compounds; Young Adult

2014
Effect of tolbutamide, glyburide and glipizide administered supraspinally on CA3 hippocampal neuronal cell death and hyperglycemia induced by kainic acid in mice.
    Brain research, 2014, May-20, Volume: 1564

    Topics: Animals; Blood Glucose; CA3 Region, Hippocampal; Cell Death; Glipizide; Glyburide; Hyperglycemia; Hypoglycemic Agents; Infusions, Intraventricular; Kainic Acid; Male; Mice; Mice, Inbred ICR; Neurons; Sulfonylurea Compounds; Tolbutamide

2014
Coadministration of co-trimoxazole with sulfonylureas: hypoglycemia events and pattern of use.
    The journals of gerontology. Series A, Biological sciences and medical sciences, 2015, Volume: 70, Issue:2

    Topics: Aged; Aged, 80 and over; Anti-Infective Agents; Cohort Studies; Diabetes Mellitus; Drug Interactions; Emergency Service, Hospital; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Medicare; Polypharmacy; Primary Health Care; Trimethoprim, Sulfamethoxazole Drug Combination; United States

2015
Hypoglycemia after antimicrobial drug prescription for older patients using sulfonylureas.
    JAMA internal medicine, 2014, Volume: 174, Issue:10

    Topics: Aged; Aged, 80 and over; Anti-Infective Agents; Ciprofloxacin; Clarithromycin; Drug Interactions; Drug Prescriptions; Female; Glipizide; Glyburide; Health Care Costs; Humans; Hypoglycemia; Hypoglycemic Agents; Levofloxacin; Logistic Models; Male; Medicare; Metronidazole; Morbidity; Odds Ratio; Retrospective Studies; Risk Factors; Sulfonylurea Compounds; Texas; Trimethoprim, Sulfamethoxazole Drug Combination; United States

2014
Metformin in combination with various insulin secretagogues in type 2 diabetes and associated risk of cardiovascular morbidity and mortality--a retrospective nationwide study.
    Diabetes research and clinical practice, 2015, Volume: 107, Issue:1

    Topics: Aged; Carbamates; Cardiovascular Diseases; Denmark; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Morbidity; Myocardial Infarction; Piperidines; Registries; Retrospective Studies; Risk Factors; Stroke; Sulfonylurea Compounds; Tolbutamide

2015
Severe hypoglycemia in users of sulfonylurea antidiabetic agents and antihyperlipidemics.
    Clinical pharmacology and therapeutics, 2016, Volume: 99, Issue:5

    Topics: Aged; Algorithms; Cohort Studies; Drug Interactions; Female; Fenofibrate; Glipizide; Glyburide; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypoglycemia; Hypoglycemic Agents; Hypolipidemic Agents; Incidence; Male; Middle Aged; Retrospective Studies; Severity of Illness Index; Sulfonylurea Compounds

2016
Biomedical Informatics Approaches to Identifying Drug-Drug Interactions: Application to Insulin Secretagogues.
    Epidemiology (Cambridge, Mass.), 2017, Volume: 28, Issue:3

    Topics: Area Under Curve; Carbamates; Cyclohexanes; Databases, Factual; Diabetes Mellitus, Type 2; Drug Interactions; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Medical Informatics; Nateglinide; Pharmacoepidemiology; Phenylalanine; Piperidines; Sulfonylurea Compounds

2017
Mechanism-based selection of stabilization strategy for amorphous formulations: Insights into crystallization pathways.
    Journal of controlled release : official journal of the Controlled Release Society, 2017, 06-28, Volume: 256

    Topics: Calorimetry, Differential Scanning; Crystallization; Drug Compounding; Drug Liberation; Drug Stability; Glipizide; Glyburide; Hydrogen Bonding; Hypromellose Derivatives; Indapamide; Metolazone; Molecular Dynamics Simulation; Povidone; Spectrum Analysis, Raman

2017
Sentinel Modular Program for Propensity Score-Matched Cohort Analyses: Application to Glyburide, Glipizide, and Serious Hypoglycemia.
    Epidemiology (Cambridge, Mass.), 2017, Volume: 28, Issue:6

    Topics: Adult; Aged; Cohort Studies; Diabetes Mellitus, Type 2; Emergency Service, Hospital; Female; Glipizide; Glyburide; Hospitalization; Humans; Hypoglycemia; Hypoglycemic Agents; Incidence; Male; Middle Aged; Propensity Score; Proportional Hazards Models; Sentinel Surveillance; Severity of Illness Index; United States

2017
Risk of Hypoglycemia Following Hospital Discharge in Patients With Diabetes and Acute Kidney Injury.
    Diabetes care, 2018, Volume: 41, Issue:3

    Topics: Acute Kidney Injury; Adult; Aged; Blood Glucose; Diabetes Mellitus; Diabetic Nephropathies; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Kidney Function Tests; Male; Middle Aged; Patient Discharge; Retrospective Studies; Risk Factors

2018
Effect of Tinospora cordifolia aqua-alcoholic extract on pharmacokinetic of Glibenclamide in rat: An herb-drug interaction study.
    Journal of pharmaceutical and biomedical analysis, 2018, Mar-20, Volume: 151

    Topics: Administration, Oral; Animals; Biological Availability; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Ethanol; Glipizide; Glyburide; Herb-Drug Interactions; Humans; Isoenzymes; Male; Metabolic Clearance Rate; Microsomes, Liver; Plant Extracts; Rats; Rats, Sprague-Dawley; Reference Standards; Tinospora; Water

2018
Comparative Safety of Sulfonylureas and the Risk of Sudden Cardiac Arrest and Ventricular Arrhythmia.
    Diabetes care, 2018, Volume: 41, Issue:4

    Topics: Aged; Arrhythmias, Cardiac; Cause of Death; Death, Sudden, Cardiac; Diabetic Angiopathies; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Middle Aged; Retrospective Studies; Risk Factors; Sulfonylurea Compounds; United States; Ventricular Dysfunction

2018
Comparison of mortality and cardiovascular event risk associated with various insulin secretagogues: A nationwide real-world analysis.
    Diabetes research and clinical practice, 2019, Volume: 152

    Topics: Aged; Carbamates; Cardiovascular Diseases; Cohort Studies; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Follow-Up Studies; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Male; Middle Aged; Mortality; Piperidines; Secretagogues; Sulfonylurea Compounds; Taiwan

2019
Computational Drug Repositioning for Chagas Disease Using Protein-Ligand Interaction Profiling.
    International journal of molecular sciences, 2020, Jun-16, Volume: 21, Issue:12

    Topics: Chagas Disease; Computer Simulation; Drug Repositioning; Folic Acid Antagonists; Glipizide; Glyburide; Humans; Ligands; Molecular Docking Simulation; Molecular Structure; Pyrimidines; Structure-Activity Relationship; Sulfonylurea Compounds; Trypanocidal Agents; Trypanosoma cruzi

2020
Risk of sudden cardiac arrest and ventricular arrhythmia with sulfonylureas: An experience with conceptual replication in two independent populations.
    Scientific reports, 2020, 06-22, Volume: 10, Issue:1

    Topics: Aged; Cohort Studies; Death, Sudden, Cardiac; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Male; Medicaid; Middle Aged; Sulfonylurea Compounds; Treatment Outcome; United States; Ventricular Fibrillation

2020
Sensitive detection of antidiabetic compounds and one degradation product in wastewater samples by a new SPE-LC-MS/MS method.
    Journal of environmental science and health. Part A, Toxic/hazardous substances & environmental engineering, 2021, Volume: 56, Issue:3

    Topics: Chromatography, Liquid; Environmental Monitoring; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Metformin; Reproducibility of Results; Solid Phase Extraction; Sulfonylurea Compounds; Tandem Mass Spectrometry; Wastewater; Water Pollutants, Chemical

2021
Angiotensin-Converting Enzyme Inhibitors Used Concomitantly with Insulin Secretagogues and the Risk of Serious Hypoglycemia.
    Clinical pharmacology and therapeutics, 2022, Volume: 111, Issue:1

    Topics: Administrative Claims, Healthcare; Aged; Aged, 80 and over; Angiotensin-Converting Enzyme Inhibitors; Carbamates; Databases, Factual; Diabetes Mellitus, Type 2; Drug Interactions; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Medicaid; Metformin; Middle Aged; Nateglinide; Pharmacoepidemiology; Piperidines; Secretagogues; Sulfonylurea Compounds; United States

2022
Total Synthesis of Glipizide and Glibenclamide in Continuous Flow.
    Chemistry (Weinheim an der Bergstrasse, Germany), 2021, Nov-17, Volume: 27, Issue:64

    Topics: Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin

2021
Comparative safety of sulfonylureas among U.S. nursing home residents.
    Journal of the American Geriatrics Society, 2023, Volume: 71, Issue:4

    Topics: Aged; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Male; Medicare; Myocardial Infarction; Nursing Homes; Retrospective Studies; Stroke; United States

2023
Analytical Method Capable of Quantifying Eight Nitrosamine Impurities from Five Different Commercially Available Metformin Formulations with Glipizide, Glibenclamide, Gliclazide, Evogliptin, and Glimepiride by Ultra High Performance Liquid Chromatography
    Journal of pharmaceutical sciences, 2023, Volume: 112, Issue:5

    Topics: Chromatography, High Pressure Liquid; Chromatography, Liquid; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Humans; Metformin; Nitrosamines; Pharmaceutical Preparations; Tandem Mass Spectrometry

2023
Analysis of Hypoglycemic Drugs by Liquid Chromatography-Tandem Mass Spectrometry.
    Methods in molecular biology (Clifton, N.J.), 2024, Volume: 2737

    Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Chromatography, Liquid; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Nateglinide; Pioglitazone; Rosiglitazone; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Tolazamide; Tolbutamide

2024