glutamine and quinazolines

glutamine has been researched along with quinazolines in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (16.67)18.2507
2000's2 (33.33)29.6817
2010's3 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Birdsall, DL; Finer-Moore, J; Huang, W; Santi, DV; Stroud, RM1
Basuroy, S; Rao, RK; Seth, A; Sheth, P1
Avissar, NE; Sax, HC; Toia, L1
Chough, C; Joung, M; Kim, ES; Lim, JW; Maeng, HJ; Shim, CK; Shim, WS1
Fan, Z; Li, X; Lu, H; Lu, Y; Qiu, S1
Aldib, I; Chikh Alard, I; De Carvalho, A; Dufrasne, F; Flemmig, J; Furtmüller, PG; Gelbcke, M; Mathieu, V; Meyer, F; Nève, J; Obinger, C; Prévost, M; Rousseau, A; Soubhye, J; Tadrent, S; Van Antwerpen, P; Zouaoui Boudjeltia, K1

Other Studies

6 other study(ies) available for glutamine and quinazolines

ArticleYear
The separate effects of E60Q in Lactobacillus casei thymidylate synthase delineate between mechanisms for formation of intermediates in catalysis.
    Protein engineering, 1998, Volume: 11, Issue:3

    Topics: Amino Acid Substitution; Asparagine; Binding Sites; Catalysis; Crystallography, X-Ray; Deoxyuracil Nucleotides; Folic Acid; Glutamic Acid; Glutamine; Lacticaseibacillus casei; Mutation; Nucleotides; Protein Binding; Protein Conformation; Pyrimidines; Quinazolines; Structure-Activity Relationship; Substrate Specificity; Thymidylate Synthase

1998
L-Glutamine ameliorates acetaldehyde-induced increase in paracellular permeability in Caco-2 cell monolayer.
    American journal of physiology. Gastrointestinal and liver physiology, 2004, Volume: 287, Issue:3

    Topics: Acetaldehyde; Actins; Adherens Junctions; Caco-2 Cells; Cell Membrane Permeability; Cytoskeletal Proteins; Dose-Response Relationship, Drug; Egtazic Acid; Endotoxins; ErbB Receptors; Glutamine; Humans; Lipopolysaccharides; Mannitol; Membrane Proteins; Occludin; Phosphorylation; Quinazolines; Tight Junctions; Tyrosine; Tyrphostins

2004
In human entrocytes, GLN transport and ASCT2 surface expression induced by short-term EGF are MAPK, PI3K, and Rho-dependent.
    Digestive diseases and sciences, 2008, Volume: 53, Issue:8

    Topics: Amino Acid Transport System ASC; Androstadienes; Blotting, Western; Caco-2 Cells; Cell Membrane; Enterocytes; Epidermal Growth Factor; ErbB Receptors; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Glutamine; Humans; Minor Histocompatibility Antigens; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Protein Transport; Protein Tyrosine Phosphatases; Quinazolines; rho GTP-Binding Proteins; RNA Interference; Signal Transduction; Sodium; Time Factors; Tyrphostins; Up-Regulation; Wortmannin

2008
Addition of amino acid moieties to lapatinib increases the anti-cancer effect via amino acid transporters.
    Biopharmaceutics & drug disposition, 2014, Volume: 35, Issue:1

    Topics: Amino Acid Transport Systems; Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Survival; Dogs; Glutamine; Humans; Lapatinib; Madin Darby Canine Kidney Cells; Protein Kinase Inhibitors; Quinazolines; Tyrosine; Valine

2014
ASCT2 (SLC1A5) is an EGFR-associated protein that can be co-targeted by cetuximab to sensitize cancer cells to ROS-induced apoptosis.
    Cancer letters, 2016, 10-10, Volume: 381, Issue:1

    Topics: Amino Acid Transport System ASC; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Carcinoma, Squamous Cell; Cell Line, Tumor; Cetuximab; Dichloroacetic Acid; Down-Regulation; Endocytosis; ErbB Receptors; Gefitinib; Glutamine; Glutathione; Head and Neck Neoplasms; Humans; Minor Histocompatibility Antigens; Oxidative Stress; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; Quinazolines; Reactive Oxygen Species; RNA Interference; Signal Transduction; Squamous Cell Carcinoma of Head and Neck; Time Factors; Transfection

2016
Discovery of Novel Potent Reversible and Irreversible Myeloperoxidase Inhibitors Using Virtual Screening Procedure.
    Journal of medicinal chemistry, 2017, 08-10, Volume: 60, Issue:15

    Topics: Benzimidazoles; Cell Line; Databases, Chemical; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Glutamic Acid; Glutamine; Guanidines; Humans; Hydrogen Peroxide; Kinetics; Lactoperoxidase; Lipoproteins, LDL; Models, Chemical; Molecular Docking Simulation; Neutrophils; Oxidation-Reduction; Peroxidase; Quinazolines; Stereoisomerism

2017