glyburide has been researched along with 4-aminopyridine in 150 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (1.33) | 18.7374 |
1990's | 59 (39.33) | 18.2507 |
2000's | 58 (38.67) | 29.6817 |
2010's | 28 (18.67) | 24.3611 |
2020's | 3 (2.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Sen, S; Sinha, N | 1 |
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Honda, H; Ishida, Y; Watanabe, TX | 1 |
Gwilt, M; Henderson, CG; Orme, J; Rourke, JD | 2 |
Kamijo, T; Kido, H; Miwa, A; Nakamura, F; Sugimoto, T; Tomaru, T; Uchida, Y | 1 |
Peers, C; Reeve, HL; Vaughan, PF | 1 |
Lazdunski, M; Schaeffer, P | 1 |
Bose, D; Elliott, DA; Gu, M; Ong, BY | 1 |
Castle, NA; Haylett, DG | 1 |
Baskin, EP; Garcia, ML; Heaney, LA; Kaczorowski, GJ; Stein, RB; Wallace, AA; Winquist, RJ | 1 |
Lang, RJ; Zhang, Y | 1 |
Kleppisch, T; Nelson, MT | 1 |
Kanwal, S; Trachte, GJ | 1 |
Antonenko, YN; Kinnally, KW; Smith, D; Tedeschi, H | 1 |
Broadley, KJ; Ford, WR; Urquhart, RA | 1 |
Ginkawa, M; Kontani, H; Sakai, T | 1 |
Devor, DC; Frizzell, RA | 1 |
Brayden, JE; McCarron, JG; Nelson, MT; Quayle, JM | 1 |
Osmanović, SS; Pan, WJ; Shefner, SA | 1 |
Peterson, VA; Strobl, JS; Wonderlin, WF; Woodfork, KA | 1 |
Cahill, AL; Perlman, RL | 1 |
Bagetta, G; Constanti, A; Libri, V | 1 |
Ebisu, H; Eda, M; Fukaya, C; Gohda, M; Hihara, M; Matzno, S; Nakamura, N; Okada, T; Sakashita, H; Takemoto, T | 1 |
Daniel, EE; Inazu, M; Zhang, H | 1 |
Aaronson, PI; Robertson, TP; Smirnov, SV; Ward, JP | 1 |
Chai, S; Kolias, TJ; Webb, RC | 1 |
Beech, DJ; Sadraei, H | 1 |
Chavkin, C; Simmons, ML | 1 |
Foster, RW; Isaac, L; McArdle, S; Miller, NM; Small, RC | 1 |
O'Rourke, ST | 1 |
Evans, AM; Gurney, AM; Osipenko, ON | 1 |
Bishop, BE; Doggrell, SA | 1 |
Katusic, ZS; Kinoshita, H | 1 |
Barber, RD; Henderson, RM; Woolf, AS | 1 |
García-Segoviano, JA; Naranjo-Rodríguez, EB; Prieto-Gómez, B; Reyes-Vázquez, C; Trujillo-Santana, JT | 1 |
Satake, N; Shibata, M; Shibata, S | 1 |
Horimoto, N; Nabekura, J; Ogawa, T | 1 |
Jánossy, A; Jurányi, Z; Orsó, E; Sperlágh, B; Szalay, KS; Vinson, GP; Vizi, ES; Windisch, K | 1 |
Bozkurt, AK; Kaynar, M; Süzer, O | 1 |
Katusic, ZS; Onoue, H | 2 |
Alper, SL; Brugnara, C; Morgan, KG; Parker, C; Rittenhouse, AR | 1 |
Buus, C; Mulvany, MJ; Nilsson, H; Prieto, D | 1 |
Ito, T; Mokuno, S; Murase, K; Okumura, K; Shinoda, M; Toki, Y | 1 |
Hiley, CR; White, R | 1 |
Bojić, M; Djukanović, B; Gojkoviíc Bukarica, L; Kazić, T; Panić, G; Perić, M; Sajić, Z | 1 |
Campos, Y; Fernandez, M; Mendoza-León, A; Moll, H; Ponte-Sucre, A | 1 |
Paul, RJ; Shimizu, S | 1 |
Li, L; Paakkari, I; Vaali, K; Vapaatalo, H | 1 |
Beech, DJ; Prior, HM; Yates, MS | 2 |
Barman, SA | 1 |
Berger, MG; Bonnet, P; Jackson, WF; Rusch, NJ; Vandier, C | 1 |
Chen, CF; Chen, J; Chiou, WF | 1 |
Puil, E; Ries, CR | 1 |
Faraci, FM; Sobey, CG | 1 |
Bryan, RM; Johnson, TD; Marrelli, SP; Mombouli, JV; You, J | 1 |
Kecskeméti, V; Losonczy, G; Mucha, I; Nánási, PP; Pacher, P; Ungvári, Z | 1 |
Broadley, KJ; Ford, WR | 1 |
Kwan, HY; Yao, X | 1 |
Caligiuri, G; Hansson, GK; Jiang, J; Pernow, J; Thorén, P | 1 |
Honda, H; Kogo, H; Unemoto, T | 1 |
Gordon, JB; Halla, TR; Madden, JA | 1 |
Hata, F; Nishio, H; Nishiwaki, H; Saitoh, N; Takeuch, T | 1 |
Damron, DS; Doi, S; Horibe, M; Murray, PA; Ogawa, K; Tanaka, S | 1 |
Kubota, I; Miyashita, T; Tomoike, H; Watanabe, T; Yamaki, M; Yamauchi, S | 1 |
Cole, WC; Dong, H; Jiang, Y; Triggle, CR | 1 |
Archer, S; Bateson, J; Michelakis, E; Olley, P; Puttagunta, L; Rebeyka, I | 1 |
Davies, PJ; Martínez-Pinna, J; McLachlan, EM | 1 |
Huddart, H; Leathard, HL; Mukerji, MS | 1 |
Aguan, K; Pinkas, G; Thompson, LP; Weiner, CP | 1 |
Miller, DV; Paterson, WG; Zhang, Y | 1 |
Dacey, RG; Dietrich, HH; Horiuchi, T; Tsugane, S | 1 |
El Haj, AJ; Gu, Y; Howl, JD; Preston, MR; Publicover, SJ | 1 |
Balogh, I; Kecskeméti, V | 1 |
Bardou, M; Dumas, J; Dumas, M; Goirand, F; Rochette, L | 1 |
Gosche, JR | 1 |
Archer, SL; Hashimoto, K; Knaus, HG; Michelakis, ED; Nsair, A; Puttagunta, L; Waite, R; Weir, EK; Wu, X | 1 |
Corriu, C; Côrtes, SF; Lemos, VS; Lopes, MJ; Medeiros, IA; Rezende, BA; Teixeira, MM | 1 |
Duarte, ID; Soares, AC | 1 |
Boachie-Ansah, G; Grainger, J | 1 |
Hempelmann, RG; Kruse, ML; Mehdorn, HM; Seebeck, J; Ziegler, A | 1 |
Imai, T; Koike, K; Okamoto, T; Shigenobu, K; Tanaka, H; Tanaka, Y; Yamamoto, Y | 1 |
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI; Rosas, R; Vidal-Cantú, GC | 1 |
Bisaccia, F; Gasbarro, AR; Lograno, MD; Ostuni, A; Tamburro, AM | 1 |
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI; Rosas, R; Torres-López, JE; Vidal-Cantú, GC | 1 |
Clapp, LH; Wilson, AJ | 1 |
Argüelles, CF; Granados-Soto, V; Ortiz, MI | 1 |
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI | 2 |
El-Mahmoudy, A; Matsuyama, H; Shimizu, Y; Takewaki, T; Thapaliya, S | 1 |
Hirosawa, J; Ishibe, Y; Liu, R; Okazaki, N; Ueda, M | 1 |
Burleigh, DE | 1 |
Liu, XS; Ni, W; Xu, YJ; Zhang, ZX | 1 |
Höhn, J; Krassói, I; Kun, A; Papp, JG; Pataricza, J | 1 |
Kang, D; Kim, D; Mariash, E | 1 |
Alves, DP; Amarante, LH; Duarte, ID | 1 |
Chang, IY; Choi, S; Jun, JY; Kim, KW; Kim, MJ; Kim, MY; Kong, ID; Lee, KP; Park, CK; So, I; Yeum, CH; You, HJ | 1 |
Dubrovska, G; Essin, K; Gollasch, M; Huang, Y; Luft, FC; Tsang, SY; Verlohren, S | 1 |
Anapolski, M; Barfield, JP; Cooper, TG; Yeung, CH | 1 |
Austin, C; Bruce, J; Taggart, M | 1 |
Chen, SX; Ni, W; Xu, YJ; Zhang, ZX; Zhao, LM | 1 |
Bisseling, TM; Borggreven, JM; Copius Peereboom-Stegeman, JJ; Russel, FG; Smits, P; Steegers, EA; van der Laak, JA; van der Wal, S; Versteegen, MG | 1 |
Fujimoto, S; Kunimatsu, M; Mori, M; Tsushima, H | 1 |
Castañeda-Hernández, G; Castro-Olguín, J; Ortiz, MI; Peña-Samaniego, N | 1 |
Granados-Soto, V; Medina-Tato, DA; Ortiz, MI; Palma-Martínez, J; Sarmiento-Heredia, D | 1 |
Djukanovic, B; Gojkovic-Bukarica, L; Heinle, H; Markovic-Lipkovski, J; Nezic, D; Novakovic, A; Peric, M | 1 |
Chu, V; Janssen, LJ; Tazzeo, T; Zhang, Y | 1 |
Bukarica, LG; Heinle, H; Kanjuh, V; Novakovic, A | 1 |
Seyrek, M; Ulusoy, HB; Yildirim, V; Yildiz, O | 1 |
Exintaris, B; Lang, RJ; Nguyen, DT | 1 |
Baggio, CH; Cipriani, TR; da Silva-Santos, JE; de Souza, LM; Freitas, CS; Graça, C; Marques, MC; Pontarolo, R; Rattmann, YD; Rieck, L; Sassaki, GL | 1 |
Bagcivan, I; Gursoy, S; Kaya Temiz, T; Turan, M; Yildirim, MK; Yildirim, S; Yilmaz, A | 1 |
Chen, G; Han, X; Iadecola, C; Ma, D; Meng, L; Song, X; Wang, F; Wang, G; Wang, S; Weng, D; Xi, L; Xing, H; Xu, G; Yao, W; Zhou, J; Zhu, T | 1 |
Akar, F; Katircioglu, SF; Manavbasi, Y; Parlar, AI; Ulus, AT | 1 |
Li, J; Liang, Y; Niu, L; Wu, D; Xue, W; Zhang, M | 1 |
Basak, F; Cehreli, SB; Cehreli, ZC; Guven, G; Kaya, E; Seyrek, M; Ulku, C; Vural, IM; Yildiz, O | 1 |
Chen, J; Chen, X; Liu, J; Wang, T; Xiao, H; Yang, J; Ye, Z; Yin, C | 1 |
Achike, FI; Mustafa, MR; Subramaniam, G | 1 |
Bayram, Z; Golbasi, I; Ozdem, SS | 1 |
Choudhury, S; Garg, SK; Mishra, SK; Singh, TU | 1 |
Assreuy, J; Fernandes, D; Sordi, R | 1 |
Achike, FI; Tan, BT; Yeo, JL | 1 |
Berwick, ZC; Dick, GM; Lynch, B; Payne, GA; Sturek, M; Tune, JD | 1 |
Cehreli, ZC; Guven, G; Seyrek, M; Vural, IM; Yildiz, O | 1 |
Hahm, KD; Jeong, SM; Kim, YK; Lee, C; Leem, JG; Park, PH; Shin, JW; Song, JG | 1 |
Kleikers, P; van der Sterren, S; Villamor, E; Zimmermann, LJ | 1 |
Chang, HH; Chen, MF; Chen, PY; Chiang, CL; Kuo, JS; Lee, TJ; Lee, YC; Liu, CH; Yeh, JI | 1 |
Arcanjo, DD; Cavalcanti, SC; Oliveira, AP; Oliveira, NN; Oliveira, Rde C; Quintans-Júnior, LJ; Santos, MR; Silva-Filho, JC | 1 |
He, GW; Jovic, M; Kanjuh, V; Milojevic, P; Nenezic, D; Novakovic, A; Pavlovic, M; Stojanovic, I; Ugresic, N; Yang, Q | 1 |
Khaertdinov, NN; Sitdikova, GF; Zefirov, AL | 1 |
Cruickshank, SF; Dospinescu, C; Rowe, I; Wainwright, C; Widmer, H | 1 |
Deja, MA; Golba, KS; Janusiewicz, P; Malinowski, M; Roleder, T; Wos, S | 1 |
Li, CY; Pi, MS; Ru, Q; Tian, X; Wu, RH; Wu, YX | 1 |
Beleslin-Cokic, B; Gojkovic-Bukarica, L; Heinle, H; Ilic, B; Novakovic, R; Radunovic, N; Scepanovic, R | 1 |
Bayram, Z; Nacitarhan, C; Ozdem, SS | 1 |
Medeiros, MA; Quintans, JS; Quintans-Júnior, LJ; Ribeiro, FP; Ribeiro, LA; Sampaio, PA; Silva, MT; Silva, YM | 1 |
Liu, Y; Lu, P; Wang, D; Zhu, D; Zhu, Y | 1 |
Cavalcante, Fde A; Correia, AC; da Silva, BA; de Souza, IL; Paredes-Gamero, EJ; Santos, BV; Silva, Mda C; Vasconcelos, LH | 1 |
Garg, SK; Hajare, SW; Nakade, UP; Saroj, VK; Sharma, A; Yadav, RS | 1 |
Baldelli, P; Benfenati, F; Cappetti, B; Forte, N; Medrihan, L | 1 |
Khin, PP; Sohn, UD; Zaw, TS | 1 |
Amano, T; Fujii, N; Kenny, GP; Louie, JC; McNeely, BD; Nishiyasu, T | 1 |
Fujii, N; Ichinose, M; Kenny, GP; McGarr, GW; Nishiyasu, T | 1 |
Altun, A; Bagcivan, I; Cakmak, E; Kahramanoglu, YE; Kurt, A; Pence, HH; Sarac, B; Soylu, S | 1 |
Al Hennawi, K; Erdem Kış, E; Tiftik, RN; Ün, İ | 1 |
Sahinturk, S | 1 |
1 trial(s) available for glyburide and 4-aminopyridine
Article | Year |
---|---|
Tetraethylammonium, glibenclamide, and 4-aminopyridine modulate post-occlusive reactive hyperemia in non-glabrous human skin with no roles of NOS and COX.
Topics: 4-Aminopyridine; Adult; Glyburide; Humans; Hyperemia; Male; Nitric Oxide Synthase; Prostaglandin-Endoperoxide Synthases; Skin; Tetraethylammonium | 2020 |
149 other study(ies) available for glyburide and 4-aminopyridine
Article | Year |
---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship | 2011 |
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain | 2016 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
Ca2+ release from isolated sarcoplasmic reticulum of guinea-pig psoas muscle induced by K(+)-channel blockers.
Topics: 4-Aminopyridine; Animals; Apamin; Calcium; Charybdotoxin; Glyburide; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Potassium Channels; Psoas Muscles; Sarcoplasmic Reticulum; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds | 1992 |
Effects of drugs on ventricular fibrillation and ischaemic K+ loss in a model of ischaemia in perfused guinea-pig hearts in vitro.
Topics: 4-Aminopyridine; Animals; Anti-Arrhythmia Agents; Benzothiazoles; Calcium Channel Blockers; Disease Models, Animal; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Myocardial Ischemia; Piperidines; Potassium; Potassium Channels; Pyrazines; Pyridines; Sympatholytics; Thiazoles; Ventricular Fibrillation | 1992 |
[The vasospasmolytic effects of nicorandil, cromakalim and pinacidil on 3,4-diaminopyridine-induced phasic contractions in canine coronary arteries as an experimental vasospasm model].
Topics: 4-Aminopyridine; Amifampridine; Animals; Benzopyrans; Coronary Vasospasm; Cromakalim; Disease Models, Animal; Dogs; Female; Glyburide; Guanidines; In Vitro Techniques; Ion Channel Gating; Male; Methylene Blue; Niacinamide; Nicorandil; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents | 1992 |
Glibenclamide inhibits a voltage-gated K+ current in the human neuroblastoma cell line SH-SY5Y.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Cadmium; Cell Line; Glyburide; Humans; Kinetics; Membrane Potentials; Neuroblastoma; Potassium Channels; Tetraethylammonium; Tetraethylammonium Compounds | 1992 |
K+ efflux pathways and neurotransmitter release associated to hippocampal ischemia: effects of glucose and of K+ channel blockers.
Topics: 4-Aminopyridine; Animals; Apamin; Aspartic Acid; Barium; Barium Compounds; Brain Ischemia; Calcium Chloride; Charybdotoxin; Chlorides; Elapid Venoms; gamma-Aminobutyric Acid; Glipizide; Glucose; Glyburide; Hippocampus; In Vitro Techniques; Kinetics; Potassium; Potassium Channels; Rats; Rats, Inbred Strains; Rubidium; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds | 1991 |
Inhibition of the acetylcholine-induced relaxation of canine isolated basilar artery by potassium-conductance blockers.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Barium; Basilar Artery; Dogs; Female; Glyburide; In Vitro Techniques; Isometric Contraction; Male; Membranes; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroprusside; Potassium Channels; Potassium Chloride; Sodium; Tetraethylammonium Compounds | 1991 |
Effect of channel blockers on potassium efflux from metabolically exhausted frog skeletal muscle.
Topics: 4-Aminopyridine; Aminopyridines; Animals; Apamin; Barium; Cell Membrane Permeability; Decamethonium Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Glyburide; In Vitro Techniques; Ion Channels; Muscles; Potassium; Quinine; Rana temporaria; Rubidium; Scorpion Venoms; Tetraethylammonium Compounds; Tolbutamide | 1987 |
Glyburide blocks the relaxation response to BRL 34915 (cromakalim), minoxidil sulfate and diazoxide in vascular smooth muscle.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Aminopyridines; Animals; Antihypertensive Agents; Benzopyrans; Charybdotoxin; Cromakalim; Diazoxide; Glyburide; Male; Minoxidil; Muscle, Smooth, Vascular; Potassium Channels; Pyrroles; Rats; Rats, Inbred Strains; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds; Vasodilation | 1989 |
The effects of K+ channel blockers on the spontaneous electrical and contractile activity in the proximal renal pelvis of the guinea pig.
Topics: 4-Aminopyridine; Action Potentials; Animals; Apamin; Charybdotoxin; Female; Glyburide; Guinea Pigs; Kidney Pelvis; Male; Muscle Contraction; Muscle, Smooth; Potassium Channel Blockers; Potassium Channels; Tetraethylammonium; Tetraethylammonium Compounds | 1996 |
ATP-sensitive K+ currents in cerebral arterial smooth muscle: pharmacological and hormonal modulation.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Cerebral Arteries; Electric Conductivity; Glyburide; Male; Muscle, Smooth, Vascular; Potassium Channel Blockers; Potassium Channels; Rabbits; Tetraethylammonium; Tetraethylammonium Compounds; Vasoconstrictor Agents; Vasodilator Agents | 1995 |
Potassium channel inhibitors attenuate neuromodulatory effects of atrial natriuretic factor in the rabbit isolated vas deferens.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Atrial Natriuretic Factor; Benzopyrans; Charybdotoxin; Cromakalim; Glyburide; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Potassium Channel Blockers; Potassium Channels; Prazosin; Pyrroles; Rabbits; Receptors, Adrenergic; Scorpion Venoms; Synaptic Transmission; Tetraethylammonium; Tetraethylammonium Compounds; Vas Deferens | 1994 |
Single-channel activity induced in mitoplasts by alkaline pH.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Glyburide; Hydrogen-Ion Concentration; Ion Channels; Mitochondria | 1994 |
Potassium channel blockade of atrial negative inotropic responses to P1-purinoceptor and muscarinic receptor agonists and to cromakalim.
Topics: 4-Aminopyridine; Adenosine; Animals; Benzopyrans; Carbachol; Cromakalim; Depression, Chemical; Glyburide; Guinea Pigs; Heart Atria; Hydrochloric Acid; In Vitro Techniques; Male; Myocardial Contraction; Parasympatholytics; Phenylisopropyladenosine; Potassium Channels; Pyrroles; Receptors, Muscarinic; Receptors, Purinergic; Rubidium Radioisotopes | 1993 |
A simple method for measurement of ureteric peristaltic function in vivo and the effects of drugs acting on ion channels applied from the ureter lumen in anesthetized rats.
Topics: 4-Aminopyridine; Anesthesia; Animals; Benzopyrans; Cromakalim; Glyburide; Ion Channels; Lidocaine; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyrroles; Rats; Rats, Sprague-Dawley; Ureter; Vasodilator Agents | 1993 |
Calcium-mediated agonists activate an inwardly rectified K+ channel in colonic secretory cells.
Topics: 4-Aminopyridine; Animals; Apamin; Barium; Calcium; Cell Line; Charybdotoxin; Colon; Cytosol; Glyburide; Hydrogen-Ion Concentration; Kinetics; Membrane Potentials; Potassium Channels; Quinine; Scorpion Venoms; Sodium; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors | 1993 |
Inward rectifier K+ currents in smooth muscle cells from rat resistance-sized cerebral arteries.
Topics: 4-Aminopyridine; Animals; Barium; Cerebral Arteries; Charybdotoxin; Female; Glyburide; Kinetics; Membrane Potentials; Muscle, Smooth, Vascular; Potassium; Potassium Channels; Rats; Rats, Inbred WKY; Scorpion Venoms | 1993 |
Characterization of the adenosine A1 receptor-activated potassium current in rat locus ceruleus neurons.
Topics: 4-Aminopyridine; Adenosine; Animals; Barium; Dose-Response Relationship, Drug; Glyburide; Locus Coeruleus; Male; Membrane Potentials; Neurons; Potassium Channels; Rats; Rats, Inbred F344; Receptors, Purinergic P1; Theophylline | 1995 |
Inhibition of ATP-sensitive potassium channels causes reversible cell-cycle arrest of human breast cancer cells in tissue culture.
Topics: 4-Aminopyridine; Breast Neoplasms; Cell Cycle; Cell Division; Glyburide; Humans; Potassium Channel Blockers; Potassium Channels; Pyrrolidines; Quinidine; Tetraethylammonium; Tetraethylammonium Compounds; Tumor Cells, Cultured | 1995 |
Tetraethylammonium selectively stimulates secretion from noradrenergic bovine chromaffin cells.
Topics: 4-Aminopyridine; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; Drug Interactions; Drug Synergism; Epinephrine; Glyburide; Nifedipine; Norepinephrine; Ouabain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tolbutamide | 1994 |
K(+)-channel blockers and coronary vasoconstriction in guinea-pig perfused hearts in-vitro.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Coronary Vessels; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Perfusion; Phentolamine; Potassium Channels; Pyrazines; Pyridines; Vasoconstriction | 1993 |
Persistent muscarinic excitation in guinea-pig olfactory cortex neurons: involvement of a slow post-stimulus afterdepolarizing current.
Topics: 4-Aminopyridine; Action Potentials; Animals; Atropine; Barium; Glyburide; Guinea Pigs; Lanthanum; Membrane Potentials; Neurons; Olfactory Pathways; Oxotremorine; Potassium Channels; Quaternary Ammonium Compounds; Receptors, Muscarinic; Tubocurarine | 1993 |
Novel potassium channel openers: synthesis and pharmacological evaluation of new N-(substituted-3-pyridyl)-N'-alkylthioureas and related compounds.
Topics: 4-Aminopyridine; Amifampridine; Animals; Antihypertensive Agents; Biomechanical Phenomena; Glyburide; Guanidines; Hypertension; Male; Molecular Structure; Norbornanes; Pinacidil; Portal Vein; Potassium Channels; Rats; Rats, Inbred SHR; Rats, Wistar; Structure-Activity Relationship | 1994 |
Properties of the LP-805-induced potassium currents in cultured bovine pulmonary artery endothelial cells.
Topics: 4-Aminopyridine; Animals; Cattle; Cells, Cultured; Endothelium, Vascular; Glyburide; Membrane Potentials; Potassium Channels; Pulmonary Artery; Pyrazoles; Pyrimidines; Quaternary Ammonium Compounds; Tetraethylammonium; Tetraethylammonium Compounds; Vasodilator Agents | 1994 |
Chronic hypoxia is associated with reduced delayed rectifier K+ current in rat pulmonary artery muscle cells.
Topics: 4-Aminopyridine; Animals; Chronic Disease; Electric Conductivity; Electrophysiology; Glyburide; Hypoxia; Male; Muscle, Smooth, Vascular; Potassium; Pulmonary Artery; Rats; Rats, Wistar | 1994 |
Potassium channel antagonists and vascular reactivity in stroke-prone spontaneously hypertensive rats.
Topics: 4-Aminopyridine; Amifampridine; Animals; Apamin; Barium; Cardiovascular System; Carotid Arteries; Cell Membrane; Cerebrovascular Disorders; Diazoxide; Female; Glyburide; Hypertension; Male; Muscle, Smooth, Vascular; Potassium Channels; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Risk Factors; Tetraethylammonium; Tetraethylammonium Compounds; Vasoconstriction; Vasodilation | 1993 |
Ionic currents and inhibitory effects of glibenclamide in seminal vesicle smooth muscle cells.
Topics: 4-Aminopyridine; Amifampridine; Animals; Barium; Biological Transport, Active; Cadmium; Calcium; Calcium Channels; Egtazic Acid; Electric Stimulation; Glyburide; Guinea Pigs; Hypoglycemic Agents; Ion Transport; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Patch-Clamp Techniques; Potassium; Potassium Channels; Potassium Chloride; Seminal Vesicles; Tetraethylammonium; Tetraethylammonium Compounds | 1995 |
k-Opioid receptor activation of a dendrotoxin-sensitive potassium channel mediates presynaptic inhibition of mossy fiber neurotransmitter release.
Topics: 4-Aminopyridine; Analgesics; Animals; Barium; Bee Venoms; Benzeneacetamides; Elapid Venoms; Evoked Potentials; Glyburide; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Nerve Fibers; Neurotoxins; Peptides; Potassium Channels; Pyrrolidines; Receptors, Opioid, kappa; Shaker Superfamily of Potassium Channels; Synapses; Tetraethylammonium; Tetraethylammonium Compounds | 1996 |
Effects of some K(+)-channel inhibitors on the electrical behaviour of guinea-pig isolated trachealis and on its responses to spasmogenic drugs.
Topics: 4-Aminopyridine; Action Potentials; Animals; Anti-Arrhythmia Agents; Atropine; Carbachol; Charybdotoxin; Electrophysiology; Female; Glyburide; Guinea Pigs; Histamine; Hypoglycemic Agents; Male; Muscle, Smooth; Parasympatholytics; Peptides; Phenethylamines; Potassium Channel Blockers; Scorpion Venoms; Sulfonamides; Trachea | 1996 |
Effects of potassium channel blockers on resting tone in isolated coronary arteries.
Topics: 4-Aminopyridine; Animals; Coronary Vessels; Dose-Response Relationship, Drug; Glyburide; In Vitro Techniques; Potassium Channel Blockers; Swine; Tetraethylammonium Compounds | 1996 |
Properties of a novel K+ current that is active at resting potential in rabbit pulmonary artery smooth muscle cells.
Topics: 4-Aminopyridine; Animals; Electrophysiology; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Ion Channel Gating; Male; Membrane Potentials; Muscle Tonus; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Potassium Channels; Pulmonary Artery; Rabbits; Tetraethylammonium Compounds | 1996 |
Effects of potassium channel blockers on the action potentials and contractility of the rat right ventricle.
Topics: 4-Aminopyridine; Action Potentials; Adrenergic beta-Agonists; Animals; Anti-Arrhythmia Agents; Dose-Response Relationship, Drug; Glyburide; Heart; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Potassium Channel Blockers; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Stimulation, Chemical | 1996 |
Role of potassium channels in relaxations of isolated canine basilar arteries to acidosis.
Topics: 4-Aminopyridine; Acidosis; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Barium Compounds; Basilar Artery; Calcium Channel Blockers; Charybdotoxin; Chlorides; Dogs; Endothelium, Vascular; Female; Glyburide; Hydrogen-Ion Concentration; Ion Channel Gating; KATP Channels; Male; Molsidomine; Muscle, Smooth, Vascular; Potassium Channels; Potassium Channels, Inwardly Rectifying; Uridine Triphosphate; Vasodilation | 1997 |
Potassium conductances and proliferation in conditionally immortalized renal glomerular mesangial cells from the H-2Kb-tsA58 transgenic mouse.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; Barium; Calcium; Cell Division; Cell Line; Cesium; Gadolinium; Glomerular Mesangium; Glyburide; H-2 Antigens; Interferon-gamma; Mice; Mice, Transgenic; Oncogenes; Osmolar Concentration; Potassium Channels | 1997 |
Apamin blocks the direct relaxant effect of melatonin on rat ileal smooth muscle.
Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Apamin; Calcium; Calcium Channel Blockers; Carbachol; Cholinergic Antagonists; Glyburide; Hexamethonium; Humans; Ileum; Male; Melatonin; Muscarinic Antagonists; Muscle Contraction; Neuromuscular Depolarizing Agents; Nitrendipine; Phentolamine; Rats; Rats, Wistar; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1997 |
The involvement of KCa, KATP and KV channels in vasorelaxing responses to acetylcholine in rat aortic rings.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Cyclic GMP; Glyburide; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Nitric Oxide; Peptides; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Vasodilation | 1997 |
Arachidonic acid activation of potassium channels in rat visual cortex neurons.
Topics: 4-Aminopyridine; Animals; Apamin; Arachidonic Acid; Barium; Charybdotoxin; Docosahexaenoic Acids; Egtazic Acid; Fatty Acids, Nonesterified; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Quinidine; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Tetraethylammonium Compounds; Visual Cortex | 1997 |
ATP and [3H]noradrenaline release and the presence of ecto-Ca(2+)-ATPases in the capsule-glomerulosa fraction of the rat adrenal gland.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Adrenal Glands; Adrenergic alpha-Antagonists; Animals; Berberine; Calcium-Transporting ATPases; Electric Stimulation; Glyburide; Histocytochemistry; Male; Microscopy, Electron; Norepinephrine; Organ Culture Techniques; Potassium Channel Blockers; Rats; Rats, Wistar; Tetrodotoxin; Tritium | 1997 |
Benefits of supplementing St Thomas' Hospital cardioplegic solution with tetraethylammonium on functional and metabolic recovery of isolated rat hearts.
Topics: 4-Aminopyridine; Animals; Bicarbonates; Calcium Chloride; Cardioplegic Solutions; Coronary Circulation; Dose-Response Relationship, Drug; Energy Metabolism; Female; Glyburide; Heart Arrest, Induced; Magnesium; Male; Myocardium; Potassium Channel Blockers; Potassium Chloride; Rats; Rats, Wistar; Sodium Chloride; Tetraethylammonium; Tetraethylammonium Compounds | 1997 |
Role of potassium channels in relaxations of canine middle cerebral arteries induced by nitric oxide donors.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; 4-Aminopyridine; Animals; Barium Compounds; Cerebral Arteries; Charybdotoxin; Chlorides; Cyclic GMP; Diltiazem; Dogs; Glyburide; In Vitro Techniques; Molsidomine; Muscle, Smooth, Vascular; Nitric Oxide; Nitroprusside; Potassium Channels; Purinones; Vasodilation; Vasodilator Agents | 1997 |
Inhibition of maxi-K currents in ferret portal vein smooth muscle cells by the antifungal clotrimazole.
Topics: 4-Aminopyridine; Animals; Antifungal Agents; Cells, Cultured; Charybdotoxin; Clotrimazole; Cytochrome P-450 Enzyme System; Electric Conductivity; Ferrets; Glyburide; Ion Channel Gating; Membrane Potentials; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Peptides; Portal Vein; Potassium Channel Blockers; Tetraethylammonium; Tetraethylammonium Compounds; Toxins, Biological | 1997 |
Interactions between neuropeptide Y and the adenylate cyclase pathway in rat mesenteric small arteries: role of membrane potential.
Topics: 4-Aminopyridine; Acetylcholine; Adenylyl Cyclases; Animals; Charybdotoxin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dichlororibofuranosylbenzimidazole; Gadolinium; Glyburide; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Nifedipine; Potassium Channels; Rats; Rats, Wistar; Thionucleotides | 1997 |
Types of potassium channels involved in coronary reactive hyperemia depend on duration of preceding ischemia in rat hearts.
Topics: 4-Aminopyridine; Adenosine Diphosphate; Animals; Apamin; Charybdotoxin; Glyburide; Hyperemia; In Vitro Techniques; Indomethacin; Male; Myocardial Ischemia; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Potassium Channels; Rats; Rats, Wistar; Regional Blood Flow; Tetraethylammonium; Tetraethylammonium Compounds | 1997 |
A comparison of EDHF-mediated and anandamide-induced relaxations in the rat isolated mesenteric artery.
Topics: 4-Aminopyridine; Animals; Apamin; Arachidonic Acids; Barium; Biological Factors; Calcium Channel Blockers; Charybdotoxin; Endocannabinoids; Enzyme Inhibitors; Glyburide; Hypoglycemic Agents; Indoles; Male; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Peptides; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Potassium; Potassium Channel Blockers; Protease Inhibitors; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Tosyl Compounds; Vasodilation; Virulence Factors, Bordetella | 1997 |
The effects of levcromakalim and pinacidil on the human internal mammary artery.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Apamin; Charybdotoxin; Coronary Artery Bypass; Coronary Disease; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Guanidines; Humans; In Vitro Techniques; Male; Mammary Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Pinacidil; Potassium Channels; Tetraethylammonium; Vasodilation; Vasodilator Agents | 1997 |
Leishmania sp.: growth and survival are impaired by ion channel blockers.
Topics: 4-Aminopyridine; Amiloride; Animals; Anthracenes; Cell Line; Cells, Cultured; Glyburide; Humans; Ion Channels; Leishmania; Macrophages; Mice | 1998 |
The endothelium-dependent, substance P relaxation of porcine coronary arteries resistant to nitric oxide synthesis inhibition is partially mediated by 4-aminopyridine-sensitive voltage-dependent K+ channels.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Animals; Apamin; Calcium; Charybdotoxin; Coronary Vessels; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Ion Transport; Isometric Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Potassium Channels; Quaternary Ammonium Compounds; Substance P; Swine | 1997 |
The effect of subarachnoid hemorrhage on mechanisms of vasodilation mediated by cyclic adenosine monophosphate.
Topics: 4-Aminopyridine; Adenylyl Cyclases; Animals; Basilar Artery; Charybdotoxin; Colforsin; Cyclic AMP; Disease Models, Animal; Dogs; Endothelium, Vascular; Enzyme Activation; Female; Glyburide; Ischemic Attack, Transient; Male; Potassium Channel Blockers; Potassium Channels; Subarachnoid Hemorrhage; Vasodilation; Vasodilator Agents | 1998 |
Relaxing effects of NO donors on guinea pig trachea in vitro are mediated by calcium-sensitive potassium channels.
Topics: 4-Aminopyridine; Animals; Calcium; Charybdotoxin; Female; Glyburide; Guinea Pigs; Male; Molsidomine; Nitric Oxide; Peptides; Potassium Channels; Trachea; Triazoles | 1998 |
Functions of large conductance Ca2+-activated (BKCa), delayed rectifier (KV) and background K+ channels in the control of membrane potential in rabbit renal arcuate artery.
Topics: 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amifampridine; Animals; Apamin; Arteries; Barium; Charybdotoxin; Glyburide; In Vitro Techniques; Kidney; Large-Conductance Calcium-Activated Potassium Channels; Male; Membrane Potentials; Muscle, Smooth, Vascular; Ouabain; Peptides; Potassium Channels; Potassium Channels, Calcium-Activated; Rabbits; Scorpion Venoms; Vasoconstriction | 1998 |
Potassium channels modulate hypoxic pulmonary vasoconstriction.
Topics: 4-Aminopyridine; Animals; Blood Pressure; Dogs; Female; Glyburide; Hypoxia; In Vitro Techniques; Male; Mathematics; Models, Cardiovascular; Potassium Channel Blockers; Potassium Channels; Pulmonary Artery; Pulmonary Circulation; Tetraethylammonium; Vascular Resistance; Vasoconstriction | 1998 |
Intracellular acidosis differentially regulates KV channels in coronary and pulmonary vascular muscle.
Topics: 4-Aminopyridine; Acidosis; Ammonium Chloride; Animals; Cell Membrane; Coronary Vessels; Elapid Venoms; Glyburide; Hydrogen-Ion Concentration; In Vitro Techniques; Membrane Potentials; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Peptides; Potassium Channel Blockers; Potassium Channels; Pulmonary Artery; Rats; Rats, Sprague-Dawley | 1998 |
Relaxation of corpus cavernosum and raised intracavernous pressure by berberine in rabbit.
Topics: 4-Aminopyridine; Animals; Apamin; Berberine; Charybdotoxin; Dose-Response Relationship, Drug; Endothelium; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Male; Muscle Relaxation; Penis; Potassium; Potassium Channel Blockers; Pressure; Rabbits | 1998 |
Role of K+ channels in A2A adenosine receptor-mediated dilation of the pressurized renal arcuate artery.
Topics: 4-Aminopyridine; Adenosine; Amifampridine; Animals; Antihypertensive Agents; Apamin; Arteries; Barium; Cromakalim; Enzyme Inhibitors; Glyburide; In Vitro Techniques; Kidney; Male; Nicardipine; Ouabain; Peptides; Phenethylamines; Potassium; Potassium Channels; Pressure; Purinergic P1 Receptor Agonists; Rabbits; Receptor, Adenosine A2A; Receptors, Purinergic P1; Vasodilation; Vasodilator Agents | 1999 |
Ionic mechanism of isoflurane's actions on thalamocortical neurons.
Topics: 4-Aminopyridine; Action Potentials; Anesthetics, Inhalation; Animals; Baclofen; Cerebral Cortex; Dose-Response Relationship, Drug; Electric Conductivity; Female; GABA Agonists; Glyburide; Hypoglycemic Agents; Isoflurane; Male; Neurons; Parasympathomimetics; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Synapses; Tacrine; Tetraethylammonium; Tetrodotoxin; Thalamus | 1999 |
Inhibitory effect of 4-aminopyridine on responses of the basilar artery to nitric oxide.
Topics: 4-Aminopyridine; Acetylcholine; Adenosine Triphosphate; Animals; Basilar Artery; Cromakalim; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Male; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Oxadiazoles; Papaverine; Potassium Channel Blockers; Quinoxalines; Rats; Rats, Sprague-Dawley; Vasodilation; Vasodilator Agents | 1999 |
P2u receptor-mediated release of endothelium-derived relaxing factor/nitric oxide and endothelium-derived hyperpolarizing factor from cerebrovascular endothelium in rats.
Topics: 4-Aminopyridine; Animals; Apamin; Barium Compounds; Cerebral Arteries; Cerebrovascular Circulation; Charybdotoxin; Chlorides; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Hypoglycemic Agents; Male; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxadiazoles; Peptides; Potassium Channels; Potassium Chloride; Quinoxalines; Rats; Rats, Long-Evans; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Tetraethylammonium; Uridine Triphosphate; Vasodilation | 1999 |
Post-partum prolongation of the atrial repolarization in rabbit.
Topics: 4-Aminopyridine; Action Potentials; Animals; Atrial Function; Electrophysiology; Estrogens; Female; Glyburide; Heart Atria; Heart Conduction System; Hypoglycemic Agents; Muscle Fibers, Skeletal; Myocardium; Pinacidil; Postpartum Period; Potassium Channels; Pregnancy; Rabbits; Vasodilator Agents | 1999 |
Effects of K(+)-channel blockers on A1-adenosine receptor-mediated negative inotropy and chronotropy of guinea-pig isolated left and right atria.
Topics: 4-Aminopyridine; Adenosine; Animals; Dose-Response Relationship, Drug; Drug Interactions; Glyburide; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Potassium Channel Blockers; Receptors, Purinergic P1; Tetraethylammonium; Vasodilator Agents | 1999 |
Activity of voltage-gated K+ channels is associated with cell proliferation and Ca2+ influx in carcinoma cells of colon cancer.
Topics: 4-Aminopyridine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Carbamates; Cell Division; Charybdotoxin; Colonic Neoplasms; Glyburide; Humans; Ion Channel Gating; Nickel; Peptides; Phenylcarbamates; Potassium; Potassium Channel Blockers; Potassium Channels; Quaternary Ammonium Compounds; RNA, Messenger; Tetraethylammonium; Tumor Cells, Cultured | 1999 |
Enhanced phenylephrine-induced rhythmic activity in the atherosclerotic mouse aorta via an increase in opening of KCa channels: relation to Kv channels and nitric oxide.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Aorta; Arteriosclerosis; Calcium; Cholera Toxin; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Indomethacin; Ion Channel Gating; Male; Mice; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; Ouabain; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Ryanodine; Tetraethylammonium Compounds | 1999 |
Different mechanisms for testosterone-induced relaxation of aorta between normotensive and spontaneously hypertensive rats.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Aorta, Thoracic; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Glyburide; Hypertension; Hypoglycemic Agents; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroarginine; Nitroprusside; Potassium Channels; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Testosterone; Tetraethylammonium; Vasodilator Agents | 1999 |
Mediators of alkalosis-induced relaxation of piglet pulmonary veins.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Alkalosis; Animals; Cyclic GMP; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Nitric Oxide; Nitroarginine; Oxadiazoles; Peptides; Potassium Channels; Pulmonary Veins; Quinoxalines; Swine; Vasoconstrictor Agents; Vasodilation | 2000 |
Possible role of potassium channels in mu-receptor-mediated inhibition and muscarinic autoinhibition in acetylcholine release from myenteric plexus of guinea pig ileum.
Topics: 4-Aminopyridine; Acetylcholine; Analgesics, Opioid; Animals; Apamin; Atropine; Drug Interactions; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Glyburide; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscarinic Antagonists; Myenteric Plexus; Naloxone; Narcotic Antagonists; Neuromuscular Junction; Peptides; Potassium Channel Blockers; Potassium Channels; Receptors, Muscarinic; Receptors, Opioid, mu; Tetraethylammonium | 2000 |
K(+) channel inhibition, calcium signaling, and vasomotor tone in canine pulmonary artery smooth muscle.
Topics: 4-Aminopyridine; Adrenergic alpha-Agonists; Animals; Calcium Signaling; Cells, Cultured; Cromakalim; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; In Vitro Techniques; Membrane Potentials; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Pulmonary Artery; Thapsigargin; Vasoconstriction; Vasodilator Agents; Vasomotor System | 2000 |
4-aminopyridine inhibits the occurrence of ventricular fibrillation but not ventricular tachycardia in the reperfused, P6olated rat heart.
Topics: 4-Aminopyridine; Animals; Anti-Arrhythmia Agents; Blood Flow Velocity; Glyburide; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Reperfusion; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Tachycardia, Ventricular; Torsades de Pointes; Ventricular Fibrillation; Verapamil | 2000 |
Comparison of the pharmacological properties of EDHF-mediated vasorelaxation in guinea-pig cerebral and mesenteric resistance vessels.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Arachidonic Acids; Biological Factors; Cerebral Arteries; Charybdotoxin; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Guinea Pigs; Imidazoles; In Vitro Techniques; Indomethacin; Male; Mesenteric Arteries; Nitric Oxide; Nitroarginine; Ouabain; Oxadiazoles; Potassium Channel Blockers; Potassium Channels; Quinoxalines; Vasodilation; Vasodilator Agents | 2000 |
Voltage-gated potassium channels in human ductus arteriosus.
Topics: 4-Aminopyridine; Charybdotoxin; Cyclooxygenase Inhibitors; Ductus Arteriosus; Ductus Arteriosus, Patent; Endothelin-1; Glyburide; Humans; Hypoxia; Ion Channel Gating; Membrane Potentials; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Oxygen Consumption; Potassium Channels | 2000 |
Diversity of channels involved in Ca(2+) activation of K(+) channels during the prolonged AHP in guinea-pig sympathetic neurons.
Topics: 4-Aminopyridine; Animals; Apamin; Calcium; Calcium Channel Blockers; Calcium Channels; Female; Ganglia, Sympathetic; Glyburide; Guinea Pigs; In Vitro Techniques; Large-Conductance Calcium-Activated Potassium Channels; Male; Membrane Potentials; Neurons; omega-Agatoxin IVA; omega-Conotoxin GVIA; Patch-Clamp Techniques; Peptides; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Small-Conductance Calcium-Activated Potassium Channels; Tetraethylammonium | 2000 |
The effects of potassium channel blockers on progesterone-induced suppression of rat portal vein contractility.
Topics: 4-Aminopyridine; Animals; Barium Compounds; Chlorides; Glyburide; Hypoglycemic Agents; Male; Muscle Contraction; Muscle, Smooth, Vascular; Peptides; Portal Vein; Potassium Channel Blockers; Progesterone; Rats; Rats, Wistar | 2000 |
Chronic hypoxia increases the NO contribution of acetylcholine vasodilation of the fetal guinea pig heart.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Coronary Vessels; Female; Fetal Hypoxia; Gene Expression Regulation; Gestational Age; Glyburide; Guinea Pigs; Heart Ventricles; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroprusside; Oxygen; Potassium Channel Blockers; Pregnancy; RNA, Messenger; Vasodilation | 2000 |
Opposing roles of K(+) and Cl(-) channels in maintenance of opossum lower esophageal sphincter tone.
Topics: 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Action Potentials; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Chloride Channels; Esophagogastric Junction; Glyburide; Isometric Contraction; Microelectrodes; Muscle, Smooth; Nifedipine; Niflumic Acid; Opossums; Potassium Channels | 2000 |
Role of potassium channels in regulation of brain arteriolar tone: comparison of cerebrum versus brain stem.
Topics: 4-Aminopyridine; Animals; Arterioles; Barium Compounds; Brain; Brain Stem; Chlorides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Nitric Oxide Synthase; Nitroarginine; Pinacidil; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Telencephalon; Tetraethylammonium; Vasoconstriction; Vasodilator Agents | 2001 |
Three types of K(+) currents in murine osteocyte-like cells (MLO-Y4).
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Apamin; Cell Differentiation; Cell Line; Cell Lineage; Cesium; Chlorides; Collagen; DNA Primers; Gene Expression; Glyburide; Guanosine Triphosphate; Hypoglycemic Agents; Membrane Potentials; Mice; Osteocytes; Patch-Clamp Techniques; Potassium Channels; Reverse Transcriptase Polymerase Chain Reaction; Sodium Chloride; Tetraethylammonium | 2001 |
The role of platelet-activating factor (PAF) antagonists and nitric oxide in cardiac actions of PAF. Electrophysiological and morphological study.
Topics: 4-Aminopyridine; Action Potentials; Animals; Azepines; Diterpenes; Electrophysiology; Fibrinolytic Agents; Ginkgolides; Glyburide; Guinea Pigs; Heart; In Vitro Techniques; Lactones; Myocardium; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Platelet Activating Factor; Platelet Aggregation Inhibitors; Potassium Channel Blockers; Reperfusion Injury; Triazoles | 2000 |
Effects of phosphodiesterase inhibitors on hypoxic pulmonary vasoconstriction. Influence of K(+) channels and nitric oxide.
Topics: 4-Aminopyridine; Animals; Apamin; Charybdotoxin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Hypoxia; In Vitro Techniques; Lung; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Potassium Channels; Purinones; Rats; Rats, Wistar; Rolipram; Theophylline; Vasoconstriction | 2001 |
Oxygen dilation in fetal pulmonary arterioles: role of K(+) channels.
Topics: 4-Aminopyridine; Animals; Arterioles; Charybdotoxin; Female; Fetus; Glyburide; Hypoglycemic Agents; Lung; Oxygen; Potassium Channel Blockers; Potassium Channels; Pregnancy; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Vasodilation | 2001 |
Potassium channels regulate tone in rat pulmonary veins.
Topics: 4-Aminopyridine; Animals; Barium; Cell Separation; Endothelium, Vascular; Glyburide; Immunohistochemistry; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardium; Patch-Clamp Techniques; Peptides; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pulmonary Circulation; Pulmonary Veins; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Vascular Resistance; Vasoconstriction; Vasodilation | 2001 |
Pharmacological evidence for the activation of potassium channels as the mechanism involved in the hypotensive and vasorelaxant effect of dioclein in rat small resistance arteries.
Topics: 4-Aminopyridine; Analgesics; Animals; Apamin; Barium Compounds; Charybdotoxin; Chlorides; Consciousness; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Flavanones; Flavonoids; Glyburide; Hemodynamics; Hypotension; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptides; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Rats; Rats, Wistar; Tetraethylammonium; Time Factors; Vascular Resistance; Vasodilation | 2001 |
Dibutyryl-cyclic GMP induces peripheral antinociception via activation of ATP-sensitive K(+) channels in the rat PGE2-induced hyperalgesic paw.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Analgesics; Animals; Apamin; Cesium; Charybdotoxin; Dibutyryl Cyclic GMP; Dinoprostone; Dose-Response Relationship, Drug; Glyburide; Hindlimb; Hyperalgesia; Male; Pain; Pain Measurement; Pain Threshold; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide | 2001 |
Anandamide-induced relaxation of sheep coronary arteries: the role of the vascular endothelium, arachidonic acid metabolites and potassium channels.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Animals; Apamin; Arachidonic Acid; Arachidonic Acids; Barium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Coronary Vessels; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Miconazole; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptides; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Potassium; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Receptors, Drug; Rimonabant; Sheep; Tetraethylammonium; Vasoconstrictor Agents; Vasodilation | 2001 |
Role of potassium channels in the relaxation induced by the nitric oxide (NO) donor DEA/NO in the isolated rat basilar artery.
Topics: 4-Aminopyridine; Animals; Anti-Arrhythmia Agents; Basilar Artery; Glyburide; Hydrazines; In Vitro Techniques; Male; Molsidomine; Nitric Oxide Donors; Nitrogen Oxides; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Vasodilation | 2001 |
Effects of different types of K+ channel modulators on the spontaneous myogenic contraction of guinea-pig urinary bladder smooth muscle.
Topics: 4-Aminopyridine; Animals; Anti-Arrhythmia Agents; Apamin; Barium; Benzimidazoles; Calcium Channel Blockers; Cation Transport Proteins; Cromakalim; Diltiazem; Ether-A-Go-Go Potassium Channels; Female; Glyburide; Guinea Pigs; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle Contraction; Muscle, Smooth; Nisoldipine; Parasympatholytics; Peptides; Periodicity; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Potassium Channels, Voltage-Gated; Pyridines; Small-Conductance Calcium-Activated Potassium Channels; Urinary Bladder | 2001 |
Evidence for a new mechanism of action of diclofenac: activation of K+ channels.
Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; ATP-Binding Cassette Transporters; Behavior, Animal; Diclofenac; Female; Formaldehyde; Glyburide; Hypoglycemic Agents; KATP Channels; Pain Measurement; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar | 2001 |
Novel properties of peptides derived from the sequence coded by exon 26A of human elastin.
Topics: 4-Aminopyridine; Animals; Aorta; Dose-Response Relationship, Drug; Elastin; Enzyme Inhibitors; Exons; Glyburide; Humans; Hypoglycemic Agents; In Vitro Techniques; Lactose; Male; Models, Biological; Muscle, Smooth, Vascular; Nitroarginine; Peptides; Phenylephrine; Potassium Channel Blockers; Rats; Rats, Wistar; Tolbutamide; Vasoconstrictor Agents; Virulence Factors, Bordetella | 2002 |
Pharmacological evidence for the activation of K(+) channels by diclofenac.
Topics: 4-Aminopyridine; Analgesics; Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Behavior, Animal; Charybdotoxin; Diclofenac; Dose-Response Relationship, Drug; Female; Formaldehyde; Glyburide; Hindlimb; Morphine; Pain; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide | 2002 |
The molecular site of action of K(ATP) channel inhibitors determines their ability to inhibit iNOS-mediated relaxation in rat aorta.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Aminopyridines; Analysis of Variance; Animals; Aorta; Arginine; Barium; Endothelium, Vascular; Glyburide; Guanidines; Lipopolysaccharides; Male; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitrites; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Tolbutamide; Vasodilator Agents | 2002 |
The peripheral antinociceptive effect of resveratrol is associated with activation of potassium channels.
Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; ATP-Binding Cassette Transporters; Charybdotoxin; Female; Glipizide; Glyburide; KATP Channels; Morphine; Narcotics; Peripheral Nervous System; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Resveratrol; Stilbenes; Tetraethylammonium; Tolbutamide | 2002 |
Possible involvement of potassium channels in peripheral antinociception induced by metamizol: lack of participation of ATP-sensitive K+ channels.
Topics: 4-Aminopyridine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apamin; Area Under Curve; ATP-Binding Cassette Transporters; Charybdotoxin; Dipyrone; Drug Interactions; Female; Formaldehyde; Glyburide; KATP Channels; Pain Measurement; Peripheral Nerves; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tetraethylammonium; Tolbutamide | 2003 |
An endothelium-derived factor modulates purinergic neurotransmission to mesenteric arterial smooth muscle of hamster.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Apamin; Biological Factors; Charybdotoxin; Cricetinae; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Epoprostenol; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Male; Membrane Potentials; Mesenteric Arteries; Mesocricetus; Muscle, Smooth, Vascular; Neuromuscular Junction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Ouabain; Pinacidil; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Synaptic Transmission; Tetraethylammonium; Time Factors; Triazines; Uridine Triphosphate; Vasodilator Agents | 2003 |
Volatile anesthetics regulate pulmonary vascular tension through different potassium channel subtypes in isolated rabbit lungs.
Topics: 4-Aminopyridine; Anesthetics, Inhalation; Animals; Female; Glyburide; Lung; Peptides; Potassium Channel Blockers; Potassium Channels; Rabbits; Vascular Resistance | 2003 |
Involvement of inwardly rectifying K+ channels in secretory responses of human ileal mucosa.
Topics: 4-Aminopyridine; Apamin; Bacterial Toxins; Barium Compounds; Charybdotoxin; Chlorides; Glyburide; Humans; Ileum; Intestinal Mucosa; Potassium Channel Blockers; Potassium Channels; Vasoactive Intestinal Peptide | 2003 |
[Effects of potassium channel blockers on the proliferation of rat bronchial smooth muscle cells].
Topics: 4-Aminopyridine; Animals; Bronchi; Calcium; Cell Division; Cells, Cultured; Glyburide; Muscle, Smooth; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Potassium Channels, Voltage-Gated; Proliferating Cell Nuclear Antigen; Rats; Rats, Sprague-Dawley; Tetraethylammonium | 2003 |
Functional role of potassium channels in the vasodilating mechanism of levosimendan in porcine isolated coronary artery.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Calcium; Coronary Vessels; Cromakalim; Glyburide; Hydrazones; In Vitro Techniques; Ion Channel Gating; Isometric Contraction; Muscle, Smooth, Vascular; Peptides; Potassium Channel Blockers; Potassium Channels; Pyridazines; Simendan; Swine; Tetraethylammonium; Vasodilator Agents | 2003 |
Functional expression of TRESK-2, a new member of the tandem-pore K+ channel family.
Topics: 4-Aminopyridine; Amino Acid Sequence; Animals; Apamin; Arachidonic Acid; Base Sequence; Blotting, Northern; Cell Membrane; Cloning, Molecular; COS Cells; Cytoplasm; DNA; DNA, Complementary; Electrophysiology; Glyburide; Humans; Male; Mice; Molecular Sequence Data; Phylogeny; Potassium Channels; Protein Structure, Tertiary; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Homology, Amino Acid; Testis; Tetraethylammonium; Time Factors; Tissue Distribution; Transfection | 2004 |
Study of the involvement of K+ channels in the peripheral antinociception of the kappa-opioid receptor agonist bremazocine.
Topics: 4-Aminopyridine; Analgesics; Animals; ATP-Binding Cassette Transporters; Benzomorphans; Charybdotoxin; Cyclic GMP; Dequalinium; Glyburide; Hyperalgesia; KATP Channels; Male; Naltrexone; Nitric Oxide; Peripheral Nervous System; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Opioid, kappa; Signal Transduction; Tetraethylammonium; Tolbutamide | 2004 |
Substance P induces inward current and regulates pacemaker currents through tachykinin NK1 receptor in cultured interstitial cells of Cajal of murine small intestine.
Topics: 4-Aminopyridine; Action Potentials; Alkaloids; Animals; Benzophenanthridines; Calcium; Cations, Divalent; Cells, Cultured; Electrophysiology; Enteric Nervous System; Female; Glyburide; Intestine, Small; Ion Channels; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nifedipine; Phenanthridines; Receptors, Neurokinin-1; Sinoatrial Node; Sodium; Substance P; Tachykinins; Tetraethylammonium; Tetrodotoxin | 2004 |
Visceral periadventitial adipose tissue regulates arterial tone of mesenteric arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Adipose Tissue; Amifampridine; Animals; Apamin; Barium; Cromakalim; Delayed Rectifier Potassium Channels; Endothelin-1; Glyburide; Male; Mesenteric Artery, Superior; Peptides; Phenylephrine; Potassium; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Quaternary Ammonium Compounds; Rats; Rats, Sprague-Dawley; Serotonin; Tetraethylammonium; Vascular Resistance; Vasodilation; Viscera | 2004 |
Volume regulation of mature and immature spermatozoa in a primate model, and possible ion channels involved.
Topics: 4-Aminopyridine; Animals; Apamin; Cell Size; Cells, Cultured; Charybdotoxin; Ejaculation; Epididymis; Glyburide; Ion Channels; Macaca fascicularis; Male; Neurotoxins; Nitrobenzoates; Potassium Channel Blockers; Quaternary Ammonium Compounds; Quinine; Scorpion Venoms; Spermatozoa; Tetraethylammonium | 2004 |
Contractile responses of isolated rat mesenteric arteries to acute episodes of severe hypoxia and subsequent reoxygenation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Adenosine Triphosphate; Animals; Anti-Arrhythmia Agents; Calcium; Endothelium, Vascular; Ethylamines; Glyburide; Hypoxia; Male; Mesenteric Arteries; Muscle Contraction; Norepinephrine; Oxygen; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Reperfusion Injury; Ryanodine | 2004 |
[Effect of potassium channel on the proliferation, apoptosis and related-gene expression in human bronchial smooth muscle cells].
Topics: 4-Aminopyridine; Apoptosis; Bronchi; Calcium; Cell Cycle; Cell Proliferation; Cells, Cultured; Fas Ligand Protein; Female; Flow Cytometry; Glyburide; Humans; Male; Middle Aged; Myocytes, Smooth Muscle; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Proliferating Cell Nuclear Antigen; Tetraethylammonium | 2004 |
Impaired KATP channel function in the fetoplacental circulation of patients with type 1 diabetes mellitus.
Topics: 4-Aminopyridine; Charybdotoxin; Diabetes Mellitus, Type 1; Endothelial Cells; Female; Glyburide; Humans; In Vitro Techniques; Placental Circulation; Potassium Channels; Pregnancy; Pregnancy in Diabetics | 2005 |
Pharmacological evidence for the activation of Ca2+-activated K+ channels by meloxicam in the formalin test.
Topics: 4-Aminopyridine; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Apamin; Behavior, Animal; Charybdotoxin; Dose-Response Relationship, Drug; Female; Formaldehyde; Glyburide; Meloxicam; Pain; Pain Measurement; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tetraethylammonium; Thiazines; Thiazoles; Tolbutamide | 2005 |
Capsaicin-induced, capsazepine-insensitive relaxation of the guinea-pig ileum.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Apamin; Barium; Benzopyrans; Caffeine; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Charybdotoxin; Diclofenac; Dimethyl Sulfoxide; Diterpenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanethidine; Guinea Pigs; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle Relaxation; Muscle, Smooth; Myosin Light Chains; Nitroarginine; Papaverine; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Protein Serine-Threonine Kinases; Pyrazoles; Receptor, Cannabinoid, CB1; rho-Associated Kinases; Tetraethylammonium; Vasodilator Agents | 2006 |
Probable activation of the opioid receptor-nitric oxide-cyclic GMP-K+ channels pathway by codeine.
Topics: 4-Aminopyridine; Analgesics, Opioid; Animals; Codeine; Cyclic GMP; Female; Glyburide; Methylene Blue; Naloxone; NG-Nitroarginine Methyl Ester; Nitric Oxide; Potassium Channels; Rats; Rats, Wistar; Receptors, Opioid; Tetraethylammonium; Tolbutamide | 2005 |
Possible activation of the NO-cyclic GMP-protein kinase G-K+ channels pathway by gabapentin on the formalin test.
Topics: 4-Aminopyridine; Amines; Analgesics; Animals; Apamin; Carbazoles; Charybdotoxin; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Cyclohexanecarboxylic Acids; Female; Gabapentin; gamma-Aminobutyric Acid; Glyburide; Indoles; Naloxone; NG-Nitroarginine Methyl Ester; Nitric Oxide; Pain Measurement; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tolbutamide | 2006 |
The mechanism of endothelium-independent relaxation induced by the wine polyphenol resveratrol in human internal mammary artery.
Topics: 4-Aminopyridine; Anti-Arrhythmia Agents; Charybdotoxin; Coronary Artery Bypass; Coronary Disease; Glyburide; Humans; Male; Mammary Arteries; Middle Aged; Muscle Relaxation; Muscle, Smooth, Vascular; Neurotoxins; Potassium Channel Blockers; Potassium Channels; Resveratrol; Scorpion Venoms; Stilbenes; Tetraethylammonium; Vasodilation; Vasodilator Agents; Wine | 2006 |
Membrane potassium currents in human radial artery and their regulation by nitric oxide donor.
Topics: 4-Aminopyridine; Adult; Aged; Aged, 80 and over; Blotting, Western; Female; Glyburide; Guanylate Cyclase; Humans; In Vitro Techniques; Ion Channel Gating; Male; Membrane Potentials; Middle Aged; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nitric Oxide Donors; Oxadiazoles; Patch-Clamp Techniques; Penicillamine; Peptides; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Potassium Channels, Voltage-Gated; Quinoxalines; Radial Artery; Tetraethylammonium Compounds | 2006 |
Potassium channels-mediated vasorelaxation of rat aorta induced by resveratrol.
Topics: 4-Aminopyridine; Animals; Antioxidants; Aorta; Charybdotoxin; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; Glyburide; In Vitro Techniques; Male; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Resveratrol; Scorpion Venoms; Stilbenes; Tetraethylammonium; Vasodilation; Vasodilator Agents | 2006 |
Testosterone relaxes isolated human radial artery by potassium channel opening action.
Topics: 4-Aminopyridine; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Humans; In Vitro Techniques; Indomethacin; NG-Nitroarginine Methyl Ester; Perfusion; Phenylephrine; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Potassium Chloride; Radial Artery; Testosterone; Tetraethylammonium; Vasoconstrictor Agents; Vasodilation | 2007 |
K+ channel modulation of slow wave activity in the guinea-pig prostate.
Topics: 4-Aminopyridine; Animals; Apamin; Benzopyrans; Calcitonin Gene-Related Peptide; Cromakalim; Cyclopentanes; Dose-Response Relationship, Drug; Electrophysiology; Glyburide; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Nitroprusside; Peptides; Potassium Channel Blockers; Potassium Channels; Prostate; Stromal Cells; Tetraethylammonium | 2007 |
In vivo assessment of safety and mechanisms underlying in vitro relaxation induced by Mikania laevigata Schultz Bip. ex Baker in the rat trachea.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Brazil; Coumarins; Dose-Response Relationship, Drug; Female; Gas Chromatography-Mass Spectrometry; Glyburide; In Vitro Techniques; Male; Mice; Mikania; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Oxadiazoles; Plant Extracts; Potassium Channel Blockers; Quinoxalines; Rats; Rats, Wistar; Tetraethylammonium; Toxicity Tests, Acute; Toxicity Tests, Chronic; Trachea | 2007 |
Investigation of relaxant effects of propofol on sheep sphincter of Oddi.
Topics: 4-Aminopyridine; Anesthetics, Intravenous; Animals; Dose-Response Relationship, Drug; Drug Combinations; Glyburide; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Propofol; Sheep; Sphincter of Oddi; Tetraethylammonium | 2007 |
Heat shock proteins and p53 play a critical role in K+ channel-mediated tumor cell proliferation and apoptosis.
Topics: 4-Aminopyridine; Alkaloids; Apoptosis; bcl-2-Associated X Protein; Benzylisoquinolines; Calcium Channel Blockers; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cyclin-Dependent Kinase Inhibitor p21; DNA Fragmentation; DNA-Binding Proteins; Glyburide; Heat-Shock Proteins; Humans; Large-Conductance Calcium-Activated Potassium Channels; Neoplasms; Oncogene Proteins, Viral; Patch-Clamp Techniques; Peptides; Potassium Channel Blockers; Tetraethylammonium; Tumor Suppressor Protein p53 | 2007 |
The gender differences in the relaxation to levosimendan of human internal mammary artery.
Topics: 4-Aminopyridine; Anti-Arrhythmia Agents; Charybdotoxin; Coronary Artery Bypass; Dose-Response Relationship, Drug; Female; Glyburide; Humans; Hydrazones; Male; Mammary Arteries; Middle Aged; Potassium Channel Blockers; Pyridazines; Sex Characteristics; Simendan; Vasodilation | 2007 |
Effects of taurine on aortic rings isolated from fructose-fed insulin resistance Sprague-Dawley rat are changed.
Topics: 4-Aminopyridine; Acetylcholine; Administration, Oral; Animals; Aorta; Blood Glucose; Blood Pressure; Cyclooxygenase Inhibitors; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Endothelium-Dependent Relaxing Factors; Endothelium, Vascular; Fructose; Glyburide; In Vitro Techniques; Indomethacin; Insulin; Insulin Resistance; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Peptides; Phenylephrine; Potassium Channel Blockers; Potassium Chloride; Rats; Rats, Sprague-Dawley; Taurine; Tetraethylammonium; Vasoconstriction; Vasodilation | 2008 |
Vasorelaxant effect of a self-etch adhesive system through calcium antagonistic action.
Topics: 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Dentin-Bonding Agents; Endothelium, Vascular; Enzyme Inhibitors; Epoprostenol; Glyburide; Indomethacin; Male; Materials Testing; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Potassium Channels, Voltage-Gated; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Time Factors; Vasoconstrictor Agents; Vasodilator Agents | 2008 |
The relaxation mechanisms of tetrandrine on the rabbit corpus cavernosum tissue in vitro.
Topics: 4-Aminopyridine; Animals; Benzylisoquinolines; Drugs, Chinese Herbal; Enzyme Inhibitors; Glyburide; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; Muscle, Smooth; Nitroarginine; Oxadiazoles; Penis; Potassium Channel Blockers; Potassium Chloride; Quinoxalines; Rabbits; Stephania tetrandra; Tetraethylammonium | 2009 |
Effect of acidosis on the mechanism(s) of insulin-induced vasorelaxation in normal Wistar-Kyoto (WKY) rat aorta.
Topics: 4-Aminopyridine; Acidosis; Animals; Aorta; Barium Compounds; Chlorides; Endothelium, Vascular; Glyburide; Hydrogen-Ion Concentration; Hypoglycemic Agents; Indomethacin; Insulin; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Ouabain; Phenylephrine; Potassium Channel Blockers; Rats; Rats, Inbred WKY; Tetraethylammonium; Vasoconstriction; Vasodilation | 2009 |
The role of nitric oxide and potassium channels in the effect of adrenomedullin in human internal thoracic arteries.
Topics: 4-Aminopyridine; Adrenomedullin; Aged; Glyburide; Humans; In Vitro Techniques; Male; Mammary Arteries; Middle Aged; NG-Nitroarginine Methyl Ester; Nitric Oxide; Potassium Channel Blockers; Potassium Channels | 2010 |
Cellular coupling of potassium channels with beta2 adrenoceptors in mediating myometrial relaxation in buffaloes (Bubalus bubalis).
Topics: 4-Aminopyridine; Adrenergic beta-Agonists; Albuterol; Animals; Buffaloes; Cromakalim; Female; Glyburide; Hypoglycemic Agents; Muscle Relaxation; Myometrium; Parasympatholytics; Potassium Channels; Receptors, Adrenergic, beta-2; Tetraethylammonium; Uterine Contraction | 2010 |
Differential involvement of potassium channel subtypes in early and late sepsis-induced hyporesponsiveness to vasoconstrictors.
Topics: 4-Aminopyridine; Animals; Apamin; Blood Pressure; Female; Glyburide; Muscle Contraction; Muscle, Smooth, Vascular; Peptides; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Sepsis; Tetraethylammonium; Time Factors; Vasoconstrictor Agents | 2010 |
Exploring the mechanism of endothelial involvement in acidosis-induced vasodilatation of aortic tissues from normal and diabetic rats.
Topics: 4-Aminopyridine; Acidosis; Animals; Aorta; Barium Compounds; Chlorides; Diabetes Mellitus; Endothelium, Vascular; Glucose Clamp Technique; Glyburide; Indomethacin; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Peptides; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Vasodilation | 2010 |
Contribution of adenosine A(2A) and A(2B) receptors to ischemic coronary dilation: role of K(V) and K(ATP) channels.
Topics: 4-Aminopyridine; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Coronary Circulation; Disease Models, Animal; Dogs; Flavins; Glyburide; Hyperemia; KATP Channels; Male; Myocardial Ischemia; Phenethylamines; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Pyrimidines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Triazoles; Vasodilation | 2010 |
Vasodilatory effect of hydroxyethyl methacrylate and triethylene glycol dimethacrylate in rat aorta through calcium antagonistic action.
Topics: 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Calcium Chloride; Composite Resins; Cyclooxygenase Inhibitors; Dental Materials; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Indomethacin; Male; Methacrylates; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide Synthase; Polyethylene Glycols; Polymethacrylic Acids; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Transducers; Vasoconstrictor Agents; Vasodilator Agents | 2011 |
Adenosine triphosphate-sensitive potassium channel blockers attenuate the antiallodynic effect of R-PIA in neuropathic rats.
Topics: 4-Aminopyridine; Adenosine; Adenosine Triphosphate; Animals; Glyburide; Humans; Hyperalgesia; Injections, Spinal; Male; Neurons; Pain; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Spinal Nerves | 2011 |
Vasoactivity of the gasotransmitters hydrogen sulfide and carbon monoxide in the chicken ductus arteriosus.
Topics: 4-Aminopyridine; Animals; Carbon Monoxide; Chick Embryo; Ductus Arteriosus; Glyburide; Hydrogen Sulfide; Models, Animal; NG-Nitroarginine Methyl Ester; Oxygen; Peptides; Sulfides; Tetraethylammonium; Vasodilation; Vasodilator Agents | 2011 |
Role of perivascular adipose tissue-derived methyl palmitate in vascular tone regulation and pathogenesis of hypertension.
Topics: 4-Aminopyridine; Adipocytes; Adipose Tissue; Angiotensin II; Animals; Aorta; Calcium; Cells, Cultured; Endothelium, Vascular; Fibroblasts; Glyburide; Hypertension; Losartan; Male; Palmitates; Peptides; Potassium Channels, Voltage-Gated; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Tetraethylammonium; Vasodilation; Vasodilator Agents | 2011 |
Investigation of mechanisms involved in (-)-borneol-induced vasorelaxant response on rat thoracic aorta.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium Chloride; Camphanes; Endothelium, Vascular; Glyburide; Phenylephrine; Potassium Channels; Potassium Chloride; Rats; Tetraethylammonium; Vasodilator Agents | 2012 |
Different potassium channels are involved in relaxation of rat renal artery induced by P1075.
Topics: 4-Aminopyridine; Animals; Endothelium, Vascular; Glyburide; Guanidines; Male; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Pyridines; Rats; Rats, Wistar; Renal Artery; Scorpion Venoms; Tetraethylammonium; Vasodilation; Vasodilator Agents | 2012 |
Role of calcium and potassium channels in effects of hydrogen sulfide on frog myocardial contractility.
Topics: 4-Aminopyridine; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Electric Stimulation; Glyburide; Heart; Hydrogen Sulfide; In Vitro Techniques; KATP Channels; Minoxidil; Myocardial Contraction; Myocardium; Nifedipine; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Rana ridibunda; Tetraethylammonium | 2011 |
Hypoxia sensitivity of a voltage-gated potassium current in porcine intrapulmonary vein smooth muscle cells.
Topics: 4-Aminopyridine; Amino Acid Sequence; Animals; Calcium Channel Blockers; Cell Hypoxia; Cells, Cultured; Conserved Sequence; Gene Expression; Glyburide; In Vitro Techniques; Membrane Potentials; Molecular Sequence Data; Mycotoxins; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Potassium Channels, Voltage-Gated; Pulmonary Veins; Sus scrofa; Tetraethylammonium; Vasoconstriction | 2012 |
Mechanisms of vasodilatatory effect of perivascular tissue of human internal thoracic artery.
Topics: 4-Aminopyridine; Adipose Tissue, White; Adventitia; Apamin; Barium Compounds; Chlorides; Glyburide; Heart Diseases; Humans; Immersion; In Vitro Techniques; Isometric Contraction; Large-Conductance Calcium-Activated Potassium Channels; Mammary Arteries; Muscle, Smooth, Vascular; Peptides; Potassium Channel Blockers; Potassium Channels; Vasodilation; Vasodilator Agents | 2013 |
Voltage-gated and ATP-sensitive K+ channels are associated with cell proliferation and tumorigenesis of human glioma.
Topics: 4-Aminopyridine; Animals; Apoptosis; Calcium; Calcium Signaling; Cell Line, Tumor; Cell Proliferation; Cell Transformation, Neoplastic; Diazoxide; G1 Phase Cell Cycle Checkpoints; Glioma; Glyburide; Humans; KATP Channels; Mice; Mice, Nude; Peptides; Phloretin; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Scorpion Venoms; Tetraethylammonium; Xenograft Model Antitumor Assays | 2014 |
The effect of resveratrol on contractility of non-pregnant rat uterus: the contribution of K(+) channels.
Topics: 4-Aminopyridine; Animals; Benzimidazoles; Female; Glyburide; Isometric Contraction; Muscle, Smooth; Oxytocin; Peptides; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Resveratrol; Stilbenes; Tetraethylammonium; Uterus | 2013 |
Effects of glucagon-like peptide-1 in diabetic rat small resistance arteries.
Topics: 4-Aminopyridine; Animals; Apamin; Arteries; Charybdotoxin; Cyclic GMP; Diabetes Mellitus, Experimental; Endothelium, Vascular; Glucagon-Like Peptide 1; Glyburide; Male; Nitric Oxide; Peptide Fragments; Peptides; Potassium Channels, Calcium-Activated; Rats; Rats, Wistar; Reactive Oxygen Species; Superoxide Dismutase | 2014 |
The vasorelaxant effect of p-cymene in rat aorta involves potassium channels.
Topics: 4-Aminopyridine; Animals; Aorta; Cesium; Chlorides; Cymenes; Dimethyl Sulfoxide; Glyburide; Male; Monoterpenes; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Vasodilation; Vasodilator Agents | 2015 |
15-oxo-ETE-induced internal carotid artery constriction in hypoxic rats is mediated by potassium channels.
Topics: 4-Aminopyridine; Animals; Arachidonic Acids; Carotid Artery, Internal; Glyburide; Hydroxyprostaglandin Dehydrogenases; Hypoxia; In Vitro Techniques; Male; Potassium Channels; Rats, Wistar; Tetraethylammonium; Vasoconstriction | 2016 |
Flavonoid galetin 3,6-dimethyl ether attenuates guinea pig ileum contraction through K(+) channel activation and decrease in cytosolic calcium concentration.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Apamin; Calcium; Calcium Chloride; Carbachol; Cell Survival; Cesium; Chlorides; Flavonoids; Glyburide; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Muscle Cells; Muscle Contraction; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Tetraethylammonium | 2015 |
Functional involvement of L-type calcium channels and cyclic nucleotide-dependent pathways in cadmium-induced myometrial relaxation in rats.
Topics: 4-Aminopyridine; Animals; Cadmium; Calcium Channels, L-Type; Cyclic GMP; Female; Glyburide; In Vitro Techniques; Muscle Relaxation; Myometrium; Phenylephrine; Propranolol; Rats; Rats, Wistar | 2017 |
2-Deoxy-d-glucose enhances tonic inhibition through the neurosteroid-mediated activation of extrasynaptic GABA
Topics: 4-Aminopyridine; Animals; Antimetabolites; Antineoplastic Agents; Bicuculline; Deoxyglucose; Enzyme Inhibitors; Female; Finasteride; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glyburide; Hippocampus; Hypoglycemic Agents; In Vitro Techniques; Iodoacetates; Isoquinolines; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Potassium Channel Blockers; Receptors, GABA; Statistics, Nonparametric | 2016 |
Signal Transduction Underlying the Inhibitory Mechanism of Fluoxetine on Electrical Field Stimulation Response in Rat Ileal Smooth Muscle.
Topics: 4-Aminopyridine; Amides; Animals; Atropine; Azepines; Benzophenanthridines; Bicuculline; Calcimycin; Drug Interactions; Electric Stimulation; Estrenes; Fluoxetine; Glyburide; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Ondansetron; Pyridines; Pyrrolidinones; Rats; Signal Transduction; Sulfonamides; Tetraethylammonium | 2017 |
Mechanisms of nicotine-induced cutaneous vasodilation and sweating in young adults: roles for K
Topics: 4-Aminopyridine; Atropine; Female; Glyburide; Humans; Male; Nicotine; Nitric Oxide; Potassium Channel Blockers; Potassium Channels; Prostaglandins; Sweating; Tetraethylammonium; Vasodilation; Young Adult | 2017 |
Investigation the relaxant effects of proton pump ınhibitors and their relaxation mechanism on sheep sphincter of Oddi.
Topics: 4-Aminopyridine; Animals; Cholangiopancreatography, Endoscopic Retrograde; Glyburide; Male; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Proton Pump Inhibitors; Sheep; Sphincter of Oddi | 2019 |
The role of potassium channels in the proliferation and migration of endometrial adenocarcinoma HEC1-A cells.
Topics: 4-Aminopyridine; Adenocarcinoma; Cell Proliferation; Endometrial Neoplasms; Female; Glyburide; Humans; Potassium Channels; Tetraethylammonium | 2022 |
Elabela relaxes rat pulmonary artery and trachea via BK
Topics: 4-Aminopyridine; Adenosine Triphosphate; Animals; Dideoxyadenosine; Endothelium, Vascular; Glyburide; Indomethacin; Male; Prostaglandins; Pulmonary Artery; Rats; Rats, Wistar; Trachea; Vascular Ring; Vasodilation; Vasodilator Agents | 2023 |