glyburide and cifenline

glyburide has been researched along with cifenline in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (50.00)18.2507
2000's5 (35.71)29.6817
2010's2 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Arita, M; Kiyosue, T; Sato, T; Wu, B1
Okamoto, K; Sakuta, H; Watanabe, Y1
Arita, M; Kiyosue, T; Nakamura, S; Sato, T; Wu, B1
Ai, T; Horie, M; Ishida, H; Ishida-Takahashi, A; Sasayama, S; Tsuura, Y1
Fujimoto, S; Horie, M; Ishida, H; Ishida-Takahashi, A; Kato, S; Mukai, E; Seino, Y; Tsuda, K; Tsuura, Y1
Arita, M; Sato, T; Shigematsu, S1
Horie, M; Ishida, H; Mukai, E; Noma, A; Seino, Y; Takano, M1
Horie, M; Ishida, H; Ishida-Takahashi, A; Sasayama, S; Seino, Y; Tsuji, K; Watanuki, M; Yuzuki, Y1
Brading, AF; Ito, Y; Masaki, I; Sueishi, K; Takano, M; Teramoto, N; Yonemitsu, Y; Yunoki, T1

Other Studies

14 other study(ies) available for glyburide and cifenline

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Blockade of 2,4-dinitrophenol induced ATP sensitive potassium current in guinea pig ventricular myocytes by class I antiarrhythmic drugs.
    Cardiovascular research, 1992, Volume: 26, Issue:11

    Topics: 2,4-Dinitrophenol; Action Potentials; Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Dinitrophenols; Disopyramide; Flecainide; Glyburide; Guinea Pigs; Heart Ventricles; Imidazoles; Lidocaine; Mexiletine; Myocardium; Piperidines; Potassium; Procainamide; Pyridines

1992
Antiarrhythmic drugs, clofilium and cibenzoline are potent inhibitors of glibenclamide-sensitive K+ currents in Xenopus oocytes.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Benzopyrans; Electrophysiology; Female; Glyburide; Imidazoles; Membrane Potentials; Oocytes; Potassium Channels; Pyridines; Quaternary Ammonium Compounds; Xenopus laevis

1993
Cibenzoline inhibits diazoxide- and 2,4-dinitrophenol-activated ATP-sensitive K+ channels in guinea-pig ventricular cells.
    British journal of pharmacology, 1993, Volume: 108, Issue:2

    Topics: 2,4-Dinitrophenol; Action Potentials; Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Diazoxide; Dinitrophenols; Glyburide; Guinea Pigs; Heart; Heart Ventricles; Imidazoles; In Vitro Techniques; Membrane Potentials; Potassium Channels

1993
Block of pancreatic ATP-sensitive K+ channels and insulinotrophic action by the antiarrhythmic agent, cibenzoline.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Animals; Anti-Arrhythmia Agents; Glyburide; Hydrogen-Ion Concentration; Hypoglycemia; Hypoglycemic Agents; Imidazoles; Insulin; Insulin Secretion; Islets of Langerhans; Male; Potassium Channels; Rats; Rats, Wistar

1996
Metabolic inhibition impairs ATP-sensitive K+ channel block by sulfonylurea in pancreatic beta-cells.
    The American journal of physiology, 1998, Volume: 274, Issue:1

    Topics: 2,4-Dinitrophenol; Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; ATP-Binding Cassette Transporters; Cells, Cultured; Glyburide; Imidazoles; Islets of Langerhans; Male; Membrane Potentials; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Drug; Sulfonylurea Receptors

1998
Class I antiarrhythmic drugs alter the severity of myocardial stunning by modulating ATP-sensitive K+ channels in guinea pig ventricular muscles.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:3

    Topics: Animals; Anti-Arrhythmia Agents; Glyburide; Guinea Pigs; Heart; Heart Ventricles; Imidazoles; Lidocaine; Male; Mexiletine; Myocardial Stunning; Potassium Channels

1998
The antiarrhythmic agent cibenzoline inhibits KATP channels by binding to Kir6.2.
    Biochemical and biophysical research communications, 1998, Oct-20, Volume: 251, Issue:2

    Topics: Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; ATP-Binding Cassette Transporters; Cloning, Molecular; COS Cells; Glyburide; Imidazoles; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptor Cross-Talk; Receptors, Drug; Recombinant Proteins; Sequence Deletion; Sulfonylurea Receptors; Transfection

1998
Blockade of cardiac ATP-sensitive K+ channel by cibenzoline targets its pore-forming subunit.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Cell Membrane Permeability; Cells, Cultured; Drug Interactions; Electrophysiology; Female; Glyburide; Guinea Pigs; Heart Ventricles; Hydrogen-Ion Concentration; Hypoglycemic Agents; Imidazoles; Male; Patch-Clamp Techniques; Pinacidil; Potassium Channels

2000
Dual action of ZD6169, a novel K(+) channel opener, on ATP-sensitive K(+) channels in pig urethral myocytes.
    British journal of pharmacology, 2001, Volume: 133, Issue:1

    Topics: Adenosine Triphosphate; Amides; Animals; Anti-Arrhythmia Agents; Benzophenones; Cells, Cultured; COS Cells; Cromakalim; Electric Conductivity; Female; Glyburide; Hypoglycemic Agents; Imidazoles; Ion Channel Gating; Membrane Potentials; Muscle, Smooth; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Swine; Time Factors; Urethra; Vasodilator Agents

2001