glyburide has been researched along with chlorpropamide in 131 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 86 (65.65) | 18.7374 |
1990's | 21 (16.03) | 18.2507 |
2000's | 12 (9.16) | 29.6817 |
2010's | 11 (8.40) | 24.3611 |
2020's | 1 (0.76) | 2.80 |
Authors | Studies |
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Hashimoto, Y; Inui, K; Saito, H; Uwai, Y | 1 |
Topliss, JG; Yoshida, F | 1 |
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M | 1 |
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Buttar, D; Colclough, N; Gerhardt, S; MacFaul, PA; Maskos, K; Phillips, SD; Plowright, A; Steinbacher, S; Steuber, H; Tam, K; Whittamore, P | 1 |
Barber, J; Dawson, S; Kenna, JG; Paul, N; Stahl, S | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Melander, A; Wåhlin-Boll, E | 2 |
Luntz, GR | 2 |
Campbell, IW; Clarke, BF | 2 |
Balant, L | 1 |
Haslbeck, M | 1 |
Macchi, IA; Zeytinoğlu, FN | 1 |
Handler, JS; Keiser, HR; Zusman, RM | 1 |
Foy, JM; Lucas, PD | 1 |
Christensen, LK; Hansen, JM | 1 |
Bloom, A; Bulpitt, CJ; Shaw, KM | 1 |
Jorgensen, KD | 1 |
Di Saverio, S; Roncaia, R; Torri, A; Zanni, A | 1 |
Balant, L; Fabre, J; Loutan, L; Samimi, H; Tillolès, M | 1 |
Biggs, PI; Owens, DR; Seldrup, J; Shetty, KJ; Wragg, KG | 1 |
Bennett, MA; Fitzgerald, MG; Malins, JM; Pentecost, BL; Soler, NG | 1 |
Bullock, I; Galloway, DB; Gilbert, JC; Petrie, JC; Watson, WA | 1 |
Haider, Z; Obaidullah, S | 1 |
Andreev, D; Pampulov, L | 1 |
Müller, WE; Wollert, U | 1 |
Brown, KF; Crooks, MJ | 2 |
Sauer, H; Schneider, B | 1 |
Madhavan, R; Sankaran, JR; Seshasaianam, C; Seshiah, V; Shanker, R; Sundaram, A; Venkataraman, S | 1 |
Friedberg, SJ; Pugh, JA; Ramirez, G; Sawyer, J; Tuley, M; Wagner, ML | 1 |
Sugarman, JR | 1 |
Harrower, AD | 2 |
Corenblum, B; Shumak, SL; Steiner, G | 1 |
Boutagy, JS; Shenfield, GM; Webb, C | 1 |
Dux, S; Huminer, D; Pitlik, SD; Rosenfeld, JB | 1 |
Morrison, AD; Shank, WA | 1 |
Bressler, R; Jackson, JE | 1 |
Balabolkin, MI; Nedosugova, LV | 1 |
Bowers, CY; Kosola, JW; Prosser, PR | 1 |
Colombo, R; Pinelli, A; Tofanetti, O; Trivulzio, S; Zecca, L | 1 |
Owens, DR | 1 |
Feldman, JM | 1 |
Fajardo, F; Ginier, P; Levin, SR; Madan, S | 1 |
Oksala, H; Pitkäjärvi, T; Ylitalo, P | 1 |
Burnett, MA; Davies, EG; Harris, EA; Hosker, JP; Turner, RC | 1 |
Hatao, K; Kaku, K; Kaneko, T; Matsuda, M; Tsuchiya, M | 1 |
Ravina, A | 1 |
Jackson, WP; Keller, P; Van Mieghem, W | 1 |
Foy, JM; Standing, VF | 1 |
Daweke, H; Fähndrich, W; Liebermeister, H; Schmitt, H | 1 |
De Baere, H; De Leeuw, I; Decraene, P; Lemmens, P; Verhaegen, H | 2 |
Stowers, JM | 1 |
Ceuterick-Goethals, AM; De Schepper, PJ; Debeer, L; Mannaerts, G | 1 |
Kain, T; Ravina, A | 1 |
Hsu, PL; Luzzi, LA; Ma, JK | 1 |
Kar, BC; Panda, NC; Parija, CR; Tej, SC; Tripathy, BB | 1 |
Tattersall, RB | 2 |
Hasselblatt, A; Panten, U; Poser, W; Schönborn, J | 1 |
Mughini, L; Polosa, P | 1 |
Scott, D; Thomas, M | 1 |
Bavel'skii, ZE; Kuts, LG; Lazaris, YA | 1 |
Alberti, KG; Ball, S; Woods, HF | 1 |
Aziz, MT; Einen, MA; el-Ebrashy, N; Higazi, AM; Mashaly, M | 1 |
Brogard, JM; Dorner, M; Kuntzmann, F; Touitou, D | 1 |
Edlén, A | 1 |
Bird, GW; Eeles, GH; Litchfield, JA; Rahman, M; Wingham, J | 1 |
Parodi, FA | 1 |
Mitra, D; Mutalik, GS; Nayak, NJ; Oak, VR | 1 |
Baigorria, L; Contreras, AR; Gabrielli, S | 1 |
Bloom, A | 1 |
Henning, H; Look, D | 1 |
Blohmé, G | 1 |
Bhatia, SK; Hadden, DR; Montgomery, DA | 1 |
Howanitz, J; Miller, M; Moses, AM | 1 |
Potitong, B | 1 |
Sigroth, K; Steen, B; Svanborg, A | 1 |
Creutzfeldt, W; Scheler, F; Wigger, W | 1 |
Consiglio, D; Hopps, V; Mantia, G | 1 |
Hellman, B; Sehlin, J; Täljedal, IB | 1 |
Bailey, CJ; Billingham, MS; Hall, RA; Simpson, S | 2 |
Lunetta, M; Mughini, L; Mughini, MT; Presti, C | 1 |
Melander, A; Sartor, G; Scherstén, B; Wåhlin-Boll, E | 2 |
Feldman, JM; Skillman, TG | 1 |
Lowy, C; Perkins, JR; Sönksen, PH; West, TE | 1 |
Bailey, CJ; Broadbent, ME | 1 |
Huupponen, R; Saarimaa, H; Viikari, J | 1 |
Beljic, T; Miric, M | 1 |
Elliott, BD; Johnson, R; Langer, O; Prihoda, T; Schenker, S | 1 |
Tammelleo, AD | 1 |
Duarte, AL; Malerbi, DA; Paiva, ES; Wajchenberg, BL | 1 |
Selvaag, E | 1 |
Abenhaim, L; Monette, J; van Staa, T | 1 |
Chan, TY; Cheung, AY | 1 |
Furuya, K; Iwata, M; Machida, Y; Onishi, H; Shirotake, S; Takahashi, Y | 1 |
Cull, CA; Holman, RR; Matthews, DR; Stratton, IM; Turner, RC | 1 |
Ikeda, T; Ochi, H | 1 |
André, P | 1 |
Galli Kienle, M; Magni, F; Marazzini, L; Monti, L; Pereira, S | 1 |
Corrall, RJ; Hattersley, AT; Liddell, WG; Pearson, ER; Shepherd, M | 1 |
Gottsäter, M; Lindberg, G; Lindwall, K; Melander, A; Olsson, J; Tisell, A | 1 |
Matthews, DR; Wallace, TM | 1 |
Saha, B | 1 |
Fatehi, M; Lang, VY; Light, PE | 1 |
Friščić, T; Mottillo, C; Štrukil, V; Tan, D | 1 |
Jannetto, PJ; Langman, LJ | 1 |
13 review(s) available for glyburide and chlorpropamide
Article | Year |
---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
["First" and "second" generation sulfonylureas: distinction or difference? (author's transl)].
Topics: Animals; Chlorpropamide; Dose-Response Relationship, Drug; Glipizide; Glyburide; Half-Life; Humans; Hypoglycemic Agents; Kinetics; Structure-Activity Relationship; Sulfonylurea Compounds; Tolbutamide | 1978 |
[New aspects of therapy with oral antidiabetic agents].
Topics: Acidosis; Biguanides; Blood Proteins; Chlorpropamide; Diabetes Mellitus; Diabetic Nephropathies; Drug Interactions; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Protein Binding; Sulfonamides; Sulfonylurea Compounds; Tolbutamide | 1979 |
Drug interactions with oral sulphonylurea hypoglycaemic drugs.
Topics: Allopurinol; Analgesics; Anticoagulants; Chloramphenicol; Chlorpropamide; Disulfiram; Drug Interactions; Ethanol; Glyburide; Humans; Hypoglycemic Agents; Hypolipidemic Agents; Kinetics; Monoamine Oxidase Inhibitors; Novobiocin; Phenylbutazone; Phenytoin; Probenecid; Propranolol; Rifampin; Sulfonamides; Sulfonylurea Compounds; Tolbutamide | 1977 |
[What is achieved by the therapy with oral antidiabetics?].
Topics: Administration, Oral; Adult; Biguanides; Chlorpropamide; Diabetes Mellitus; Diabetic Angiopathies; Drug Interactions; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Obesity; Phenformin; Prospective Studies; Retrospective Studies | 1976 |
Is combination sulfonylurea and insulin therapy useful in NIDDM patients? A metaanalysis.
Topics: Blood Glucose; C-Peptide; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; MEDLINE; Meta-Analysis as Topic; Middle Aged; Periodicals as Topic; Sulfonylurea Compounds; Tolazamide; Treatment Outcome; United States | 1992 |
Inadvertent sulfonylurea-induced hypoglycemia. A dangerous, but preventable condition.
Topics: Aged; Chlorpropamide; Female; Glyburide; Humans; Hypoglycemia; Male; Medication Errors | 1989 |
Oral sulfonylureas for the treatment of type II diabetes: an update.
Topics: Administration, Oral; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Hypersensitivity; Glipizide; Glyburide; Humans; Insulin Resistance; Kinetics; Liver; Nausea; Patient Education as Topic; Sulfonylurea Compounds | 1986 |
Effects of oral sulfonylureas on the spectrum of defects in non-insulin-dependent diabetes mellitus.
Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Clinical Trials as Topic; Combined Modality Therapy; Diabetes Mellitus, Type 2; Energy Intake; Glyburide; Humans; Insulin; Insulin Resistance; Insulin Secretion; Islets of Langerhans; Kinetics; Middle Aged; Physical Exertion; Prospective Studies; Sulfonylurea Compounds; United Kingdom | 1985 |
Review of glyburide after one year on the market.
Topics: Chlorpropamide; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Evaluation Studies as Topic; Glyburide; Humans; Insulin; Intestinal Absorption | 1985 |
Oral treatment in diabetes.
Topics: Acetohexamide; Acidosis; Administration, Oral; Animals; Biguanides; Cardiovascular Diseases; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Glyburide; Humans; Hypoglycemia; Liver; Obesity; Structure-Activity Relationship; Sulfonylurea Compounds; Tolazamide; Tolbutamide | 1972 |
Glibenclamide: a review.
Topics: Administration, Oral; Adolescent; Adult; Aged; Animals; Biguanides; Blood Glucose; Carbon Isotopes; Child; Chlorpropamide; Diabetes Mellitus; Dogs; Drug Interactions; Drug Synergism; Female; Fibrinolysis; Glucagon; Glucose; Glyburide; Guinea Pigs; Humans; Hypoglycemia; In Vitro Techniques; Insulin; Islets of Langerhans; Lipids; Liver Glycogen; Pancreas; Pregnancy; Protein Binding; Rabbits; Rats; Stimulation, Chemical; Sulfonylurea Compounds | 1971 |
[25 years of diabetic treatment by oral hypoglycemic agents: successes and failures].
Topics: Aged; Aging; Blood Glucose; Cardiovascular Diseases; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diet, Reducing; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Middle Aged; Phenformin; Sulfonylurea Compounds; Tolbutamide | 1984 |
17 trial(s) available for glyburide and chlorpropamide
Article | Year |
---|---|
Repeated blood glucose and plasma insulin levels in normal volunteer subjects receiving isocaloric meals, before and after chlorpropamide and glibenclamide.
Topics: Adolescent; Adult; Blood Glucose; Chlorpropamide; Diet; Glyburide; Humans; Insulin; Male | 1977 |
[Therapeutic effect of glibenclamide contrasted with other oral antidiabetic agents].
Topics: Administration, Oral; Adult; Biguanides; Chlorpropamide; Chronic Disease; Clinical Trials as Topic; Diabetes Mellitus; Drug Evaluation; Drug Therapy, Combination; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Tolbutamide | 1975 |
Is combination sulfonylurea and insulin therapy useful in NIDDM patients? A metaanalysis.
Topics: Blood Glucose; C-Peptide; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; MEDLINE; Meta-Analysis as Topic; Middle Aged; Periodicals as Topic; Sulfonylurea Compounds; Tolazamide; Treatment Outcome; United States | 1992 |
Efficacy of gliclazide in comparison with other sulphonylureas in the treatment of NIDDM.
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Diet, Diabetic; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Tolbutamide | 1991 |
U.K. prospective diabetes study. II. Reduction in HbA1c with basal insulin supplement, sulfonylurea, or biguanide therapy in maturity-onset diabetes. A multicenter study.
Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Diabetes Mellitus, Type 2; Female; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Insulin, Long-Acting; Male; Metformin; Middle Aged; Obesity; Random Allocation | 1985 |
The 24-hour effects of glyburide and chlorpropamide after chronic treatment of type II diabetic patients.
Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Cholesterol; Diabetes Mellitus, Type 2; Drug Evaluation; Female; Glucagon; Glyburide; Growth Hormone; Humans; Insulin; Male; Middle Aged; Radioimmunoassay; Random Allocation; Time Factors; Triglycerides | 1985 |
Effects of oral sulfonylureas on the spectrum of defects in non-insulin-dependent diabetes mellitus.
Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Clinical Trials as Topic; Combined Modality Therapy; Diabetes Mellitus, Type 2; Energy Intake; Glyburide; Humans; Insulin; Insulin Resistance; Insulin Secretion; Islets of Langerhans; Kinetics; Middle Aged; Physical Exertion; Prospective Studies; Sulfonylurea Compounds; United Kingdom | 1985 |
Once-daily use of glyburide.
Topics: Blood Glucose; Body Weight; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Administration Schedule; Glucagon; Glyburide; Glycosuria; Humans; Insulin | 1985 |
Comparison of acute and prolonged effects of glibenclamide and chlorpropamide in patients with non-insulin-dependent diabetes.
Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Creatinine; Diabetes Mellitus, Type 2; Electrolytes; Female; Glyburide; Humans; Insulin; Male; Middle Aged; Sex Factors; Time Factors | 1985 |
Comparison of diabetic control in type 2 (non-insulin dependent) diabetic patients treated with different sulphonylureas.
Topics: Aged; Chlorpropamide; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Middle Aged; Random Allocation; Sulfonylurea Compounds | 1985 |
[Clinical testing of a sulfonylurea preparation (glibenclamide)].
Topics: Adult; Aged; Chlorpropamide; Clinical Trials as Topic; Diabetes Mellitus; Diet Therapy; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Tolbutamide | 1969 |
Improved metabolic control does not reverse left ventricular filling abnormalities in newly diagnosed non-insulin-dependent diabetes patients.
Topics: Adult; Blood Glucose; Blood Pressure; C-Peptide; Chlorpropamide; Cholesterol; Diabetes Mellitus, Type 2; Diet, Diabetic; Echocardiography, Doppler; Female; Follow-Up Studies; Glucagon; Glyburide; Glycated Hemoglobin; Heart Rate; Humans; Male; Middle Aged; Reference Values; Triglycerides; Ventricular Function, Left | 1994 |
United Kingdom Prospective Diabetes Study (UKPDS). 13: Relative efficacy of randomly allocated diet, sulphonylurea, insulin, or metformin in patients with newly diagnosed non-insulin dependent diabetes followed for three years.
Topics: Adult; Aged; Blood Glucose; Body Weight; Chlorpropamide; Diabetes Mellitus; Diabetes Mellitus, Type 2; Female; Follow-Up Studies; Glyburide; Glycated Hemoglobin; Humans; Insulin; Male; Metformin; Middle Aged; Obesity; Patient Compliance; Sulfonylurea Compounds | 1995 |
UKPDS 28: a randomized trial of efficacy of early addition of metformin in sulfonylurea-treated type 2 diabetes. U.K. Prospective Diabetes Study Group.
Topics: Blood Glucose; Blood Pressure; Chlorpropamide; Cholesterol; Clinical Protocols; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Patient Compliance; Sulfonylurea Compounds; Triglycerides; United Kingdom | 1998 |
UKPDS 26: Sulphonylurea failure in non-insulin-dependent diabetic patients over six years. UK Prospective Diabetes Study (UKPDS) Group.
Topics: Adult; Blood Glucose; Body Mass Index; Chlorpropamide; Diabetes Mellitus, Type 2; Fasting; Female; Glyburide; Humans; Hypoglycemic Agents; Islets of Langerhans; Male; Middle Aged; Prospective Studies; Treatment Failure; United Kingdom | 1998 |
Intensive blood-glucose control with sulphonylureas or insulin compared with conventional treatment and risk of complications in patients with type 2 diabetes (UKPDS 33). UK Prospective Diabetes Study (UKPDS) Group.
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Prospective Studies; Risk Factors; Sulfonylurea Compounds | 1998 |
Effect of intensive blood-glucose control with metformin on complications in overweight patients with type 2 diabetes (UKPDS 34). UK Prospective Diabetes Study (UKPDS) Group.
Topics: Chlorpropamide; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Obesity; Prospective Studies; Risk Factors | 1998 |
103 other study(ies) available for glyburide and chlorpropamide
Article | Year |
---|---|
Inhibitory effect of anti-diabetic agents on rat organic anion transporter rOAT1.
Topics: Animals; Anion Transport Proteins; Binding, Competitive; Carbon Radioisotopes; Carrier Proteins; Chlorpropamide; Cyclohexanes; Dose-Response Relationship, Drug; Female; Glyburide; Hypoglycemic Agents; Kinetics; Nateglinide; Oocytes; p-Aminohippuric Acid; Phenylalanine; Rats; RNA, Complementary; Sulfonylurea Compounds; Tolbutamide; Xenopus | 2000 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Cheminformatic models to predict binding affinities to human serum albumin.
Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids | 2001 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship | 2008 |
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions.
Topics: Binding Sites; Crystallography, X-Ray; Drug Interactions; Humans; Pharmaceutical Preparations; Protein Binding; Protein Structure, Tertiary; Serum Albumin; Spectrometry, Fluorescence | 2010 |
In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Cholestasis; Drug-Related Side Effects and Adverse Reactions; Humans; Insecta; Rats; Risk Factors | 2012 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
High-performance liquid chromatographic determination of glipizide and some other sulfonylurea drugs in serum.
Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Glipizide; Glyburide; Humans; Hydrogen-Ion Concentration; Sulfonylurea Compounds; Tolbutamide | 1979 |
Letter: Treatment of maturity-onset diabetes.
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus; Diet, Diabetic; Glyburide; Humans | 1975 |
Letter: Treatment of maturity-onset diabetes.
Topics: Adult; Age Factors; Aged; Blood Glucose; Body Weight; Chlorpropamide; Diabetes Mellitus; Diet, Diabetic; Glyburide; Humans; Middle Aged | 1975 |
Letter: Treatment of maturity-onset diabetes.
Topics: Adult; Blood Glucose; Body Weight; Chlorpropamide; Diabetes Mellitus; Glyburide; Humans | 1975 |
Hyaluronidase-induced inhibition of the insulinotropic action of sulfonylureas, leucine, and glucagon in rodent isolated pancreatic islets.
Topics: Animals; Chlorpropamide; Cricetinae; Female; Glucagon; Glucose; Glyburide; Hyaluronoglucosaminidase; Insulin; Islets of Langerhans; Leucine; Mice; Microbial Collagenase; Rats; Species Specificity; Sulfonylurea Compounds; Tolbutamide | 1976 |
Inhibition of vasopressin-stimulated prostaglandin E biosynthesis by chlorpropamide in the toad urinary bladder. Mechanism of enhancement of vasopressin-stimulated water flow.
Topics: Animals; Anura; Arginine Vasopressin; Chlorpropamide; Chromatography, Thin Layer; Cyclic AMP; Glyburide; Lipid Metabolism; Permeability; Prostaglandins E; Stimulation, Chemical; Structure-Activity Relationship; Theophylline; Tolbutamide; Urinary Bladder; Vasopressins; Water | 1977 |
Modification of diuresis in the rat by chlorpropamide, glibenclamide and tolbutamide.
Topics: Administration, Oral; Animals; Body Water; Chlorpropamide; Diabetes Mellitus; Diuresis; Glyburide; Hydrogen-Ion Concentration; Male; Potassium; Rats; Sodium; Streptozocin; Time Factors; Tolbutamide | 1975 |
Side effects of therapy in diabetes evaluated by a self-administered questionnaire.
Topics: Chlorpropamide; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Patient Acceptance of Health Care; Phenformin; Surveys and Questionnaires; Tolbutamide | 1977 |
The pharmacology of a new hypoglycaemic agent N-[4-(2-(2,3-dihydrobenzo(b)furan-7-carboxamid o)-ethyl)-benzenesulphonyl]-N'-cyclohexlurea (NOVO CS 476). III. General pharmacological studies.
Topics: Animals; Blood Pressure; Cats; Chlorpropamide; Diuresis; Dogs; Female; Glyburide; Guinea Pigs; Heart; Hypoglycemic Agents; Male; Muscle Contraction; Muscle, Smooth; Papillary Muscles; Rats; Sulfonylurea Compounds; Tolbutamide | 1977 |
[Clinico-statistical studies of the use of oral hypoglycemic agents in the therapy of diabetes: critical evaluation of their effectiveness and tolerance].
Topics: Adult; Aged; Chlorpropamide; Diabetes Mellitus; Drug Evaluation; Drug Therapy, Combination; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Phenformin; Tolbutamide | 1977 |
[Hypoglycemic sulfonylurea metabolites: clinical interest. Experiences with glibenclamide in the rat].
Topics: Animals; Biotransformation; Blood Glucose; Chlorpropamide; Glyburide; Injections, Intraperitoneal; Rats; Tolbutamide | 1977 |
Myocardial infarction in diabetics.
Topics: Administration, Oral; Adult; Aged; Chlorpropamide; Coronary Care Units; Diabetes Complications; Diabetes Mellitus; Diabetic Retinopathy; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Myocardial Infarction; Phenformin; Sex Factors; Sulfonylurea Compounds; Tolbutamide | 1975 |
In vivo cytogenetic activity of sulphonylurea drugs in man.
Topics: Adult; Chlorpropamide; Chromosome Aberrations; Chromosome Deletion; Diabetes Mellitus; Female; Glyburide; Humans; Lymphocytes; Male; Middle Aged; Pregnancy; Sulfonylurea Compounds; Tolazamide; Translocation, Genetic | 1976 |
Comparative study of glibenclamide & chlorpropamide in newly diagnosed maturity onset diabetics.
Topics: Adult; Aged; Blood Glucose; Body Weight; Chlorpropamide; Diabetes Mellitus; Drug Evaluation; Female; Follow-Up Studies; Glyburide; Humans; Male; Middle Aged; Time Factors | 1976 |
Glyburide.
Topics: Chlorpropamide; Diabetes Mellitus; Drug Evaluation; Glyburide; Humans; Hypoglycemia; Insulin; Insulin Secretion; Islets of Langerhans | 1976 |
Circular dichroism studies on the interaction of sulfonylureas with bovine and human serum albumin.
Topics: Binding Sites; Binding, Competitive; Carbutamide; Chlorpropamide; Circular Dichroism; Glipizide; Glyburide; Humans; In Vitro Techniques; Optical Rotatory Dispersion; Protein Binding; Serum Albumin; Serum Albumin, Bovine; Sulfonylurea Compounds; Tolbutamide | 1976 |
Displacement of tolbutamide, glibencalmide and chlorpropamide from serum albumin by anionic drugs.
Topics: Acetaminophen; Animals; Cattle; Chlorpropamide; Dialysis; Glyburide; Humans; Phenylbutazone; Protein Binding; Salicylates; Serum Albumin; Serum Albumin, Bovine; Sulfaphenazole; Tolbutamide; Warfarin | 1976 |
Effect of bed time intermediate acting insulin in NIDDM subjects refractory to a combination of sulphonylureas and biguanides.
Topics: Biguanides; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Combinations; Female; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Injections, Subcutaneous; Insulin, Long-Acting; Lipids; Male; Metformin; Middle Aged; Phenformin; Sulfonylurea Compounds; Time Factors | 1992 |
Hypoglycemia associated hospitalizations in a population with a high prevalence of non-insulin-dependent diabetes mellitus.
Topics: Arizona; Chlorpropamide; Diabetes Mellitus, Type 2; Glyburide; Hospitalization; Humans; Hypoglycemia; Indians, North American; Insulin; New Mexico; Prevalence; Retrospective Studies; Utah | 1991 |
Recurrent hypoglycemia secondary to drug-dispensing error.
Topics: Aged; Chlorpropamide; Drug Labeling; Glyburide; Humans; Hypoglycemia; Male; Medication Errors; Middle Aged | 1991 |
A screening test for detecting sulfonylureas in plasma.
Topics: Aged; Aged, 80 and over; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide | 1990 |
Use oral hypoglycemics with caution...
Topics: Aged; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Interactions; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Sulfonylurea Compounds | 1988 |
[Effect of long-term therapy with sulfanylurea preparations on the relation of insulin secretion and the insulin-binding capacity of its receptors].
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Evaluation; Female; Gliclazide; Glucose Tolerance Test; Glyburide; Glycosuria; Humans; Hypoglycemic Agents; Insulin; Insulin Antibodies; Insulin Secretion; Leukocytes; Male; Middle Aged; Receptor, Insulin; Sulfonylurea Compounds | 1988 |
Determination of glibenclamide, chlorpropamide and tolbutamide in plasma by high-performance liquid chromatography with ultraviolet detection.
Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Diabetes Mellitus; Dinitrofluorobenzene; Gas Chromatography-Mass Spectrometry; Glyburide; Humans; Spectrophotometry, Ultraviolet; Tolbutamide | 1985 |
Sulphonylurea therapy doubles B-cell response to glucose in type 2 diabetic patients.
Topics: Aged; Blood Glucose; C-Peptide; Chlorpropamide; Diabetes Mellitus, Type 2; Glucose; Glyburide; Humans; Hyperglycemia; Insulin; Insulin Resistance; Islets of Langerhans; Middle Aged; Sulfonylurea Compounds | 1985 |
Sulfonylurea stimulates liver fructose-2,6-bisphosphate formation in proportion to its hypoglycemic action.
Topics: Acetohexamide; Animals; Buformin; Chlorpropamide; Fructosediphosphates; Gliclazide; Gluconeogenesis; Glyburide; Glycolysis; Hexosediphosphates; In Vitro Techniques; Liver; Male; Rats; Rats, Inbred Strains; Stimulation, Chemical; Sulfamethoxazole; Sulfonylurea Compounds; Tolbutamide | 1985 |
Antidiuretic action of chlorpropamide.
Topics: Chlorpropamide; Diuresis; Female; Glyburide; Humans; Male; Tolbutamide | 1973 |
The binding of sulphonylureas to serum albumin.
Topics: Animals; Carbon Radioisotopes; Cattle; Chlorpropamide; Glyburide; Humans; Hydrogen-Ion Concentration; Protein Binding; Serum Albumin; Serum Albumin, Bovine; Sulfonylurea Compounds; Tolazamide; Tolbutamide | 1974 |
Observations of the mechanism of action of the sulfonylureas under clinical conditions.
Topics: Adult; Aged; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Fasting; Female; Glyburide; Humans; Hypoglycemia; Insulin; Male; Middle Aged; Time Factors; Tolbutamide | 1973 |
The effect of glibenclamide on non-esterified fatty acid levels in the plasma of the severely alloxan diabetic rat.
Topics: Animals; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Experimental; Fatty Acids, Nonesterified; Glyburide; Insulin; Male; Rats; Tolbutamide | 1973 |
[A comparison of intravenous tolbutamide and insulin administration during and after operation in patients with maturity-onset diabetes (author's transl)].
Topics: Administration, Oral; Age Factors; Aged; Anesthesia, General; Blood Glucose; Carbohydrates; Carbutamide; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Diet Therapy; Fructose; Glyburide; Glycosuria; Humans; Injections, Intravenous; Insulin; Ketone Bodies; Plasma Substitutes; Postoperative Care; Preoperative Care; Surgical Procedures, Operative; Tolbutamide | 1974 |
An open comparative study of the efficacy and tolerance of a new antidiabetic agent: glipizide.
Topics: Blood Glucose; Chlorpropamide; Cyclohexanes; Diabetes Mellitus; Diet, Diabetic; Female; Glyburide; Glycosuria; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Nausea; Phenformin; Pyrazines; Sulfonylurea Compounds | 1973 |
Metabolic effects of hypoglycemic sulfonylureas. IV. Interference of sulfonylureas with mitochondrial oxidative phosphorylation.
Topics: Adenosine Triphosphate; Animals; Carbutamide; Chlorpropamide; Dinitrophenols; Dose-Response Relationship, Drug; Glyburide; Hypoglycemic Agents; Male; Mitochondria, Liver; Oligomycins; Oxidative Phosphorylation; Oxygen Consumption; Rats; Succinates; Sulfonylurea Compounds | 1974 |
[Hypoglycemia caused by oral antidiabetic agents].
Topics: Adult; Aged; Chlorpropamide; Delayed-Action Preparations; Diet; Female; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Kidney Diseases; Liver Diseases; Male; Middle Aged; Phenformin; Tolazamide; Tolbutamide | 1973 |
[Chlorpropamide, thiazides and congestive heart failure].
Topics: Aged; Chlorpropamide; Diabetes Mellitus; Diuresis; Diuretics; Glyburide; Heart Failure; Humans; Hydrochlorothiazide; Insulin; Male; Pulmonary Edema | 1974 |
Interactions of sulfonylureas with plasma proteins.
Topics: Acetohexamide; Acridines; Aniline Compounds; Animals; Binding Sites; Blood Proteins; Cattle; Chlorpropamide; Cyclohexanes; Glyburide; Humans; Hypoglycemic Agents; Naphthalenesulfonates; Protein Binding; Pyrazines; Serum Albumin; Serum Albumin, Bovine; Spectrometry, Fluorescence; Sulfonylurea Compounds; Tolbutamide; Warfarin | 1974 |
Clinical assessment of glybenclamide (daonil) in diabetes mellitus.
Topics: Chlorpropamide; Diabetes Mellitus; Female; Glyburide; Humans; Male; Tolbutamide | 1973 |
Mild familial diabetes with dominant inheritance.
Topics: Acetohexamide; Adolescent; Adult; Aged; Blood Glucose; Carbohydrates; Child; Chlorpropamide; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diet Therapy; Female; Genes, Dominant; Glucose Tolerance Test; Glyburide; Glycosuria; Humans; Insulin; Insulin Secretion; Ketone Bodies; Male; Metformin; Middle Aged; Pregnancy; Pregnancy in Diabetics; Radioimmunoassay; Sulfonylurea Compounds | 1974 |
Effect of hypoglycemic sulfonylureas on hepatic fructose metabolism in the rat.
Topics: Acetoacetates; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Chlorpropamide; Fasting; Flavoproteins; Fructose; Gluconeogenesis; Glyburide; Hydrogen-Ion Concentration; Hydroxybutyrates; Hypoglycemia; Ketone Bodies; Liver; Male; Mitochondria, Liver; Oxidation-Reduction; Perfusion; Rats; Spectrometry, Fluorescence; Sulfonylurea Compounds; Time Factors; Tolbutamide | 1974 |
[The glibenclamide-phenformin combination in the therapy of diabetes mellitus].
Topics: Adult; Aged; Biguanides; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Drug Combinations; Drug Evaluation; Drug Synergism; Female; Glyburide; Humans; Insulin; Male; Middle Aged; Phenformin; Tolbutamide | 1974 |
Letter: The dangers of hypoglycaemia on oral hypoglycaemia agents.
Topics: Aged; Chlorpropamide; Glyburide; Humans; Hypoglycemia; Middle Aged | 1974 |
Zinc and insulin content in pancreatic islets of rats after administration of hypoglycemic sulfonamides.
Topics: Animals; Blood Glucose; Chlorpropamide; Glyburide; Histocytochemistry; Hypoglycemic Agents; Insulin; Islets of Langerhans; Male; Rats; Tolbutamide; Zinc | 1974 |
Lacticacidosis, ketoacidosis, and hyperalaninaemia in a phenformintreated diabetic patient.
Topics: Acetoacetates; Alanine; Amitriptyline; Bicarbonates; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Diabetic Ketoacidosis; Glucose; Glyburide; Hemiplegia; Humans; Hydrogen-Ion Concentration; Hydroxybutyrates; Insulin; Ketone Bodies; Lactates; Male; Middle Aged; Phenformin | 1974 |
Oral management of uncomplicated maturity onset diabetes.
Topics: Adult; Aged; Biguanides; Chlorpropamide; Diabetes Mellitus; Diet; Drug Combinations; Glucose Tolerance Test; Glyburide; Humans; Hypoglycemic Agents; Insulin; Middle Aged; Obesity; Sulfonylurea Compounds; Tolbutamide | 1974 |
[Hypoglycemic accidents during treatment with antidiabetic sulfamides. Apropos of 5 cases of hypoglycemic coma in aged subjects].
Topics: Aged; Blood Glucose; Carbutamide; Chlorpropamide; Diabetes Mellitus; Diabetic Coma; Diet Therapy; Female; Glucose; Glyburide; Humans; Hypoglycemic Agents; Male; Medication Errors; Sulfonylurea Compounds | 1973 |
[Glibenclamide, a new oral antidiabetic].
Topics: Administration, Oral; Adult; Aged; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Female; Glyburide; Humans; Insulin; Male; Metformin; Middle Aged; Phenformin; Sulfonylurea Compounds | 1972 |
Haemolytic anaemia associated with antibodies to tolbutamide and phenacetin.
Topics: Anemia, Hemolytic; Antibodies; Chlorpropamide; Coombs Test; Cross Reactions; Female; Glyburide; Humans; Middle Aged; Phenacetin; Tolbutamide | 1972 |
[Role of glibenclamide in the therapy of diabetes].
Topics: Adult; Chlorpropamide; Diabetes Mellitus; Evaluation Studies as Topic; Glyburide; Glycosuria; Humans; Insulin; Insulin Secretion; Sulfonylurea Compounds; Tolbutamide | 1972 |
A dose equivalence study of glybenclamide (daonil)--a new hypoglycaemic agent.
Topics: Adult; Chlorpropamide; Diabetes Mellitus; Female; Glyburide; Humans; Male; Sulfonylurea Compounds; Therapeutic Equivalency; Tolbutamide | 1972 |
[Glibenclamide and diabetes mellitus. 1. Year's clinical experience].
Topics: Administration, Oral; Adult; Aged; Chlorpropamide; Diabetes Mellitus; Female; Glyburide; Humans; Male; Middle Aged; Sulfonylurea Compounds | 1972 |
Oral therapy in diabetes.
Topics: Acetohexamide; Administration, Oral; Animals; Chlorpropamide; Diabetes Mellitus; Diet Therapy; Evaluation Studies as Topic; Glyburide; Humans; Hypoglycemic Agents; Insulin; Metformin; Obesity; Phenformin; Pyrimidines; Sulfonamides; Time Factors; Tolbutamide | 1972 |
[Reaction of diabetic carbohydrate metabolism on the change from chlorpropamide to glibenclamide].
Topics: Adult; Chlorpropamide; Diabetes Complications; Diabetes Mellitus; Female; Glyburide; Humans; Hypoglycemia; Male; Middle Aged | 1972 |
[Glibenclamide--a better antidiabetic agent?].
Topics: Aged; Blood Glucose; Body Weight; Chlorpropamide; Cholesterol; Diabetes Mellitus; Female; Glyburide; Glycosuria; Humans; Male; Middle Aged; Time Factors; Triglycerides | 1972 |
Diabetes mellitus: the thin maturity-onset diabetic.
Topics: Acetohexamide; Body Weight; Chlorpropamide; Diabetes Mellitus; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Middle Aged; Tolazamide; Tolbutamide | 1972 |
Clinical observations on the mechanism of the antidiuretic action of chlorpropamide in vasopressin-sensitive diabetes insipidus and in normal subjects.
Topics: Adolescent; Adult; Blood Glucose; Child; Child, Preschool; Chlorpropamide; Diabetes Insipidus; Drug Synergism; Ethanol; Glyburide; Humans; Hypoglycemia; Metformin; Middle Aged; Osmolar Concentration; Sodium; Thiazines; Vasopressins; Water | 1972 |
Diuretic action of three sulfonylurea drugs.
Topics: 11-Hydroxycorticosteroids; Acetohexamide; Adrenal Glands; Adult; Autoanalysis; Blood Glucose; Chlorpropamide; Creatinine; Diuresis; Evaluation Studies as Topic; Glyburide; Humans; Male; Natriuresis; Photometry; Potassium; Radioimmunoassay; Tolazamide; Vasopressins; Water | 1973 |
Study on a new antidiabetic agent, glibenclamide (HB419). A clinical evaluation and comparative study.
Topics: Adult; Aged; Chlorpropamide; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged | 1971 |
[ADH-like mechanism of action of chlorpropamide in diabetes insipidus (a comparison with the antidiuretic effect of other blood glucose decreasing sulfonamides and hydrochlorothiazide)].
Topics: Aged; Blood Glucose; Body Weight; Chlorpropamide; Depression, Chemical; Diabetes Insipidus; Diuresis; Female; Glyburide; Humans; Hydrochlorothiazide; Hypoglycemic Agents; Male; Middle Aged; Natriuresis; Osmolar Concentration; Potassium; Sulfonylurea Compounds; Tolbutamide; Vasopressins | 1970 |
[Synergism between oral diabetics and insulin].
Topics: Animals; Biguanides; Blood Glucose; Chlorpropamide; Columbidae; Drug Synergism; Glyburide; Hypoglycemia; Hypoglycemic Agents; Insulin; Tolbutamide | 1971 |
Glibenclamide is exceptional among hypoglycaemic sulphonylureas in accumulating progressively in beta-cell-rich pancreatic islets.
Topics: Animals; Carbutamide; Chlorpropamide; Glipizide; Glyburide; Islets of Langerhans; Mice; Mice, Obese; Sulfonylurea Compounds; Tolbutamide | 1984 |
Clinical pharmacology of glipizide.
Topics: Biological Availability; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Half-Life; Humans; Kinetics; Structure-Activity Relationship; Sulfonylurea Compounds; Tolbutamide | 1983 |
Lack of effect of glibenclamide, chlorpropamide and metformin on plasma cholesterol and HDL-cholesterol in non-diabetic rats.
Topics: Animals; Chlorpropamide; Cholesterol; Glyburide; Lipoproteins, HDL; Male; Metformin; Rats | 1980 |
[Behavior of lactate and pyruvate in diabetics treated with a combination of fenformin and sulfonylurea in varying doses. I].
Topics: Adult; Aged; Chlorpropamide; Diabetes Mellitus; Diabetic Ketoacidosis; Drug Combinations; Female; Glyburide; Humans; Lactates; Male; Middle Aged; Phenformin; Pyruvates; Sulfonylurea Compounds | 1980 |
Kinetics-effect relations of glipizide and other sulfonylureas.
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus; Dose-Response Relationship, Drug; Fasting; Feeding Behavior; Glipizide; Glyburide; Humans; Kidney; Sulfonylurea Compounds; Tolbutamide | 1980 |
Comparative single-dose kinetics and effects of four sulfonylureas in healthy volunteers.
Topics: Adult; Blood Glucose; Chlorpropamide; Fasting; Glipizide; Glyburide; Humans; Insulin; Kinetics; Male; Sulfonylurea Compounds; Time Factors; Tolbutamide | 1980 |
The pharmacology of sulfonylureas.
Topics: Acetohexamide; Blood Glucose; Chlorpropamide; Diabetes Mellitus; Glyburide; Humans; Insulin; Sulfonylurea Compounds; Tolazamide; Tolbutamide | 1981 |
Hormonal and metabolic effects of chlorpropamide, glibenclamide and placebo in a cross-over study in diabetics not controlled by diet alone.
Topics: Adult; Aged; Body Weight; Chlorpropamide; Diabetes Mellitus; Diet, Diabetic; Fatty Acids, Nonesterified; Female; Glucose Tolerance Test; Glyburide; Glycerol; Growth Hormone; Humans; Insulin; Ketone Bodies; Lactates; Lipids; Male; Middle Aged; Pyruvates | 1981 |
Chronic effects of glibenclamide, chlorpropamide and metformin on plasma glucose and insulin in non-diabetic rats.
Topics: Animals; Blood Glucose; Chlorpropamide; Glucose Tolerance Test; Glyburide; Insulin; Male; Metformin; Rats; Rats, Inbred Strains; Time Factors | 1981 |
Plasma high density lipoprotein cholesterol in streptozotocin diabetic and non-diabetic mice after prolonged administration of glibenclamide, chlorpropamide and metformin.
Topics: Animals; Blood Glucose; Body Weight; Chlorpropamide; Cholesterol; Cholesterol, HDL; Diabetes Mellitus, Experimental; Glyburide; Kinetics; Lipoproteins, HDL; Male; Metformin; Mice | 1981 |
Chlorpropamide and glibenclamide serum concentrations in hospitalized patients.
Topics: Aged; Body Weight; Chlorpropamide; Diabetes Mellitus; Dose-Response Relationship, Drug; Female; Glyburide; Humans; Male; Middle Aged | 1982 |
Comparative placental transport of oral hypoglycemic agents in humans: a model of human placental drug transfer.
Topics: Administration, Oral; Analysis of Variance; Antipyrine; Biological Transport; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Maternal-Fetal Exchange; Models, Biological; Molecular Weight; Placenta; Pregnancy; Regression Analysis; Tolbutamide | 1994 |
Nurse liability for dispensing meds "as ordered". Case in point: Navarro v. George 615A. 2d 890--PA (1992).
Topics: Chlorpropamide; Diabetes Mellitus; Glyburide; Humans; Male; Malpractice; Medication Errors; Nursing Staff; Pennsylvania; Prisons | 1993 |
Long-term comparative trial of glibenclamide and chlorpropamide in diet-failed, maturity-onset diabetics.
Topics: Adult; Blood Glucose; Body Weight; Chlorpropamide; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemia; Middle Aged; Treatment Failure | 1975 |
Metabolic effects of dietary sucrose and fructose in type II diabetic subjects.
Topics: Adult; Aged; Blood Glucose; Blood Proteins; Body Weight; C-Peptide; Chlorpropamide; Cholesterol; Cholesterol, HDL; Cholesterol, LDL; Diabetes Mellitus, Type 2; Dietary Carbohydrates; Dietary Sucrose; Energy Intake; Female; Fructose; Glyburide; Glycated Serum Proteins; Glycoproteins; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Postprandial Period; Triglycerides | 1996 |
Photohemolytic potency of oral antidiabetic drugs in vitro: effects of antioxidants and a nitrogen atmosphere.
Topics: Antioxidants; Ascorbic Acid; Carbutamide; Chlorpropamide; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glyburide; Hemolysis; Humans; Hypoglycemic Agents; Nitrogen; Radiation-Sensitizing Agents; Reactive Oxygen Species; Sulfonamides; Sulfonylurea Compounds; Superoxide Dismutase; Tolazamide; Tolbutamide; Ultraviolet Rays; Vitamin E | 1996 |
Rates of hypoglycemia in users of sulfonylureas.
Topics: Adult; Aged; Chlorpropamide; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Incidence; Male; Middle Aged; Poisson Distribution; Risk; Risk Factors; Sulfonylurea Compounds; Surveys and Questionnaires; Time Factors; Tolbutamide | 1997 |
Predictors of relapse in elderly diabetic patients admitted with sulphonylurea-induced severe hypoglycaemic attacks.
Topics: Aged; Aged, 80 and over; Chlorpropamide; Diabetes Mellitus, Type 2; Female; Geriatric Assessment; Glyburide; Hong Kong; Hospitalization; Humans; Hypoglycemia; Male; Middle Aged; Recurrence; Sulfonylurea Compounds | 1997 |
[Trial for transdermal administration of sulfonylureas].
Topics: Animals; Blood Glucose; Chemical Phenomena; Chemistry, Physical; Chlorpropamide; Glyburide; Hypoglycemic Agents; Male; Ointments; Rats; Rats, Wistar; Skin Absorption | 1997 |
Sulfonylureas stimulate renin secretion from the perfused kidney of the rat.
Topics: Animals; Blood Pressure; Chlorpropamide; Cyclic AMP; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Kidney; Male; Perfusion; Rats; Rats, Wistar; Renin; Stimulation, Chemical; Sulfonylurea Compounds; Tolbutamide | 1999 |
[Impact of intensive blood glucose control with hypoglycemic sulfamides, metformin or insulin on complications of non-insulin dependent diabetes].
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Metformin; Multicenter Studies as Topic; Randomized Controlled Trials as Topic; Risk Factors | 1999 |
Identification of sulfonylureas in serum by electrospray mass spectrometry.
Topics: Calibration; Chlorpropamide; Chromatography, Liquid; Glipizide; Glyburide; Humans; Mass Spectrometry; Models, Chemical; Sulfonylurea Compounds; Tolbutamide; Ultraviolet Rays | 2000 |
Sensitivity to sulphonylureas in patients with hepatocyte nuclear factor-1alpha gene mutations: evidence for pharmacogenetics in diabetes.
Topics: Adult; Amino Acid Substitution; Chlorpropamide; Diabetes Mellitus, Type 2; DNA Transposable Elements; DNA-Binding Proteins; Female; Glyburide; Hepatocyte Nuclear Factor 1; Hepatocyte Nuclear Factor 1-alpha; Hepatocyte Nuclear Factor 1-beta; Humans; Hypoglycemic Agents; Insulin; Metformin; Middle Aged; Nuclear Proteins; Point Mutation; Sulfonylurea Compounds; Transcription Factors | 2000 |
Differences in pharmacotherapy and in glucose control of type 2 diabetes patients in two neighbouring towns: a longitudinal population-based study.
Topics: Aged; Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Longitudinal Studies; Male; Retrospective Studies; Sweden; Time Factors; Urban Population | 2001 |
Coefficient of failure: a methodology for examining longitudinal beta-cell function in Type 2 diabetes.
Topics: Chlorpropamide; Diabetes Mellitus, Type 2; Female; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Islets of Langerhans; Least-Squares Analysis; Longitudinal Studies; Male; Middle Aged; Predictive Value of Tests; Regression Analysis; Time Factors; Treatment Failure; Treatment Outcome | 2002 |
Hypogycaemia without coma.
Topics: Butylscopolammonium Bromide; Chlorpropamide; Female; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Middle Aged; Prochlorperazine | 2007 |
Pharmacogenomic analysis of ATP-sensitive potassium channels coexpressing the common type 2 diabetes risk variants E23K and S1369A.
Topics: ATP-Binding Cassette Transporters; Chlorpropamide; Cyclohexanes; Diabetes Mellitus, Type 2; Gene Expression Regulation; Gliclazide; Glyburide; Haplotypes; Homozygote; Humans; Isoindoles; Nateglinide; Patch-Clamp Techniques; Phenylalanine; Polymorphism, Single Nucleotide; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Structure-Activity Relationship; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide | 2012 |
Mechanosynthesis of pharmaceutically relevant sulfonyl-(thio)ureas.
Topics: Catalysis; Chlorpropamide; Copper; Glyburide; Hypoglycemic Agents; Isothiocyanates; Molecular Structure; Sulfonamides; Tolbutamide | 2014 |
Analysis of Hypoglycemic Drugs by Liquid Chromatography-Tandem Mass Spectrometry.
Topics: Chlorpropamide; Chromatography, High Pressure Liquid; Chromatography, Liquid; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Nateglinide; Pioglitazone; Rosiglitazone; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Tolazamide; Tolbutamide | 2024 |