glyburide and clonidine

glyburide has been researched along with clonidine in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.33)18.7374
1990's10 (33.33)18.2507
2000's16 (53.33)29.6817
2010's3 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Barnes, PJ; Belvisi, MG; Miura, M; Stretton, D1
Burnham, BL; Chick, WL; Clark, SA1
Ammälä, C; Arkhammar, P; Berggren, PO; Bokvist, K; Larsson, O; Rorsman, P; Wåhlander, K1
Angus, JA; McPherson, GA1
Altszuler, N; Cherksey, B1
Faber, JE; Tateishi, J1
Edwards, G; Ibbotson, T; Weston, AH1
Cooper, JR; Zoltay, G1
Lodge, NJ; Smith, MA1
Dohi, S; Iida, H; Ishiyama, T1
Foldes, FF; Matkó, I; Nagashima, H; Oe, K; Sántha, E; Sperlágh, B; Vizi, ES1
Bell, K; Favaloro, J; Iskander, MM; Khalil, V; McPherson, GA1
Hashimoto, S; Makita, T; Saito, M; Sakai, K; Shibata, O; Sumikawa, K1
Fülöp, K; Fürst, S; Gyires, K; Müllner, K; Rónai, AZ1
Koga, Y; Okuda, T; Yamazumi, I1
García-Barrado, MJ; Iglesias-Osma, MC; Martín, M; Moratinos, J; Rodríguez, R1
Eckhardt, K; Feuerstein, TJ; Günter, T; Roth, P; Schmidt, S1
Carvalho, LC; de Moura, RS; Madeira, SV; Miranda, DZ; Pinto, AC; Rangel, BM; Resende, AC; Rubenich, LM; Sicca, RF; Souza, MA; Tano, T1
Dkhar, SA; Naveen, AT; Peddyreddy, MK; Ramaswamy, S; Shewade, DG1

Reviews

1 review(s) available for glyburide and clonidine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

29 other study(ies) available for glyburide and clonidine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Calcium-activated potassium channels mediate prejunctional inhibition of peripheral sensory nerves.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Feb-15, Volume: 89, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Apamin; Bronchi; Bronchoconstriction; Calcium; Cation Transport Proteins; Charybdotoxin; Clonidine; Cricetinae; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Glyburide; In Vitro Techniques; Ion Channel Gating; Male; Neural Inhibition; Neurons, Afferent; Neuropeptide Y; Potassium Channels; Pyrrolidines; Scorpion Venoms

1992
Modulation of glucose-induced insulin secretion from a rat clonal beta-cell line.
    Endocrinology, 1990, Volume: 127, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Alanine; Animals; Carbachol; Cell Line; Clone Cells; Clonidine; Colforsin; Dose-Response Relationship, Drug; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Potassium; Rats; Stereoisomerism

1990
Activation by adrenaline of a low-conductance G protein-dependent K+ channel in mouse pancreatic B cells.
    Nature, 1991, Jan-03, Volume: 349, Issue:6304

    Topics: Animals; Clonidine; Epinephrine; Glucose; Glyburide; Islets of Langerhans; Membrane Potentials; Mice; Potassium Channels; Tolbutamide; Yohimbine

1991
Characterization of responses to cromakalim and pinacidil in smooth and cardiac muscle by use of selective antagonists.
    British journal of pharmacology, 1990, Volume: 100, Issue:2

    Topics: Animals; Aorta, Thoracic; Benzopyrans; Clonidine; Coronary Vessels; Cromakalim; Dogs; Electric Stimulation; Glyburide; Guanidines; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Myocardial Contraction; Phentolamine; Pinacidil; Potassium Channels; Pyrroles; Rats

1990
Tolbutamide and glyburide differ in effectiveness to displace alpha- and beta-adrenergic radioligands in pancreatic islet cells and membranes.
    Diabetes, 1984, Volume: 33, Issue:5

    Topics: Alprenolol; Animals; Cell Membrane; Clonidine; Dihydroalprenolol; Epinephrine; Glyburide; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tolbutamide

1984
ATP-sensitive K+ channels mediate alpha 2D-adrenergic receptor contraction of arteriolar smooth muscle and reversal of contraction by hypoxia.
    Circulation research, 1995, Volume: 76, Issue:1

    Topics: Adenosine Triphosphate; Animals; Brimonidine Tartrate; Cell Hypoxia; Clonidine; Glyburide; In Vitro Techniques; Muscle, Smooth, Vascular; Nitroprusside; Phenylephrine; Potassium Channels; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction

1995
Antagonism of levcromakalim by imidazoline- and guanidine-derivatives in rat portal vein: involvement of the delayed rectifier.
    British journal of pharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Antazoline; Benzopyrans; Clonidine; Cromakalim; Glyburide; Guanabenz; Imidazoline Receptors; Male; Phentolamine; Portal Vein; Potassium Channels; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Drug

1993
Dendrotoxin blocks a class of potassium channels that are opened by inhibitory presynaptic modulators in rat cortical synaptosomes and slices.
    Cellular and molecular neurobiology, 1993, Volume: 13, Issue:1

    Topics: 2-Chloroadenosine; Acetylcholine; Animals; Carbachol; Cerebral Cortex; Clonidine; Elapid Venoms; Glyburide; Ion Channel Gating; Morphine; Potassium Channels; Rats; Rats, Sprague-Dawley; Synaptosomes; Tetraethylammonium; Tetraethylammonium Compounds; Veratridine

1993
The novel cardioprotective agent BMS-180448 activates a potassium conductance in cardiac and vascular smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:4

    Topics: Animals; Aorta, Thoracic; Benzopyrans; Cardiotonic Agents; Cardiovascular Agents; Cells, Cultured; Clonidine; Glyburide; Guanidines; Guinea Pigs; Heart Ventricles; Male; Muscle, Smooth, Vascular; Myocardium; Patch-Clamp Techniques; Potassium Channels; Rabbits; Rubidium Radioisotopes

1996
The vascular effects of topical and intravenous alpha2-adrenoceptor agonist clonidine on canine pial microcirculation.
    Anesthesia and analgesia, 1998, Volume: 86, Issue:4

    Topics: Adjuvants, Anesthesia; Administration, Topical; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Blood Glucose; Cerebrovascular Circulation; Clonidine; Craniotomy; Dogs; Dose-Response Relationship, Drug; Glyburide; Heart Rate; Injections, Intravenous; Microcirculation; Pentobarbital; Pia Mater; Potassium; Potassium Channel Blockers; Receptors, Adrenergic, alpha-2; Vasoconstrictor Agents; Vasodilator Agents; Veins; Yohimbine

1998
Modulation of norepinephrine release by ATP-dependent K(+)-channel activators and inhibitors in guinea-pig and human isolated right atrium.
    Cardiovascular research, 1999, Volume: 43, Issue:1

    Topics: Adenosine; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Analysis of Variance; Animals; Clonidine; Cromakalim; Decanoic Acids; Diazoxide; Dose-Response Relationship, Drug; Glyburide; Guinea Pigs; Heart Atria; Humans; Hydroxy Acids; In Vitro Techniques; Male; Muscarinic Agonists; Norepinephrine; Oxotremorine; Pinacidil; Potassium Channel Blockers; Potassium Channels; Stimulation, Chemical; Sympathetic Nervous System

1999
The identification of a potent imidazoline-based vascular K(ATP) channel antagonist.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 362, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; ATP-Binding Cassette Transporters; Cattle; Clonidine; Coronary Vessels; Cromakalim; Glyburide; Guanidines; Heart Atria; Heart Rate; Hypoglycemic Agents; Imidazoles; In Vitro Techniques; KATP Channels; Muscle, Smooth, Vascular; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyridines; Radioligand Assay; Rats; Swine; Vasodilator Agents

2000
Clonidine attenuates the carbachol-induced contractile and phosphatidylinositol responses of rat trachea.
    The Journal of pharmacy and pharmacology, 2000, Volume: 52, Issue:12

    Topics: Aluminum Compounds; Analgesics; Animals; Carbachol; Clonidine; Dose-Response Relationship, Drug; Fluorides; Glyburide; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Rats; Rats, Wistar; Trachea

2000
Involvement of central K(ATP) channels in the gastric antisecretory action of alpha2-adrenoceptor agonists and beta-endorphin in rats.
    European journal of pharmacology, 2002, Jan-25, Volume: 435, Issue:2-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; beta-Endorphin; Central Nervous System; Clonidine; Gastric Acid; Gastric Mucosa; Glyburide; Hypoglycemic Agents; Ligation; Male; Membrane Proteins; Oxymetazoline; Potassium Channels; Pylorus; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Stomach

2002
Involvement of potassium channels in spinal antinociceptions induced by fentanyl, clonidine and bethanechol in rats.
    Japanese journal of pharmacology, 2001, Volume: 87, Issue:4

    Topics: Adenosine Triphosphatases; Adrenergic alpha-Agonists; Analgesics, Opioid; Animals; Bethanechol; Charybdotoxin; Clonidine; Enzyme Inhibitors; Fentanyl; Glyburide; Injections, Spinal; Male; Motor Activity; Muscarinic Antagonists; Nicorandil; Pain Measurement; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Reaction Time; Spinal Cord

2001
Role of mu-opioid receptors in insulin release in the presence of inhibitory and excitatory secretagogues.
    European journal of pharmacology, 2002, Jul-12, Volume: 448, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Brimonidine Tartrate; Clonidine; Drug Interactions; Female; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Naloxone; Quinoxalines; Receptors, Opioid, mu; Somatostatin

2002
Differential effects of K(ATP) channel blockers on [(3)H]-noradrenaline overflow after short- and long-term exposure to (+)-oxaprotiline or desipramine.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:2

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Animals; Antidepressive Agents; Autoreceptors; Clonidine; Desipramine; Drug Interactions; Glyburide; In Vitro Techniques; Male; Maprotiline; Neocortex; Norepinephrine; Potassium Channel Blockers; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Time Factors

2003
Mechanism of the endothelium-dependent vasodilation and the antihypertensive effect of Brazilian red wine.
    Journal of cardiovascular pharmacology, 2004, Volume: 44, Issue:3

    Topics: Acetylcholine; Administration, Oral; Alcohol Drinking; Animals; Apamin; Atropine; Blood Pressure; Bradykinin; Brazil; Charybdotoxin; Clonidine; Deoxycholic Acid; Drug Therapy, Combination; Endothelium, Vascular; Flavonoids; Glyburide; Guanylate Cyclase; Hypertension; Indomethacin; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitroglycerin; Norepinephrine; Oxadiazoles; Perfusion; Phenols; Polyphenols; Potassium Chloride; Pressure; Pyrilamine; Quinazolines; Quinoxalines; Rats; Rats, Wistar; Vasoconstriction; Vasodilation; Wine; Yohimbine

2004
An inherent acceleratory effect of insulin on small intestinal transit and its pharmacological characterization in normal mice.
    World journal of gastroenterology, 2006, Apr-28, Volume: 12, Issue:16

    Topics: Animals; Atropine; Calcium Channels; Clonidine; Gastrointestinal Transit; Glyburide; Insulin; Insulin Secretion; Intestine, Small; Male; Mice; Naloxone; Ondansetron; Receptors, Opioid; Verapamil

2006