glyburide and carbamates

glyburide has been researched along with carbamates in 67 studies

Research

Studies (67)

TimeframeStudies, this research(%)All Research%
pre-19901 (1.49)18.7374
1990's19 (28.36)18.2507
2000's28 (41.79)29.6817
2010's18 (26.87)24.3611
2020's1 (1.49)2.80

Authors

AuthorsStudies
Camerini-Davalos, RA; Ehrenreich, TH; Oppermann, W; Reddi, AS; Strugatz, LH1
Ampudia-Blasco, FJ; Bender, R; Berger, M; Heinemann, L; Heise, T; Schmidt, A; Starke, AA1
Kruseman, AC; Menheere, PP; Müller, PG; Nijst, L; Sels, JP; Wolffenbuttel, BH1
Dissing, S; Frøkjaer-Jensen, J; Gromada, J; Kofod, H1
Brasseur, R; Lins, L; Malaisse, WJ1
Kikuchi, M1
Grell, W; Mark, M1
Fuhlendorff, J; Ladrière, L; Malaisse, WJ; Malaisse-Lagae, F2
Brand, CL; Carr, RD; Fuhlendorff, J; Kofod, H; MacKay, P; Rolin, B; Rorsman, P; Shymko, R1
Balfour, JA; Faulds, D1
Grell, W; Griss, G; Hurnaus, R; Luger, P; Mark, M; Müller, P; Nar, H; Rupprecht, E; Sauter, R; Wittneben, H1
Mooradian, AD; Thurman, JE1
Landgraf, R; Wolffenbuttel, BH1
Clauson, P; Damsbo, P; Marbury, TC; Windfeld, K1
Huang, WC; Lebovitz, H; Marbury, T; Strange, P1
Bilo, HJ; Landgraf, R; Müller, PG1
Kwan, HY; Yao, X1
Cai, Z; Lansdell, KA; Sheppard, DN1
Dunning, BE; Hu, S; Wang, S1
Riddle, M1
Bell, PA; Boettcher, BR; Dunning, BE; Fanelli, B; Geisse, S; Hu, S; Schmitz, R; Wang, S1
Landgraf, R1
Rutten, GE1
Hu, S; Wang, S1
Hu, S1
Cozma, LS; Dunseath, GJ; Langendorg, KW; Luzio, SD; Owens, DR; Pieber, T1
Mafauzy, M1
Ashcroft, SJ; Mikhailov, MV; Mikhailova, EA1
Ambrosi, F; Boemi, M; Carle, F; Filipponi, P; Gregorio, F1
Bell, CF; Botteman, MF; Braunstein, SN; Devine, ST; Ramsdell, JW; Stephens, JM1
Nicklasson, L; Stockl, K; Vanderplas, AM1
Carr, RD; Degn, KB; Gall, MA; Rizza, RA; Schmitz, O; Thomsen, MK; Veldhuis, JD; Østergård, T1
Haslbeck, M; Jakob, S; Kellerer, M; Linn, T1
Abrahamson, MJ1
Corll, C; Martin, RJ; Porter, JR; Roane, DS; Zhang, Y; Zhou, J1
Esposito, K; Giugliano, D; Marfella, R; Nappo, F1
Bae, JH; Cho, CH; Han, J; Jang, BC; Kim, SP; Kim, SS; Lee, HY; Lim, JG; Park, JW; Park, MJ; Song, DK; Suh, SI; Yun, JE1
Berney, T; Bosco, D; Carr, RD; Donath, MY; Maedler, K; Zuellig, RA1
Abbatecola, AM; Grella, R; Manzella, D; Paolisso, G1
Hjemdahl, P; Ostenson, CG; Wallén, NH; Yngen, M1
Choudhury, H; Harisudhan, T; Mullangi, R; Srinivas, NR; Venkatesh, P1
Kühner, P; Quast, U; Russ, U; Stephan, D; Winkler, M1
Fedele, V; Fioravanti, M; Leotta, C; Paolisso, G; Papa, G; Purrello, F; Rizzo, MR; Solerte, SB1
Erkent, U; Ertunc, M; Guc, MO; Ilhan, M; Iskit, AB; Onur, R1
Jin, SH; Li, ZR; Shi, YQ; Yao, J1
Bieger, S; Kühner, P; Quast, U; Stephan, D; Winkler, M; Wolff, F1
Gupta, A; Jain, S; Kumar, N; Tiwary, AK1
Meneilly, GS1
Bain, SC; Bodvarsdottir, TB; Bracken, RM; Deacon, CF; Dunseath, G; Holst, JJ; Lowe, GD; Luzio, S; Prior, SL; Rumley, A; Stephens, JW; Wareham, K1
Abdelmoneim, AS; Brocks, DR; Hasenbank, SE; Light, PE; Seubert, JM; Simpson, SH1
Bryan, J; Kühner, P; Ortiz, D; Prager, R; Quast, U; Russ, U; Stephan, D; Winkler, M1
Amato, S; Baiocco, E; Curione, M; Di Bona, S; Gatti, A; Mandosi, E; Morano, S; Rossetti, M; Salvatore, S; Tarquini, G; Turinese, I; Varrenti, M1
Andersson, C; Fosbøl, EL; Gislason, G; Køber, L; Mogensen, UM; Scheller, NM; Schramm, TK; Torp-Pedersen, C; Vaag, A1
Abdelmoneim, AS; Huang, Y; Light, P; Qiu, W; Simpson, SH1
Benoit-Biancamano, MO; Fortin, JS1
Chinwuba Okoye, T; Chukwunonso Obi, B; Nonye Igwe, C; Okpashi, VE; Olisah Alumanah, E1
Berggren, PO; Zaitsev, SV; Zaitseva, II1
Bilker, WB; Brensinger, CM; Chiang, C; Han, X; Hennessy, S; Leonard, CE; Li, L1
Areosa Sastre, A; González-Colaço Harmand, M; Martínez, G; Vernooij, RW1
Dehpour, AR; Moradi, A; Nikoui, V; Ostadhadi, S; Zolfaghari, S1
Aoyama, S; Fujino, R; Hashizume, K; Ito, K; Lee, W; Maeda, K; Ninomiya, SI; Sugiyama, Y; Toshimoto, K1
Bachmann, HS; Besser, M; Koester, V; Severing, AL; Stuermer, EK; Terberger, N1
Huang, HK; Yeh, JI1
David, LL; Innes, LM; Kandasamy, B; Martin, GM; Shyng, SL; Sung, MW; Yang, Z; Yoshioka, C1
Asaumi, R; Imawaka, H; Kusuhara, H; Lee, W; Menzel, K; Nunoya, KI; Sugiyama, Y1
Bilker, WB; Brensinger, CM; Flory, JH; Hee Nam, Y; Hennessy, S; Leonard, CE1

Reviews

9 review(s) available for glyburide and carbamates

ArticleYear
Modulation of insulin secretion in non-insulin-dependent diabetes mellitus by two novel oral hypoglycaemic agents, NN623 and A4166.
    Diabetic medicine : a journal of the British Diabetic Association, 1996, Volume: 13, Issue:9 Suppl 6

    Topics: Administration, Oral; Biological Availability; Blood Glucose; Carbamates; Cyclohexanes; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Intestinal Absorption; Molecular Structure; Nateglinide; Phenylalanine; Piperidines; Reference Values; Stereoisomerism

1996
Repaglinide.
    Drugs & aging, 1998, Volume: 13, Issue:2

    Topics: Animals; Carbamates; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemic Agents; Islets of Langerhans; Piperidines; Randomized Controlled Trials as Topic; Stereoisomerism

1998
Drug therapy of postprandial hyperglycaemia.
    Drugs, 1999, Volume: 57, Issue:1

    Topics: 1-Deoxynojirimycin; Acarbose; Amyloid; Carbamates; Diabetes Mellitus; Enzyme Inhibitors; Glucosamine; Glyburide; Humans; Hyperglycemia; Hypoglycemic Agents; Imino Pyranoses; Inositol; Insulin; Insulin Lispro; Islet Amyloid Polypeptide; Piperidines; Postprandial Period; Trisaccharides

1999
Combining sulfonylureas and other oral agents.
    The American journal of medicine, 2000, Apr-17, Volume: 108 Suppl 6a

    Topics: Acarbose; Administration, Oral; Carbamates; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Drug Therapy, Combination; Glyburide; Humans; Hypoglycemic Agents; Metformin; Piperidines; Sulfonylurea Compounds

2000
Meglitinide analogues in the treatment of type 2 diabetes mellitus.
    Drugs & aging, 2000, Volume: 17, Issue:5

    Topics: Benzamides; Carbamates; Cyclohexanes; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemic Agents; Molecular Structure; Nateglinide; Phenylalanine; Piperidines

2000
[Repaglinide, potentially a therapeutic improvement for diabetes mellitus type 2].
    Nederlands tijdschrift voor geneeskunde, 2001, Aug-11, Volume: 145, Issue:32

    Topics: Carbamates; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Insulin Secretion; Metformin; Piperidines; Therapeutic Equivalency

2001
[Continuation 50. Type 2 diabetes: possibilities and limitations of pharmacological therapy].
    MMW Fortschritte der Medizin, 2003, Dec-18, Volume: 145, Issue:51-52

    Topics: 1-Deoxynojirimycin; Acarbose; Aged; Blood Glucose; Carbamates; Contraindications; Cyclohexanes; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Enzyme Inhibitors; Fasting; Follow-Up Studies; Germany; Glucosamine; Glyburide; Glycated Hemoglobin; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemia; Hypoglycemic Agents; Imino Pyranoses; Insulin; Metformin; Middle Aged; Nateglinide; Obesity; Patient Compliance; Phenylalanine; Pioglitazone; Piperidines; Practice Guidelines as Topic; Risk Factors; Rosiglitazone; Sulfonylurea Compounds; Thiazolidinediones; Time Factors

2003
Variations in tissue selectivity amongst insulin secretagogues: a systematic review.
    Diabetes, obesity & metabolism, 2012, Volume: 14, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Cardiovascular Diseases; Cricetinae; Cyclohexanes; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Ischemic Preconditioning, Myocardial; Isoindoles; Mice; Muscle, Smooth, Vascular; Myocytes, Cardiac; Nateglinide; Phenylalanine; Piperidines; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Risk Factors; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide

2012
Effect of the treatment of Type 2 diabetes mellitus on the development of cognitive impairment and dementia.
    The Cochrane database of systematic reviews, 2017, 06-15, Volume: 6

    Topics: Carbamates; Cause of Death; Cognition Disorders; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemic Agents; Memory Disorders; Metformin; Piperidines; Randomized Controlled Trials as Topic; Rosiglitazone; Thiazolidinediones

2017

Trials

17 trial(s) available for glyburide and carbamates

ArticleYear
Comparative dose-related time-action profiles of glibenclamide and a new non-sulphonylurea drug, AG-EE 623 ZW, during euglycaemic clamp in healthy subjects.
    Diabetologia, 1994, Volume: 37, Issue:7

    Topics: Administration, Oral; Adult; Blood Glucose; Carbamates; Dose-Response Relationship, Drug; Glucose; Glucose Clamp Technique; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Male; Piperidines; Time Factors

1994
Effects of a new oral hypoglycaemic agent, repaglinide, on metabolic control in sulphonylurea-treated patients with NIDDM.
    European journal of clinical pharmacology, 1993, Volume: 45, Issue:2

    Topics: Aged; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Female; Fructosamine; Gliclazide; Glyburide; Glycated Hemoglobin; Hexosamines; Humans; Hypoglycemic Agents; Lipids; Male; Middle Aged; Piperidines; Tolbutamide

1993
Modulation of insulin secretion in non-insulin-dependent diabetes mellitus by two novel oral hypoglycaemic agents, NN623 and A4166.
    Diabetic medicine : a journal of the British Diabetic Association, 1996, Volume: 13, Issue:9 Suppl 6

    Topics: Administration, Oral; Biological Availability; Blood Glucose; Carbamates; Cyclohexanes; Diabetes Mellitus, Type 2; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Intestinal Absorption; Molecular Structure; Nateglinide; Phenylalanine; Piperidines; Reference Values; Stereoisomerism

1996
A 1-year multicenter randomized double-blind comparison of repaglinide and glyburide for the treatment of type 2 diabetes. Dutch and German Repaglinide Study Group.
    Diabetes care, 1999, Volume: 22, Issue:3

    Topics: Adult; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Double-Blind Method; Fasting; Female; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Male; Middle Aged; Piperidines

1999
A double-blind randomized comparison of meal-related glycemic control by repaglinide and glyburide in well-controlled type 2 diabetic patients.
    Diabetes care, 1999, Volume: 22, Issue:5

    Topics: Adult; Aged; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Diet, Diabetic; Double-Blind Method; Drug Administration Schedule; Eating; Energy Intake; Fasting; Glyburide; Humans; Hypoglycemic Agents; Middle Aged; Piperidines

1999
Repaglinide versus glyburide: a one-year comparison trial.
    Diabetes research and clinical practice, 1999, Volume: 43, Issue:3

    Topics: Adult; Aged; Blood Glucose; C-Peptide; Carbamates; Cholesterol; Cholesterol, HDL; Cholesterol, LDL; Diabetes Mellitus, Type 2; Double-Blind Method; Female; Fibrinogen; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Piperidines; Prospective Studies; Triglycerides; United States; United States Food and Drug Administration

1999
A comparison of repaglinide and glibenclamide in the treatment of type 2 diabetic patients previously treated with sulphonylureas.
    European journal of clinical pharmacology, 1999, Volume: 55, Issue:3

    Topics: Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Double-Blind Method; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Piperidines; Sulfonylurea Compounds

1999
Comparison of the effects of three insulinotropic drugs on plasma insulin levels after a standard meal.
    Diabetes care, 2002, Volume: 25, Issue:8

    Topics: Aged; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Double-Blind Method; Eating; Female; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Middle Aged; Piperidines

2002
Repaglinide versus glibenclamide treatment of Type 2 diabetes during Ramadan fasting.
    Diabetes research and clinical practice, 2002, Volume: 58, Issue:1

    Topics: Biomarkers; Carbamates; Diabetes Mellitus, Type 2; Fasting; Feeding Behavior; Female; Fructosamine; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Islam; Malaysia; Male; Middle Aged; Piperidines; Risk Factors; Safety; Time Factors

2002
The insulin secretagogues glibenclamide and repaglinide do not influence growth hormone secretion in humans but stimulate glucagon secretion during profound insulin deficiency.
    The Journal of clinical endocrinology and metabolism, 2004, Volume: 89, Issue:1

    Topics: Blood Glucose; C-Peptide; Carbamates; Diabetes Mellitus, Type 1; Fatty Acids, Nonesterified; Glucagon; Glucose Clamp Technique; Glyburide; Growth Hormone-Releasing Hormone; Human Growth Hormone; Humans; Hypoglycemic Agents; Insulin; Piperidines; Placebos; Potassium Channel Blockers; Somatostatin

2004
Regression of carotid atherosclerosis by control of postprandial hyperglycemia in type 2 diabetes mellitus.
    Circulation, 2004, Jul-13, Volume: 110, Issue:2

    Topics: Adult; Aged; Biomarkers; Blood Glucose; Carbamates; Carotid Artery Diseases; Cross-Sectional Studies; Diabetes Mellitus, Type 2; Fasting; Female; Glyburide; Glycated Hemoglobin; Humans; Hyperglycemia; Hypoglycemic Agents; Inflammation; Insulin; Lipids; Male; Middle Aged; Piperidines; Postprandial Period; Single-Blind Method; Tunica Intima; Tunica Media; Ultrasonography

2004
Repaglinide administration improves brachial reactivity in type 2 diabetic patients.
    Diabetes care, 2005, Volume: 28, Issue:2

    Topics: Aged; Blood Glucose; Brachial Artery; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Endothelium, Vascular; Female; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Oxidative Stress; Piperidines

2005
Meal-induced platelet activation in Type 2 diabetes mellitus: effects of treatment with repaglinide and glibenclamide.
    Diabetic medicine : a journal of the British Diabetic Association, 2006, Volume: 23, Issue:2

    Topics: Adenosine Diphosphate; Blood Glucose; C-Reactive Protein; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Eating; Fasting; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Intercellular Adhesion Molecule-1; Male; Middle Aged; P-Selectin; Piperidines; Platelet Activation; Platelet Function Tests; Postprandial Period; Treatment Outcome; von Willebrand Factor

2006
Safety of type 2 diabetes treatment with repaglinide compared with glibenclamide in elderly people: A randomized, open-label, two-period, cross-over trial.
    Diabetes care, 2006, Volume: 29, Issue:8

    Topics: Aged; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Glyburide; Humans; Piperidines

2006
Effect of repaglinide versus glyburide on postprandial glucose and insulin values in elderly patients with type 2 diabetes.
    Diabetes technology & therapeutics, 2011, Volume: 13, Issue:1

    Topics: Aged; Area Under Curve; Blood Glucose; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Piperidines; Postprandial Period

2011
Effects of short-term therapy with glibenclamide and repaglinide on incretin hormones and oxidative damage associated with postprandial hyperglycaemia in people with type 2 diabetes mellitus.
    Diabetes research and clinical practice, 2011, Volume: 94, Issue:2

    Topics: Adult; Aged; Analysis of Variance; Biomarkers; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Drug Administration Schedule; Drug Therapy, Combination; E-Selectin; F2-Isoprostanes; Female; Gastric Inhibitory Polypeptide; Glucagon-Like Peptide 1; Glyburide; Glycated Hemoglobin; Humans; Hyperglycemia; Hypoglycemic Agents; Incretins; Insulin; Intercellular Adhesion Molecule-1; Interleukin-6; Male; Metformin; Middle Aged; Oxidative Stress; Piperidines; Postprandial Period; Time Factors; Treatment Outcome; Wales

2011
Lack of the QTc physiologic decrease during cardiac stress test in patients with type 2 diabetes treated with secretagogues.
    Acta diabetologica, 2014, Volume: 51, Issue:1

    Topics: Aged; Arrhythmias, Cardiac; Carbamates; Diabetes Mellitus, Type 2; Electrocardiography; Exercise Test; Female; Glyburide; Heart Rate; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Piperidines

2014

Other Studies

42 other study(ies) available for glyburide and carbamates

ArticleYear
Diabetic glomerulosclerosis in KK mice and its prevention by glyburide and pyridinolcarbamate.
    Advances in experimental medicine and biology, 1979, Volume: 119

    Topics: Animals; Blood Glucose; Carbamates; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Glucose Tolerance Test; Glyburide; Kidney; Mice; Mice, Inbred Strains; Pyridinolcarbamate; Species Specificity

1979
Effects of the hypoglycaemic drugs repaglinide and glibenclamide on ATP-sensitive potassium-channels and cytosolic calcium levels in beta TC3 cells and rat pancreatic beta cells.
    Diabetologia, 1995, Volume: 38, Issue:9

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Calcium; Carbamates; Cell Line; Cells, Cultured; Cytosol; Dose-Response Relationship, Drug; Glyburide; Hypoglycemic Agents; Ion Channel Gating; Islets of Langerhans; Kinetics; Membrane Potentials; Mice; Patch-Clamp Techniques; Piperidines; Potassium Channels; Rats; Serum Albumin; Time Factors; Verapamil

1995
Conformational analysis of non-sulfonylurea hypoglycemic agents of the meglitinide family.
    Biochemical pharmacology, 1995, Nov-27, Volume: 50, Issue:11

    Topics: Benzamides; Carbamates; Cyclohexanes; Drug Design; Glyburide; Hypoglycemic Agents; Indoles; Isoindoles; Molecular Conformation; Nateglinide; Phenylalanine; Piperidines; Stereoisomerism; Structure-Activity Relationship; Sulfonylurea Compounds

1995
Hypoglycaemic effects of the novel antidiabetic agent repaglinide in rats and dogs.
    British journal of pharmacology, 1997, Volume: 121, Issue:8

    Topics: Animals; Carbamates; Dogs; Female; Glyburide; Hypoglycemic Agents; Piperidines; Rats; Rats, Wistar; Stereoisomerism; Sulfonylurea Compounds

1997
Repaglinide, glibenclamide and glimepiride administration to normal and hereditarily diabetic rats.
    European journal of pharmacology, 1997, Sep-24, Volume: 335, Issue:2-3

    Topics: Administration, Oral; Animals; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Fasting; Female; Glyburide; Hypoglycemic Agents; Insulin; Male; Piperidines; Rats; Rats, Wistar; Sulfonylurea Compounds

1997
Effect of antidiabetic agents on the increase in glycemia and insulinemia caused by refeeding in hereditarily diabetic rats.
    Research communications in molecular pathology and pharmacology, 1997, Volume: 97, Issue:1

    Topics: Animals; Blood Glucose; Carbamates; Diabetes Mellitus, Experimental; Food; Glyburide; Hypoglycemic Agents; Insulin; Male; Piperidines; Rats; Starvation

1997
Stimulation of insulin release by repaglinide and glibenclamide involves both common and distinct processes.
    Diabetes, 1998, Volume: 47, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Blood Glucose; Carbamates; Cohort Studies; Culture Techniques; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Evoked Potentials; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred Strains; Osmolar Concentration; Patch-Clamp Techniques; Perfusion; Piperidines; Rats; Rats, Sprague-Dawley; Time Factors; Tritium

1998
Repaglinide and related hypoglycemic benzoic acid derivatives.
    Journal of medicinal chemistry, 1998, Dec-17, Volume: 41, Issue:26

    Topics: Administration, Oral; Animals; ATP-Binding Cassette Transporters; Benzoates; Blood Glucose; Carbamates; Crystallography, X-Ray; Female; Glyburide; Hypoglycemic Agents; Models, Molecular; Molecular Conformation; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship; Sulfonylurea Compounds; Sulfonylurea Receptors

1998
Activity of voltage-gated K+ channels is associated with cell proliferation and Ca2+ influx in carcinoma cells of colon cancer.
    Life sciences, 1999, Volume: 65, Issue:1

    Topics: 4-Aminopyridine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Carbamates; Cell Division; Charybdotoxin; Colonic Neoplasms; Glyburide; Humans; Ion Channel Gating; Nickel; Peptides; Phenylcarbamates; Potassium; Potassium Channel Blockers; Potassium Channels; Quaternary Ammonium Compounds; RNA, Messenger; Tetraethylammonium; Tumor Cells, Cultured

1999
Inhibition of heterologously expressed cystic fibrosis transmembrane conductance regulator Cl- channels by non-sulphonylurea hypoglycaemic agents.
    British journal of pharmacology, 1999, Volume: 128, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzamides; Carbamates; Cell Line; Chloride Channels; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Electric Conductivity; Epithelial Cells; Glyburide; Humans; Hypoglycemic Agents; Indoles; Ion Channel Gating; Isoindoles; Kinetics; Mice; Patch-Clamp Techniques; Piperidines; Sulfonylurea Compounds; Transfection

1999
Tissue selectivity of antidiabetic agent nateglinide: study on cardiovascular and beta-cell K(ATP) channels.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:3

    Topics: Animals; Aorta, Thoracic; Carbamates; Cardiovascular System; Coronary Vessels; Cyclohexanes; Glyburide; Heart; Hypoglycemic Agents; Islets of Langerhans; Male; Muscle, Smooth, Vascular; Nateglinide; Phenylalanine; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Swine

1999
Pancreatic beta-cell K(ATP) channel activity and membrane-binding studies with nateglinide: A comparison with sulfonylureas and repaglinide.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Binding, Competitive; Carbamates; Cell Membrane; Cell Separation; Cells, Cultured; Cyclohexanes; Glucose; Glyburide; Glycosyltransferases; Humans; Hypoglycemia; Hypoglycemic Agents; In Vitro Techniques; Insulin; Islets of Langerhans; KATP Channels; Kinetics; Male; Membrane Proteins; Nateglinide; Patch-Clamp Techniques; Phenylalanine; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Repressor Proteins; Saccharomyces cerevisiae Proteins; Sulfonylurea Compounds

2000
Effect of insulinotropic agent nateglinide on Kv and Ca(2+) channels in pancreatic beta-cell.
    European journal of pharmacology, 2001, Sep-14, Volume: 427, Issue:2

    Topics: Animals; Calcium Channels; Carbamates; Cyclohexanes; Dose-Response Relationship, Drug; Electric Stimulation; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Membrane Potentials; Nateglinide; Patch-Clamp Techniques; Phenylalanine; Piperidines; Potassium Channels; Rats; Rats, Sprague-Dawley

2001
Interaction of nateglinide with K(ATP) channel in beta-cells underlies its unique insulinotropic action.
    European journal of pharmacology, 2002, May-03, Volume: 442, Issue:1-2

    Topics: Adenosine Triphosphate; Animals; Carbamates; Cyclohexanes; Dose-Response Relationship, Drug; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Membrane Potentials; Nateglinide; Phenylalanine; Piperidines; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Sulfonylurea Compounds; Time Factors

2002
A novel simple method for the investigation of drug binding to the K(ATP) channel sulfonylurea receptor.
    Analytical biochemistry, 2002, Aug-15, Volume: 307, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Gliclazide; Glyburide; Hypoglycemic Agents; Kinetics; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Rats; Receptors, Drug; Spodoptera; Sulfonylurea Receptors; Tolbutamide

2002
Effects of S 21403 on hormone secretion from isolated rat pancreas at different glucose concentrations.
    European journal of pharmacology, 2002, Dec-05, Volume: 456, Issue:1-3

    Topics: Animals; Carbamates; Dose-Response Relationship, Drug; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Indoles; Insulin; Insulin Secretion; Isoindoles; Male; Pancreas; Piperidines; Rats; Rats, Sprague-Dawley; Time Factors

2002
Economic model of first-line drug strategies to achieve recommended glycaemic control in newly diagnosed type 2 diabetes mellitus.
    PharmacoEconomics, 2003, Volume: 21, Issue:11

    Topics: Carbamates; Cohort Studies; Decision Trees; Diabetes Mellitus, Type 2; Direct Service Costs; Drug Costs; Drug Therapy, Combination; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Managed Care Programs; Markov Chains; Metformin; Models, Economic; Piperidines; Rosiglitazone; Thiazoles; Thiazolidinediones; United States

2003
A comparison of costs for four oral antidiabetic regimens within a managed care population.
    Managed care interface, 2003, Volume: 16, Issue:7

    Topics: Administration, Oral; Adolescent; Adult; Aged; California; Carbamates; Cohort Studies; Data Interpretation, Statistical; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glyburide; Health Care Costs; Humans; Hypoglycemic Agents; Insulin; Insurance Claim Review; Male; Managed Care Programs; Metformin; Middle Aged; Piperidines; Retrospective Studies

2003
Optimal glycemic control in type 2 diabetes mellitus: fasting and postprandial glucose in context.
    Archives of internal medicine, 2004, Mar-08, Volume: 164, Issue:5

    Topics: Antihypertensive Agents; Blood Glucose; Blood Glucose Self-Monitoring; Carbamates; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Disease Progression; Drug Therapy, Combination; Glyburide; Glycated Hemoglobin; Glycoside Hydrolase Inhibitors; Humans; Hyperglycemia; Hypoglycemic Agents; Metformin; Piperidines; Postprandial Period

2004
Evidence for hypothalamic K+(ATP) channels in the modulation of glucose homeostasis.
    European journal of pharmacology, 2004, May-10, Volume: 492, Issue:1

    Topics: Animals; Blood Glucose; Carbamates; Chromatography, High Pressure Liquid; Epinephrine; Glucagon; Glyburide; Homeostasis; Hypoglycemic Agents; Hypothalamus; Male; Norepinephrine; Piperidines; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley

2004
Taurine block of cloned ATP-sensitive K+ channels with different sulfonylurea receptor subunits expressed in Xenopus laevis oocytes.
    Biochemical pharmacology, 2004, Sep-01, Volume: 68, Issue:5

    Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Drug Interactions; Female; Gene Expression; Gliclazide; Glyburide; Hypoglycemic Agents; Membrane Proteins; Mice; Oocytes; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Subunits; Rats; Receptors, Drug; Sulfonylurea Receptors; Taurine; Tolbutamide; Xenopus laevis

2004
Sulfonylurea induced beta-cell apoptosis in cultured human islets.
    The Journal of clinical endocrinology and metabolism, 2005, Volume: 90, Issue:1

    Topics: Adult; Aged; Apoptosis; Calcium; Carbamates; Cells, Cultured; Cyclohexanes; Dose-Response Relationship, Drug; Glyburide; Humans; Hypoglycemic Agents; Insulin; Islets of Langerhans; Middle Aged; Nateglinide; Phenylalanine; Piperidines

2005
Simultaneous estimation of six anti-diabetic drugs--glibenclamide, gliclazide, glipizide, pioglitazone, repaglinide and rosiglitazone: development of a novel HPLC method for use in the analysis of pharmaceutical formulations and its application to human p
    Biomedical chromatography : BMC, 2006, Volume: 20, Issue:10

    Topics: Carbamates; Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Molecular Structure; Pioglitazone; Piperidines; Reproducibility of Results; Rosiglitazone; Thiazolidinediones

2006
Selectivity of repaglinide and glibenclamide for the pancreatic over the cardiovascular K(ATP) channels.
    Diabetologia, 2006, Volume: 49, Issue:9

    Topics: Adenosine Triphosphate; ATP-Binding Cassette Transporters; Binding, Competitive; Carbamates; Cardiovascular System; Cell Line; Dose-Response Relationship, Drug; Glyburide; Humans; Hypoglycemic Agents; Membrane Potentials; Molecular Structure; Pancreas; Patch-Clamp Techniques; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors

2006
Glibenclamide attenuates the antiarrhythmic effect of endotoxin with a mechanism not involving K(ATP) channels.
    Vascular pharmacology, 2007, Volume: 46, Issue:2

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Arrhythmias, Cardiac; Blood Pressure; Carbamates; Cyclohexanes; Disease Models, Animal; Drug Interactions; Endotoxemia; Glyburide; Heart Atria; Heart Conduction System; Lipopolysaccharides; Male; Myocardial Ischemia; Nateglinide; Phenylalanine; Piperidines; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Tachycardia, Ventricular; Tetraethylammonium; Time Factors; Ventricular Fibrillation; Ventricular Premature Complexes

2007
Development of a RP-HPLC method for screening potentially counterfeit anti-diabetic drugs.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2007, Jun-15, Volume: 853, Issue:1-2

    Topics: Carbamates; Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Molecular Structure; Piperidines; Reproducibility of Results; Sulfonylurea Compounds

2007
Testing the bipartite model of the sulfonylurea receptor binding site: binding of A-, B-, and A + B-site ligands.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:2

    Topics: Amino Acid Substitution; Animals; ATP-Binding Cassette Transporters; Binding Sites; Binding, Competitive; Carbamates; Cell Line; Cyclohexanes; Dose-Response Relationship, Drug; Glyburide; Hypoglycemic Agents; KATP Channels; Ligands; Mice; Molecular Structure; Nateglinide; Phenylalanine; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Radioligand Assay; Rats; Receptors, Drug; Sulfonylurea Compounds; Sulfonylurea Receptors; Transfection

2007
Spermicidal activity of sulfonylureas and meglitinide analogues: role of intrasperm Ca2+ elevation.
    The Journal of pharmacy and pharmacology, 2008, Volume: 60, Issue:3

    Topics: Adult; Benzamides; Calcium; Carbamates; Cross-Over Studies; Dose-Response Relationship, Drug; Gliclazide; Glyburide; Homeostasis; Humans; Hypoglycemic Agents; KATP Channels; Male; Piperidines; Sperm Motility; Spermatocidal Agents; Spermatozoa; Sulfonylurea Compounds; Time Factors

2008
Importance of the Kir6.2 N-terminus for the interaction of glibenclamide and repaglinide with the pancreatic K(ATP) channel.
    Naunyn-Schmiedeberg's archives of pharmacology, 2012, Volume: 385, Issue:3

    Topics: Animals; ATP-Binding Cassette Transporters; Binding Sites; Carbamates; Glyburide; HEK293 Cells; Humans; Hypoglycemic Agents; Pancreas; Patch-Clamp Techniques; Piperidines; Potassium Channels, Inwardly Rectifying; Protein Binding; Rats; Receptors, Drug; Sulfonylurea Receptors

2012
Metformin in combination with various insulin secretagogues in type 2 diabetes and associated risk of cardiovascular morbidity and mortality--a retrospective nationwide study.
    Diabetes research and clinical practice, 2015, Volume: 107, Issue:1

    Topics: Aged; Carbamates; Cardiovascular Diseases; Denmark; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Morbidity; Myocardial Infarction; Piperidines; Registries; Retrospective Studies; Risk Factors; Stroke; Sulfonylurea Compounds; Tolbutamide

2015
Comparative cardiovascular safety of insulin secretagogues following hospitalization for ischemic heart disease among type 2 diabetes patients: a cohort study.
    Journal of diabetes and its complications, 2015, Volume: 29, Issue:2

    Topics: Aged; Aged, 80 and over; Alberta; Blue Cross Blue Shield Insurance Plans; Carbamates; Cardiovascular Diseases; Cohort Studies; Databases, Factual; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Diabetic Cardiomyopathies; Female; Gliclazide; Glyburide; Hospitalization; Humans; Hypoglycemic Agents; Male; Myocardial Ischemia; Piperidines; Proportional Hazards Models; Retrospective Studies; Risk; Universal Health Insurance

2015
In vitro evaluation of hypoglycemic agents to target human islet amyloid polypeptide: a key protein involved in amyloid deposition and beta-cell loss.
    Canadian journal of diabetes, 2015, Volume: 39, Issue:5

    Topics: Amyloid; Amyloidosis; Animals; Carbamates; Cell Survival; Chromans; Circular Dichroism; Glyburide; Humans; Hypoglycemic Agents; Insulin-Secreting Cells; Islet Amyloid Polypeptide; Piperidines; Protein Structure, Secondary; Rats; Thiazolidinediones; Troglitazone

2015
Comparative Study of the Antioxidant Effects of Metformin, Glibenclamide, and Repaglinide in Alloxan-Induced Diabetic Rats.
    Journal of diabetes research, 2016, Volume: 2016

    Topics: Alloxan; Animals; Antioxidants; Biomarkers; Blood Glucose; Carbamates; Catalase; Diabetes Complications; Diabetes Mellitus, Experimental; Glutathione; Glyburide; Hypoglycemic Agents; Lipid Peroxidation; Male; Malondialdehyde; Metformin; Oxidative Stress; Piperidines; Rats; Superoxide Dismutase

2016
Insulinotropic compounds decrease endothelial cell survival.
    Toxicology in vitro : an international journal published in association with BIBRA, 2016, Volume: 33

    Topics: Benzofurans; Carbamates; Cell Proliferation; Cell Survival; Cells, Cultured; Dimethyl Sulfoxide; Glucose; Glyburide; Human Umbilical Vein Endothelial Cells; Humans; Hypoglycemic Agents; Imidazoles; Indoles; Nitric Oxide; Piperidines; Vascular Endothelial Growth Factor A

2016
Biomedical Informatics Approaches to Identifying Drug-Drug Interactions: Application to Insulin Secretagogues.
    Epidemiology (Cambridge, Mass.), 2017, Volume: 28, Issue:3

    Topics: Area Under Curve; Carbamates; Cyclohexanes; Databases, Factual; Diabetes Mellitus, Type 2; Drug Interactions; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Medical Informatics; Nateglinide; Pharmacoepidemiology; Phenylalanine; Piperidines; Sulfonylurea Compounds

2017
Cromakalim, a Potassium Channel Opener, Ameliorates the Organophosphate and Carbamate-Induced Seizure in Mice.
    Acta medica Iranica, 2018, Volume: 56, Issue:1

    Topics: Animals; Anticonvulsants; Carbamates; Cromakalim; Dichlorvos; Dose-Response Relationship, Drug; Glyburide; Male; Mice; Organophosphate Poisoning; Physostigmine; Potassium Channels; Seizures

2018
Strategies to improve the prediction accuracy of hepatic intrinsic clearance of three antidiabetic drugs: Application of the extended clearance concept and consideration of the effect of albumin on CYP2C metabolism and OATP1B-mediated hepatic uptake.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2018, Dec-01, Volume: 125

    Topics: Albumins; Carbamates; Cytochrome P-450 Enzyme System; Glyburide; HEK293 Cells; Hepatocytes; Humans; Hypoglycemic Agents; Liver; Liver-Specific Organic Anion Transporter 1; Metabolic Clearance Rate; Microsomes, Liver; Models, Biological; Nateglinide; Piperidines; Solute Carrier Organic Anion Transporter Family Member 1B3

2018
Side effects of frequently used oral antidiabetics on wound healing in vitro.
    Naunyn-Schmiedeberg's archives of pharmacology, 2019, Volume: 392, Issue:3

    Topics: Administration, Oral; Apoptosis; Carbamates; Caspases; Cell Line; Endopeptidases; Fibroblasts; Gelatinases; Glyburide; Humans; Hypoglycemic Agents; Keratinocytes; Membrane Proteins; Metformin; Piperidines; Receptors, CXCR4; Serine Endopeptidases; Sitagliptin Phosphate; Wound Healing

2019
Comparison of mortality and cardiovascular event risk associated with various insulin secretagogues: A nationwide real-world analysis.
    Diabetes research and clinical practice, 2019, Volume: 152

    Topics: Aged; Carbamates; Cardiovascular Diseases; Cohort Studies; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Follow-Up Studies; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Male; Middle Aged; Mortality; Piperidines; Secretagogues; Sulfonylurea Compounds; Taiwan

2019
Mechanism of pharmacochaperoning in a mammalian K
    eLife, 2019, 07-25, Volume: 8

    Topics: Animals; Binding Sites; Carbamates; Cell Line; Cricetinae; Cryoelectron Microscopy; Cysteine; Glyburide; Humans; KATP Channels; Mammals; Models, Molecular; Mutation; Pharmaceutical Preparations; Piperidines; Potassium Channels, Inwardly Rectifying; Protein Binding; Rats

2019
Expanded Physiologically-Based Pharmacokinetic Model of Rifampicin for Predicting Interactions With Drugs and an Endogenous Biomarker via Complex Mechanisms Including Organic Anion Transporting Polypeptide 1B Induction.
    CPT: pharmacometrics & systems pharmacology, 2019, Volume: 8, Issue:11

    Topics: Biomarkers; Carbamates; Computer Simulation; Coproporphyrins; Drug Interactions; Glyburide; Humans; Models, Biological; Organic Anion Transporters; Piperidines; Rifampin

2019
Angiotensin-Converting Enzyme Inhibitors Used Concomitantly with Insulin Secretagogues and the Risk of Serious Hypoglycemia.
    Clinical pharmacology and therapeutics, 2022, Volume: 111, Issue:1

    Topics: Administrative Claims, Healthcare; Aged; Aged, 80 and over; Angiotensin-Converting Enzyme Inhibitors; Carbamates; Databases, Factual; Diabetes Mellitus, Type 2; Drug Interactions; Female; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Medicaid; Metformin; Middle Aged; Nateglinide; Pharmacoepidemiology; Piperidines; Secretagogues; Sulfonylurea Compounds; United States

2022